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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 145 / 252
Larcaviximab DB17775
biotech | CAS: 1792982-56-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laromustine DB05817
small molecule | CAS: 173424-77-6

VNP40101M is a novel alkylating agent that has been used in trials studying the treatment of Leukemia, Lymphoma, Lung Cancer, Small Intestine Cancer, and Myelodysplastic Syndromes, among others.

Kategori:
AmidesSulfonesSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laronidase Approved DB00090
biotech | CAS: 210589-09-6

Human recombinant alpha-L-iduronidase, 628 residues (mature form), produced by recombinant DNAtechnology in a Chinese hamster ovary cell line. Laronidase is a glycoprotein with a molecular weight of approximately 83 kD. The predicted amino acid sequence of th…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Iduronic acid
Waktu Paruh1.5-3.6 hrs
Vol. Distribusi-
Klirens-
Genetik -
Laropiprant Approved DB11629
small molecule | CAS: 571170-77-9

Laropiprant is an ingredient in the EMA-withdrawn product Pelzont.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prostaglandin E2 receptor EP2 subtype3-hydroxy-3-methylglutaryl-coenzyme A reductaseThromboxane A2 receptor +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Larotaxel DB12984
small molecule | CAS: 156294-36-9

Larotaxel has been used in trials studying the treatment of Cancer, Metastases, Breast Cancer, Breast Neoplasms, and Pancreatic Neoplasms, among others.

Kategori:
CyclodecanesCycloparaffinsDiterpenes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Larotrectinib Approved DB14723
small molecule | CAS: 1223403-58-4

Larotrectinib is an orally administered inhibitor of tropomyosin receptor kinase (Trk), a receptor tyrosine kinase activated by neurotrophins which is mutated in a variety of cancer cell types and plays an important role in tumor cell growth and survival.[L49…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +8
Target Protein:
High affinity nerve growth factor receptorBDNF/NT-3 growth factors receptorNT-3 growth factor receptor
Waktu ParuhIn healthy subjects…
Vol. DistribusiFollowing intraveno…
KlirensThe mean clearance …
Genetik -
Larsucosterol DB18079
small molecule | CAS: 884905-07-1

Deskripsi belum tersedia.

Kategori:
CholestanesCholestenesFused-Ring Compounds +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lartesertib DB19045
small molecule | CAS: 2495096-26-7

Lartesertib is under investigation in clinical trial NCT06433219 (Tuvusertib Combined With Niraparib or Lartesertib in Participants With Epithelial Ovarian Cancer (Ddriver EOC 302)).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2425817-08-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAS-191954 DB17816
small molecule | CAS: 1403947-26-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lasalocid DB11423
small molecule | CAS: 25999-31-9

Lasalocid is an agent that presents antibacterial and coccidiostat activities. It is produced by strains of _Streptomyces lasaliensis_.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntiparasitic Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lasmiditan Approved DB11732
small molecule | CAS: 439239-90-4

Lasmiditan is an oral medication used in the termination of migraine headaches that was first approved for use in the United States in October 2019.[L9338,L9356] It was also approved by the European Commission on August 17, 2022.[L43997] Traditionally, the…

Kategori:
AmidesAnalgesicsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 1F
Waktu ParuhThe mean eliminatio…
Vol. DistribusiLasmiditan has been…
Klirens-
Genetik -
Lasofoxifene Approved DB06202
small molecule | CAS: 180916-16-9

Lasofoxifene is a non-steroidal 3rd generation selective estrogen receptor modulator (SERM) that selectively binds to both ER? and ER? with high affinity. It is a naphthalene derivative marketed for prevention and treatment of osteoporosis and for the treatme…

Kategori:
Genito Urinary System and Sex HormonesNaphthalenesSelective Estrogen Receptor Modulators +1
Target Protein:
Fusion glycoprotein F0Estrogen receptorEstrogen receptor beta +1
Waktu ParuhElimination half-li…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Latamoxef Approved DB04570
small molecule | CAS: 64952-97-2

Latamoxef is a broad- spectrum beta-lactam antibiotic similar in structure to the cephalosporins except for the substitution of an oxaazabicyclo moiety for the thiaazabicyclo moiety of certain cephalosporins. It has been proposed especially for the meningitid…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 3Penicillin-binding protein 1A +2
Waktu Paruh1.6 hours
Vol. Distribusi8.51 L
Klirens-
Genetik -
Latanoprost Approved DB00654
small molecule | CAS: 130209-82-4

Latanoprost is a prodrug analog of prostaglandin F2 alpha that is used to treat elevated intraocular pressure (IOP). It was initially approved by the FDA in 1998. Latanoprost is the first topical prostaglandin F2 alpha analog used for glaucoma treatment.[A184…

