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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 144 / 252
Lacnotuzumab DB14928
biotech | CAS: 1831128-32-5

Lacnotuzumab is under investigation in clinical trial NCT01643850 (MCS110 in Patients With Pigmented Villonodular Synovitis (PVNS)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
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Lacosamide Approved DB06218
small molecule | CAS: 175481-36-4

Lacosamide is an antiepileptic drug used to treat seizures. As a chiral functionalized amino acid, it works by blocking slowly inactivating components of voltage-gated sodium currents. Lacosamide exhibits a stereoselective mode of interaction with sodium chan…

Kategori:
AcetamidesAcetatesAcids, Acyclic +21
Target Protein:
Dihydropyrimidinase-related protein 2Sodium channel protein type 11 subunit alphaSodium channel protein type 9 subunit alpha +2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
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Lacripep DB18921
biotech | CAS: 2243095-21-6

Lacripep is under investigation in clinical trial NCT03226444 (Lacripep™ in Subjects With Dry Eye Associated With Primary Sjögren's Syndrome).

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Lactaldehyde DB03776
small molecule | CAS: 598-35-6

Deskripsi belum tersedia.

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Lactic acid Approved DB04398
small molecule | CAS: 50-21-5

A normal intermediate in the fermentation (oxidation, metabolism) of sugar. The concentrated form is used internally to prevent gastrointestinal fermentation. (From Stedman, 26th ed) Sodium lactate is the sodium salt of lactic acid, and has a mild saline tast…

Kategori:
Basic Ointments and ProtectantsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +6
Target Protein:
Bifunctional protein PutANimA-related protein
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Lactide, L- DB19115
small molecule | CAS: 4511-42-6

Lactide, L- is under investigation in clinical trial NCT05450471 (Effectiveness of Endonasal Polymeric Implant for Chronic Rhinosinusitis).

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Lactitol Approved DB12942
small molecule | CAS: 585-86-4

Lactitol, also known as 4-?-D-galactopyranosyl-D-glucitol, is a sugar alcohol synthesized from [lactose].[A190918] It is used in food manufacturing as a nutritive sweetener and is approximately 35% as sweet as table sugar (i.e. [sucrose]).[A190912] Clinically…

Kategori:
AlcoholsAlimentary Tract and MetabolismCarbohydrates +15
Waktu ParuhThe average half-li…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lactobacillus acidophilus Approved DB15823
biotech | CAS: 68333-16-4

Deskripsi belum tersedia.

Kategori:
CarbohydratesCarbon Compounds, InorganicCarbonates +7
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biotech

Deskripsi belum tersedia.

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Lactobacillus casei Approved DB16541
biotech | CAS: 68333-14-2

Deskripsi belum tersedia.

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biotech

Lactobacillus is a common bacteria found in the gut with Lactobacillus coryniformis K8 being originally isolated from artisan goat cheese.

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biotech

Deskripsi belum tersedia.

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small molecule

Deskripsi belum tersedia.

Kategori:
Probiotics
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biotech

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biotech

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biotech

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biotech

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Lactoferrin DB16555
biotech | CAS: 151186-19-5

Lactoferrin is under investigation in clinical trial NCT03748043 (The Effectiveness of Lactoferrin in Treatment of Iron Deficiency Anemia in Children With Chronic Tonsillitis).

Kategori:
Amino Acids, Peptides, and ProteinsAnimal Proteins, DietaryAnti-Infective Agents +22
Target Protein:
Tryptase alpha/beta-1
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Lactose Approved DB04465
small molecule | CAS: 63-42-3

A disaccharide of glucose and galactose in human and cow milk. It is used in pharmacy for tablets, in medicine as a nutrient, and in industry.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +9
Target Protein:
Galectin-3SialidaseBeta-galactosidase +5
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Lactuca sativa whole Approved DB15604
biotech

Lactuca sativa whole allergenic extract is used in allergenic testing.

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Lactulose Approved DB00581
small molecule | CAS: 4618-18-2

Lactulose is a synthetic disaccharide derivative of lactose that is most commonly used as a laxative agent despite also being formally indicated to serve as an adjunct therapy in treating portal-systemic encephalopathy (PSE).[FDA Label,L6199,L6202] Despite be…

Kategori:
Acidifying ActivityAlimentary Tract and MetabolismAmmonia Detoxicants +8
Target Protein:
Evolved beta-galactosidase subunit alpha
Waktu ParuhThe data regarding …
Vol. DistribusiNegligible amounts …
KlirensNegligible amounts …
Genetik -
Lacutamab DB15322
biotech | CAS: 2187368-16-5

Lacutamab is under investigation in clinical trial NCT02593045 (Study of IPH4102 in Patients With Relapsed/Refractory Cutaneous T-cell Lymphomas (CTCL)).

