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12560

Total database: 17430
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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 149 / 252
Lisocabtagene maraleucel Approved DB16582
biotech

Lisocabtagene maraleucel is a chimeric antigen receptor (CAR) T-cell therapy, similar to [brexucabtagene autoleucel] and [axicabtagene ciloleucel].[A228493,L31588] Lisocabtagene maraleucel is a genetically modified autologous T-cell therapy that targets CD19,…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Target Protein:
B-lymphocyte antigen CD19
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Lisuride Approved DB00589
small molecule | CAS: 18016-80-3

An ergot derivative that acts as an agonist at dopamine D2 receptors (dopamine agonists). It may also act as an antagonist at dopamine D1 receptors, and as an agonist at some serotonin receptors (serotonin agonists).

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +27
Target Protein:
D(2) dopamine receptorD(3) dopamine receptorD(4) dopamine receptor +12
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Lithium carbonate Approved DB14509
small molecule | CAS: 554-13-2

Lithium has been used to treat manic episodes since the 19th century[A176642]. Though it is widely used, its mechanism of action is still unknown[FDA Label][A14585,A176642,A176651,L5843]. Lithium carbonate has a narrow therapeutic range and so careful monitor…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +26
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu ParuhThe half life of li…
Vol. DistribusiApparent volume of …
KlirensClearance is genera…
Genetik -
Lithium cation DB01356
small molecule | CAS: 7439-93-2

Lithium was used during the 19th century to treat gout. Lithium salts such as lithium carbonate (Li2CO3), lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drug…

Kategori:
Antidepressive AgentsAntimanic AgentsAntipsychotic Agents +11
Target Protein:
Glycogen synthase kinase-3 betaInositol monophosphatase 1Inositol monophosphatase 2 +1
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Lithium citrate Approved DB14507
small molecule | CAS: 919-16-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntidepressive AgentsAntimanic Agents +12
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
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Lithium hydroxide Approved DB14506
small molecule | CAS: 1310-65-2

Used for tryptophan determinations in proteins & foods.

Kategori:
Lithium CompoundsNarrow Therapeutic Index Drugs
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small molecule | CAS: 29126-50-9

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDermatologicalsDicarboxylic Acids +2
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
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Litifilimab DB18864
biotech | CAS: 2407378-48-5

Litifilimab is under investigation in clinical trial NCT05531565 (A Study to Assess the Efficacy and Safety of BIIB059 (Litifilimab) in Participants With Active Subacute Cutaneous Lupus Erythematosus (SCLE) And/or Chronic Cutaneous Lupus Erythematosus (CCLE) …

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Litoxetine DB15038
small molecule | CAS: 86811-09-8

Litoxetine is under investigation in clinical trial NCT03397771 (DBPC Trial to Evaluate the Safety, Tolerability and Efficacy of Oral Litoxetine in Subjects With Urinary Incontinence).

Target Protein:
Sodium-dependent serotonin transporter
Waktu Paruh-
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Lividomycin A DB04728
small molecule | CAS: 36441-41-5

Deskripsi belum tersedia.

Target Protein:
Telomerase reverse transcriptase
Waktu Paruh-
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Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

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Livoletide DB15188
small molecule | CAS: 1088543-62-7

Livoletide is under investigation in clinical trial NCT03790865 (Effects of Livoletide (AZP-531) on Food-related Behaviors in Patients With Prader-Willi Syndrome).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +3
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Lixadesiran DB17295
biotech | CAS: 1152798-49-6

Deskripsi belum tersedia.

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Lixisenatide Approved DB09265
biotech | CAS: 320367-13-3

Lixisenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist used in the treatment of type II diabetes mellitus (T2DM). It is sold by Sanofi-Aventis under the brand name Adlyxin in the US[L763] and Lyxumia in the EU.[L764] Adlyxin recieved FDA approval …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhFollowing the admin…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
biotech | CAS: 2461531-19-9

Lixmabegagene relduparvovec, formerly known as LYS-GM101, is a recombinant adeno-associated virus vector serotype rh.10 (AAVrh.10) carrying the human ?-galactosidase gene (GBL1). It is under development for the treatment of GM1 gangliosidosis.[L45929]

Kategori:
Adeno-associated Viral Vector Therapies
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Lixudebart DB19244
biotech | CAS: 2749515-10-2

Lixudebart, an investigational first-in-class monoclonal antibody, aims to reverse fibrosis.[L50833]

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Lixumistat DB18748
small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

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LJ-2698 DB18018
small molecule | CAS: 945457-84-1

Deskripsi belum tersedia.

