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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 144 / 315
small molecule | CAS: 53861-57-7

Deskripsi belum tersedia.

Kategori:
1-Carboxyglutamic AcidAcids, AcyclicAmino Acids +5
Target Protein:
ProthrombinCoagulation factor IXCoagulation factor X +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
gamma-Hydroxybutyric acid Approved DB01440
small molecule | CAS: 591-81-1

Gamma hydroxybutyric acid, commonly abbreviated GHB, is a therapeutic drug which is illegal in multiple countries. It is currently regulated in the US and sold by Jazz Pharmaceuticals under the name Xyrem. However, it is important to note that GHB is a design…

Kategori:
Acids, AcyclicAdjuvants, AnesthesiaAnesthetics +12
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2GABA(B) Receptor +1
Waktu Paruh30 to 60 minutes
Vol. Distribusi* 190 to 384 mL/kg
Klirens* apparent oral cl=…
Genetik -
small molecule | CAS: 54-28-4

gamma-Tocopherol is under investigation in clinical trial NCT00836368 (In Vitro Basophil Responsiveness to Allergen Challenge After Gamma-tocopherol Supplementation in Allergic Asthmatics).

Kategori:
AntioxidantsBenzopyransBiological Factors +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gamolenic acid Approved DB13854
small molecule | CAS: 506-26-3

Gamolenic acid, or gamma-linolenic acid (?-Linolenic acid) or GLA, is an essential fatty acid (EFA) comprised of 18 carbon atoms with three double bonds [F27] that is most commonly found in human milk and other botanical sources [A32848]. It is an omega-6 pol…

Kategori:
Agents that reduce seizure thresholdDermatologicalsFatty Acids +5
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Ganaplacide DB16173
small molecule | CAS: 1261113-96-5

Ganaplacide is under investigation in clinical trial NCT03167242 (Efficacy and Safety of KAF156 in Combination With LUM-SDF in Adults and Children With Uncomplicated Plasmodium Falciparum Malaria).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganaxolone Approved DB05087
small molecule | CAS: 38398-32-2

Ganaxolone is the 3?-methylated synthetic analog of [allopregnanolone],[L41130] a metabolite of [progesterone].[A3197] Ganaxolone belongs to a class of compounds referred to as neurosteroids.[A3197] Endogenous neurosteroids, which comprise certain metabolites…

Kategori:
AnticonvulsantsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Substrates +14
Target Protein:
GABA(A) Receptor
Waktu ParuhThe terminal half-l…
Vol. DistribusiBoth ganaxolone and…
Klirens-
Genetik -
Ganciclovir Approved DB01004
small molecule | CAS: 82410-32-0

An acyclovir analog that is a potent inhibitor of the Herpesvirus family including cytomegalovirus. Ganciclovir is used to treat complications from AIDS-associated cytomegalovirus infections.

Kategori:
Agents Causing Muscle ToxicityAgents that reduce seizure thresholdAnti-Infective Agents +23
Target Protein:
DNA polymerase catalytic subunitDNAThymidine kinase
Waktu Paruh2.5 to 3.6 hours (m…
Vol. Distribusi* 0.74 ± 0.15 L/kg
Klirens* 128 +/- 63 mL/min…
Genetik -
Gancotamab DB14784
biotech | CAS: 1509928-00-0

Gancotamab is under investigation in clinical trial NCT02213744 (MM-302 Plus Trastuzumab vs. Chemotherapy of Physician's Choice Plus Trastuzumab in HER2-Positive Locally Advanced/Metastatic Breast Cancer Patients).

Kategori:
Amino Acids, Peptides, and ProteinsAnthracyclinesAntibodies +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gandotinib DB13040
small molecule | CAS: 1229236-86-5

Gandotinib has been used in trials studying the treatment of Myelofibrosis, Polycythemia Vera, Primary Myelofibrosis, Thrombocythemia, Essential, and Myeloproliferative Disorders, among others.