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +18
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Latanoprost acid Approved DB19360
small molecule | CAS: 41639-83-2

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latanoprostene bunod Approved DB11660
small molecule | CAS: 860005-21-6

Latanoprostene Bunod has been used in trials studying the treatment of Glaucoma, Ocular Hypertension, Open-Angle Glaucoma, Open Angle Glaucoma, and Intraocular Pressure. As of November 2, 2017 the FDA approved Bausch + Lomb's Vyzulta (latanoprostene bunod …

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +12
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUnfortunately there…
KlirensSince latanoprost a…
Genetik -
Latiglutenase DB06326
biotech | CAS: 1360452-96-5

Deskripsi belum tersedia.

Kategori:
Celiac Disease, drug therapyEnzymesEnzymes and Coenzymes +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latozinemab DB16978
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latrepirdine DB11725
small molecule | CAS: 3613-73-8

Latrepirdine has been investigated for the treatment of Alzheimer's Disease and Huntington's Disease.

Kategori:
Alzheimer DiseaseHeterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 6Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Latrunculin A DB02621
small molecule | CAS: 76343-93-6

Latrunculin A is an actin binding macrolide purified from the red sea sponge Latrunculia magnifica. It is under investigation for the treatment of cancer. It disrupts actin polymerization, prevents mitotic spindle formation and thus cell replication.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleGelsolinIota toxin component Ia
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laurocapram Approved DB17308
small molecule | CAS: 59227-89-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAVA-051 DB18395
biotech

LAVA-051 is a humanized V?9V?2-T cell-engaging bispecific antibody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavender oil Approved DB14566
biotech | CAS: 8000-28-0

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin A DB16768
small molecule | CAS: 125697-92-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEnzyme InhibitorsTyrosine Kinase Inhibitors
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase Lck
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavendustin b DB16760
small molecule | CAS: 125697-91-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lavoltidine DB12884
small molecule | CAS: 76956-02-0

Lavoltidine has been used in trials studying the diagnostic of Reflux, Gastroesophageal and Gastroesophageal Reflux Disease.

Kategori:
Gastric Acid Lowering AgentsHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LAX-101 DB05301
small molecule | CAS: 909712-41-0

LAX-101 treats hungtington’s disease, not just the symptoms but the disease itself. The active molecule in LAX-101 is Eicosapentaenoic Acid (EPA). All molecules of EPA are identical. The molecules of EPA found in LAX-101 are identical to the molecules of EPA …

Target Protein:
Phospholipase D1Caspase-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lazertinib Approved DB16216
small molecule | CAS: 1903008-80-9

Lazertinib is an oral, third-generation, epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI).[A264299, A264304] Lazertinib was first approved in South Korea on January 18, 2021, for the treatment of _EGFR_ T790M mutation-positive non-small…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Lazuvapagon DB19046
small molecule | CAS: 2379889-71-9

Lazuvapagon is under investigation in clinical trial NCT03116191 (Trial of SK-1404 for Nocturia Due to Nocturnal Polyuria in Japanese Subjects).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-001 DB17685
biotech

LB-001 is a gene editing therapy designed to incorporate a functioning version of the faulty methylmalonyl-COA mutase (MUT) gene into the genome of patients with methylmalonic acidemia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-100 DB15412
small molecule | CAS: 1632032-53-1

LB-100 is under investigation in clinical trial NCT03886662 (A Study of LB-100 in Patients With Low or Intermediate-1 Risk Myelodysplastic Syndromes (MDS)).

Kategori:
Antineoplastic AgentsEnzyme Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-102 DB19214
small molecule | CAS: 2227154-23-4

LB-102 is under investigation in clinical trial NCT06179108 (Randomized, Double-blinded, Placebo-controlled, Evaluating the Treatment With LB-102 in Patients With Acute Schizophrenia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB-P8 DB18535
biotech

LB-P8 is an investigational live biotherapeutic product consisting of a single bacterial strain (_Leuconostoc citreum_).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LB54640 DB18331
small molecule

LB54640 is orally-administered small molecule agonist of the melanocortin 4 receptor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LC16M8 DB05019
biotech

LC16m8 is a next-generation, attenuated smallpox vaccine that is designed to have a better safety profile, yet be equally effective, compared to conventional smallpox vaccines. It is the only attenuated vaccine to be licensed for use in humans to prevent smal…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LCL-161 DB12085
small molecule | CAS: 1005342-46-0

LCL161 has been used in trials studying the treatment of Leukemia, Neoplasms, Solid Tumors, Breast Cancer, and Ovarian Cancer, among others.

