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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Halaman 148 / 252
Lidorestat DB07063
small molecule | CAS: 245116-90-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1401812-88-1

Lifastuzumab vedotin is under investigation in clinical trial NCT01363947 (Safety and Pharmacokinetics of Escalating Doses of DNIB0600A in Participants With Non-Small Cell Lung Cancer (NSCLC) and Platinum Resistant Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifileucel Approved DB17107
biotech | CAS: 2306267-74-1

Lifileucel is a tumour-derived autologous T cell immunotherapy composed of a suspension of tumour-derived T cells from the patient [L50171] which undergo isolation, ex vivo expansion, and activation[A263341] Lifileucel was granted accelerated approval by the …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifirafenib DB14773
small molecule | CAS: 1446090-79-4

Lifirafenib is under investigation in clinical trial NCT03641586 (The Study of BGB-283 in Chinese Subjects With Local Advanced or Metastatic Malignant Solid Tumor).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase B-raf
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lifitegrast Approved DB11611
small molecule | CAS: 1025967-78-5

Lifitegrast is a FDA approved drug for the treatment of keratoconjunctivitis sicca (dry eye syndrome). It is a tetrahydroisoquinoline derivative and lymphocyte function-associated antigen-1 ( LFA-1) antagonist that was discovered through the rational design p…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +18
Target Protein:
Intercellular adhesion molecule 1Integrin alpha-L
Waktu ParuhNot possible to cal…
Vol. Distribusi-
KlirensNot possible to cal…
Genetik -
Ligandrol DB13934
small molecule | CAS: 1165910-22-4

Ligandrol is an investigational selective androgen receptor modulator (SARM) for treatment of conditions such as muscle wasting and osteoporosis.

Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ligelizumab DB11856
biotech | CAS: 1322627-61-1

Ligelizumab is a humanized IgG1k monoclonal antibody targeted against immunoglobulin E (IgE). Similar in mechanism to [omalizumab], another IgE-directed monoclonal antibody, ligelizumab has a distinct binding epitope as compared to its peer (with a small degr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Immunoglobulin heavy constant epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Light green SF yellowish Approved DB11183
small molecule | CAS: 5141-20-8

Light green SF yellowish is a green triarylmethane dye that is used in the preparation of the staining solution which is widely used as a counterstain. It is used in histological applications and other labratory settings, and usually exists as a disodium salt…

Kategori:
AminesArylsulfonatesArylsulfonic Acids +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Light mineral oil Approved DB11579
small molecule | CAS: 92062-35-6

Deskripsi belum tersedia.

Kategori:
Basic Ointments and Protectants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ligufalimab DB17542
biotech | CAS: 2428381-55-7

Ligufalimab is a humanized immunoglobulin G4 (IgG4) monoclonal antibody targeting leukocyte surface antigen CD47. It is under investigation in clinical trial NCT04900350 (A Trial of AK117 (Anti-cd47) in Patients With Myelodysplastic Syndrome).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ligustrazine DB19074
small molecule | CAS: 1124-11-4

Ligustrazine is under investigation in clinical trial NCT05942352 (Clinical Study of Ligustrazine in Treating Alcohol Addiction).

Kategori:
Antiplatelet agentsCardiovascular AgentsVasodilating Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lilotomab DB19076
biotech | CAS: 1453362-55-4

Lilotomab is under investigation in clinical trial NCT01796171 (A Phase 1/2 Study of Betalutin for Treatment of Relapsed Non-hodgkin Lymphoma).

Waktu Paruh-
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Lima bean Approved DB10540
biotech

Lima bean allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Limaprost DB09211
small molecule | CAS: 74397-12-9

Limaprost (as Limaprost alfadex; CAS number 88852-12-4) is an oral prostaglandin E1 analog. Prostaglandins act on a variety of cells such as vascular smooth muscle cells causing constriction or dilation, on platelets causing aggregation or disaggregation and …

Kategori:
AnticoagulantsAutacoidsBiological Factors +11
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype +1
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensMean total clearanc…
Genetik -
Lime (citrus) Approved DB10635
biotech

Lime (citrus) allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 138-86-3

Limonene, (+/-)- is under investigation in clinical trial NCT05525260 (Limonene for Pulmonary Nodule Chemoprevention).

