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11778

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8554 (72.6%)
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6383 (54.2%)
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11778 (100.0%)

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Halaman 144 / 236
MDX-1303 DB05945
biotech | CAS: 915947-57-8

MDX-1303 is a fully human antibody against the inhalation anthrax, the most lethal form of illness in humans caused by the Bacillus anthracis bacterium, and targets a protein component of these lethal toxins known as the anthrax protective antigen.

Target Protein:
Anthrax toxin receptor 2Anthrax toxin receptor 1
Waktu Paruh-
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MDX-1379 DB05329
biotech

MDX-1379 vaccine consists of two gp100 melanoma peptides. This drug is underinvestigation to treat malignant melanoma.

Waktu Paruh-
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MDX-210 DB17250
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
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Genetik -
ME-344 DB13062
small molecule | CAS: 1374524-68-1

ME-344 has been used in trials studying the treatment of Solid Tumors.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTOR
Waktu Paruh-
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Me-4(18F)DG DB19207
small molecule | CAS: 915776-36-2

Me-4(18F)DG is under investigation in clinical trial NCT05558904 (An Investigational Scan (Me-4fdg PET/CT) for the Detection of Sodium-glucose Transport for Early Diagnosis of Lung Cancer).

Kategori:
CarbohydratesFluorine RadioisotopesGlycosides
Waktu Paruh-
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Mebendazole Approved DB00643
small molecule | CAS: 31431-39-7

A benzimidazole that acts by interfering with carbohydrate metabolism and inhibiting polymerization of microtubules. [PubChem]

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +11
Target Protein:
Tubulin alpha-1A chainTubulin beta-4B chain
Waktu Paruh2.5 to 5.5 hours (r…
Vol. Distribusi-
Klirens-
Genetik -
Mebenil DB14728
small molecule | CAS: 7055-03-0

An obsolete fungicide used to control various pathogens on cereals and seed potatoes.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
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Mebeverine Approved DB12554
small molecule | CAS: 3625-06-7

Mebeverine has been investigated for the treatment of Irritable Bowel Syndrome and Post-cholecystectomy Gastrointestinal Spasms.

Kategori:
Agents Causing Muscle ToxicityAgents producing tachycardiaAlimentary Tract and Metabolism +10
Target Protein:
Muscarinic acetylcholine receptor M5
Waktu Paruh-
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Mebrofenin Approved DB15779
small molecule | CAS: 78266-06-5

Deskripsi belum tersedia.

Kategori:
AminesAmino AcidsAmino Acids, Peptides, and Proteins
Waktu Paruh-
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Mebutamate Approved DB06797
small molecule | CAS: 64-55-1

Mebutamate is a sedative and anxiolytic drug with anti-hypertensive (blood pressure lowering) effects comparable to those of other barbiturates but is only around 1/3rd the potency of secobarbital as a sedative. Side effects include dizziness and headaches.

Kategori:
Anti-Anxiety AgentsCarbamatesCentral Nervous System Depressants +2
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3
Waktu Paruh-
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Mecamylamine Approved DB00657
small molecule | CAS: 60-40-2

A nicotinic antagonist that is well absorbed from the gastrointestinal tract and crosses the blood-brain barrier. Mecamylamine has been used as a ganglionic blocker in treating hypertension, but, like most ganglionic blockers, is more often used now as a rese…

Kategori:
Agents that produce neuromuscular block (indirect)Antiadrenergic Agents, Ganglion-BlockingAnticholinergic Agents +15
Target Protein:
Neuronal acetylcholine receptor subunit alpha-2Neuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-4 +1
Waktu Paruh-
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biotech | CAS: 1570067-55-8

Mecapegfilgrastim is under investigation in clinical trial NCT05463601 (Mecapegfilgrastim for the Prevention of Dalpiciclib -Induced Neutropenia in Advanced Breast Cancer).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +13
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Mecasermin Approved DB01277
biotech | CAS: 68562-41-4

