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17430

Total database: 17430
Struktur (SMILES)
12313 (70.6%)
Target
9368 (53.7%)
Genomik
112 (0.6%)
Referensi
17430 (100.0%)

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Halaman 147 / 349
biotech | CAS: 944130-77-2

Eptacog alfa pegol (activated) has been used in trials studying the prevention and treatment of Haemophilia A, Haemophilia B, Congenital Bleeding Disorder, Haemophilia B With Inhibitors, and Haemophilia A With Inhibitors.

Kategori:
Pegylated agents
Waktu Paruh-
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Genetik -
Eptifibatide Approved DB00063
biotech | CAS: 188627-80-7

Synthetic cyclic hexapeptide that binds to platelet receptor glycoprotein and inhibits platelet aggregation. Derived from venom of the Southeastern pygmy rattlesnake (Sistrurus miliarus barbouri), eptifibatide is a cyclic heptapeptide that belongs to the clas…

Kategori:
Amino Acids, Peptides, and ProteinsAntiplatelet agentsBlood and Blood Forming Organs +5
Target Protein:
Integrin beta-3Integrin alpha-IIbVoltage-dependent N-type calcium channel
Waktu ParuhApproximately 2.5 h…
Vol. Distribusi-
Klirens* 55 mL/kg/h [patie…
Genetik -
Eptinezumab Approved DB14040
biotech | CAS: 1644539-04-7

Eptinezumab is a fully-humanized IgG1 antibody manufactured using yeast (_Pichia pastoris_) and developed by Lundbeck Seattle Biopharmaceuticals.[L12318] Eptinezumab has been specifically designed to bind to both alpha and beta forms of the human calcitonin g…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe central volume …
KlirensThe apparent cleara…
Genetik -
Eptotermin alfa Approved DB11631
biotech | CAS: 129805-33-0

A bone morphogenetic protein that is widely expressed during EMBRYONIC DEVELOPMENT. It is both a potent osteogenic factor and a specific regulator of nephrogenesis. Eptotermin alfa is an ingredient in the EMA-withdrawn product Osigraft.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBone Morphogenetic Proteins +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EQ101 DB17396
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Deskripsi belum tersedia.

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Equilenin DB03515
small molecule | CAS: 517-09-9

Equilenin is an estrogenic steroid produced by horses. It has a total of five double bonds in the A- and B-ring. High concentration of equilenin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
Steroid Delta-isomeraseSteroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equilin DB02187
small molecule | CAS: 474-86-2

An estrogenic steroid produced by horses. It has a total of four double bonds in the A- and B-ring. High concentration of equilin is found in the urine of pregnant mares.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesCytochrome P-450 CYP3A Substrates +12
Target Protein:
17-beta-hydroxysteroid dehydrogenase type 1Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Equine Botulinum Neurotoxin A Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype A. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
BoNT/A
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin B Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype B. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type B
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin C Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype C. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type C1
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin D Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype D. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type D
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin E Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype E. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type E
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin F Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype F. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type F
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
biotech

Equine Botulinum Neurotoxin G Immune FAB2 is composed of a mixture of immune globulin fragments purified from plasma of horses that were previously immunized with botulinum toxin serotype G. It is intravenously administered for the treatment of symptomatic bo…

Target Protein:
Botulinum neurotoxin type G
Waktu ParuhEquine Botulinum Ne…
Vol. DistribusiEquine Botulinum Ne…
KlirensEquine Botulinum Ne…
Genetik -
Equine collagen DB16613
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Equisetum arvense top Approved DB14349
biotech

Equisetum arvense top is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Equol DB11674
small molecule | CAS: 531-95-3

Equol has been used in trials studying the treatment of Breast Cancer.

Kategori:
BenzopyransChromonesEstrogens +7
Target Protein:
Estrogen receptor betaSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equus caballus dander Approved DB11021
biotech

Equus caballus dander is the dander of Equus caballus. Equus caballus dander is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equus caballus hair Approved DB10880
biotech

Horse hair is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Equus caballus skin Approved DB10410
biotech

Equus caballus skin allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ER-176 C-11 DB19181
small molecule | CAS: 1623028-18-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ER2001 DB18165
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Eragidomide DB19242
small molecule | CAS: 1860875-51-9

Eragidomide is under investigation in clinical trial NCT04297124 (A Study to Evaluate the Metabolism and Excretion of [14C]-CC-90009 in Healthy Male Subjects).