Kategori:
Adenosine A3 Receptor AntagonistsNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +5
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LJP 1082 DB05446
small molecule

LJP 1082 is a Toleragen that is designed to shut down the B cells that produce antibodies to ß2 GP1. LJP 1082 is undergoing trial for for the treatment of stroke, deep-vein thrombosis and other conditions associated with antibody-mediated thrombosis. Antibody…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsCarbohydrates +7
Target Protein:
Beta-2-glycoprotein 1
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LJP-538 DB17810
biotech

Deskripsi belum tersedia.

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LJP-539 DB17811
biotech

Deskripsi belum tersedia.

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LL-37 DB16532
biotech

LL-37 is a human cathelicidin that inhibits viral replication and while also playing a role in host defense against infection.

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LLL-3348 DB05771
biotech

The botanical drug product LLL-3348 is a once-daily oral formulation for treatment of chronic stable plaque type psoriasis.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Interleukin-10
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LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

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LM-609 DB05787
biotech

LM-609 (Vitaxin) is an artificial antibody that targets a protein on the surface of newly forming blood vessels, as well as on certain tumors. In addition to cancer, the protein has been implicated in bone destruction in rheumatoid arthritis and the inflammat…

Target Protein:
Integrin beta-3
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LMB-100 DB18591
biotech | CAS: 1841500-93-3

LMB-100 is a is an antibody-toxin conjugate with an antimesothelin Fab linked to a 24-kilodalton portion of Pseudomonas exotoxin A with mutations that decrease immunogenicity.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Genetik -
biotech

LNP-nCoVsaRNA is a purified, synthetic mRNA vaccine candidate encoding the S glycoprotein of SARS-CoV-2, which is used primarily by the virus to attach to and invade human cells. The vaccine was developed in and tested by the Medical Research Council Clinical…

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LNS-8801 DB18091
small molecule | CAS: 881639-98-1

Deskripsi belum tersedia.

Target Protein:
G-protein coupled estrogen receptor 1
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Lobaplatin DB13049
small molecule | CAS: 135558-11-1

Lobaplatin has been used in trials studying the treatment of Breast Cancer, Hepatocellular Carcinoma, and Lobaplatin and Gemcitabine in Combination, Second-line Treatments on Advanced Osteosarcoma.

Kategori:
CycloparaffinsOrganometallic Compounds
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Lobeline DB05137
small molecule | CAS: 90-69-7

An alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has been proposed for a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation. …

Kategori:
AlkaloidsAutonomic AgentsCholinergic Agents +7
Target Protein:
Synaptic vesicular amine transporterNeuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-9 +1
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Lobster Approved DB10541
biotech

Lobster allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Lobucavir DB12531
small molecule | CAS: 127759-89-1

Lobucavir has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +10
Target Protein:
Gag-Pol polyprotein
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small molecule | CAS: 398507-55-6

Lodenafil carbonate has been used in trials studying the treatment of Coronaropathy and Erectile Dysfunction.

Kategori:
AlkaliesAnionsCarbon Compounds, Inorganic +3
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Lodoxamide Approved DB06794
small molecule | CAS: 53882-12-5

Lodoxamide is a mast-cell stabilizer for topical administration into the eye. Mast-cell stabilizers, first one approved being cromolyn sodium, are used in treatment of ocular hypersensitivity reactions such as vernal conjunctivitis. These conditions often req…

Kategori:
Acids, AldehydicAlcoholsAmino Acids +13
Waktu ParuhElimination half-li…
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Lofepramine DB13411
small molecule | CAS: 23047-25-8

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
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Lomefloxacin Approved DB00978
small molecule | CAS: 98079-51-7

Lomefloxacin is a fluoroquinolone antibiotic, used to treat bacterial infections including bronchitis and urinary tract infections (UTIs). Additionally, it has been employed for the prophylaxis of UTIs prior to surgery as well.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA topoisomerase 2-betaDNA topoisomerase 4 subunit A +1
Waktu Paruh8 hours
Vol. Distribusi-
Klirens* 271 mL/min/1.73 m…
Genetik -
Lomerizine DB14065
small molecule | CAS: 101477-55-8

Lomerizine is a diphenylmethylpiperazine calcium channel blocker[A245378, A245383] with relatively selective central nervous system (CNS) effects.[A245383] This drug is used to prophylactically treat migraines[A245368, A245373] and is also being investigated…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Sodium channel protein type 5 subunit alphaVoltage-dependent N-type calcium channel subunit alpha-1BATP-dependent translocase ABCB1
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Lomibuvir DB11954
small molecule | CAS: 1026785-55-6

Lomibuvir has been used in trials studying the treatment of Chronic Hepatitis C Virus and Chronic Hepatitis C Virus Infection.