Mecasermin contains recombinant-DNA-engineered human insulin-like growth factor-1 (rhIGF-1)[FDA Label]. IGF-1 consists of 70 amino acids in a single chain with three intramolecular disulfide bridges and a molecular weight of 7649 daltons. The amino acid seque…

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesBiological Factors +15
Target Protein:
Insulin-like growth factor 1 receptorInsulin-like growth factor-binding protein 3Insulin receptor +1
Waktu ParuhMean half life of 5…
Vol. Distribusi* 0.257 ± 0.073 L/k…
KlirensClearance of Mecase…
Genetik -
Mecasermin rinfabate Approved DB14751
biotech | CAS: 478166-15-3

Mecasermin rinfabate is approved for severe primary insulin-like growth factor (IGF) deficiency or in patients with GH gene deletion who have developed antibodies to growth hormone (GH)[A176020]. Mecasermin rinfabate is similar to [DB01277] in that both drugs…

Kategori:
Anterior Pituitary Lobe Hormones and AnaloguesPituitary and Hypothalamic Hormones and AnaloguesSomatropin and Somatropin Agonists +1
Target Protein:
Insulin-like growth factor 1 receptorInsulin receptorCation-independent mannose-6-phosphate receptor
Waktu ParuhHalf life ranges fr…
Vol. DistribusiApproximately 1000m…
KlirensClearance ranges fr…
Genetik -
biotech | CAS: 2460400-64-8

Mecbotamab vedotin is an anti-Axl humanized monoclonal antibody conjugated to monomethyl auristatin E using a cleavable linker (CAB-Axl-ADC).[A255212]

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Mechlorethamine Approved DB00888
small molecule | CAS: 51-75-2

A vesicant and necrotizing irritant destructive to mucous membranes, mechlorethamine is an alkylating drug. It was formerly used as a war gas. The hydrochloride is used as an antineoplastic in Hodgkin's disease and lymphomas. It causes severe gastrointestinal…

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +16
Target Protein:
DNA
Waktu Paruh15 minutes
Vol. Distribusi-
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Meclinertant DB06455
small molecule | CAS: 146362-70-1

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, Neurotensin, antagonists & inhibitors
Target Protein:
Neurotensin receptor type 1
Waktu Paruh-
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Meclizine Approved DB00737
small molecule | CAS: 569-65-3

Meclizine is a histamine H1 antagonist with antiemetic and antivertigo properties. It is used in the symptomatic treatment of motion sickness and control of vertigo associated with vestibular system diseases. It also exhibits anticholinergic, central nervous …

Kategori:
Anti-Allergic AgentsAnticholinergic AgentsAntiemetics +19
Target Protein:
Histamine H1 receptorNuclear receptor subfamily 1 group I member 3
Waktu ParuhMeclizine has a pla…
Vol. DistribusiThe volume of distr…
KlirensThere is limited da…
Genetik -
Meclocycline DB13092
small molecule | CAS: 2013-58-3

Meclocycline is under investigation in clinical trial NCT00385515 (Efficacy of SNX-1012 in the Treatment of Oral Mucositis) [L797].

Kategori:
Anti-Acne PreparationsAnti-Acne Preparations for Topical UseAnti-Bacterial Agents +5
Target Protein:
30S ribosomal protein S7
Waktu ParuhHalf life estimated…
Vol. DistribusiEstimated Vd of 121…
Klirens-
Genetik -
Meclofenoxate DB13758
small molecule | CAS: 51-68-3

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicCentral Nervous System Agents +10
Waktu Paruh-
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Mecloxamine DB15790
small molecule | CAS: 5668-06-4

Deskripsi belum tersedia.

Waktu Paruh-
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Medazepam DB13437
small molecule | CAS: 2898-12-6

Deskripsi belum tersedia.

