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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 148 / 236
Methyltestosterone Approved DB06710
small molecule | CAS: 58-18-4

A synthetic anabolic steroid used for treating men with testosterone deficiency or similar androgen replacement therapies. Also, has antineoplastic properties and so has been used secondarily in women with advanced breast cancer. Methyltestosterone is a sched…

Kategori:
3-Oxoandrosten (4) DerivativesAnabolic AgentsAndrogens +20
Target Protein:
Androgen receptorEstrogen receptor
Waktu Paruh6-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7060-82-4

Deskripsi belum tersedia.

Kategori:
Oxidation-Reduction ActivityOxidation-Reduction AgentSerotonergic Drugs Shown to Increase Risk of Serotonin Syndrome
Target Protein:
AcetylcholinesteraseTranscriptional regulator
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 59322-44-0

Deskripsi belum tersedia.

Target Protein:
Trans-sialidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Methyprylon Approved DB01107
small molecule | CAS: 125-64-4

Methyprylon is a sedative of the piperidinedione derivative family that was previously used for the treatment of insomnia. However, with the introduction of newer drugs with fewer side effects, such as benzodiazepines, the clinical use of methyprylon is now l…

Kategori:
Central Nervous System DepressantsHypnotics and SedativesNervous System +3
Target Protein:
GABA(A) ReceptorGamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh6-16 hours
Vol. Distribusi-
Klirens-
Genetik -
Methysergide Approved DB00247
small molecule | CAS: 361-37-5

An ergot derivative that is a congener of lysergic acid diethylamide. It antagonizes the effects of serotonin in blood vessels and gastrointestinal smooth muscle, but has few of the properties of other ergot alkaloids. Methysergide is used prophylactically i…

Kategori:
Agents that produce hypertensionAlkaloidsAnalgesics +20
Target Protein:
5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C5-hydroxytryptamine receptor 2A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metiamide DB08805
small molecule | CAS: 34839-70-8

Metiamide is an H-2 receptor antagonist derived from burimamide. It was an intermediate product on the path to developing cimetidine.

Kategori:
Acid ReducersAmidesAnti-Ulcer Agents +8
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meticillin Approved DB01603
small molecule | CAS: 61-32-5

One of the penicillins which is resistant to penicillinase but susceptible to a penicillin-binding protein. It is inactivated by gastric acid so administered by injection.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
MecA PBP2' (penicillin binding protein 2')Penicillin-binding protein 2aPenicillin-binding protein 1b +3
Waktu Paruh25-60 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meticrane Approved DB13284
small molecule | CAS: 1084-65-7

Meticrane is a diuretic medication. It has been marketed in Japan under the trade name Arresten and is used to lower blood pressure [L5647].

Kategori:
DiureticsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metipranolol Approved DB01214
small molecule | CAS: 22664-55-7

A beta-adrenergic antagonist effective for both beta-1 and beta-2 receptors. It is used as an antiarrhythmic, antihypertensive, and antiglaucoma agent.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +23
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metizoline DB13614
small molecule | CAS: 17692-22-7

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoclopramide Approved DB01233
small molecule | CAS: 364-62-5

Diabetic gastroparesis is a condition that causes frequent nausea and vomiting, which has a negative impact on quality of life and poses a significant burden on the healthcare system.[A184934] Metoclopramide is a dopamine antagonist used to treat nausea and v…

Kategori:
Acids, CarbocyclicAgents Causing Muscle ToxicityAlimentary Tract and Metabolism +35
Target Protein:
5-hydroxytryptamine receptor 45-hydroxytryptamine receptor 3AMuscarinic acetylcholine receptor M1 +1
Gen Terkait:
KCNH2 ADRA1D CYP2D6 +4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
KlirensThe renal clearance…
Genetik 7 Varian
Metocurine Approved DB01336
small molecule | CAS: 5152-30-7

Dimethyltubocurarinium (INN) or metocurine (USAN), also known as dimethyltubocurarine, is a non-depolarizing muscle relaxant. Patients on chronic anticonvulsant drugs are relatively resistant to metocurine. [A2393]

Kategori:
Agents producing tachycardiaAlkaloidsAmines +18
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metocurine iodide Approved DB00416
small molecule | CAS: 7601-55-0

Metocurine iodide is a benzylisoquinolinium competitive nondepolarizing neuromuscular blocking agent. It is used as an anesthesia adjunct to induce skeletal muscle relaxation and to reduce the intensity of muscle contractions in convulsive therapy Metocurine …

