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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Halaman 146 / 321
Fibrinogen human Approved DB09222
biotech | CAS: 9001-32-5

Fibrinogen concentrate (human) is a hematological agent. It works by replacing a specific protein in the blood, fibrinogen (factor I), that helps with blood clotting. It is a soluble plasma glycoprotein with a molecular weight of about 340 kDa and is a physi…

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsBiological Factors +8
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Fibrinolysin DB05254
biotech | CAS: 9004-09-5

Fibrinolysin consists of two polypeptide chains, one light and one heavy, linked by a disulfide bond. The light chain has a molecular weight of approximately 27,000 Da and contains the active center of Fibrinolysin; the heavy chain has a molecular weight of a…

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCardiovascular Agents +11
Target Protein:
Plasminogen activator inhibitor 1Urokinase-type plasminogen activator
Waktu ParuhAlmost completely i…
Vol. Distribusi-
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Genetik -
biotech | CAS: 106096-92-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 1 +4
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Ficlatuzumab DB11680
biotech | CAS: 1174900-84-5

Ficlatuzumab has been used in trials studying the treatment of Acute Myeloid Leukemia, Non-small Cell Lung Cancer, Mullerian Mixed Tumor of Ovary, Relapsed Acute Myeloid Leukemia, and Refractory Acute Myeloid Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Ficonalkib DB18774
small molecule | CAS: 2233574-95-1

Deskripsi belum tersedia.

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Fidanacogene elaparvovec Approved DB16783
biotech | CAS: 1954659-47-2

Fidanacogene elaparvovec is a liver-specific adeno-associated virus (AAV) vector containing a codon-optimized human coagulation FIX gene that was investigated as a potential treatment for hemophilia B.[L46691] Hemophilia B is a rare X-linked genetic disorder …

Kategori:
Adeno-associated Viral Vector TherapiesHepatotoxic Agents
Target Protein:
Coagulation factor IX (F9)
Waktu Paruh-
Vol. DistribusiIn a monkey biodist…
KlirensClearance of vector…
Genetik -
Fidarestat DB02021
small molecule | CAS: 136087-85-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member B10
Waktu Paruh-
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Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Fidrisertib DB18064
small molecule | CAS: 2141955-96-4

Deskripsi belum tersedia.

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Figitumumab DB11685
biotech | CAS: 943453-46-1

Figitumumab has been used in trials studying the treatment of Sarcoma, Solid Tumor, Breast Cancer, Lung Neoplasms, and Advanced Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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Figopitant DB12122
small molecule | CAS: 502422-74-4

Figopitant is under investigation in clinical trial NCT02209714 (Safety, Tolerability and Pharmacodynamics After Oral Administration of BIIF 1149 BS in Healthy Male Volunteers).

Kategori:
AcetamidesAmidesBenzene Derivatives
Target Protein:
Substance-P receptor
Waktu Paruh-
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Filaminast DB02660
small molecule | CAS: 141184-34-1

Filaminast is a phosphodiesterase 4 inhibitor (PDE4 inhibitor). As such, has potential in the treatment of asthma and chronic obstructive pulmonary disease (COPD).

Kategori:
AminesHydroxylamines
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
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Filanesib DB06040
small molecule | CAS: 885060-09-3

Filanesib is a potent Kinesin Spindle Protein (KSP) inhibitor that caused marked tumor regression in preclinical models of human solid tumors and human leukemias, often leading to durable responses.

Kategori:
Antimitotic AgentsAntineoplastic AgentsMitosis Modulators +2
Target Protein:
Kinesin-like protein KIF11
Waktu Paruh-
Vol. Distribusi-
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Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
Klirens-
Genetik -
Filgrastim Approved DB00099
biotech | CAS: 121181-53-1

Filgrastim is a short-acting recombinant, non-pegylated human granulocyte colony-stimulating factor (G-CSF) analog produced by recombinant DNA technology. It has an amino acid sequence identical to endogenous G-CSF, but it is non-glycosylated unlike the endog…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBiological Factors +10
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhAfter intravenous a…
Vol. DistribusiAfter intravenous a…
KlirensClearance rates of …
Genetik -
Filibuvir DB11878
small molecule | CAS: 877130-28-4

Filibuvir has been used in trials studying the treatment of Hepatitis, Hepatitis C, and Chronic Hepatitis C.

Kategori:
PyransRNA Replicase, antagonists & inhibitorsRNA-Dependent RNA Polymerase, antagonists & inhibitors
Target Protein:
Genome polyprotein
Waktu Paruh-
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Filociclovir DB12438
small molecule | CAS: 632325-71-4

Filociclovir is under investigation in clinical trial NCT01433835 (Safety and Pharmacokinetics of Single Oral Doses of Filociclovir in Healthy Volunteers).

