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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 147 / 252
Levallorphan Approved DB00504
small molecule | CAS: 152-02-3

An opioid antagonist with properties similar to those of naloxone; in addition it also possesses some agonist properties. It should be used cautiously; levallorphan reverses severe opioid-induced respiratory depression but may exacerbate respiratory depressio…

Kategori:
AlkaloidsCentral Nervous System AgentsHeterocyclic Compounds, Fused-Ring +6
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Mu-type opioid receptor
Waktu Paruh1 hour
Vol. Distribusi-
Klirens-
Genetik -
Levetiracetam Approved DB01202
small molecule | CAS: 102767-28-2

Levetiracetam is a drug within the pyrrolidine class that is used to treat various types of seizures stemming from epileptic disorders. It was first approved for use in the United States in 1999 and is structurally and mechanistically unrelated to other anti-…

Kategori:
AcetamidesAmidesAnticonvulsants +8
Target Protein:
5-hydroxytryptamine receptor 3AVoltage-dependent N-type calcium channel subunit alpha-1BSynaptic vesicle glycoprotein 2A
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe volume of distr…
KlirensThe total plasma cl…
Genetik -
Levilimab DB16387
biotech | CAS: 2035008-70-7

Levilimab is under investigation in clinical trial NCT04227366 (Study of the Efficacy and Safety of BCD-089 in Combination With Methotrexate in Patients With Active Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levmetamfetamine Approved DB09571
small molecule | CAS: 33817-09-3

Levomethamphetamine, the L-enantiomer of methamphetamine is a sympathomimetic vasoconstrictor used in some over-the-counter (OTC) nasal decongestant inhalers in the United States.

Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Levobetaxolol Approved DB09351
small molecule | CAS: 93221-48-8

Levobetaxolol is a beta-blocker used to lower the pressure in the eye to treat conditions such as glaucoma. It was marketed as a 0.5% ophthalmic solution of levobetaxolol hydrochloride under the trade name Betaxon but has been discontinued.

Kategori:
Adrenergic AntagonistsAdrenergic beta-AntagonistsAgents causing hyperkalemia +3
Target Protein:
Beta-1 adrenergic receptor
Waktu ParuhThe mean half life …
Vol. Distribusi-
Klirens-
Genetik -
Levobunolol Approved DB01210
small molecule | CAS: 47141-42-4

A nonselective beta-adrenoceptor antagonist used in the treatment of glaucoma.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +22
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
Levocabastine Approved DB01106
small molecule | CAS: 79516-68-0

Levocabastine is a selective second-generation H1-receptor antagonist used for allergic conjunctivitis. Levocabastine was discovered at Janssen Pharmaceutica in 1979.

Kategori:
Anti-Allergic AgentsAntiallergic Agents, Excl. CorticosteroidsCentral Nervous System Depressants +11
Target Protein:
Histamine H1 receptorNeurotensin receptor type 2
Waktu Paruh36 hours (after ora…
Vol. Distribusi-
Klirens-
Genetik -
Levocarnitine Approved DB00583
small molecule | CAS: 541-15-1

Constituent of striated muscle and liver. It is used therapeutically to stimulate gastric and pancreatic secretions and in the treatment of hyperlipoproteinemias.

Kategori:
Alimentary Tract and MetabolismAminesAmino Acids and Derivatives +9
Target Protein:
Carnitine O-palmitoyltransferase 1, muscle isoformXanthine dehydrogenase/oxidaseLiver carboxylesterase 1 +9
Waktu Paruh17.4 hours (elimina…
Vol. DistribusiThe steady state vo…
KlirensTotal body clearanc…
Genetik -
small molecule | CAS: 20064-19-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levocetirizine Approved DB06282
small molecule | CAS: 130018-77-8

Levocetirizine is a selective histamine H<sub>1</sub> antagonist used to treat a variety of allergic symptoms.[A181748,A181790,L7694] It is the R enantiomer of [cetirizine].[L7694] Levocetirizine has greater affinity for the histamine H<sub>1</sub> receptor t…

Kategori:
Antihistamines for Systemic UseCentral Nervous System DepressantsCytochrome P-450 CYP3A Substrates +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe average half li…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Levodopa Approved DB01235
small molecule | CAS: 59-92-7

Levodopa is a prodrug of dopamine that is administered to patients with Parkinson's due to its ability to cross the blood-brain barrier[Label]. Levodopa can be metabolised to dopamine on either side of the blood-brain barrier and so it is generally administer…

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +21
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +2
Waktu Paruh2.3 hours for orall…
Vol. Distribusi168L for orally inh…
KlirensIntravenously admin…
Genetik -
small molecule | CAS: 99291-25-5

Levodropropizine is under investigation in clinical trial NCT01573663 (A Drug-Drug Interaction Study of Ambroxol and Levodropropizine).

