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12560

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9109 (72.5%)
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6912 (55.0%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 146 / 252
Lemborexant Approved DB11951
small molecule | CAS: 1369764-02-2

Lemborexant is a novel dual orexin receptor antagonist used in the treatment of insomnia characterized by difficulties with sleep onset and/or sleep maintenance.[L10863] Recent research in the field of sleep disorders has revealed that insomnia is likely driv…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Inducers +17
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhThe half-life for l…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Lemon Approved DB10538
biotech

Lemon allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lemuteporfin DB04980
small molecule | CAS: 215808-49-4

Lemuteporfin, under development by QLT Incorporated, is a benzoporphyrin-derived chlorin-like photosensitizer. It is intended for the treatment of beign prostatic hyperplasia.

Kategori:
AlcoholsBiological FactorsGlycols +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lemzoparlimab DB17572
biotech | CAS: 2377483-71-9

Lemzoparlimab is under investigation in clinical trial NCT04912063 (Study to Evaluate Adverse Events and Movement of Lemzoparlimab in Body When Used Intravenously (IV) With Azacitidine Subcutaneously or IV and Venetoclax Orally in Participants With Acute Myel…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenabasum DB12193
small molecule | CAS: 137945-48-3

Ajulemic acid has been used in trials studying the treatment of Cystic Fibrosis, Dermatomyositis, and Diffuse Cutaneous Systemic Sclerosis.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +5
Target Protein:
Tumor necrosis factor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenacapavir Approved DB15673
small molecule | CAS: 2189684-44-2

HIV/AIDS remains an area of concern despite the introduction of numerous successful therapies, mainly due to the emergence of multidrug resistance and patient difficulty in adhering to treatment regimens.[A244170, A244175] Lenacapavir is a first-in-class caps…

Kategori:
AcetatesAcids, AcyclicAmides +17
Target Protein:
Gag-Pol polyprotein
Waktu ParuhThe median half-lif…
Vol. DistribusiThe steady state vo…
KlirensLenacapavir clearan…
Genetik -
Lenalidomide Approved DB00480
small molecule | CAS: 191732-72-6

Lenalidomide (previously referred to as CC-5013) is an immunomodulatory drug with potent antineoplastic, anti-angiogenic, and anti-inflammatory properties.[A228553] It is a 4-amino-glutamyl analogue of [thalidomide] [A228543] and like thalidomide, lenalidomid…

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +18
Target Protein:
Tumor necrosis factorProtein cereblonTumor necrosis factor ligand superfamily member 11 +2
Waktu ParuhIn healthy subjects…
Vol. DistribusiIn healthy male sub…
KlirensThe renal clearance…
Genetik -
Leniolisib Approved DB16217
small molecule | CAS: 1354690-24-6

Leniolisib is a potent and selective inhibitor of phosphoinositide 3-kinase ? (PI3K?). The FDA approved leniolisib on March 24, 2023, making it the first treatment for activated phosphoinositide 3-kinase delta syndrome (APDS).[L45758] APDS is a primary immuno…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe effective half-…
Vol. DistribusiThe systemic decay …
KlirensIn one study, healt…
Genetik -
Lenograstim Approved DB13144
biotech | CAS: 135968-09-1

Lenograstim is a recombinant granulocyte colony-stimulating factor used as an immunostimulating agent.

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +13
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiApparent distributi…
KlirensPlasma clearance of…
Genetik -
Lenomorelin DB11895
biotech | CAS: 258279-04-8

Lenomorelin has been investigated for the treatment and basic science of Cancer, Alcoholism, Metabolism, Hypopituitarism, and Frailty Syndrome, among others.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lentil Approved DB10645
biotech

Lentil allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lentinan DB13480
small molecule | CAS: 37339-90-5

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenvatinib Approved DB09078
small molecule | CAS: 417716-92-8