Kategori:
AlkaloidsAminesAnticholinergic Agents +12
Target Protein:
Neuronal acetylcholine receptor subunit alpha-4Neuronal acetylcholine receptor subunit beta-2Neuronal acetylcholine receptor subunit alpha-2
Waktu Paruh3 to 4 hours
Vol. Distribusi-
Klirens-
Genetik -
Metolazone Approved DB00524
small molecule | CAS: 17560-51-9

A quinazoline-sulfonamide that is considered a thiazide-like diuretic which is long-acting so useful in chronic renal failure. It also tends to lower blood pressure and increase potassium loss.

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +21
Target Protein:
Solute carrier family 12 member 3
Waktu ParuhApproximately 14 ho…
Vol. Distribusi-
Klirens-
Genetik -
Metopimazine DB13591
small molecule | CAS: 14008-44-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAntiemetics and Antinauseants +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprine DB04655
small molecule | CAS: 7761-45-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsFolic Acid Antagonists +1
Target Protein:
Peptide deformylase, mitochondrialHistamine N-methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metoprolol Approved DB00264
small molecule | CAS: 51384-51-1

Metoprolol is a selective beta-1 blocker commonly employed as the succinate and tartrate derivatives depending if the formulation is designed to be of immediate release or extended release.[A175159, L5530] The possibility of the generation of these formulatio…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-1 Receptor Antagonists +29
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptorBeta adrenergic receptor
Gen Terkait:
ADRB1 CYP2D6 ADRB1
Waktu ParuhThe immediate relea…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik 3 Varian
Metoserpate DB11530
small molecule | CAS: 1178-28-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingIndole Alkaloids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metribolone DB02998
small molecule | CAS: 965-93-5

A synthetic non-aromatizable androgen and anabolic steroid. It binds strongly to the androgen receptor and has therefore also been used as an affinity label for this receptor in the prostate and in prostatic tumors.

Kategori:
EstranesEstrenesFused-Ring Compounds +1
Target Protein:
Progesterone receptorAndrogen receptorNuclear receptor coactivator 2 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrifonate DB11473
small molecule | CAS: 52-68-6

Metrifonate or trichlorfon is an irreversible organophosphate acetylcholinesterase inhibitor. It is a prodrug which is activated non-enzymatically into 2,2-dichlorovinyl dimethyl phosphate.

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizamide DB01578
small molecule | CAS: 31112-62-6

Metrizamide is a solute for density gradient centrifugation offering higher maximum solution density without the problems of increased viscosity. It is also used as a resorbable, non-ionic contrast medium.

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metrizoic acid Approved DB09346
small molecule | CAS: 1949-45-7

Metrizoic acid is a molecule used as a contrast medium. It present a higher risk of allergic reactions due to its high osmolality. Its approval has been discontinued by the FDA. One study in 1976 demonstrated that metrizoic acid, when used for cardiac angiog…

Kategori:
Acids, CarbocyclicBenzene DerivativesBenzoates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metronidazole Approved DB00916
small molecule | CAS: 443-48-1

Metronidazole is a commonly used antibiotic, belonging to the nitroimidazole class of antibiotics.[L3754] It is frequently used to treat gastrointestinal infections as well as trichomoniasis and giardiasis, and amebiasis which are parasitic infections.[A18103…

Kategori:
Agents that reduce seizure thresholdAlimentary Tract and MetabolismAnti-Bacterial Agents +38
Target Protein:
Oxygen-insensitive NADPH nitroreductaseAnaerobic bacterial DNAProtozoal DNA
Waktu ParuhThe elimination hal…
Vol. DistribusiMetronidazole is wi…
KlirensDose adjustments ma…
Genetik -
small molecule | CAS: 13182-89-3

Deskripsi belum tersedia.

Kategori:
ImidazolesNitro CompoundsNitroimidazoles
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Metyrosine Approved DB00765
small molecule | CAS: 672-87-7

An inhibitor of the enzyme tyrosine 3-monooxygenase, and consequently of the synthesis of catecholamines. It is used to control the symptoms of excessive sympathetic stimulation in patients with pheochromocytoma. (Martindale, The Extra Pharmacopoeia, 30th ed)

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +6
Target Protein:
Tyrosine 3-monooxygenase
Waktu Paruh3.4 to 3.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Mevalonic acid DB03518
small molecule | CAS: 150-97-0

Deskripsi belum tersedia.