Kategori:
AlcoholsAntitussive AgentsCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levofloxacin Approved DB01137
small molecule | CAS: 100986-85-4

Levofloxacin is a fluoroquinolone antibiotic and the optical S-(-) isomer of racemic [ofloxacin].[A190663] It reportedly carries 8 to 128-fold more activity against both gram-negative and gram-positive bacteria compared to R-(+)-ofloxacin[A190663] and remains…

Kategori:
4-QuinolonesAlimentary Tract and MetabolismAnti-Bacterial Agents +35
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu ParuhThe average termina…
Vol. DistribusiLevofloxacin is wid…
KlirensThe average apparen…
Genetik -
Levoketoconazole Approved DB05667
small molecule | CAS: 142128-57-2

Cushing's syndrome (CS) is underpinned by chronic hypercortisolism leading to multisystem morbidity, including effects on the cardiovascular and endocrine systems, metabolic syndrome with accompanying changes in body composition, neuropsychiatric effects, cha…

Kategori:
Adrenal Cortex HormonesAntiadrenal PreparationsAnticorticosteroids +32
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyaseCytochrome P450 11B1, mitochondrialCytochrome P450 11B2, mitochondrial +2
Waktu ParuhLevoketoconazole ha…
Vol. DistribusiLevoketoconazole ha…
Klirens-
Genetik -
Levoleucovorin Approved DB11596
small molecule | CAS: 68538-85-2

Levoleucovorin is the enantiomerically active form of Folinic Acid (also known as 5-formyl tetrahydrofolic acid or leucovorin). Commercially available leucovorin is composed of a 1:1 racemic mixture of the dextrorotary and levorotary isomers, while levoleucov…

Kategori:
AntidotesCoenzymesCompounds used in a research, industrial, or household setting +14
Target Protein:
Serine hydroxymethyltransferase
Waktu ParuhThe mean terminal h…
Vol. DistribusiData can't be found.
KlirensData can't be found.
Genetik -
Levomefolic acid Approved DB11256
small molecule | CAS: 31690-09-2

Levomefolic acid (INN) is the metabolite of folic acid (Vitamin B9) and it is a predominant active form of folate found in foods and in the blood circulation, accounting for 98% of folates in human plasma [A19276]. It is transported across the membranes inclu…

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +10
Waktu ParuhThe mean eliminatio…
Vol. DistribusiCirculates in its f…
Klirens-
Genetik -
Levomenol Approved DB13153
small molecule | CAS: 23089-26-1

Bisabolol, or more formally ?-(?)-bisabolol or also known as levomenol, (-)-alpha-Bisabolol is found in fats and oils. (-)-alpha-Bisabolol is isolated from essential oil of Matricaria chamomilla (German chamomile) (-)-alpha-Bisabolol belongs to the family of …

Kategori:
Biological ProductsComplex MixturesLipids +7
Waktu Paruh-
Vol. DistribusiTo demonstrate the …
Klirens-
Genetik -
Levomenthol Approved DB00825
small molecule | CAS: 2216-51-5

Menthol is a covalent organic compound made synthetically or obtained from peppermint or other mint oils. Forming clear or white waxy, crystalline substance, menthol is typically solid at room temperature. (-)-Menthol is the naturally-occurring and main form …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsAntipruritics +16
Target Protein:
Transient receptor potential cation channel subfamily M member 8Transient receptor potential cation channel subfamily A member 1Transient receptor potential cation channel subfamily V member 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomethadone DB13515
small molecule | CAS: 125-58-6

Deskripsi belum tersedia.