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Ladarixin DB16212
small molecule | CAS: 849776-05-2

Ladarixin is under investigation in clinical trial NCT04628481 (A Study of Oral Ladarixin in New-onset Type 1 Diabetes and a Low Residual ?-Cell Function).

Kategori:
AmidesReceptors, Interleukin-8A, antagonists & inhibitorsSulfones +1
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Lademirsen DB17611
biotech | CAS: 1404019-95-9

Deskripsi belum tersedia.

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biotech | CAS: 1629760-29-7

Ladiratuzumab vedotin is under investigation in clinical trial NCT01969643 (A Safety Study of SGN-LIV1A in Breast Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Lamb Approved DB10537
biotech

Lamb allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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small molecule

Deskripsi belum tersedia.

Target Protein:
Camphor 5-monooxygenase
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Lamivudine Approved DB00709
small molecule | CAS: 134678-17-4

A reverse transcriptase inhibitor and zalcitabine analog in which a sulfur atom replaces the 3' carbon of the pentose ring. It is used to treat Human Immunodeficiency Virus Type 1 (HIV-1) and hepatitis B (HBV).

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +26
Target Protein:
Gag-Pol polyproteinReverse transcriptase/RNaseHDNA +1
Waktu Paruh5 to 7 hours (healt…
Vol. DistribusiApparent volume of …
Klirens* Renal clearance =…
Genetik -
Lamotrigine Approved DB00555
small molecule | CAS: 84057-84-1

Lamotrigine is an antiepileptic drug belonging in the phenyltriazine class. It is used in the treatment of both epilepsy and as a mood stabilizer in bipolar disorder. Lamotrigine is the first medication since lithium granted Food and Drug Administration (FDA)…

Kategori:
Agents causing hyperkalemiaAgents producing tachycardiaAnti-epileptic Agent +31
Target Protein:
Voltage-dependent R-type calcium channel subunit alpha-1ESodium channel protein type 11 subunit alphaVoltage-gated sodium channel alpha subunit +15
Waktu ParuhThe average elimina…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent p…
Genetik -
Lanadelumab Approved DB14597
biotech | CAS: 1426055-14-2

Lanadelumab, also known as DX-2930, is a human IgG1 monoclonal antibody designed for subcutaneous self-injection.[L4538] It is a fully human immunoglobulin, k-light-chain made in recombinant Chinese Hamster Ovary cells.[L4537] It has been granted priority rev…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Plasma kallikrein
Waktu ParuhLanadelumab has a h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Lanatoside C DB13467
small molecule | CAS: 17575-22-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesCardanolidesCardenolides +6
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Lancovutide DB05029
small molecule | CAS: 1391-36-2

Lancovutide, a peptide antibiotic, is in clinical development for the treatment of cystic fibrosis. Lancovutide is a 19-amino-acid tetracyclic peptide produced by Streptoverticillium cinnamoneus and is closely related to cinnamycin (Ro09-0198). It belongs to …

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Landiolol Approved DB12212
small molecule | CAS: 133242-30-5

Landiolol is a rapid-acting beta-blocker used for rapid ventricular rate control.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +11
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Landipirdine DB16214
small molecule | CAS: 1000308-25-7

Landipirdine is under investigation in clinical trial NCT02258152 (SYN120 Study to Evaluate Its Safety, Tolerability and Efficacy in Parkinson's Disease Dementia (SYNAPSE)).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 65-hydroxytryptamine receptor 2A
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Lanicemine DB11889
small molecule | CAS: 153322-05-5

Lanicemine has been used in trials studying the treatment and basic science of Depression, Major Depressive Disorder, and Treatment Resistant Major Depressive Disorder.

Kategori:
AminesAntidepressive AgentsCentral Nervous System Depressants +2
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Lanimostim DB06559
small molecule | CAS: 117276-75-2

Deskripsi belum tersedia.

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Laniquidar DB12799
small molecule | CAS: 197509-46-9

Laniquidar has been used in trials studying the treatment of Breast Cancer.

Kategori:
Carbon RadioisotopesDrug Resistance, MultipleHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylcholine translocator ABCB4
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Lanolin Approved DB11112
small molecule | CAS: 8006-54-0

Lanolin is a yellow fat obtained from sheep's wool. It is used as an emollient, cosmetic, and pharmaceutic aid [L2580]. The US federal code of regulations states that lanolin in the concentration range of 12-50% may be included in over the counter skin ointme…

Kategori:
Basic Ointments and ProtectantsCompounds used in a research, industrial, or household settingCosmetics +3
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Lanopepden DB11912
small molecule | CAS: 1152107-25-9

Lanopepden has been used in trials studying the treatment of Pneumonia, Infections, Bacterial, Skin Diseases, Infectious, and Skin Infections, Bacterial.

