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11778

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Halaman 143 / 236
Margetuximab Approved DB14967
biotech | CAS: 1350624-75-7

The HER2 oncoprotein, the product of the human _ERBB2_/mouse _neu_ genes, is a member of the HER family of receptor tyrosine kinases that includes the epidermal growth factor receptor (EGFR). Of the various subtypes of breast cancer, HER2-positive breast canc…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Receptor tyrosine-protein kinase erbB-2
Waktu ParuhMargetuximab has a …
Vol. DistribusiMargetuximab has a …
KlirensMargetuximab has a …
Genetik -
Maribavir Approved DB06234
small molecule | CAS: 176161-24-3

Maribavir is an inhibitor of the cytomegalovirus (CMV; HHV5) pUL97 kinase which is used to treat CMV infections in patients post-transplantation.[L39322] Most standard CMV therapies, such as [ganciclovir] or [foscarnet], target CMV DNA polymerase - while gene…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +14
Target Protein:
Serine/threonine protein kinase UL97
Waktu ParuhIn post-transplant …
Vol. DistribusiThe mean apparent s…
KlirensIn post-transplant …
Genetik -
biotech | CAS: 2760218-55-9

Maridebart Cafraglutide is under investigation in clinical trial NCT05669599 (Dose-ranging Study to Evaluate the Efficacy, Safety, and Tolerability of AMG 133 in Adult Subjects With Overweight or Obesity, With or Without Type 2 Diabetes Mellitus).

Waktu Paruh-
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Marimastat DB00786
small molecule | CAS: 154039-60-8

Used in the treatment of cancer, Marmiastat is an angiogenesis and metastasis inhibitor. As an angiogenesis inhibitor it limits the growth and production of blood vessels. As an antimetatstatic agent it prevents malignant cells from breaching the basement mem…

Kategori:
AminesEnzyme InhibitorsHydroxy Acids +2
Target Protein:
Interstitial collagenase72 kDa type IV collagenaseStromelysin-1 +20
Waktu Paruh-
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Genetik -
biotech | CAS: 9007-34-5

Marine collagen, soluble is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
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Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntioxidantsAntiplatelet agents +14
Waktu Paruh-
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Marizomib DB11762
small molecule | CAS: 437742-34-2

Marizomib has been used in trials studying the treatment of Cancer, Melanoma, Lymphoma, Glioblastoma, and Malignant Glioma, among others.

Waktu Paruh-
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Maropitant DB11427
small molecule | CAS: 147116-67-4

Maropitant, used as maropitant citrate, is a neurokinin receptor antagonist, which was developed by Zoetis specifically for the treatment of motion sickness and vomiting in dogs. It was approved by the FDA in 2007 for use in dogs, and more recently has also b…

Kategori:
AntiemeticsAutonomic AgentsBenzene Derivatives +3
Waktu Paruh-
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Genetik -
Marstacimab Approved DB17725
biotech | CAS: 1985638-39-8

Marstacimab is a human monoclonal immunoglobulin G Type 1 (IgG1) antibody produced by Chinese hamster ovary (CHO) cells by recombinant DNA technology.[L51803] It is a tissue factor pathway inhibitor (TFPI) antagonist, which is an endogenous anticoagulant.[A26…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Tissue factor pathway inhibitor
Waktu ParuhIn a study consisti…
Vol. DistribusiIn patients with he…
KlirensIn a study consisti…
Genetik -
Martinostat DB14979
small molecule | CAS: 1629052-58-9

Martinostat is under investigation in clinical trial NCT03721211 (Imaging With [11C]Martinostat in Breast Cancer).

Kategori:
AminesBridged-Ring CompoundsCarbon Radioisotopes +3
Target Protein:
Histone deacetylase 7Histone deacetylase 9Histone deacetylase 8 +6
Waktu Paruh-
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Genetik -
biotech | CAS: 1600492-21-4

Marzeptacog alfa (activated) is under investigation in clinical trial NCT01439971 (Phase 1 Safety, Pharmacokinetics And Pharmacodynamics Study Of Recombinant Factor VIIa Variant (813d) In Adult Subjects With Hemophilia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +10
Waktu Paruh-
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Genetik -
Masilukast DB16227
small molecule | CAS: 136564-68-6

Masilukast is under investigation in clinical trial NCT01740986 (Safety and Efficacy of SA09012 in Asthma).