Kategori:
Drugs Used in Addictive DisordersDrugs Used in Opioid DependenceNervous System
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levomilnacipran Approved DB08918
small molecule | CAS: 96847-54-0

Levomilnacipran is a selective serotonin and norepinephrine reuptake inhibitor (SNRI), although it is a more potent inhibitor of norepinephrine reuptake than serotonin reuptake.[A261181, A38560] Levomilnacipran is the more active 1S,2R-enantiomer in the racem…

Kategori:
Adrenergic Uptake InhibitorsAgents producing tachycardiaAntidepressive Agents +27
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporter
Waktu ParuhThe apparent termin…
Vol. DistribusiLevomilnacipran is …
KlirensFollowing oral admi…
Genetik -
small molecule | CAS: 154357-42-3

Levonadifloxacin is under investigation in clinical trial NCT03405064 (Comparative Study of Levonadifloxacin (IV and Oral) With Linezolid (IV and Oral) in Acute Bacterial Skin and Skin Structure Infections (ABSSSI)).

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levonorgestrel Approved DB00367
small molecule | CAS: 797-63-7

Levonorgestrel (LNG) is a synthetic progestogen similar to [Progesterone] used in contraception and hormone therapy.[A181988,T659] Also known as Plan B, it is used as a single agent in emergency contraception, and as a hormonal contraceptive released from an …

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +23
Target Protein:
Progesterone receptor3-oxo-5-alpha-steroid 4-dehydrogenase 1Estrogen receptor +3
Waktu ParuhThe elimination hal…
Vol. DistribusiOne pharmacokinetic…
KlirensClearance was found…
Genetik -
small molecule | CAS: 230313-75-4

Levophencynonate is under investigation in clinical trial NCT02299804 (A Clinical Trial to Evaluate Efficacy and Safety of Levophencynonate Hydrochloride in Patient With Vertigo).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levorphanol Approved DB00854
small molecule | CAS: 77-07-6

A narcotic analgesic that may be habit-forming. It is nearly as effective orally as by injection.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +11
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu Paruh11-16 hours
Vol. Distribusi* 10 to 13 L/kg
Klirens* 0.78 to 1.1 L/kg/…
Genetik -
Levosimendan Approved DB00922
small molecule | CAS: 141505-33-1

Levosimendan increases calcium sensitivity to myocytes by binding to troponin C in a calcium dependent manner. This increases contractility without raising calcium levels. It also relaxes vascular smooth muscle by opening adenosine triphosphate sensitive pota…

Kategori:
Antiarrhythmic agentsCardiac Stimulants Excl. Cardiac GlycosidesCardiac Therapy +14
Target Protein:
Troponin C, slow skeletal and cardiac musclesATP-sensitive inward rectifier potassium channel 11ATP-sensitive inward rectifier potassium channel 8 +1
Waktu ParuhEliminination half-…
Vol. Distribusi-
Klirens-
Genetik -
Levothyroxine Approved DB00451
small molecule | CAS: 51-48-9

Levothyroxine is a synthetically produced form of thyroxine, a major endogenous hormone secreted by the thyroid gland.[F4633] Also known as L-thyroxine or the brand name product Synthroid, levothyroxine is used primarily to treat hypothyroidism, a condition w…

Kategori:
Agents used to treat hypothyroidismAmino AcidsAmino Acids, Aromatic +16
Target Protein:
Integrin alpha-VIntegrin beta-3Thyroid hormone receptor alpha +1
Waktu ParuhT<sub>4</sub> half-…
Vol. Distribusi-
Klirens-
Genetik -
Levotofisopam DB19073
small molecule | CAS: 82059-51-6

Levotofisopam is under investigation in clinical trial NCT01519687 (Study of Levotofisopam 50 Mg Three Times a Day (TID) Administered for 7 Days on Hyperuricemia and Gout).

Kategori:
Antidepressive AgentsBenzazepinesCentral Nervous System Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levovirin DB06523
small molecule | CAS: 206269-27-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexacalcitol DB03451
small molecule | CAS: 131875-08-6

Lexacalcitol is a solid. This compound belongs to the vitamin D and derivatives class of chemicals. These are compounds containing a secosteroid backbone, usually secoergostane or secocholestane. It is known to target the vitamin D3 receptor.

Kategori:
Antineoplastic AgentsCholestanesCholestenes +11
Target Protein:
Vitamin D3 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexanersen DB17933
biotech | CAS: 2073015-40-2

Lexanersen is an antisense oligonucleotide under investigation for use as a disease-modifying therapy in Huntington's disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1390631-57-8

Lexaptepid pegol has been used in trials studying the treatment of Anemia, Inflammation, Chronic Diseases, End Stage Renal Disease, and Anemia of Chronic Disease.