Kategori:
AcetatesAcids, AcyclicAmides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eravacycline Approved DB12329
small molecule | CAS: 1207283-85-9

Eravacycline, known as _Xerava_ by Tetraphase Pharmaceuticals, is a fully synthetic fluorocycline antibiotic of the tetracycline class with activity against clinically significant gram-negative, gram-positive aerobic, and facultative bacteria. This includes m…

Kategori:
Anti-Bacterial AgentsAntibacterials for Systemic UseAntiinfectives for Systemic Use +6
Target Protein:
30S ribosomal protein S4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe volume of distr…
Klirens17.82 L/min (standa…
Genetik -
ERB-196 DB06875
small molecule | CAS: 550997-55-2

Deskripsi belum tersedia.

Kategori:
Estrogen Receptor beta, agonistsNaphthalenes
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erbumine DB18019
small molecule | CAS: 1919888-06-4

Deskripsi belum tersedia.

Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ERC-1671 DB17431
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erdafitinib Approved DB12147
small molecule | CAS: 1346242-81-6

In early April of 2019, the US FDA approved Janssen Pharmaceutical Companies' brand name Balversa (erdafitinib) as the first-ever fibroblast growth factor receptor (FGFR) kinase inhibitor indicated for patients with locally advanced or metastatic urothelial c…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C9 Substrates +25
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +7
Waktu ParuhThe mean effective …
Vol. DistribusiThe mean apparent v…
KlirensThe mean total appa…
Genetik -
Erdosteine Approved DB05057
small molecule | CAS: 84611-23-4

Erdosteine is a drug that causes a breakdown of mucus, also known as a _mucolytic_ agent. It is a _thiol_ derivative produced for the clinical management of chronic obstructive bronchitis, in addition to infective exacerbations of chronic bronchitis. This dru…

Kategori:
AcetatesAcids, AcyclicCough and Cold Preparations +4
Target Protein:
Chymotrypsin-like elastase family member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erenumab Approved DB14039
biotech | CAS: 1582205-90-0

Erenumab (AMG-334) (INN; trade name Aimovig) is a human monoclonal antibody designed specifically to bind and antagonize the calcitonin gene-related peptide receptor (CGRPR) as a means to prevent migraines. Aimovig, as released and marketed by Novartis and Am…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +14
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhErenumab exhibits n…
Vol. DistribusiAfter a single 140 …
KlirensCertain studies sho…
Genetik -
Erfonrilimab DB17446
biotech | CAS: 2367013-69-0

Erfonrilimab is a bispecific monoclonal antibody directed against both the programmed cell death-1 ligand 1 (PD-L1) and cytotoxic T-lymphocyte-associated antigen 4 (CTLA4).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergidina DB18565
biotech

Ergidina is a recombinant human minibody against complement component C5 fused with RGD-motif.

Waktu Paruh-
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Ergocalciferol Approved DB00153
small molecule | CAS: 50-14-6

Ergocalciferol is an inactivated vitamin D analog.[A177526] It is synthesized by some plants in the presence of UVB light.[T577] The production of ergocalciferol was prompted by the identification of dietary deficiency, more specifically vitamin D, as the mai…

Kategori:
Alimentary Tract and MetabolismBone Density Conservation AgentsCalcium-Regulating Hormones and Agents +11
Target Protein:
Vitamin D3 receptorVoltage-dependent calcium channel
Waktu ParuhErgocalciferol can …
Vol. DistribusiThe amount of circu…
KlirensThere are no formal…
Genetik -
Ergoloid mesylate Approved DB01049
small molecule | CAS: 8067-24-1

Ergoloid Mesylate is an equiproportional preparation of three different ergotamantriones: dihydroergocornine, dihydroergocristine, and dihydroergocryptine.[A32912] All these components are produced by the fungus _Claviceps purpurea_ and are all derivatives of…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +24
Target Protein:
Dopamine receptorAlpha adrenergic receptorBeta adrenergic receptor +1
Waktu ParuhThe reported plasma…
Vol. DistribusiThe volume of distr…
KlirensTo know more about …
Genetik -
Ergometrine Approved DB01253
small molecule | CAS: 60-79-7

An ergot alkaloid with uterine and vascular smooth muscle contractile properties.

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-Agonists +20
Target Protein:
Alpha-1A adrenergic receptorD(2) dopamine receptor
Waktu Paruht<sub>1/2 &alpha;</…
Vol. Distribusi-
Klirens-
Genetik -
Ergosterol Approved DB04038
small molecule | CAS: 57-87-4

A steroid of interest both because its biosynthesis in FUNGI is a target of ANTIFUNGAL AGENTS, notably AZOLES, and because when it is present in SKIN of animals, ULTRAVIOLET RAYS break a bond to result in ERGOCALCIFEROL.