Kategori:
AminesAnti-Bacterial AgentsEnzyme Inhibitors +2
Target Protein:
Peptide deformylase
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Lanoteplase DB06245
biotech | CAS: 171870-23-8

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsBiological Factors +10
Target Protein:
Urokinase plasminogen activator surface receptorFibrinogen alpha chainKallikrein-1 +14
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Lanraplenib DB14770
small molecule | CAS: 1800046-95-0

Lanraplenib is under investigation in clinical trial NCT03285711 (Safety and Efficacy of Filgotinib and Lanraplenib in Adults With Lupus Membranous Nephropathy (LMN)).

Target Protein:
Tyrosine-protein kinase SYK
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Lanreotide Approved DB06791
small molecule | CAS: 108736-35-2

Lanreotide is a drug employed in the management of acromegaly (a hormonal condition caused by excess growth hormone) in addition to symptoms caused by neuroendocrine tumors, especially carcinoid syndrome. This drug is a long-acting analog of the drug somatost…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5
Waktu ParuhHalf-life is approx…
Vol. DistribusiEstimated Volume of…
KlirensEstimated Clearance…
Genetik -
Lansoprazole Approved DB00448
small molecule | CAS: 103577-45-3

Lansoprazole marketed under the brand Prevacid, is a proton pump inhibitor (PPI) and is structurally classified as a substituted benzimidazole.[A177065] It reduces gastric acid secretion by targeting gastric H,K-ATPase pumps and is thus effective at promoting…

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +39
Target Protein:
Potassium-transporting ATPase alpha chain 1Microtubule-associated protein tau
Gen Terkait:
CYP2C19 CYP2C19 ABCB1
Waktu ParuhOne source reports …
Vol. DistribusiThe apparent volume…
KlirensThe reported cleara…
Genetik 3 Varian
Lanthanum carbonate Approved DB06792
small molecule | CAS: 587-26-8

Lanthanum carbonate is a phosphate binder marketed under the trade name _Fosrenol_ by Shire Pharmaceuticals. It is a large pill that requires thorough chewing to avoid choking and other gastrointestinal adverse effects. It is used to treat elevated phosphate …

Kategori:
Drugs for Treatment of Hyperkalemia and HyperphosphatemiaElementsKidney Failure, Chronic +6
Target Protein:
Phosphate
Waktu ParuhThe elimination hal…
Vol. Distribusi-
KlirensIn healthy voluntee…
Genetik -
small molecule | CAS: 16096-89-2

Deskripsi belum tersedia.

Kategori:
Metal cationsPhosphate BinderPhosphate Chelating Activity
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Lapaquistat DB16215
small molecule | CAS: 189059-71-0

Lapaquistat is under investigation in clinical trial NCT00256178 (Efficacy of Lapaquistat Acetate and Simvastatin in Subjects With Primary Dyslipidemia.).

Kategori:
AzepinesFarnesyl-Diphosphate Farnesyltransferase, antagonists & inhibitors
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Lapatinib Approved DB01259
small molecule | CAS: 231277-92-2

Lapatinib is an anti-cancer drug developed by GlaxoSmithKline (GSK) as a treatment for solid tumours such as breast and lung cancer. It was approved by the FDA on March 13, 2007, for use in patients with advanced metastatic breast cancer in conjunction with t…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +22
Target Protein:
Epidermal growth factor receptorEukaryotic elongation factor 2 kinaseReceptor tyrosine-protein kinase erbB-2
Gen Terkait:
HLA-DQA1 HLA-DRB1 HLA-DQB1 +1
Waktu ParuhSingle-dose termina…
Vol. Distribusi-
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Genetik 4 Varian
Lapuleucel-t DB19117
biotech | CAS: 845680-07-1

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines
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Laquinimod DB06685
small molecule | CAS: 248281-84-7

Laquinimod is an immunomodulator developed by Active Biotech and produced by Teva Pharmaceutical Industries. It is currently under development in phase III trials for treatment of multiple sclerosis as an oral therapy, like fingolimod. It has been shown to re…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +3
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
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Larazotide DB05645
small molecule | CAS: 258818-34-7

An octapeptide inhibitor of paracellular permeability whose structure is derived from a protein (zonula occludens toxin) secreted by Vibrio cholerae for treatment of Coeliac disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Haptoglobin
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