Kategori:
AlcoholsCyclohexanesCycloparaffins +4
Target Protein:
Genome polyprotein
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Lomifylline Approved DB18002
small molecule | CAS: 10226-54-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsDrugs for Obstructive Airway DiseasesHeterocyclic Compounds, Fused-Ring +3
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Lomitapide Approved DB08827
small molecule | CAS: 182431-12-5

Lomitapide is a microsomal triglyceride transfer protein (MTP) inhibitor used in homozygous familial hypercholesterolemia (HoFH) patients. It is marketed under the name Juxtapid (R).

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +17
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu ParuhLomitapide half-lif…
Vol. DistribusiThe steady state vo…
Klirens-
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Lomvastomig DB19060
biotech | CAS: 2648840-52-0

Lomvastomig is under investigation in clinical trial NCT04785820 (A Study of Lomvastomig (RO7121661) and Tobemstomig (RO7247669) Compared With Nivolumab in Participants With Advanced or Metastatic Squamous Cell Carcinoma of the Esophagus).

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Lonafarnib Approved DB06448
small molecule | CAS: 193275-84-2

Hutchinson-Gilford progeria syndrome (HGPS) is a rare autosomal dominant disorder estimated to affect approximately one in 20 million individuals resulting in adverse symptoms associated with premature ageing: skeletal dysplasia, joint contractures, atheroscl…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBenzocycloheptenes +30
Target Protein:
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta
Waktu ParuhLonafarnib has a me…
Vol. DistribusiIn healthy patients…
Klirens-
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Lonapegsomatropin Approved DB16220
biotech | CAS: 1934255-39-6

Lonapegsomatropin, also known as TransCon hGH or ACP 001, is a methoxypegylated prodrug of human growth hormone ([somatropin]) indicated for the treatment of children 1 year and older, weighing at least 11.5 kg, with growth failure due to insufficient growth …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesCytochrome P-450 CYP1A2 Inducers +18
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhThe half life of lo…
Vol. DistribusiLonapegsomatropin-t…
KlirensIn pediatric patien…
Genetik -
Lonaprisan DB16221
small molecule | CAS: 211254-73-8

Lonaprisan is under investigation in clinical trial NCT00555919 (ZK 230211 in Postmenopausal Woman With Metastatic Breast Cancer).

Kategori:
EstranesFused-Ring CompoundsHydrocarbons, Fluorinated +2
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor
Waktu Paruh-
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Lonazolac DB13432
small molecule | CAS: 53808-88-1

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +13
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Loncastuximab tesirine Approved DB16222
biotech | CAS: 1879918-31-6

Relapsed and refractory B-cell acute lymphoblastic leukemia (B-ALL) are a therapeutic challenge for patients who have undergone prior systemic therapies with limited success.[A234439] Prognosis is poor and more effective therapies are needed to treat relapsed…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe half-life of lo…
Vol. DistribusiIn clinical studies…
KlirensIn pharmacokinetic …
Genetik -
Londamocitinib DB19190
small molecule | CAS: 2241039-81-4

Londamocitinib is under investigation in clinical trial NCT06020014 (Phase 2a Study to Assess the Efficacy and Safety of AZD4604 in Adult Patients With Moderate-to-severe Asthma Uncontrolled on Medium-high Dose ICS-LABA).

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Lonidamine DB06266
small molecule | CAS: 50264-69-2

Lonidamine (LND) is a drug that interferes with energy metabolism of cancer cells, principally inhibiting aerobic glycolytic activity, by its effect on mitochondrially-bound hexokinase (HK). In such way LND could impair energy-requiring processes, as recovery…

Kategori:
Adrenal Cortex HormonesAnti-Infective AgentsAntineoplastic Agents +11
Target Protein:
Cystic fibrosis transmembrane conductance regulatorHexokinase-1
Waktu Paruh-
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Lonigutamab DB18940
biotech | CAS: 2362015-67-4

Lonigutamab is under investigation in clinical trial NCT05683496 (Efficacy and Safety of Lonigutamab in Subjects With Thyroid Eye Disease (TED)).

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Loperamide Approved DB00836
small molecule | CAS: 53179-11-6

Loperamide is an anti-diarrheal agent that is available as an over-the-counter product for treating diarrhea.[L42785] The drug was first synthesized in 1969 and used medically in 1976.[A251610] It is a highly lipophilic synthetic phenylpiperidine opioid that …

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAntiarrhythmic agents +20
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe apparent elimin…
Vol. DistribusiLoperamide has a la…
Klirens-
Genetik -
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