Lenvatinib is a receptor tyrosine kinase (RTK) inhibitor that inhibits the kinase activities of vascular endothelial growth factor (VEGF) receptors VEGFR1 (FLT1), VEGFR2 (KDR), and VEGFR3 (FLT4). Lenvatinib also inhibits other RTKs that have been implicated i…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +7
Waktu ParuhThe terminal elimin…
Vol. Distribusi-
Klirens-
Genetik -
Lenvervimab DB17814
biotech | CAS: 2055006-79-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenzilumab DB15148
biotech | CAS: 1229575-09-0

Lenzilumab is under investigation in clinical trial NCT02546284 (Study of Lenzilumab in Previously Treated Patients With Chronic Myelomonocytic Leukemia (CMML)).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lepirudin Approved DB00001
biotech | CAS: 138068-37-8

Lepirudin is a recombinant hirudin formed by 65 amino acids that acts as a highly specific and direct thrombin inhibitor.[L41539,L41569] Natural hirudin is an endogenous anticoagulant found in _Hirudo medicinalis_ leeches.[L41539] Lepirudin is produced in yea…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Target Protein:
Prothrombin
Waktu ParuhLepirudin has an in…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of le…
Genetik -
Leptazoline A DB15551
small molecule

Leptazoline A is a polar oxazoline from the Cyanobacterium Leptolyngbya sp. Also see [Leptazoline B], [Leptazoline C], and [Leptazoline D].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leptazoline B DB15552
small molecule

Leptazoline B is a polar oxazoline from the Cyanobacterium Leptolyngbya sp. Also see [Leptazoline A], [Leptazoline C], and [Leptazoline D].

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Leptazoline C DB15553
small molecule

Leptazoline C is a polar oxazoline from the Cyanobacterium Leptolyngbya sp. Also see [Leptazoline A], [Leptazoline B], and [Leptazoline D].

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Leptazoline D DB15554
small molecule

Leptazoline D is a polar oxazoline from the Cyanobacterium Leptolyngbya sp. Also see [Leptazoline A], [Leptazoline B], and [Leptazoline C].

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Leptin DB05098
small molecule | CAS: 169494-85-3

Although leptin is a circulating signal that reduces appetite, in general, obese people have an unusually high circulating concentration of leptin. These people are said to be resistant to the effects of leptin, in much the same way that people with type 2 di…

Kategori:
AdipokinesAmino Acids, Peptides, and ProteinsBiological Factors +6
Target Protein:
Leptin receptor
Waktu Paruh24.9+/-4.4 min
Vol. Distribusi-
Klirens-
Genetik -
Lepunafusp alfa DB19011
biotech | CAS: 2396411-71-3

Lepunafusp alfa is under investigation in clinical trial NCT04453085 (An Extension Study of JR-171-101 Study in Patients With MPS I).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lercanidipine Approved DB00528
small molecule | CAS: 100427-26-7

Lercanidipine is a calcium channel blocker of the dihydropyridine class. It is sold under various commercial names including Zanidip.

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAgents Causing Muscle Toxicity +25
Target Protein:
Voltage-dependent calcium channel gamma-1 subunitVoltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerdelimumab DB06557
biotech | CAS: 285985-06-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leridistim DB15095
biotech | CAS: 193700-51-5

Leridistim is under investigation in clinical trial NCT00004215 (Leridistim Compared With Filgrastim in Treating Older Patients With Acute Myeloid Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leriglitazone DB15021
small molecule | CAS: 146062-44-4

Leriglitazone is under investigation in clinical trial NCT03917225 (A Clinical Study to Evaluate the Effect of MIN-102 on the Progression of Friedreich's Ataxia in Male and Female Patients).

Kategori:
Alimentary Tract and MetabolismSulfur CompoundsThiazoles +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerisetron DB12964
small molecule | CAS: 143257-98-1

Lerisetron has been used in trials studying the supportive care of Nausea and Vomiting and Testicular Germ Cell Tumor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerociclib DB16218
small molecule | CAS: 1628256-23-4

Lerociclib is under investigation in clinical trial NCT02983071 (G1T38, a CDK 4/6 Inhibitor, in Combination With Fulvestrant in Hormone Receptor-positive, Her2-negative Locally Advanced or Metastatic Breast Cancer).

Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerodalcibep DB19071
biotech | CAS: 2250073-78-8

Lerodalcibep is under investigation in clinical trial NCT05004675 (Trial to Evaluate Efficacy and Safety of LIB003 and Inclisiran in High-risk CVD Patients).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leronlimab DB05941
biotech | CAS: 674782-26-4

Leronlimab, or PRO-140, is a human monoclonal antibody developed by CytoDyn.[L12684] It was first described in the literature in 2001.[A3922] This antibody binds to CCR5, which may be useful in treating HIV, cancers, and severely ill COVID-19 patients.[A19284…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +17
Target Protein:
C-C chemokine receptor type 5
Waktu ParuhThe half life of a …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lesinidase alfa DB15267
biotech | CAS: 1522433-40-4

Lesinidase alfa is under investigation in clinical trial NCT02324049 (Safety, Pharmacokinetics, and Pharmacodynamics/Efficacy of SBC-103 in Mucopolysaccharidosis III, Type B (MPS IIIB)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lesinurad Approved DB11560
small molecule | CAS: 878672-00-5

Lesinurad is an oral uric acid transporter 1 (URAT1) inhibitor indicated for the treatment of hyperuricemia associated with gout. It reduces serum uric acid concentration through the inhibition of URAT1, an enzyme responsible for reuptake of uric acid from th…

Kategori:
AcetatesAcids, AcyclicAntigout Preparations +15
Target Protein:
Solute carrier family 22 member 12Solute carrier family 22 member 11
Waktu Paruh-
Vol. DistribusiThe mean steady sta…
Klirens-
Genetik -
Lesopitron DB04970
small molecule | CAS: 132449-46-8

Lesopitron is an anxiolytic with pre- and post-synaptic 5-HT1A agonist activity, which is under development by Esteve.

Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh1.1 to 5.6 hours
Vol. Distribusi-
Klirens-
Genetik -
Lestaurtinib DB06469
small molecule | CAS: 111358-88-4

Deskripsi belum tersedia.

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 InhibitorsCytochrome P-450 CYP3A4 Inhibitors (strength unknown) +4
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letaplimab DB16679
biotech | CAS: 2283356-07-8

Letaplimab is under investigation in clinical trial NCT04485052 (Efficacy and Safety Evaluation of IBI188 in Combination With Azacitidine in Treatment of Patients With Acute Myeloid Leukemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LetibotulinumtoxinA Approved DB16820
biotech | CAS: 1800016-51-6

The aesthetic utility of botulinum toxin was discovered incidentally following its initial use in the treatment of facial spasmodic disorders in the early 1970s.[A249920] The first aesthetic use of botulinum toxin was reported in 1989, when [onabotulinumtoxin…

Kategori:
Acetylcholine Release InhibitorsBotulinum Toxins, Type ACentral Nervous System Depressants +2
Target Protein:
Synaptosomal-associated protein 25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letolizumab DB19072
biotech | CAS: 1450981-87-9

Letolizumab is under investigation in clinical trial NCT02273960 (Study to Evaluate Safety and Efficacy in Adult Subjects With ITP).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letosteine DB08939
small molecule | CAS: 53943-88-7

Letosteine is a mucolytic used in the treatment of chronic bronchopneumopathies and related conditions.