Kategori:
Anti-Anxiety AgentsAnticonvulsantsBenzazepines +17
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
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Medetomidine DB11428
small molecule | CAS: 86347-14-0

Medetomidine is a synthetic compound used as a surgical anesthetic and analgesic. It is normally found as its hydrochloride salt, medetomidine hydrochloride. Medetomidine is an intravenously available alpha-2 adrenergic agonist. The drug has been developed by…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +12
Target Protein:
Alpha-2A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +3
Waktu Paruh-
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MEDI-491 DB17859
biotech

MEDI-491 is a recombinant human parvovirus B19 vaccine composed of the VP1 and VP2 capsid proteins.

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MEDI-547 DB18360
biotech

MEDI-547 is an anti-EphA1 monoclonal antibody conjugated to mcMMAF

Kategori:
Acids, CarbocyclicAmino Acids, Peptides, and ProteinsAntibodies +8
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MEDI-6469 DB15306
biotech | CAS: 1715924-11-0

MEDI-6469 is a monoclonal antibody under investigation in clinical trial NCT02205333 (A Phase 1b/2 Safety and Tolerability of MEDI6469 in Combination With Therapeutic Immune Agents or Monoclonal Antibodies).

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MEDI0680 DB15768
biotech

Deskripsi belum tersedia.

Kategori:
Immune Checkpoint Inhibitors
Target Protein:
Programmed cell death protein 1
Waktu Paruh-
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MEDI3506 DB16473
biotech | CAS: 2376858-66-9

Tozorakimab (MEDI3506), developed by AstraZeneca, was investigated in multiple clinical trials to evaluate its safety, tolerability, efficacy, and pharmacokinetics across various conditions. These trials include NCT03096795 (completed; healthy participants, C…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
Interleukin-33
Waktu Paruh-
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MEDI6012 DB14833
biotech

Recombinant human lecithin:cholesterol acyltransferase is under investigation in clinical trial NCT03578809 (A Study to Evaluate the Safety and Efficacy of MEDI6012 in Acute ST Elevation Myocardial Infarction).

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Medical air Approved DB09337
small molecule | CAS: 132259-10-0

Medical air is supplied by a special air compressor to patient care areas using clean outside air.

Kategori:
Medical GasesOther Miscellaneous Therapeutic Agents
Waktu Paruh-
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Genetik -
biotech

The use of the plant species _Cannabis sativa_ and _Cannabis indica_, popularly known as marijuana, has gained popularity in recent years for the management of a wide variety of medical conditions as a wave of legalization in North America has changed public …

Kategori:
Agents producing tachycardiaBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Inducers +51
Target Protein:
Cannabinoid receptor 1Cannabinoid receptor 2G-protein coupled receptor 12 +38
Waktu ParuhThe half life of TH…
Vol. DistribusiAs a very lipophili…
KlirensOne study reported …
Genetik -
Medifoxamine Approved DB13219
small molecule | CAS: 32359-34-5

Medifoxamine was marketed as an atypical antidepressant, with anxiolyitc properties in France, Spain, and Morrocco in the 1990s but was later withdrawn from the market due to it causing cases of hepatotoxicity [L5461, A174976].

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
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Medrogestone Approved DB09124
small molecule | CAS: 977-79-7

Medrogestone (INN), also known as 6,17?-dimethyl-6-dehydroprogesterone, is a progestational agent derived from 17-methylprogesterone. It was conceived as an alternative for an orally effective contraceptive option.[A31526] It was developed by Ayerst, approved…

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +10
Target Protein:
Progesterone receptor
Waktu ParuhThe half-life of me…
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Medronic acid Approved DB14078
small molecule | CAS: 1984-15-2

Deskripsi belum tersedia.