Kategori:
Antineoplastic AgentsProto-Oncogene Proteins c-bcl-2, antagonists & inhibitorsSulfur Compounds
Target Protein:
E3 ubiquitin-protein ligase XIAPBaculoviral IAP repeat-containing protein 2Baculoviral IAP repeat-containing protein 3 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LCP-AtorFen DB05769
small molecule

LCP-AtorFen is a fixed-dose combination therapy for the treatment of high cholesterol levels combining atorvastatin (the active ingredient of Lipitor®) and the lowest dose of fenofibrate without food effect. LCP-AtorFen is designed to be a once daily tablet o…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LDN-193189 DB18051
small molecule | CAS: 1062368-24-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lebrikizumab Approved DB11914
biotech | CAS: 953400-68-5

Lebrikizumab is a monoclonal antibody that binds to IL-13 with high affinity and slow off-rate.[L51374] It binds to a different epitope compared [tralokinumab].[A262874,A262879] On November 17, 2023, lebrikizumab was approved by the EMA under the brand nam…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-13
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a populati…
KlirensIn the population P…
Genetik -
Lecanemab Approved DB14580
biotech | CAS: 1260393-98-3

Lecanemab is a recombinant humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against aggregated soluble and insoluble forms of amyloid beta (A?), which are implicated in the pathophysiology of Alzheimer’s disease.[L44537] Lecanemab works to…

Kategori:
Alzheimer DiseaseAlzheimer Disease, drug therapyAmino Acids, Peptides, and Proteins +12
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean value (95%…
KlirensThe clearance of le…
Genetik -
Lecithin DB15834
small molecule | CAS: 8002-43-5

A complex mixture of phospholipids, glycolipids, triglycerides, phosphatidylcholines, phosphatidylethanolamines, and phosphatidylinositols.

Kategori:
Biological ProductsComplex MixturesCompounds used in a research, industrial, or household setting +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lecozotan DB12540
small molecule | CAS: 434283-16-6

Lecozotan has been used in trials studying the treatment of Alzheimer Disease.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT1 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 15-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ledipasvir Approved DB09027
small molecule | CAS: 1256388-51-8

Ledipasvir is a direct acting antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized int…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +10
Target Protein:
Genome polyproteinNonstructural protein 5A
Waktu ParuhThe median terminal…
Vol. Distribusi-
Klirens-
Genetik -
Leek Approved DB10659
biotech

Leek allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lefamulin Approved DB12825
small molecule | CAS: 1061337-51-6

Lefamulin is a pleuromutilin antibiotic used for the treatment of bacterial community-acquired pneumonia. A pleuromotilin is a more recently developed type of antibiotic that is derived from the fungus, Pleurotus mutilus.[A183206] Lefamulin is available in in…

Kategori:
AcetatesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
50S ribosomal protein L22
Waktu ParuhThe average elimina…
Vol. DistribusiThe average volume …
KlirensThe total body clea…
Genetik -
Lefitolimod DB15061
biotech | CAS: 1548439-51-5

Lefitolimod is under investigation in clinical trial NCT03837756 (Combining TLR9 Agonist With bNAbs for Reservoir Reduction and Immunological Control of HIV).

Kategori:
Nucleic AcidsNucleic Acids, Nucleotides, and Nucleosides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leflunomide Approved DB01097
small molecule | CAS: 75706-12-6

Leflunomide is a pyrimidine synthesis inhibitor belonging to the DMARD (disease-modifying antirheumatic drug) class of drugs, which are chemically and pharmacologically very heterogeneous. Leflunomide was approved by FDA and in many other countries (e.g., Can…

Kategori:
AdjuvantsAgents Causing Muscle ToxicityAntineoplastic and Immunomodulating Agents +16
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrialAryl hydrocarbon receptor +1
Gen Terkait:
CYP1A2
Waktu Paruh2 weeks
Vol. Distribusi* 0.13 L/kg
Klirens-
Genetik 1 Varian
Leflutrozole DB19047
small molecule | CAS: 143030-47-1

Leflutrozole is under investigation in clinical trial NCT02908074 (A 6 Month Safety Extension Study of MBGS205).

Kategori:
Aromatase Inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lefradafiban DB04863
small molecule | CAS: 149503-79-7

Lefradafiban is an oral platelet glycoprotein IIb/IIIa receptor antagonist being investigated in the treatment of angina.

Kategori:
Antianginal AgentsBenzene DerivativesPlatelet Glycoprotein GPIIb-IIIa Complex, antagonists & inhibitors +1
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 7201–7250 dari 12560
Sebelumnya Halaman 145 / 252 Berikutnya