Kategori:
Cough and Cold PreparationsExpectorantsRespiratory System Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Letrozole Approved DB01006
small molecule | CAS: 112809-51-5

Letrozole, or CGS 20267, is an oral non-steroidal type II aromatase inhibitor first described in the literature in 1990.[A190543,A1559,L11623,L11626] It is a third generation aromatase inhibitor like [exemestane] and [anastrozole], meaning it does not signifi…

Kategori:
Agents Causing Muscle ToxicityAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +21
Target Protein:
Aromatase
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe average clearan…
Genetik -
Lettuce Approved DB10539
biotech

Lettuce allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leucanthemum vulgare pollen Approved DB15529
biotech

Leucanthemum vulgare pollen allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leucine DB00149
small molecule | CAS: 61-90-5

An essential branched-chain amino acid important for hemoglobin formation.

Kategori:
Amino AcidsAmino Acids, Branched-ChainAmino Acids, Essential +4
Target Protein:
Leucine--tRNA ligase, mitochondrialtRNA wybutosine-synthesizing protein 4Leucine carboxyl methyltransferase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leucovorin Approved DB00650
small molecule | CAS: 58-05-9

Folinic Acid (also known as 5-formyl tetrahydrofolic acid or leucovorin) is the 5-formyl derivative of tetrahydrofolic acid, a necessary co-factor in the body. Commercially available leucovorin is composed of a 1:1 racemic mixture of the dextrorotary and levo…

Kategori:
AntidotesCoenzymesCompounds used in a research, industrial, or household setting +15
Target Protein:
Proton-coupled folate transporterDihydrofolate reductase
Waktu Paruh6.2 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene C4 DB08855
small molecule | CAS: 72025-60-6

The conjugation product of LEUKOTRIENE A4 and glutathione. It is the major arachidonic acid metabolite in macrophages and human mast cells as well as in antigen-sensitized lung tissue. It stimulates mucus secretion in the lung, and produces contractions of no…

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2Multidrug resistance-associated protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leukotriene D4 DB11858
small molecule | CAS: 73836-78-9

Leukotriene D4 has been used in trials studying the diagnostic of Asthma and Allergic Rhinitis.

Kategori:
Arachidonic AcidsAutacoidsBiological Factors +8
Target Protein:
Cysteinyl leukotriene receptor 1Cysteinyl leukotriene receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leupeptin DB16961
small molecule | CAS: 55123-66-5

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCathepsins, antagonists & inhibitorsCysteine Proteinase Inhibitors +4
Target Protein:
Plasmepsin-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leuprolide Approved DB00007
biotech | CAS: 53714-56-0

Leuprolide is a synthetic 9-residue peptide analogue of gonadotropin-releasing hormone (GnRH). Unlike the endogenous decapeptide GnRH, leuprolide contains a single D-amino acid (D-leucyl) residue, which helps to increase its circulating half-life from three t…

Kategori:
Adrenal Cortex HormonesAgents Causing Muscle ToxicityAmino Acids, Peptides, and Proteins +25
Target Protein:
Gonadotropin-releasing hormone receptorProgonadoliberin-1
Waktu ParuhLeuprolide has a te…
Vol. DistribusiLeuprolide has an a…
KlirensLeuprolide administ…
Genetik -
Leuvectin DB17303
biotech

Leuvectin (formerly known as VCL-1102) is a component of gene therapy along with cationic lipid 1,2-dimyristyloxypropyl-3-dimethyl-hydroxyethyl ammonium bromide/dioleyl-phosphatidyl-ethanolamine (DMRIE/DOPE).[A254711]

Kategori:
Biological ProductsComplex MixturesGene Transfer Techniques +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Levacetylmethadol Approved DB01227
small molecule | CAS: 1477-40-3

Levacetylmethadol is a narcotic analgesic with a long onset and duration of action. It is used mainly in the treatment of narcotic dependence. Levacetylmethadol was withdrawn from use in the European Union due to its high risk of QT interval prolongation.…

Kategori:
AnalgesicsAnticholinergic AgentsCentral Nervous System Agents +20
Target Protein:
Mu-type opioid receptorNeuronal acetylcholine receptor subunit beta-4Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh2.6 days
Vol. Distribusi-
Klirens-
Genetik -
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