Kategori:
Cyclohexane MonoterpenesCyclohexanesCyclohexenes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linaclotide Approved DB08890
small molecule | CAS: 851199-59-2

Linaclotide is a synthetic 14-amino acid cyclic peptide [A260271] and first-in-class guanylate cyclase-C (G-CC) agonist.[A260271, L47211] Linaclotide is structurally related to human guanylin and uroguanylin, paracrine peptide hormones that are endogenous act…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +7
Target Protein:
Guanylyl cyclase C
Waktu ParuhThere is no availab…
Vol. DistribusiGiven that linaclot…
KlirensNo information is a…
Genetik -
Linafexor DB18031
small molecule | CAS: 2499656-04-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linagliptin Approved DB08882
small molecule | CAS: 668270-12-0

Linagliptin is a DPP-4 inhibitor developed by Boehringer Ingelheim for the treatment of type II diabetes [L9557]. Linagliptin differs from other DPP-4 inhibitors in that it has a non-linear pharmacokinetic profile, is not primarily eliminated by the renal sys…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +24
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe terminal half l…
Vol. DistribusiA single intravenou…
KlirensTotal clearance of …
Genetik -
Lincomycin Approved DB01627
small molecule | CAS: 154-21-2

Lincomycin is a lincosamide antibiotic first isolated from the soil bacterium _Streptomyces lincolnensis_ in Lincoln, Nebraska.[A190621] Clinical use of lincomycin has largely been superseded by its semisynthetic derivative [clindamycin] due to its higher eff…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
23S ribosomal RNA
Waktu ParuhLincomycin has a bi…
Vol. DistribusiLincomycin administ…
KlirensLincomycin administ…
Genetik -
Lindane Approved DB00431
small molecule | CAS: 58-89-9

An organochlorine insecticide that has been used as a pediculicide and a scabicide. Lindane has been banned in California, United Kingdom, Australia, and many western countries due to concerns about neurotoxicity and adverse effects on the environment. In Can…

Kategori:
Agents that reduce seizure thresholdAgrochemicalsAntiparasitic Products, Insecticides and Repellents +9
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-1Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2 +7
Waktu Paruh18 hours
Vol. Distribusi-
Klirens-
Genetik -
Linerixibat DB11729
small molecule | CAS: 1345982-69-5

GSK2330672 has been investigated for the treatment of Diabetes Mellitus, Type 2.

Kategori:
AminesAzepinesSulfur Compounds +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linezolid Approved DB00601
small molecule | CAS: 165800-03-3

Linezolid is a synthetic antibiotic which is used for the treatment of infections caused by aerobic Gram-positive bacteria. Its effects are bacteriostatic against both enterococci and staphylococci and bactericidal against most isolates of streptococci.[L3296…

Kategori:
AcetamidesAcetatesAcids, Acyclic +22
Target Protein:
23S ribosomal RNA
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady-state, th…
KlirensTotal clearance of …
Genetik -
Linifanib DB06080
small molecule | CAS: 796967-16-3

Linifanib (ABT-869) is a small molecule vascular endothelial growth factor (VEGF) receptor-based kinase inhibitor that is designed to suppress tumor growth by preventing the formation of new blood vessels that supply the tumor with oxygen and nutrients and by…

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Vascular endothelial growth factor receptor 3Receptor-type tyrosine-protein kinase FLT3Vascular endothelial growth factor receptor 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linopirdine DB13806
small molecule | CAS: 105431-72-9

Deskripsi belum tersedia.

Kategori:
Cardiovascular AgentsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +8
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linopristin DB19296
small molecule | CAS: 325965-23-9

Linopristin is an antibiotic of the streptogramin B class. It is one part of the combination product NXL 103, along with [Virginiamycin M1]. The combination product was under investigation in clinical trials NCT00653172 and NCT00949130 for treatment of variou…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linperlisib DB17235
small molecule | CAS: 1702816-75-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linseed oil DB11357
biotech | CAS: 66071-03-2

Linseed oil is a rich source of ?-Linolenic acid extracted from the dried, ripened seeds of the flax plant *Linum usitatissimum*. Other fatty acids contained in linseed oil include palmitic acid, stearic acid, oleic acid and linolenic acid. Linseed oil is par…

Kategori:
Biological ProductsComplex MixturesFats +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linsitinib DB06075
small molecule | CAS: 867160-71-2

An orally bioavailable small molecule inhibitor of the insulin-like growth factor 1 receptor (IGF-1R) with potential antineoplastic activity. IGF-1R inhibitor OSI-906 selectively inhibits IGF-1R, which may result in the inhibition of tumor cell proliferation …

Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lintitript DB04867
small molecule | CAS: 136381-85-6

Lintitript is a new, highly specific and potent CCK-A receptor antagonist.