Kategori:
CholestanesCholestenesDiet, Food, and Nutrition +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ergotamine Approved DB00696
small molecule | CAS: 113-15-5

A vasoconstrictor found in ergot of Central Europe. It is an alpha-1 selective adrenergic agonist and is commonly used in the treatment of migraine disorders.

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +39
Target Protein:
5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 2A +11
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
Ergothioneine DB17614
small molecule | CAS: 497-30-3

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, CyclicAmino Acids, Peptides, and Proteins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eribaxaban DB06920
small molecule | CAS: 536748-46-6

Deskripsi belum tersedia.

Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eribulin Approved DB08871
small molecule | CAS: 253128-41-5

Eribulin is a microtubule inhibitor indicated for the treatment of patients with metastatic breast cancer who have previously received at least two chemotherapeutic regimens for the treatment of metastatic disease. Eribulin was isolated from the marine sponge…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEthers +10
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2
Waktu Paruhabout 40 hours
Vol. Distribusi43 L/m2 to 114 L/m2
Klirens1.16 L/hr/m2 to 2.4…
Genetik -
Eritoran DB04933
small molecule | CAS: 185955-34-4

Eritoran is a structural analogue of the lipid A portion of lipopolysaccharide (LPS). It is being developed by Eisai Research Institute of Boston for the treatment of severe sepsis.

Kategori:
AntigensAntigens, BacterialBacterial Toxins +11
Target Protein:
Toll-like receptor 4
Waktu Paruh50.4 to 62.7 hours
Vol. Distribusi-
Klirens-
Genetik -
Erlotinib Approved DB00530
small molecule | CAS: 183321-74-6

Erlotinib is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase that is used in the treatment of non-small cell lung cancer, pancreatic cancer and several other types of cancer. It is typically marketed under the trade name Tarceva. E…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +33
Target Protein:
Nuclear receptor subfamily 1 group I member 2Epidermal growth factor receptor
Gen Terkait:
EGFR EGFR EGFR
Waktu ParuhMedian half-life of…
Vol. DistribusiApparent volume of …
KlirensSmokers have a 24% …
Genetik 3 Varian
Ersodetug DB18182
biotech | CAS: 2410976-61-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ertapenem Approved DB00303
small molecule | CAS: 153832-46-3

Ertapenem is a 1-? methyl-carbapenem that is structurally related to beta-lactam antibiotics.[L14339] It was first authorized for use in the US in November 2001 and in Europe in April 2002.[A447] Shown to be effective against a wide range of Gram-positive and…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Penicillin-binding protein 1APenicillin-binding protein 1BPenicillin-binding protein 2 +5
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe apparent volume…
KlirensThe mean plasma cle…
Genetik -
Erteberel DB07933
small molecule | CAS: 533884-09-2

Erteberel is an estrogen receptor beta agonist that has been used in trials studying the treatment of Benign Prostatic Hyperplasia.

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptor betaEstrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ertiprotafib DB06521
small molecule | CAS: 251303-04-5

Ertiprotafib belongs to a novel class of insulin sensitizers developed for treatment of type 2 diabetes. In insulin-resistant rodent models, ertiprotafib and a close analog lowered both fasting blood glucose and insulin levels and improved glycemic excursion …

Kategori:
Acids, CarbocyclicSulfur Compounds
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1Inhibitor of nuclear factor kappa-B kinase subunit betaPeroxisome proliferator-activated receptor alpha +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ertugliflozin Approved DB11827
small molecule | CAS: 1210344-57-2

Ertugliflozin is a sodium-dependent glucose cotransporter-2 (SGLT2) inhibitor used to treat type II diabetes mellitus. It works to block glucose reabsorption from the glomerulus.[A31581] Ertugliflozin was first approved by the FDA in December 2017.[A26195…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 SubstratesBlood Glucose Lowering Agents +9
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensIn one clinical inv…
Genetik -
Ertumaxomab DB18923
biotech | CAS: 509077-99-0

Ertumaxomab is under investigation in clinical trial NCT00522457 (Phase II Study With the Trifunctional Antibody Ertumaxomab to Treat Metastatic Breast Cancer After Progression on Trastuzumab Therapy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Bispecific +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Erythritol DB04481
small molecule | CAS: 149-32-6

Erythritol is a four-carbon sugar that is found in algae, fungi, and lichens. It is twice as sweet as sucrose and can be used as a coronary vasodilator.

Kategori:
AlcoholsCarbohydratesCardiovascular Agents +2
Target Protein:
5-methyltetrahydropteroyltriglutamate--homocysteine methyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7301–7350 dari 17430
Sebelumnya Halaman 147 / 349 Berikutnya