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Filorexant DB12158
small molecule | CAS: 1088991-73-4

Filorexant has been used in trials studying the prevention and treatment of Migraine, Headache, Polysomnography, Diabetic Neuropathy, Painful, and Major Depressive Disorder, Recurrent.

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Fimaporfin DB17253
small molecule | CAS: 1443547-43-0

Deskripsi belum tersedia.

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Fimasartan DB09279
small molecule | CAS: 247257-48-3

Fimasartan is an angiotensin II receptor antagonist (ARB) drug employed in the treatment of both hypertension and heart failure. It has been found to be safe when administered with hydrochlorothiazide (a diuretic) in clinical trials. Fimasartan was initially …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin II receptor blockers (ARBs) and calcium channel blockers +8
Target Protein:
Type-1 angiotensin II receptor
Waktu ParuhThe half life of el…
Vol. Distribusi-
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Fimepinostat DB11891
small molecule | CAS: 1339928-25-4

Fimepinostat (CUDC-907) has been used in trials studying the treatment of lymphoma, solid tumors, breast cancer, multiple myeloma, and NUT midline carcinoma, among others.

Kategori:
Antineoplastic AgentsHistone Deacetylase InhibitorsOxazines +3
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
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Finafloxacin Approved DB09047
small molecule | CAS: 209342-40-5

Finafloxacin is a fluoroquinolone antibiotic indicated in the treatment of acute otitis externa (swimmer's ear) caused by the bacteria Pseudomonas aeruginosa and Staphylococcus aureus. Finafloxacin is marketed by Novartis under the brand Xtoro™, and was appro…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu Paruh-
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Finasteride Approved DB01216
small molecule | CAS: 98319-26-7

Finasteride is a synthetic 4-azasteroid compound [L10565] and specific inhibitor of steroid Type II 5?-reductase, which is an intracellular enzyme that converts the androgen testosterone into 5?-dihydrotestosterone (DHT). It works in a similar fashion as [dut…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +22
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 2Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 1 +1
Waktu ParuhIn healthy young su…
Vol. DistribusiThe volume of distr…
KlirensIn healthy young su…
Genetik -
Finerenone Approved DB16165
small molecule | CAS: 1050477-31-0

Finerenone, or BAY 94-8862, is a mineralocorticoid receptor antagonist indicated to reduce the risk of sustained decline in glomerular filtration rate, end stage kidney disease, cardiovascular death, heart attacks, and hospitalization due to heart failure in …

Kategori:
Agents causing hyperkalemiaCytochrome P-450 CYP2C8 SubstratesCytochrome P-450 CYP3A Substrates +6
Target Protein:
Mineralocorticoid receptor
Waktu ParuhThe half life of a …
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Fingolimod Approved DB08868
small molecule | CAS: 162359-55-9

Multiple sclerosis, or MS, is a devastating inflammatory disease that often progresses and causes severe neurological, physical, and cognitive effects.[A176474] Fingolimod is a sphingosine 1-phosphate receptor modulator for the treatment of relapsing-remittin…

Kategori:
AlcoholsAminesAmino Alcohols +16
Target Protein:
D(3) dopamine receptorSphingosine kinase 1Sphingosine 1-phosphate receptor 5 +4
Waktu ParuhThe half-life of fi…
Vol. DistribusiThe volume of distr…
KlirensFingolimod blood cl…
Genetik -
FINLAY-FR-1 DB16524
biotech

FINLAY-FR-1, also known as Soberana 01, is a vaccine candidate for COVID-19 that is being led developmentally by the Finlay Vaccine Institute[L31373]. It is currently being tested in the clinical trial RPCEC00000332 (Phase I / II, randomized, controlled, adap…

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Finotonlimab DB18859
biotech | CAS: 2350298-85-8

Finotonlimab is under investigation in clinical trial NCT04560894 (SCT-I10A Plus SCT510 Versus Sorafenib as First-line Therapy for Advanced Hepatocellular Carcinoma).

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Fipamezole DB06585
small molecule | CAS: 150586-58-6

Deskripsi belum tersedia.

Kategori:
Indenes
Waktu Paruh-
Vol. Distribusi-
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Fipaxalparant DB18124
small molecule | CAS: 1195941-38-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysophosphatidic acid receptor 1Lysophosphatidic acid receptor 3
Waktu Paruh-
Vol. Distribusi-
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Fipexide DB13790
small molecule | CAS: 34161-24-5

Deskripsi belum tersedia.