Kategori:
Anti-Inflammatory AgentsNucleic Acids, Nucleotides, and NucleosidesNucleotides +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lexatumumab DB06599
biotech | CAS: 845816-02-6

Lexatumumab is a fully humanized, high-affinity immunoglobulin G(1 lambda) monoclonal antibody (mAb).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +7
Target Protein:
Tumor necrosis factor receptor superfamily member 10B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LFF-571 DB13013
small molecule | CAS: 1160959-55-6

LFF571 has been used in trials studying the treatment of Moderate Clostridium Difficile Infection.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LG-100268 DB01941
small molecule | CAS: 153559-76-3

LG-100268 is a retinoid X receptor (RXR) selective compound.

Kategori:
LigandsNaphthalenesPyridines
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-1550 DB05785
small molecule | CAS: 178600-20-9

LGD-1550 is an orally-active synthetic aromatic retinoic acid agent with potential antineoplastic and chemopreventive activities.

Kategori:
AlkenesBiological FactorsCarotenoids +8
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD-3303 DB13937
small molecule | CAS: 917891-35-1

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGD2941 DB05234
small molecule

LGD2941 is a non-steroidal, selective androgen receptor modulator (SARM) developed jointly by Ligand and TAP.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LGH-447 DB14943
small molecule | CAS: 1210608-43-7

LGH-447 is under investigation in clinical trial NCT02160951 (Dose Escalation Study of LGH447 in Japanese Patients With Relapsed and/or Refractory Hematologic Malignancies).

Target Protein:
Serine/threonine-protein kinase pim-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LH-708 DB17636
small molecule | CAS: 1616758-14-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LI-301 DB05509
small molecule

LI 301 is an orally bio-available compound delivered in a fast melt mechanism with taste masking enabling it to be taken anytime without water. It has a novel mode of action combining both the light effect of a Selective Serotonin Reuptake Inhibitor ("SSRI")(…

Target Protein:
Mu-type opioid receptor5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liafensine DB14878
small molecule | CAS: 1198790-53-2

Liafensine is under investigation in clinical trial NCT00892840 (Multiple-Ascending Dose Study).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liarozole DB13066
small molecule | CAS: 115575-11-6

Liarozole has been used in trials studying the treatment of Ichthyosis, Lamellar.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalDermatologicals +3
Target Protein:
Cytochrome P450 26A1Aromatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Libivirumab DB17748
biotech | CAS: 569658-79-3

Libivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LIC-477 DB05363
small molecule

LIC-477is indicated to be suitable for the treatment of psychosomatic disturbances, epilepsy, trigeminal neuralgia and cerebral spasticity.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licaminlimab DB18936
biotech | CAS: 1688648-13-6

Licaminlimab is under investigation in clinical trial NCT05896670 (Safety and Efficacy of Licaminlimab Ophthalmic Suspension for the Treatment of Dry Eye Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licochalcone A DB19281
small molecule | CAS: 58749-22-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFabaceae +5
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licofelone DB04725
small molecule | CAS: 156897-06-2

Developed by the German pharmaceutical company, Merckle GmbH, together with EuroAlliance partners Alfa Wassermann and Lacer, licofelone (ML3000) is a dual COX/LOX inhibitor and the first member of this new class of analgesic and anti-inflammatory drugs. It is…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +15
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseProstaglandin G/H synthase 2Group IIE secretory phospholipase A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licogliflozin DB15048
small molecule | CAS: 1291094-73-9

Licogliflozin is under investigation in clinical trial NCT03320941 (A Dose-finding Study to Evaluate the Change in Weight After Treatment With LIK066 in Japanese Patients With Obesity).

Kategori:
AlcoholsBlood Glucose Lowering AgentsCarbohydrates +2
Target Protein:
Sodium/glucose cotransporter 1Sodium/glucose cotransporter 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Licorice Approved DB10675
biotech

Licorice allergenic extract is used in allergenic testing.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lidocaine Approved DB00281
small molecule | CAS: 137-58-6

Ever since its discovery and availability for sale and use in the late 1940s, lidocaine has become an exceptionally commonly used medication [T583]. In particular, lidocaine's principal mode of action in acting as a local anesthetic that numbs the sensations …

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAgents that reduce seizure thresholdAmides +49
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein type 10 subunit alphaSodium channel protein type 9 subunit alpha +5
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe mean systemic c…
Genetik -
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