Kategori:
Hydroxy Acids
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevastatin DB06693
small molecule | CAS: 73573-88-3

Mevastatin or compactin is a cholesterol-lowering agent isolated from <i>Penicillium citinium</i>. It was the first discovered agent belonging to the class of cholesterol-lowering medications known as statins. During a search for antibiotic compounds produced…

Kategori:
Agents Causing Muscle ToxicityAnti-Infective AgentsAnticholesteremic Agents +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevidalen DB19034
small molecule | CAS: 1638667-79-4

Mevidalen is under investigation in clinical trial NCT03305809 (A Study of LY3154207 in Participants With Dementia Due to Lewy Body Dementia (LBD) Associated With Idiopathic Parkinson's Disease (PD) or Dementia With Lewy Bodies (DLB)).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75225-51-3

Deskripsi belum tersedia.

Kategori:
Naphthalenes
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mevonlerbart DB19416
biotech | CAS: 2453195-99-6

Mevonlerbart is under investigation in clinical trial NCT06602726 (A Study to Demonstrate How Well REGN1908-1909 Works in Reducing Ocular Allergy Signs and Symptoms in Adult Participants With Cat Allergy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mexiletine Approved DB00379
small molecule | CAS: 31828-71-4

Antiarrhythmic agent pharmacologically similar to lidocaine. It may have some anticonvulsant properties.

Kategori:
AminesAntiarrhythmic agentsAntiarrhythmics, Class I +20
Target Protein:
Sodium channel protein type 5 subunit alphaAryl hydrocarbon receptor
Waktu Paruh10-12 hours
Vol. Distribusi* 5 to 7 L/lg
Klirens-
Genetik -
Mezagitamab DB16370
biotech | CAS: 2227490-52-8

Mezagitamab is under investigation in clinical trial NCT04278924 (Study to Evaluate Safety, Tolerability, and Efficacy of TAK-079 in Participants With Persistent/chronic Primary Immune Thrombocytopenia).

Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezigdomide DB17584
small molecule | CAS: 2259648-80-9

Mezigdomide is under investigation in clinical trial NCT05372354 (A Study to Evaluate Safety, Drug Levels and Effectiveness of CC-92480 (BMS-986348) in Combination With Other Treatments in Participants With Relapsed or Refractory Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mezlocillin Approved DB00948
small molecule | CAS: 51481-65-3

Semisynthetic ampicillin-derived acylureido penicillin. It has been proposed for infections with certain anaerobes and may be useful in inner ear, bile, and CNS infections.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 1APeptidoglycan synthase FtsIPenicillin-binding protein 3 +1
Waktu Paruh1.3 to 4.4 hours
Vol. Distribusi-
Klirens-
Genetik -
MGB-BP-3 DB12892
small molecule | CAS: 1000277-08-6

Mgb Bp 3 is under investigation in clinical trial NCT02518607 (Safety, Blood Levels and Effects of MGB-BP-3).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGD-024 DB17265
biotech

MGD-024 is an anti-CD123/anti-CD3 bispecific DART molecule.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MGN-4893 DB17338
biotech

MGN-4893 is an inhibitor of microRNA-451. In February 2011, it was granted FDA orphan designation for the treatment of polycythemia vera.[L47356]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mianserin Approved DB06148
small molecule | CAS: 24219-97-4

A tetracyclic compound with antidepressant effects. Mianserin was previously available internationally, however in most markets it has been phased out in favour of [mirtazapine].

Kategori:
Adrenergic AgentsAgents that produce hypertensionAntidepressive Agents +29
Target Protein:
Alpha-2A adrenergic receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2C +17
Waktu Paruh10-17 hours
Vol. Distribusi-
Klirens-
Genetik -
Mibampator DB12717
small molecule | CAS: 375345-95-2

Mibampator has been used in trials studying the treatment of Alzheimer's Disease.

Kategori:
AmidesBenzene DerivativesSulfones +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibavademab DB16673
biotech | CAS: 2305770-44-7

Mibavademab is under investigation in clinical trial NCT04159415 (Study of REGN4461, a Leptin Receptor Agonist Antibody, in Patients With Generalized Lipodystrophy).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibenratide DB15195
small molecule | CAS: 1239011-83-6

Mibenratide is under investigation in clinical trial NCT01798745 (A Study to Assess the Pharmacokinetics and Pharmacodynamics of JNJ-54452840 in Participants With Heart Failure and Anti-beta1-adrenergic Receptor Autoantibodies).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mibolerone DB11429
small molecule | CAS: 3704-09-4

Mibolerone is a potent anabolic steroid which is both higher affinity and more selective for the androgen receptor than metribolone.

