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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 147 / 321
Flaviolin DB02521
small molecule | CAS: 479-05-0

Deskripsi belum tersedia.

Kategori:
NaphthalenesQuinones
Target Protein:
PrenyltransferaseBiflaviolin synthase CYP158A2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavone Approved DB07776
small molecule | CAS: 525-82-6

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
AromataseGamma-aminobutyric acid receptor subunit alpha-1Androgen receptor +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flavoxate Approved DB01148
small molecule | CAS: 15301-69-6

A drug that has been used in various urinary syndromes and as an antispasmodic. Its therapeutic usefulness and its mechanism of action are not clear. It may have local anesthetic activity and direct relaxing effects on smooth muscle as well as some activity a…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsAutonomic Agents +15
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M5Muscarinic acetylcholine receptor M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flecainide Approved DB01195
small molecule | CAS: 54143-55-4

Flecainide is a Class I anti-arrhythmic agent like [encainide] and [propafenone].[A186880] Flecainide’s development began in 1966 and was first synthesized in 1972 as an attempt to generate new anesthetics.[A186931] It is used to prevent supraventricular and …

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +27
Target Protein:
Sodium channel protein type 4 subunit alphaSodium channel protein type 5 subunit alphaVoltage-gated inwardly rectifying potassium channel KCNH2 +1
Waktu ParuhIn healthy subjects…
Vol. DistribusiThe average volume …
KlirensThe average clearan…
Genetik -
Fleroxacin DB04576
small molecule | CAS: 79660-72-3

Fleroxacin is a broad-spectrum antimicrobial fluoroquinolone. It strongly inhibits the DNA-supercoiling activity of DNA gyrase. Fleroxacin is not an inhibitor of CYP1A2.[A39048]

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +12
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fletikumab DB12356
biotech | CAS: 1357158-22-5

Fletikumab is under investigation in clinical trial NCT01038674 (Safety and Tolerability of Anti-IL-20 in Subjects With Rheumatoid Arthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flibanserin Approved DB04908
small molecule | CAS: 167933-07-5

Flibanserin is the first drug to be approved for hypoactive sexual desire disorder (HSDD) in premenopausal women by the FDA in August 2015. It was originally developed as an antidepressant medication by Boehringer Ingelheim, but showed lack of efficacy in tri…

Kategori:
Agents that produce hypertensionAntidepressive AgentsCentral Nervous System Depressants +15
Target Protein:
5-hydroxytryptamine receptor 1A5-hydroxytryptamine receptor 2AD(4) dopamine receptor
Waktu Paruh?11 hours
Vol. Distribusi-
Klirens-
Genetik -
Flindokalner DB16908
small molecule | CAS: 187523-35-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Floctafenine Approved DB08976
small molecule | CAS: 23779-99-9

Floctafenine is an anti-inflammatory analgesic similar in action to aspirin. Floctafenine inhibits prostaglandin synthesis.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flomoxef DB11935
small molecule | CAS: 99665-00-6

Flomoxef has been used in trials studying the treatment of Urinary Tract Infection.

Kategori:
AmidesAnti-Bacterial AgentsAntibacterials for Systemic Use +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Florantyrone DB08975
small molecule | CAS: 519-95-9

Florantyrone is used in the treatment of biliary dyskinesia

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Florasulam DB15316
small molecule | CAS: 145701-23-1

Florasulam is under investigation in clinical trial NCT01193465 (Temperature and Humidity Among Different Anesthesia Work-station).

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 956903-29-0

Florbenazine F-18 is under investigation in clinical trial NCT01515384 (A Trial of 18F-AV-133 Positron Emission Tomography (PET)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Florbetaben F-18 Approved DB09148
small molecule | CAS: 902143-01-5

Florbetaben is a fluorine-18 (18F)-labeled stilbene derivative used for Positron Emission Tomography (PET) imaging of the brain. It is used for the non-invasive detection of the density of ß-amyloid neuritic plaques in the brain of adult patients with cogniti…

Kategori:
AminesBenzene DerivativesBenzylidene Compounds +6
Target Protein:
Amyloid-beta precursor protein
Waktu Paruh1 hr
Vol. Distribusi-
Klirens-
Genetik -
Florbetapir F-18 Approved DB09149
small molecule | CAS: 956103-76-7

Florbetapir (18F) is a radiopharmaceutical compound containing the radionuclide fluorine-18 bound to the compound florbetapir, a molecule that binds with high affinity to beta amyloid plaque, a peptide that plays a key role in Alzheimer's Disease pathogenesis…

Kategori:
AlcoholsAminesCentral Nervous System +6
Target Protein:
Amyloid-beta precursor proteinBeta amyloid plaque
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Florfenicol DB11413
small molecule | CAS: 73231-34-2

Florfenicol is a fluorinated synthetic analog of thiamphenicol.

Kategori:
AlcoholsAnti-Bacterial AgentsAnti-Infective Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1196963-74-2

Florilglutamic acid F-18 is under investigation in clinical trial NCT02370563 (PET Imaging of Intracranial Cancers With 18F-FSPG).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1841444-25-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flortaucipir DB15033
small molecule | CAS: 1415379-56-4

Flortaucipir is under investigation in clinical trial NCT03507257 (Longitudinal Early-onset Alzheimer's Disease Study Protocol).