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Medroxyprogesterone acetate Approved DB00603
small molecule | CAS: 71-58-9

Medroxyprogesterone acetate (MPA) is a [progesterone] derivative that is more resistant to metabolism for improved pharmacokinetic properties.[A14848] MPA can be use to treat secondary amenorrhea, endometrial hyperplasia, abnormal uterine bleeding, osteoporos…

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +46
Target Protein:
Progesterone receptorEstrogen receptorATP-dependent translocase ABCB1 +1
Waktu ParuhOral medroxyprogest…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Mefenamic acid Approved DB00784
small molecule | CAS: 61-68-7

A non-steroidal anti-inflammatory agent with analgesic, anti-inflammatory, and antipyretic properties. It is an inhibitor of cyclooxygenase.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +37
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu Paruh2 hours
Vol. Distribusi* 1.06 L/kg [Normal…
Klirens* Oral cl=21.23 L/h…
Genetik -
Mefenorex DB13852
small molecule | CAS: 17243-57-1

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAlimentary Tract and Metabolism +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Mefloquine Approved DB00358
small molecule | CAS: 53230-10-7

Malaria is a protozoan disease that places an enormous burden on human health in endemic areas around the world. The 2020 World Health Organization malaria report indicates a 60% decrease in the global malaria fatality rate between 2000 to 2019.[L30618] Despi…

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAminoquinolines +20
Target Protein:
Fe(II)-protoporphyrin IX80S ribosomal subunitAdenosine receptor A2a
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThe systemic cleara…
Genetik -
Mefruside DB13405
small molecule | CAS: 7195-27-9

Deskripsi belum tersedia.

Kategori:
AmidesDiureticsLow-Ceiling Diuretics, Excl. Thiazides +4
Waktu Paruh-
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Klirens-
Genetik -
Mefuparib DB18248
small molecule | CAS: 1392502-82-7

Deskripsi belum tersedia.

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Megestrol Approved DB19378
small molecule | CAS: 3562-63-8

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +19
Target Protein:
Progesterone receptor
Waktu Paruh-
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Megestrol acetate Approved DB00351
small molecule | CAS: 595-33-5

17-Hydroxy-6-methylpregna-3,6-diene-3,20-dione. A progestational hormone used most commonly as the acetate ester. As the acetate, it is more potent than progesterone both as a progestagen and as an ovulation inhibitor. It has also been used in the palliative …

Kategori:
Adrenal Cortex HormonesAntineoplastic AgentsAntineoplastic Agents, Hormonal +31
Target Protein:
Progesterone receptorGlucocorticoid receptor
Waktu Paruh34 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 133-51-7

Deskripsi belum tersedia.

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAlcoholsAmino Sugars +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Meglutol DB04377
small molecule | CAS: 503-49-1

An antilipemic agent which lowers cholesterol, triglycerides, serum beta-lipoproteins and phospholipids. It acts by interfering with the enzymatic steps involved in the conversion of acetate to hydroxymethylglutaryl coenzyme A as well as inhibiting the activi…

Kategori:
Acids, AcyclicAnticholesteremic AgentsAntimetabolites +7
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductase
Waktu Paruh-
Vol. Distribusi-
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Meladrazine DB13272
small molecule | CAS: 13957-36-3

Deskripsi belum tersedia.

Kategori:
Drugs for Urinary Frequency and IncontinenceGenito Urinary System and Sex HormonesUrologicals
Waktu Paruh-
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Melagatran DB13616
small molecule | CAS: 159776-70-2

Deskripsi belum tersedia.

Kategori:
AminesAnticoagulantsAntithrombins +8
Target Protein:
ProthrombinPlasminogenSerine protease 1 +1
Waktu Paruh-
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Genetik -
biotech

Melaleuca alternifolia leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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biotech

Melaleuca quinquenervia pollen is the pollen of the Melaleuca quinquenervia plant. Melaleuca quinquenervia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
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Genetik -
biotech

Melanoma antigen recognized by T-cells 1 is under investigation in clinical trial NCT01748747 (Vaccine Therapy and Resiquimod in Treating Patients With Stage II-IV Melanoma That Has Been Removed By Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +4
Waktu Paruh-
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Melarsomine DB11528
small molecule | CAS: 128470-15-5

Melarsomine is a trypanocidal agent marketed by Merial under the trade name Immiticide. It is the only FDA-approved treatment for adult heartworm infection in dogs, however, is is not approved for use in dogs with late-stage infection.

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