Kategori:
Janus Kinase 2, antagonists & inhibitorsJanus Kinases, antagonists & inhibitors
Target Protein:
Tyrosine-protein kinase JAK2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganetespib DB12047
small molecule | CAS: 888216-25-9

Ganetespib is under investigation for the treatment of BREAST CANCER, Small Cell Lung Cancer, Acute Myeloid Leukaemia, and Myelodysplastic Syndrome.

Kategori:
HSP90 Heat-Shock Proteins, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganglioside GM1 DB16948
small molecule | CAS: 116950-37-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganirelix Approved DB06785
small molecule | CAS: 124904-93-4

Ganirelix is a synthetic decapeptide and a competitive gonadotropin-releasing hormone (GnRH) antagonist. Derived from endogenous GnRH, ganirelix has amino acid substitutions. Ganirelix is indicated for controlled ovarian hyperstimulation in assisted reproduct…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Gonadotropin-Releasing HormonesDecreased GnRH Secretion +16
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe mean (SD) volum…
KlirensClearance following…
Genetik -
Ganitumab DB12205
biotech | CAS: 905703-97-1

Ganitumab has been used in trials studying the treatment of Colon Cancer, Rectal Cancer, Breast Cancer, Breast Tumors, and Breast Neoplasms, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ganstigmine DB06525
small molecule | CAS: 457075-21-7

Ganstigmine is an orally active, geneserine derived, carbamate-based acetylcholinesterase inhibitor developed for the treatment of Alzheimer's disease.

Kategori:
Acids, AcyclicCarbamates
Target Protein:
Acetylcholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gantacurium DB05710
small molecule | CAS: 758669-50-0

Gantacurium chloride is a new, investigational, non-depolarizing ultra-short acting neuromuscular blocker. It is being developed by Avera Pharmaceuticals.

Kategori:
Anticholinergic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh3.09±0.21 minutes
Vol. Distribusi-
Klirens-
Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
Klirens-
Genetik -
Garadacimab DB15629
biotech | CAS: 2162134-62-3

Garadacimab is under investigation in clinical trial NCT04281524 (A Clinical Study to Test the Efficacy and Safety of CSL312 on Catheter-associated Blood Clot Formation in Subjects With Cancer Who Receive Chemotherapy Through a PICC Line).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Garcinia gummi-gutta fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Garden snail mucin is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garenoxacin DB06160
small molecule | CAS: 194804-75-6

Garenoxacin, a quinolone antibiotic, is being investigated for the treatment of gram-positive and gram-negative bacterial infections.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garetosmab DB16379
biotech | CAS: 2097125-54-5

Fibrodysplasia ossificans progressiva (FOP) is a rare autosomal dominant disorder of episodic, progressive heterotropic ossification. FOP is characterized by episodic inflammatory episodes, which may be precipitated by trauma, including immunizations and mino…

Target Protein:
Inhibin beta A chain
Waktu Paruh-
Vol. DistribusiGaretosmab had a st…
KlirensWhen administered a…
Genetik -
Garivulimab DB16670
biotech | CAS: 2342597-81-1

Garivulimab is under investigation in clinical trial NCT03379259 (Study of BGB-A333 Alone and in Combination With Tislelizumab in Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garlic Approved DB10532
biotech | CAS: 8008-99-9

Garlic allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityHerbs and Natural ProductsIncreased Histamine Release +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garlic oil DB15989
biotech | CAS: 8000-78-0

Deskripsi belum tersedia.

Kategori:
AlkenesAnionsAnticarcinogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gartisertib DB18770
small molecule | CAS: 1613191-99-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 100040-31-1

Gastric inhibitory polypeptide is under investigation in clinical trial NCT03081676 (The Effect of GIP and GLP-1 on Insulin and Glucagon Secretion in Patients With HNF1A-diabetes Treated With or Without Sulphonylurea).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gastric intrinsic factor Approved DB09349
biotech

Intrinsic factor (IF), also known as gastric intrinsic factor (GIF), is a glycoprotein produced by the parietal cells of the stomach that is necessary for the absorption of vitamin B12 (cobalamin) later on in the small intestine. When vitamin B12 is provided …