Target Protein:
Cysteinyl leukotriene receptor 1
Waktu Paruh-
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Masitinib DB11526
small molecule | CAS: 790299-79-5

Masitinib is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in dogs. It has been available in Europe since 2009, under the brand name Masivet. In the USA it is distributed under the name Kinavet and has been available for veterinaries s…

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +5
Target Protein:
Proto-oncogene tyrosine-protein kinase Src
Waktu Paruh-
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Masoprocol Approved DB00179
small molecule | CAS: 27686-84-6

A potent lipoxygenase inhibitor that interferes with arachidonic acid metabolism. The compound also inhibits formyltetrahydrofolate synthetase, carboxylesterase, and cyclooxygenase to a lesser extent. It also serves as an antioxidant in fats and oils. [PubChe…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +16
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseReceptor tyrosine-protein kinase erbB-2Transient receptor potential cation channel subfamily M member 7 +1
Waktu Paruh-
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Matairesinol DB04200
small molecule | CAS: 580-72-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzyl CompoundsPlants
Target Protein:
Dehydrogenase/reductase SDR family member 4-like 2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Matrix-M DB16369
biotech

Matrix-M is a saponin-based adjuvant made of nanometer particles, cholesterol, and phospholipid that is developed by Novavax.[L27981] This compound is administered alongside vaccines to enhance biological functions: creating robust and long-lasting immune res…

Kategori:
CarbohydratesGlycosidesNanostructures
Waktu Paruh-
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Genetik -
Matuzumab DB05101
biotech | CAS: 339186-68-4

Matuzumab (formerly known as the experimental drug, EMD 72000) is a humanized monoclonal antibody used in cancer treatment. It has a high affinity for EGFR (epithelial growth factor receptor), frequently associated with the growth of blood vessels in malignan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Epidermal growth factor receptor
Waktu Paruh196 hours
Vol. Distribusi-
Klirens-
Genetik -
Mavacamten Approved DB14921
small molecule | CAS: 1642288-47-8

Mavacamten is a myosin inhibitor indicated for the treatment of adults with symptomatic New York Heart Association (NYHA) class II-III obstructive hypertrophic cardiomyopathy (HCM). It received initial US FDA approval in 2022, and it is one of the first myosi…

Kategori:
AminesBenzene DerivativesBenzyl Compounds +21
Target Protein:
Myosin-7
Waktu ParuhMavacamten has a va…
Vol. DistribusiThrough the use of …
KlirensMavacamten demonstr…
Genetik -
Mavatrep DB12875
small molecule | CAS: 956274-94-5

Mavatrep has been used in trials studying the treatment of Osteoarthritis, Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Mavelertinib DB16228
small molecule | CAS: 1776112-90-3

Mavelertinib is under investigation in clinical trial NCT02349633 (Study for Patients With NSCLC EGFR Mutations (Del 19 or L858R +/- T790M)).

Waktu Paruh-
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Maveropepimut-S DB17339
biotech

Maveropepimut-S is a T cell activating immunotherapy.

Waktu Paruh-
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Mavodelpar DB17662
small molecule | CAS: 942594-93-6

Deskripsi belum tersedia.

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Mavorixafor Approved DB05501
small molecule | CAS: 558447-26-0

Mavorixafor is a CXC chemokine receptor 4 (CXCR4) antagonist.[L50642] It was first approved by the FDA on April 30, 2024, for the treatment of warts, hypogammaglobulinemia, infections, and myelokathexis (WHIM) syndrome, a genetic immunodeficiency disorder cha…

Kategori:
AlkanesAminesButanes +38
Target Protein:
C-X-C chemokine receptor type 4
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiMavorixafor volume …
KlirensThe mean (CV%) appa…
Genetik -
Mavrilimumab DB12534
biotech | CAS: 1085337-57-0

Mavrilimumab has been investigated for the treatment of Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
MAX-40279 DB15191
small molecule | CAS: 2070931-57-4

MAX-40279 is under investigation in clinical trial NCT03412292 (MAX-40279 in Subjects With Acute Myelogenous Leukemia (AML)).

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Maxacalcitol DB06272
small molecule | CAS: 103909-75-7

Deskripsi belum tersedia.

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsCholestanes +13
Waktu Paruh-
Vol. Distribusi-
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Genetik -
MaxAdFVIII DB17713
biotech

MaxAdFVIII is an adenoviral vector that expresses the full-length human Factor VIII (hFVIII) cDNA. First developed by GenStar, it is being investigated for the treatment of hemophilia.

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Maxy-G34 DB05718
biotech

MAXY-G34 is a pegylated variant of human granulocyte-colony stimulating factor (G-CSF). This variant contains multiple non-naturally occurring lysines that have been introduced into alpha helixes of wild type human G-CSF as PEGylation sites, and from which mu…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +15
Waktu Paruh-
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Genetik -
Mazindol Approved DB00579
small molecule | CAS: 22232-71-9

Mazindol is a tricyclic anorexigenic agent that is unrelated to and less toxic than [amphetamine], but with some similar side effects. It inhibits uptake of catecholamines and blocks the binding of cocaine to the dopamine uptake transporter. Mazindol is only …

Kategori:
Adrenergic AgentsAdrenergic Uptake InhibitorsAlimentary Tract and Metabolism +19
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent dopamine transporterSodium-dependent serotonin transporter +1
Waktu Paruh10-13 hours
Vol. Distribusi-
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Genetik -
Mazorelvimab DB17767
biotech | CAS: 2419087-89-9

Deskripsi belum tersedia.