Kategori:
Heterocyclic Compounds, Fused-RingHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lintuzumab DB14877
biotech | CAS: 166089-32-3

Lintuzumab is under investigation in clinical trial NCT00016159 (Chemotherapy Plus Monoclonal Antibody in Treating Patients With Acute Promyelocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2209911-94-2

Lintuzumab actinium Ac-225 is under investigation in clinical trial NCT00672165 (Targeted Atomic Nano-Generators (Actinium-225-Labeled Humanized Anti-CD33 Monoclonal Antibody HuM195) in Patients With Advanced Myeloid Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Linzagolix Approved DB17083
small molecule | CAS: 935283-04-8

Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other…

Kategori:
Anti-Gonadotropin-Releasing HormonesBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Inhibitors +18
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe half-life of li…
Vol. DistribusiAfter seven days of…
KlirensThe geometric mean …
Genetik -
Liothyronine Approved DB00279
small molecule | CAS: 6893-02-3

Liothyronine is a thyroidal hormone T3 which is normally produced by the thyroid gland in a ratio 4:1 when compared with T4: T3. Liothyronine is the active form of thyroxine which is composed in a basic chemical structure by a tyrosine with bound iodine.[T457…

Kategori:
Agents used to treat hypothyroidismDrugs that are Mainly Renally ExcretedHormones +12
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaProliferating cell nuclear antigen
Waktu ParuhThe half-life of li…
Vol. DistribusiThe reported volume…
KlirensThere are no report…
Genetik -
small molecule | CAS: 20196-64-9

Liothyronine I-131 has been used in trials studying the treatment of Tricuspid Atresia and Heart Defects, Congenital.

Kategori:
Thyroxine-binding globulin substrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liotrix Approved DB01583
small molecule | CAS: 8065-29-0

Liotrix is a synthetically derived thyroid hormone replacement preparation. It consists of levothyroxine sodium (thyroxine, T4) and liothyronine sodium (triiodothyronine, T3) in a 4 to 1 ratio by weight. Liotrix was developed when it was believed that serum l…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +19
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipegfilgrastim Approved DB13200
biotech | CAS: 1117844-87-7

Lipegfilgrastim, previously known as XM22, is a pegylated, recombinant granulocyte colony-stimulating factor (G-CSF) that was synthetized using a highly site-specific glycoPEGylation technology [A32665]. It is used as an alternate to [DB00019] for prophylacti…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +17
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe average termina…
Vol. DistribusiLipegfilgrastim has…
KlirensIn a phase 1, multi…
Genetik -
small molecule

Liposome-encapsulated form of prostaglandin E1 (Liprostin) is known to be a potent vasodilator and platelet inhibitor as well as an anti-inflammatory and anti-thrombotic agent. The liposomal formulation of PGE-1 changes the drug’s dynamics and improve its the…

Target Protein:
Platelet glycoprotein Ib alpha chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Carboxylic Ester HydrolasesEnzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 118731-97-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Liquidambar styraciflua pollen is the pollen of the Liquidambar styraciflua plant. Liquidambar styraciflua pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lirafugratinib DB18300
small molecule | CAS: 2549174-42-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lirilumab DB11754
biotech | CAS: 1000676-41-4

Lirilumab has been used in trials studying the treatment of Leukemia, CANCER,NOS, Multiple Myeloma, Lymphocytic Leukemia, and Acute Myeloid Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisaftoclax DB18054
small molecule | CAS: 2180923-05-9

Lisaftoclax is a novel, orally active, selective and potent BCL-2 inhibitor

Kategori:
Benzene DerivativesNitro Compounds
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisavanbulin DB15224
small molecule | CAS: 1263384-43-5

Lisavanbulin is under investigation in clinical trial NCT02895360 (Phase 1/2a Study of BAL101553 as 48-hour Infusions in Patients With Advanced Solid Tumors or Recurrent Glioblastoma).

Kategori:
Antineoplastic AgentsAntineoplastic Agents, ImmunologicalHeterocyclic Compounds, Fused-Ring +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Lisinopril Approved DB00722
small molecule | CAS: 76547-98-3

Lisinopril is an angiotensin converting enzyme inhibitor (ACEI) used to treat hypertension, heart failure, and myocardial infarction.[L8384,L8387,L8390] Lisinopril and [captopril] are the only ACEIs that are not prodrugs.[A184853] It functions by inhibition o…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +20
Target Protein:
Angiotensin-converting enzymeRenin
Waktu ParuhLisinopril has an e…
Vol. DistribusiThe apparent volume…
KlirensA 30kg child has a …
Genetik -
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