Kategori:
Compounds used in a research, industrial, or household settingContrast MediaDiagnostic Uses of Chemicals +4
Target Protein:
Microtubule-associated protein tau
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flortaucipir F-18 Approved DB14914
small molecule | CAS: 1522051-90-6

Flortaucipir F-18, also known as <sup>18</sup>F-T807 and <sup>18</sup>F-AV-1451, is a small indole molecule synthesized with a radioactive fluorine isotope.[A203933] It is used as a marker in positron emission tomography (PET) imaging of patients suspected of…

Kategori:
Central Nervous SystemCompounds used in a research, industrial, or household settingContrast Media +6
Target Protein:
Microtubule-associated protein tauAmine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
Waktu ParuhFlortaucipir F-18 p…
Vol. DistribusiFlortaucipir F-18 i…
Klirens-
Genetik -
small molecule | CAS: 1565797-57-0

PMPBB3 F-18 is under investigation in clinical trial NCT04305210 (Alzheimer's Disease: Clinical Investigation and Neuroimage Studies Including 18F-PM-PBB3 and 18f-florbetapir (AV-45) PET Examination).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flosequinan Approved DB13228
small molecule | CAS: 76568-02-0

Flosequinan was approved in the USA and the UK for a year prior to being withdrawn from the market due to increased mortality in chronic heart failure patients, found in drug trials.[A174979,L43942]

Kategori:
Cardiac TherapyCardiovascular AgentsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1010702-75-6

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flotetuzumab DB15223
biotech | CAS: 1664355-28-5

Flotetuzumab is under investigation in clinical trial NCT02152956 (Safety Study of MGD006 in Relapsed/Refractory Acute Myeloid Leukemia (AML) or Intermediate-2/High Risk MDS).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flotufolastat F-18 Approved DB17851
small molecule | CAS: 2639294-14-5

Flotufolastat F-18 (<sup>18</sup>F-rhPSMA-7.3) is an <sup>18</sup>F-labeled ligand that targets the prostate-specific membrane antigen (PSMA).[A259846,L46731] In patients with recurrent prostate cancer that require localized treatment, the use of <sup>18</sup…

Kategori:
Diagnostic RadiopharmaceuticalsFluorine RadioisotopesPositron Emitting Activity +1
Target Protein:
Glutamate carboxypeptidase 2
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Flovagatran DB05714
small molecule | CAS: 871576-03-3

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +3
Target Protein:
Prothrombin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Floxuridine Approved DB00322
small molecule | CAS: 50-91-9

An antineoplastic antimetabolite that is metabolized to fluorouracil when administered by rapid injection. Floxuridine is available as a sterile, nonpyrogenic, lyophilized powder for reconstitution. When administered by slow, continuous, intra-arterial infusi…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +18
Target Protein:
Thymidylate synthaseThymidylate synthase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FLT190 DB18420
biotech

FLT190 is a recombinant adeno-associated viral vector serotype S3 containing DNA encoding for human alpha-galactosidase A.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FLT201 DB18419
biotech

FLT201 is a recombinant adeno-associated viral vector serotype S3 containing codon optimised expression cassette encoding human beta (?)-glucocerebrosidase variant 85 (GCasevar85)

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluanisone DB13665
small molecule | CAS: 1480-19-9

Deskripsi belum tersedia.

Kategori:
Antipsychotic AgentsButyrophenone DerivativesCentral Nervous System Agents +8
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptor5-hydroxytryptamine receptor 2A +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluasterone DB06250
small molecule | CAS: 112859-71-9

Has antiproliferative effects on HIV-1 and reduces HIV-1 replication.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesAndrostanes +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluazuron DB15583
small molecule | CAS: 86811-58-7

Fluazuron is a benzoyl phenylurea compound.

Kategori:
AmidesBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flubendazole DB08974
small molecule | CAS: 31430-15-6

Flubendazole is an anthelmintic that is used to treat worm infection in humans. It is available OTC in Europe.

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flubentylosin DB17769
small molecule | CAS: 1809266-03-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1037359-47-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluciclatide DB14842
small molecule | CAS: 879894-00-5

Fluciclatide, an investigational radiotracer intended for PET imaging, was under investigation in clinical trials NCT00565721 and NCT01961583 to evaluate its ability to detect tumors and angiogenesis. The conditions targeted by [18F]Fluciclatide in these stud…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsEthylene Glycols +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluciclovine DB15237
small molecule | CAS: 222727-43-7

Fluciclovine is under investigation in clinical trial NCT03036943 (Fluciclovine (18F) Imaging of Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluciclovine (18F) Approved DB13146
small molecule | CAS: 222727-39-1

Fluciclovine is a [18F]-tagged synthetic analog of the amino acid L-leucine. It presents excellent diagnostic properties to be used in positron emission tomography (PET) imaging.[A31384] The structure of fluciclovine allows it to be uptaken by the tumoral cel…

Kategori:
CycloparaffinsDiagnostic RadiopharmaceuticalsPositron Emitting Activity +2
Target Protein:
Neutral amino acid transporter B(0)Y+L amino acid transporter 1Cationic amino acid transporter 3 +5
Waktu ParuhFluciclovine is a c…
Vol. DistribusiThe compartmental v…
KlirensFluciclovine renal …
Genetik -
Fluclorolone DB13856
small molecule | CAS: 3693-38-7

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids, Dermatological Preparations +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fluclorolone acetonide Approved DB08973
small molecule | CAS: 3693-39-8

Fluclorolone acetonide (INN) or flucloronide (USAN) is a topical corticosteroid. It is marketed under the brand names Cutanit and Topicon.

