Hasil Filter

11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (11778)

Halaman 145 / 236
Melarsoprol DB12864
small molecule | CAS: 494-79-1

Melarsoprol is under investigation in clinical trial NCT00330148 (Randomized Clinical Trial of Three Drug Combinations for Late-Stage Gambiense Human African Trypanosomiasis).

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAnti-Infective AgentsAntiparasitic Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melatonin Approved DB01065
small molecule | CAS: 73-31-4

Melatonin is a biogenic amine that is found in animals, plants and microbes. Aaron B. Lerner of Yale University is credited for naming the hormone and for defining its chemical structure in 1958. In mammals, melatonin is produced by the pineal gland. The pin…

Kategori:
AminesAntioxidantsBiogenic Amines +21
Target Protein:
Melatonin receptor type 1AMelatonin receptor type 1BRibosyldihydronicotinamide dehydrogenase [quinone] +7
Waktu Paruh35 to 50 minutes
Vol. Distribusi-
Klirens-
Genetik -
Meldonium DB13723
small molecule | CAS: 76144-81-5

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicCardiac TherapyCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Melevodopa DB13313
small molecule | CAS: 7101-51-1

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Aromatic +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meloxicam Approved DB00814
small molecule | CAS: 71125-38-7

Meloxicam is a nonsteroidal anti-inflammatory drug (NSAID) used to relieve various types of pain, including pain caused by musculoskeletal conditions, osteoarthritis, and rheumatoid arthritis.[A190189] With a longer half-life than most other NSAIDS, it is a f…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +28
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe half-life of me…
Vol. DistribusiThe volume of distr…
KlirensAfter an oral dose,…
Genetik -
Melperone DB09224
small molecule | CAS: 3575-80-2

Melperone is an atypical antipsychotic of the butyrophenone chemical class, making it structurally related to the typical antipsychotic haloperidol. Melperone has been used for a span of greater than 30 years in the European Union [L1316]. It has been well e…

Kategori:
Antiarrhythmic agentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +17
Target Protein:
D(2) dopamine receptor
Waktu ParuhApproximately 3-4 h…
Vol. Distribusi-
Klirens-
Genetik -
Melphalan Approved DB01042
small molecule | CAS: 148-82-3

Melphalan is a nitrogen mustard or bischloroethylamine type alkylating agent.[L40928] It was first synthesized in the early 1950s by substituting L-phenylalanine for the methyl group on nitrogen mustard.[A261150, A261155] Melphalan is used in the treatment of…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +17
Target Protein:
DNA
Waktu ParuhIn patients given a…
Vol. DistribusiThe volume of distr…
KlirensAverage total body …
Genetik -
Melphalan flufenamide Approved DB16627
small molecule | CAS: 380449-51-4

Melphalan flufenamide, also known as melflufen or J1, is a prodrug of [melphalan].[A230123,L32173] Melphalan flufenamide is more readily uptaken by cells than melphalan, and is cleaved to the active metabolite by aminopeptidases.[A230123] _In vitro_ models sh…

Kategori:
Alkylating ActivityAlkylating DrugsAmino Acids +12
Target Protein:
DNA
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Melrilimab DB16373
biotech | CAS: 2222865-46-3

Melrilimab is under investigation in clinical trial NCT03207243 (Efficacy and Safety Study of GSK3772847 in Subjects With Moderately Severe Asthma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEM 1003 DB05547
small molecule

MEM 10003 was under investigation in clinical trial NCT00257673 (Safety and Efficacy of MEM 1003 Versus Placebo in Patients With Mild to Moderate Alzheimer's Disease) for the treatment of Alzheimer's Disease.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MEM136 DB17321
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Memantine Approved DB01043
small molecule | CAS: 19982-08-2

Initially approved by the FDA in 2013, memantine is an N-methyl-D-aspartate (NMDA) receptor antagonist used in the management of Alzheimer's Disease (AD). It is different from many other Alzheimer's Disease medications, as it works by a different mechanism t…

Kategori:
Anti-Dementia DrugsAnti-Dyskinesia AgentsAnti-Parkinson Drugs +20
Target Protein:
Glutamate (NMDA) receptor5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +3
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThis drug is cleare…
Genetik -
Menadione Approved DB00170
small molecule | CAS: 58-27-5

A synthetic naphthoquinone without the isoprenoid side chain and biological activity, but can be converted to active vitamin K2, menaquinone, after alkylation in vivo.

Kategori:
Antifibrinolytic AgentsBlood and Blood Forming OrgansCoagulants +45
Target Protein:
Aldehyde oxidaseVitamin K-dependent gamma-carboxylaseVitamin K epoxide reductase complex subunit 1 +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menaquinone 6 DB14936
small molecule | CAS: 84-81-1

Menaquinone 6 is under investigation in clinical trial NCT01194778 (Comparison of Efficacy of Different Dosages Vitamin K2).