Kategori:
Nervous SystemPsychoanalepticsPsychostimulants, Agents Used for ADHD and Nootropics
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Firategrast DB12732
small molecule | CAS: 402567-16-2

Firategrast has been used in trials studying the treatment of Multiple Sclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +5
Waktu Paruh-
Vol. Distribusi-
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Firazorexton DB19440
small molecule | CAS: 2274802-95-6

Firazorexton is under investigation in clinical trial NCT04096560 (A Study of TAK-994 in Adults With Type 1 and Type 2 Narcolepsy).

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Firocoxib DB09217
small molecule | CAS: 189954-96-9

Firocoxib is a cycooxygenase-2 (COX-2) selective non-steroidal anti-inflammatory drug. It currently approved for veterinary use in dogs and horses under the brand names Equioxx and Previcox. Firocoxib was the first COX-2 inhibitor approved by the U.S. Food an…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +6
Target Protein:
Prostaglandin G/H synthase 2
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biotech

Deskripsi belum tersedia.

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Firsocostat DB16166
small molecule | CAS: 1434635-54-7

Firsocostat is under investigation in clinical trial NCT02781584 (Safety, Tolerability, and Efficacy of Selonsertib, Firsocostat, and Cilofexor in Adults With Nonalcoholic Steatohepatitis (NASH)).

Kategori:
Acids, AcyclicButyratesEnzyme Inhibitors +5
Waktu Paruh-
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Firtecan pegol DB14953
small molecule | CAS: 946062-05-1

Firtecan pegol is under investigation in clinical trial NCT01036113 (A Phase 2 Study of EZN-2208 in Patients With Metastatic Breast Cancer).

Kategori:
AlcoholsAlkaloidsEthylene Glycols +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Fisetin DB07795
small molecule | CAS: 528-48-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Cyclin-dependent kinase 6Fatty acid synthaseCyclin homolog
Waktu Paruh-
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Fish liver oil Approved DB15481
biotech | CAS: 8009-00-5

Deskripsi belum tersedia.

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Fish oil Approved DB13961
biotech

Fish oil is a component of SMOFLIPID, which was FDA approved in July 2016. It is indicated in adults as a source of calories and essential fatty acids for parenteral nutrition when oral or enteral nutrition is not possible, insufficient, or contraindicated. …

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Diacylglycerol O-acyltransferase 2Prostaglandin G/H synthase 2Free fatty acid receptor 4 +8
Waktu ParuhThe half-life of EP…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of EP…
Genetik -
Fisogatinib DB16167
small molecule | CAS: 1707289-21-1

Fisogatinib is under investigation in clinical trial NCT04194801 (A Phase Ib/ii Study of Fisogatinib(blu-554) in Subjects With Hepatocellular Carcinoma).

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
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Fispemifene DB06640
small molecule | CAS: 341524-89-8

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsStilbenes
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Fitusiran DB15002
biotech | CAS: 1499251-18-1

Fitusiran is under investigation in clinical trial NCT02554773 (An Open-label Extension Study of an Investigational Drug, ALN-AT3SC, in Patients With Moderate or Severe Hemophilia A or B).

Kategori:
Amino SugarsAntisense Elements (Genetics)Carbohydrates +7
Waktu Paruh-
Vol. Distribusi-
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FK-614 DB12557
small molecule | CAS: 193012-35-0

FK614 has been used in trials studying the treatment of Diabetes Mellitus.

Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
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FK-960 DB06465
small molecule | CAS: 133920-70-4

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
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FK352B DB06484
small molecule | CAS: 143881-08-7

FK352B is a adenosine A1 antagonist that is developed for the treatment of dialysis-induced hypotension.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
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FKB-001 DB02888
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
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Genetik -
Flavin adenine dinucleotide Approved DB03147
small molecule | CAS: 146-14-5

A condensation product of riboflavin and adenosine diphosphate. The coenzyme of various aerobic dehydrogenases, e.g., D-amino acid oxidase and L-amino acid oxidase. (Lehninger, Principles of Biochemistry, 1982, p972) Flavin adenine dinucleotide is approved f…

Kategori:
Adenine NucleotidesBiological FactorsCoenzymes +13
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]Nitric oxide synthase 1Dihydropyrimidine dehydrogenase [NADP(+)] +83
Waktu Paruh-
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Flavin mononucleotide Approved DB03247
small molecule | CAS: 146-17-8

A coenzyme for a number of oxidative enzymes including NADH DEHYDROGENASE. It is the principal form in which RIBOFLAVIN is found in cells and tissues.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +11
Target Protein:
Flavin reductase (NADPH)2-Hydroxyacid oxidase 1Pyridoxine-5'-phosphate oxidase +51
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
D-amino-acid oxidase
Waktu Paruh-
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small molecule

Deskripsi belum tersedia.

Target Protein:
Cholesterol oxidase
Waktu Paruh-
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