Kategori:
EstranesEstrenesFused-Ring Compounds +7
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Miconazole Approved DB01110
small molecule | CAS: 22916-47-8

Miconazole is a broad-spectrum azole antifungal with some activity against Gram-positive bacteria as well.[A203636] It is widely used to treat mucosal yeast infections, including both oral and vaginal infections; although intravenous miconazole is no longer a…

Kategori:
14-alpha Demethylase InhibitorsAnti-Infective AgentsAntifungal Agents +41
Target Protein:
Lanosterol 14-alpha demethylaseNitric oxide synthase 3Nitric oxide synthase, inducible +5
Waktu ParuhMiconazole has a te…
Vol. DistribusiA 1200 mg miconazol…
Klirens-
Genetik -
Micronomicin Approved DB13274
small molecule | CAS: 52093-21-7

Micronomicin is an aminoglycoside antibiotic which is marketed in Japan, and sold under the brand names Sagamicin and Luxomicina.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Midazolam Approved DB00683
small molecule | CAS: 59467-70-8

Midazolam is a short-acting hypnotic-sedative drug with anxiolytic, muscle relaxant, anticonvulsant, sedative, hypnotic, and amnesic properties.[A173842] It belongs to a class of drugs called _benzodiazepines_. This drug is unique from others in this class du…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnti-Anxiety Agents +27
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site +1
Waktu Paruh**Intravenous**: …
Vol. DistribusiFemale gender, old …
Klirens**Intramuscular** …
Genetik -
Midecamycin DB13456
small molecule | CAS: 35457-80-8

Midecamycin is a naturally occurring 16-membered macrolide[A33072] that fits under the category of acetoxy-substituted macrolide antibiotics. In this molecule, an acetoxy group is substituted on the position 9 of the 16-member ring and on position 4 of the te…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +12
Waktu ParuhThe half-life of mi…
Vol. DistribusiThe reported appare…
KlirensMidecamycin present…
Genetik -
Midodrine Approved DB00211
small molecule | CAS: 42794-76-3

An ethanolamine derivative that is an adrenergic alpha agonist. It is used as a vasoconstrictor agent in the treatment of hypotension.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +19
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor
Waktu ParuhThe metabolites dis…
Vol. Distribusi-
Klirens* Renal cl=385 mL/m…
Genetik -
Midostaurin Approved DB06595
small molecule | CAS: 120685-11-2

Midostaurin (as Rydapt) is a multitarget kinase inhibitor for the treatment for adult patients with newly diagnosed acute myeloid leukemia (AML) who have a specific genetic mutation called FLT3. It was initially characterized as a potential broad-spectrum ant…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +53
Target Protein:
Protein kinase C gamma typeProtein kinase C alpha typeVascular endothelial growth factor receptor 2 +4
Waktu ParuhElimination half li…
Vol. DistribusiThe Vd of midostaur…
KlirensThe clearance value…
Genetik -
Mifamurtide Approved DB13615
small molecule | CAS: 83461-56-7

Mifamurtide is an immunomodulator with antitumor activity via activation of macrophages and monocytes. Also called L-MTP-PE, mifamurtide may be a liposomal form of of the active ingredient MTP-PE, which is a synthetic, less pyrogenic, and longer-acting deriva…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAmino Sugars +15
Target Protein:
Toll-like receptor 4Nucleotide-binding oligomerization domain-containing protein 2
Waktu ParuhFollowing intraveno…
Vol. DistribusiThe mean volume of …
KlirensThe clearance from …
Genetik -
Mifepristone Approved DB00834
small molecule | CAS: 84371-65-3

Mifepristone is a progestational and glucocorticoid hormone antagonist. Its inhibition of progesterone induces bleeding during the luteal phase and in early pregnancy by releasing endogenous prostaglandins from the endometrium or decidua. As a glucocorticoid …

Kategori:
Abortifacient AgentsAbortifacient Agents, SteroidalAdrenal Cortex Hormones +49
Target Protein:
Progesterone receptorGlucocorticoid receptorProstate-specific antigen +1
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7351–7400 dari 11778
Sebelumnya Halaman 148 / 236 Berikutnya