Kategori:
CoagulantsDiet, Food, and NutritionDiterpenes +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menaquinone 7 DB13075
small molecule | CAS: 2124-57-4

Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).

Kategori:
CoagulantsDiterpenesHematologic Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menglytate DB15983
small molecule | CAS: 579-94-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Meningococcal (groups A, C, Y and W-135) oligosaccharide diphtheria CRM197 conjugate vaccine is used to prevent invasive meningococcal disease, which is caused by bacteria _Neisseria meningitidis_ entering the bloodstream and invading the blood-brain barrier …

Kategori:
Diphtheria VaccinesMeningococcal VaccinesVaccines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Meningococcal group C polysaccharide is group-specific polysaccharide antigens extracted and purified from *Neisseria meningitidis* serogroup C. *N. meningitidis* is a bacteria that causes endemic and epidemic diseases including meningitis and meningococcemia…

Kategori:
Actively Acquired ImmunityAntigensAntigens, Bacterial +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Meningococcal group W-135 polysaccharide is group-specific polysaccharide antigens extracted and purified from *Neisseria meningitidis* serogroup W-135. *N. meningitidis* is a bacteria that causes endemic and epidemic diseases including meningitis and meningo…

Kategori:
Actively Acquired ImmunityInactivated Meningococcal Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepartricin DB13633
small molecule | CAS: 11121-32-7

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAlkenesAnti-Bacterial Agents +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meperidine Approved DB00454
small molecule | CAS: 57-42-1

A narcotic analgesic that can be used for the relief of most types of moderate to severe pain, including postoperative pain and the pain of labor. Prolonged use may lead to dependence of the morphine type; withdrawal symptoms appear more rapidly than with mor…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that reduce seizure threshold +34
Target Protein:
Kappa-type opioid receptorGlutamate receptor ionotropic, NMDA 1Glutamate receptor ionotropic, NMDA 2B +9
Waktu ParuhInitial distributio…
Vol. DistribusiMeperidine crosses …
Klirens-
Genetik -
Mephenesin Approved DB13583
small molecule | CAS: 59-47-2

Mephenesin is a synthetic cresol glyceryl ether which produces transient muscle relaxation and paralysis via central nervous system depression [A32760]. It first entered use in the 1950s.

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mephenoxalone DB13754
small molecule | CAS: 70-07-5

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsCentral Nervous System DepressantsMuscle Relaxants +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepindolol DB13530
small molecule | CAS: 23694-81-7

Mepindolol is a 2-methyl derivative of pindolol. It is a beta blocker.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +12
Target Protein:
Beta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepiprazole DB09197
small molecule | CAS: 20326-12-9

Mepiprazole is a minor tranquilizer with a phenylpiperazine structure. It is a pyrazolyl-alkyl-piperazine derivative. Mepiprazole mediates a weak inhibitory action on the uptake of 5-HT on hypothalamic neurons [A7816]. Mepiprazole is marketed in Spain for th…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepixanox DB13579
small molecule | CAS: 17854-59-0

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingRespiratory System AgentsXanthenes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meplazumab DB16465
biotech

Meplazumab is a humanized anti-CD147 antibody being investigated as an add-on therapy in patients with COVID-19 pneumonia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntibodies +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mepolizumab Approved DB06612
biotech | CAS: 196078-29-2

Eosinophils are involved in inflammatory immune responses, and prolonged hypereosinophilia (typically defined as absolute eosinophil levels of 1500/mm<sup>3</sup> or more) is associated with a spectrum of diseases, including severe asthma, eosinophilic granul…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Interleukin-5
Waktu ParuhMepolizumab has a m…
Vol. DistribusiMepolizumab has a p…
KlirensMepolizumab has an …
Genetik -
Meprednisone Approved DB09383
small molecule | CAS: 1247-42-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesCorticosteroidsCorticosteroids for Systemic Use +20
Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meprobamate Approved DB00371
small molecule | CAS: 57-53-4

A carbamate with hypnotic, sedative, and some muscle relaxant properties, although in therapeutic doses reduction of anxiety rather than a direct effect may be responsible for muscle relaxation. Meprobamate has been reported to have anticonvulsant actions aga…

Kategori:
Acids, AcyclicAnti-Anxiety AgentsCarbamates +10
Target Protein:
Peptide deformylase, mitochondrialProtein kinase C epsilon typeGABA(A) Receptor +6
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Meptazinol DB13478
small molecule | CAS: 54340-58-8

Deskripsi belum tersedia.