Kategori:
Adrenal Cortex HormonesCorticosteroidsFused-Ring Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flucloxacillin Approved DB00301
small molecule | CAS: 5250-39-5

Antibiotic analog of [cloxacillin].

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +17
Target Protein:
Penicillin-binding protein 1A
Waktu Paruh0.75–1 hour
Vol. Distribusi-
Klirens-
Genetik -
Fluconazole Approved DB00196
small molecule | CAS: 86386-73-4

Fluconazole, commonly known as _Diflucan_, is an antifungal drug used for the treatment of both systemic and superficial fungal infections in a variety of tissues. It was initially approved by the FDA in 1990. This drug is an _azole_ antifungal, in the same …

Kategori:
14-alpha Demethylase InhibitorsAgents causing hyperkalemiaAnti-Infective Agents +29
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThis drug is mainly…
Genetik -
Flucytosine Approved DB01099
small molecule | CAS: 2022-85-7

A fluorinated cytosine analog that is used as an antifungal agent.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +17
Target Protein:
DNAThymidylate synthaseDNA (cytosine-5)-methyltransferase 1
Waktu Paruh2.4 to 4.8 hours.
Vol. Distribusi-
Klirens-
Genetik -
Fludarabine Approved DB01073
small molecule | CAS: 21679-14-1

Fludarabine is a chemotherapeutic agent used in the treatment of hematological malignancies. It is commonly marketed under the brand name Fludara.

Kategori:
Adenine NucleotidesAntimetabolitesAntineoplastic Agents +22
Target Protein:
DNAAdenosine deaminaseDeoxycytidine kinase +2
Waktu Paruh20 hours
Vol. Distribusi-
Klirens* 117-145 mL/min [p…
Genetik -
Fludeoxyglucose DB15107
small molecule | CAS: 29702-43-0

Fludeoxyglucose is under investigation in clinical trial NCT03262389 (Comparison of F-18 FDG and C-11 Acetate PET in Multiple Myeloma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fludeoxyglucose (18F) Approved DB09502
small molecule | CAS: 63503-12-8

Fludeoxyglucose F 18 Injection is a positron emitting radiopharmaceutical containing no-carrier added radioactive 2-deoxy-2-[18F]fluoro-D-g1ucose, which is used for diagnostic purposes in conjunction with Positron Emission Tomography (PET). It is administered…

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDeoxy Sugars +10
Waktu Paruh10-13 minutes
Vol. DistribusiFludeoxyglucose F 1…
KlirensFludeoxyglucose F 1…
Genetik -
Fludiazepam DB01567
small molecule | CAS: 3900-31-0

Fludiazepam is a drug which is a benzodiazepine derivative. It possesses anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. It is a scheduled drug in the U.S., but is approved for use in Japan.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +11
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Translocator proteinGamma-aminobutyric acid receptor subunit alpha-2 +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fludrocortisone Approved DB00687
small molecule | CAS: 127-31-1

Fludrocortisone is a synthetic mineralocorticoid used in conjunction with [hydrocortisone] to replace missing endogenous corticosteroids in patients with adrenal insufficiency.[A187169,A187187] It is functionally similar to [aldosterone], the body's primary e…

Kategori:
11-Hydroxycorticosteroids17-HydroxycorticosteroidsAdrenal Cortex Hormones +18
Target Protein:
Androgen receptorMineralocorticoid receptorGlucocorticoid receptor
Waktu ParuhThe plasma half-lif…
Vol. DistribusiThe apparent volume…
KlirensPopulation pharmaco…
Genetik -
Flufenamic acid Approved DB02266
small molecule | CAS: 530-78-9

An anthranilic acid derivative with analgesic, anti-inflammatory, and antipyretic properties. It is used in musculoskeletal and joint disorders and administered by mouth and topically. (From Martindale, The Extra Pharmacopoeia, 30th ed, p16)

Kategori:
Acids, CarbocyclicAminobenzoatesAnti-Inflammatory Agents +8
Target Protein:
Androgen receptorProstaglandin G/H synthase 2Prostaglandin G/H synthase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Flufenoxuron DB15006
small molecule | CAS: 101463-69-8

Flufenoxuron is under investigation in clinical trial NCT00922870 (Evaluation of Hemodynamic Effects of Cascade Hemofiltration in Septic Shock).

Kategori:
AmidesBenzene Derivatives
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7301–7350 dari 16004
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