Waktu Paruh-
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MB-07803 DB05053
small molecule | CAS: 882757-24-6

MB07803 is a second generation gluconeogenesis inhibitor for the treatment of type 2 diabetes. It is designed to block the metabolic pathway in the liver that is responsible for producing glucose.

Target Protein:
Fructose-1,6-bisphosphatase isozyme 2Fructose-1,6-bisphosphatase 1
Waktu Paruh-
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Genetik -
biotech

MB-102 are autologous T cells genetically modified to express CD123-specific, hinge-optimized CD28-costimulatory chimeric receptor and a truncated human epidermal growth factor receptor.

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MB-107 DB18566
biotech

MB-107 consists of mobilized peripheral blood-derived autologous CD34+ hematopoietic stem cells that are genetically modified to express the IL2RG gene.

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MB07133 DB17139
small molecule | CAS: 685111-92-6

Deskripsi belum tersedia.

Kategori:
ArabinonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
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MB07811 DB05192
small molecule

MB07811 is the first of a novel class of product candidates discovered by Metabasis designed to lower serum cholesterol and triglycerides. MB07811, a small molecule that is administered orally, has been extensively studied preclinically and is currently under…

Kategori:
Organophosphorus Compounds
Target Protein:
Thyroid hormone receptor beta
Waktu Paruh-
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Genetik -
MBL-HCV1 DB17776
biotech

MBL-HCV1 is a monoclonal antibody developed to prevent the recurrence of hepatitis C virus (HCV) in patients receiving a liver transplant.

Waktu Paruh-
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MBO7133 DB04999
small molecule

MB07133 is a HepDirect prodrug of an activated form of cytarabine (araC), an anti-cancer drug that is used to treat leukemia but is ineffective against primary liver cancer. AraC's anti-cancer activity is associated with its ability to be converted to its bio…

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MBP-091 DB17741
biotech

MBP-091 is a monoclonal antibody being investigated for the treatment of Marburg virus disease (MVD) caused by infection with Marburg virus (MARV).[L46212]

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MBS-2320 DB18059
small molecule | CAS: 1642602-54-7

Deskripsi belum tersedia.

Waktu Paruh-
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MBX-2044 DB05598
small molecule

MBX-2044 was under investigation in clinical trial NCT00422487 (Safety and Tolerability Study of MBX-2044 in Patients With Type 2 Diabetes).

Waktu Paruh-
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MBX-2982 DB12345
small molecule | CAS: 1037792-44-1

MBX-2982 has been used in trials studying the treatment of Diabetes.

Kategori:
Sulfur Compounds
Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
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Genetik -
MC-16 DB18005
small molecule | CAS: 2036329-47-0

Deskripsi belum tersedia.

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MCMV3068A DB17764
biotech

MCMV3068A is an anticytomegalovirus monoclonal IgG1 antibody used in combination with [MCMV5322A] to form RG7667.[A259362]

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MCMV5322A DB17763
biotech

MCMV5322A is an anticytomegalovirus monoclonal IgG1 antibody used in combination with [MCMV3068A] to form RG7667.[A259362]

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MD-0727 DB05948
small molecule

MD-0727 is a novel, potent cholesterol absorption inhibitor (CAI) under investigation for the treatment of hypercholesterolemia (high cholesterol.

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MD05 DB06375
small molecule

MD05 is a beta-tricalcium phosphate (beta-TCP) coated with recombinant human growth/differentiation factor-5 (rhGDF-5).

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Mdl 101,146 DB02341
small molecule | CAS: 149859-17-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsHydrocarbons, FluorinatedHydrocarbons, Halogenated +3
Target Protein:
Neutrophil elastaseChymotrypsin-like elastase family member 1
Waktu Paruh-
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Mdl-29951 DB04175
small molecule | CAS: 101861-63-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Fructose-1,6-bisphosphatase 1
Waktu Paruh-
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MDL72527 DB04188
small molecule | CAS: 99207-33-7

Deskripsi belum tersedia.

Kategori:
AminesBiogenic AminesBiogenic Polyamines +3
Target Protein:
Spermine oxidase
Waktu Paruh-
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MDX-1097 DB18383
biotech

MDX-1097 is a chimeric monoclonal antibody directed against the kappa myeloma antigen (KMA).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
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