Kategori:
AnalgesicsAzepinesCentral Nervous System Agents +10
Target Protein:
Cholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mequinol Approved DB09516
small molecule | CAS: 150-76-5

Mequinol is a phenol used in various applications. It is used as an inhibitor for acrylic monomers and acrylonitirles, as a stabilizer for chlorinated hydrocarbons and ethyl cellulose, as an ultraviolet inhibitor, as a chemical intermediate in the manufacture…

Kategori:
AntioxidantsBenzene DerivativesBiological Factors +11
Waktu ParuhMequinol demonstrat…
Vol. DistribusiThe volume of distr…
KlirensReadily accessible …
Genetik -
Mequitazine DB01071
small molecule | CAS: 29216-28-2

Mequitazine is a histamine H1 antagonist (antihistamine). It competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract. It provides effective, temporary relief of sneezing, wa…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBronchodilator Agents +15
Target Protein:
Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meradimate Approved DB11096
small molecule | CAS: 134-09-8

Meradimate, before known as menthyl anthranilate, is used in a maximal concentration of 5% in different products as a UV filter.[T200] It is currently required to be named as meradimate in all FDA approved OTC products. Meradimate is approved by the FDA and H…

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Waktu ParuhAs meradimate is no…
Vol. DistribusiAs meradimate is no…
KlirensAs meradimate is no…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase IMP-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2Divalent-cation tolerance protein CutA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7487-94-7

Mercury chloride (HgCl2) is a highly toxic compound that volatizes slightly at ordinary temperature and appreciably at 100 degrees C. It is corrosive to mucous membranes and used as a topical antiseptic and disinfectant. Mercuric chloride was used to disinfec…

Kategori:
Anti-Infective AgentsAnti-Infective Agents, LocalAntiseptics and Disinfectants +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mercuric iodide DB04445
small molecule | CAS: 7774-29-0

Deskripsi belum tersedia.

Kategori:
AnionsAntiseptics and DisinfectantsDermatologicals +4
Target Protein:
Sulfotransferase 2A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Merestinib DB12381
small molecule | CAS: 1206799-15-6

Merestinib has been used in trials studying the treatment of Cancer, Solid Tumor, Advanced cancer, ColoRectal Cancer, and Metastatic Cancer, among others.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingNicotinic Acids +3
Target Protein:
Hepatocyte growth factor receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mericitabine DB12045
small molecule | CAS: 940908-79-2

Mericitabine has been investigated for the treatment of Hepatitis C, Chronic. Mericitabine is a polymerase inhibitor being developed for the treatment of chronic hepatitis C. Mericitabine is a prodrug of PSI-6130, which demonstrated excellent potency in p…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Merimepodib DB04862
small molecule | CAS: 198821-22-6

Merimepodib (VX-497) is a novel noncompetitive inhibitor of IMPDH. Merimepodib is orally bioavailable and inhibits the proliferation of primary human, mouse, rat, and dog lymphocytes at concentrations of approximately 100 nM.

Kategori:
Acids, AcyclicAmidesBenzene Derivatives +1
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Receptor tyrosine-protein kinase erbB-2Epidermal growth factor receptor +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meropenem Approved DB00760
small molecule | CAS: 96036-03-2

Meropenem is a broad-spectrum carbapenem antibiotic. It is active against Gram-positive and Gram-negative bacteria. Meropenem exerts its action by penetrating bacterial cells readily and interfering with the synthesis of vital cell wall components, which lead…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
D-alanyl-D-alanine carboxypeptidase DacB
Waktu ParuhApproximately 1 hou…
Vol. Distribusi-
Klirens-
Genetik -
Merotocin DB12932
biotech | CAS: 1190083-57-8

Merotocin has been used in trials studying the treatment of Preterm Delivery.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mersalyl DB09338
small molecule | CAS: 486-67-9

Mersalyl is the sodium salt form of mersalyl acid, a mercurial diuretic. It is an outdated drug, and its approval has been discontinued by the FDA. Mersalyl acid is currently replaced by less toxic non-mercury containing diuretics [L1575, L1577]. The sodium s…

Kategori:
Alkylmercury CompoundsDiureticsDrugs that are Mainly Renally Excreted +5
Target Protein:
Alkaline phosphatase, tissue-nonspecific isozymeAquaporin-1Monocarboxylate transporter 1
Waktu Paruh-
Vol. Distribusi-
KlirensThe hepatobiliary e…
Genetik -
Mertiatide DB15780
small molecule | CAS: 66516-09-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Mesalazine Approved DB00244
small molecule | CAS: 89-57-6

An anti-inflammatory agent, structurally related to the salicylates and non-steroidal anti-inflammatory drugs like acetylsalicylic acid, which is active in inflammatory bowel disease [A174022]. Although demonstrably effective in treating and maintaining remis…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAminosalicylate +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Polyunsaturated fatty acid 5-lipoxygenase +4
Waktu ParuhFor the delayed-rel…
Vol. DistribusiFor the extended-re…
KlirensThe mean (SD) renal…
Genetik -
Mesdopetam DB16229
small molecule | CAS: 1403894-72-3

Mesdopetam is under investigation in clinical trial NCT04435431 (A Clinical Study of Mesdopetam in Patients With Parkinson's Disease Experiencing Levodopa Induced Dyskinesia).

Kategori:
AminesBenzene DerivativesDopamine Agents +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 147-73-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7201–7250 dari 11778
Sebelumnya Halaman 145 / 236 Berikutnya