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsAsparagalesBiological Products +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gatifloxacin Approved DB01044
small molecule | CAS: 112811-59-3

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh7-14 hours
Vol. Distribusi-
Klirens-
Genetik -
Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gatralimab DB16528
biotech | CAS: 1826020-80-7

Gatralimab is under investigation in clinical trial NCT02389452 (Study of Safety and Efficacy of 6 Ml Synvisc-one (Hylan G-F 20) in Indian Patients With Symptomatic Osteoarthritis of Knee(s) After Initial and Repeat Treatment).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavestinel DB06741
small molecule | CAS: 153436-22-7

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Gavestinel displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites and is o…

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsGlycine Agents +5
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Gavocabtagene autoleucel is a novel cell therapy consisting of autologous genetically engineered T cells expressing a single-domain antibody that recognizes human Mesothelin, fused to the CD3-epsilon subunit which, upon expression, is incorporated into the en…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavorestat DB16707
small molecule | CAS: 2170729-29-8

Gavorestat is under investigation in clinical trial NCT04902781 (Clinical Benefit, Safety, PK and PD Study of AT-007 in Pediatric Subjects With Classic Galactosemia).

Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gaxilose Approved DB12767
small molecule | CAS: 14087-31-1

Gaxilose has been used in trials studying the diagnostic of Lactose Intolerance.

Kategori:
CarbohydratesOligosaccharidesPolysaccharides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB-115 DB19204
small molecule | CAS: 678996-63-9

GB-115 is under investigation in clinical trial NCT05586789 (A Study of the Efficacy and Safety of Ranquilon Tablets in Patients With Anxiety in Neurasthenia and Adjustment Disorders).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB-13 DB18387
biotech

GB-13 is a genetically engineered recombinant protein consisting of an IL13Ra2-targeted genetically engineered mutant of IL-13 and PE4E, a derivative of Pseudomonas exotoxin A.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB1211 DB17499
small molecule | CAS: 1978336-95-6

GB1211 is an orally active galectin-3 (Gal-3) inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GBR-12783 DB17027
small molecule | CAS: 145428-33-7

A selective inhibitor of dopamine uptake.[A252997]

Kategori:
Dopamine AgentsDopamine AgonistsDopamine Uptake Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GBR-12879 DB17028
small molecule | CAS: 67469-43-6

Deskripsi belum tersedia.

Kategori:
Piperazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC-373 DB15797
small molecule

GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, [GC-376 free acid][A219031,A219036]. It is an inhibitor of M<sup>pro</sup> (otherwise known as 3CL<sup>pro</sup>), a viral encoded protease that cleaves and activates functional prot…

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +3
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1417031-79-8

GC-376 is a 3C-like protease (3CL<sup>pro</sup> or M<sup>pro</sup>) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells[A219036]. The compound is known as a direct acting antiv…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +15
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC5107 DB17604
biotech

GC5107 is an investigational intravenous immunoglobulin. It is marketed as IVIG-SN.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GCS-100 DB17566
biotech

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0134 DB17079
small molecule | CAS: 1637394-01-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0152 DB12380
small molecule | CAS: 873652-48-3

GDC-0152 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Cycloparaffins
Target Protein:
E3 ubiquitin-protein ligase XIAP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0349 DB13072
small molecule | CAS: 1207360-89-1

GDC-0349 has been used in trials studying the treatment of Non-Hodgkin's Lymphoma, Solid Tumor.

Kategori:
AmidesBenzene Derivatives
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0623 DB11982
small molecule | CAS: 1168091-68-6

GDC-0623 has been used in trials studying the treatment of Solid Cancers.

Kategori:
Nicotinic AcidsPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0810 DB12253
small molecule | CAS: 1365888-06-7

ARN-810 has been used in trials studying the basic science and treatment of Breast Cancer.

Kategori:
Acids, CarbocyclicHeterocyclic Compounds, Fused-RingPyrazoles
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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