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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Halaman 140 / 236
Lufenuron DB11424
small molecule | CAS: 103055-07-8

Lufenuron is used in veterinary for the control of flea.

Kategori:
Acids, CarbocyclicAgrochemicalsAmides +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luliconazole Approved DB08933
small molecule | CAS: 187164-19-8

Luliconazole is a topical antifungal agent that acts by unknown mechanisms but is postulated to involve altering the synthesis of fungi cell membranes. It was approved by the FDA (USA) in November 2013 and is marketed under the brand name Luzu. Luliconazole i…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +10
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhThe half life of lu…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lu…
Genetik -
LuLym-T DB17405
biotech

LuLym-T is an investigational autologous immune cell therapy consisting of activated T Lymphocytes. Developed by Lukas Biomedical, Inc., it is currently being investigated in hepatocellular carcinoma.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lumacaftor Approved DB09280
small molecule | CAS: 936727-05-8

Lumacaftor is a drug used in combination with [DB08820] as the fixed dose combination product Orkambi for the management of Cystic Fibrosis (CF) in patients aged 6 years and older. Cystic Fibrosis is an autosomal recessive disorder caused by one of several di…

Kategori:
AminesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +21
Target Protein:
Cystic fibrosis transmembrane conductance regulator
Waktu ParuhThe half-life of lu…
Vol. DistribusiFollowing oral admi…
KlirensThe typical apparen…
Genetik -
Lumasiran Approved DB15935
biotech | CAS: 1834610-13-7

Lumasiran is a small interfering RNA used in the treatment of primary hyperoxaluria type 1 (PH1).[L23554] This condition, caused by a deficiency in the enzyme alanine-glyoxylate aminotransferase, leads to an accumulation of oxalate, causing calcium crystal fo…

Kategori:
Alimentary Tract and MetabolismAntisense Elements (Genetics)Cytochrome P-450 CYP2C8 Inhibitors +12
Target Protein:
2-Hydroxyacid oxidase 1
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent centra…
KlirensThe apparent plasma…
Genetik -
Lumateperone Approved DB06077
small molecule | CAS: 313368-91-1

Schizophrenia is a complex mental illness and impacts approximately 1% of the population.[L10902] Although there are several antipsychotics including [aripiprazole], [paliperidone] and [clozapine] available for clinical use, they are generally accompanied by …

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (Second Generation [Atypical]) +21
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2AD(2) dopamine receptor +1
Waktu ParuhLumateperone's half…
Vol. DistribusiThe volume of distr…
KlirensLumateperone's clea…
Genetik -
Lumefantrine Approved DB06708
small molecule | CAS: 82186-77-4

Lumefantrine is an antimalarial agent used to treat acute uncomplicated malaria. It is administered in combination with artemether for improved efficacy. This combination therapy exerts its effects against the erythrocytic stages of <i>Plasmodium spp.</i> and…

Kategori:
Anti-Infective AgentsAntimalarialsAntiparasitic Agents +11
Target Protein:
Sodium/potassium-transporting ATPase subunit alpha-1
Waktu Paruh~ 4.5 days
Vol. Distribusi-
Klirens-
Genetik -
Lumichrome DB04345
small molecule | CAS: 1086-80-2

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Target Protein:
Flavin reductase (NADPH)Riboflavin biosynthesis protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumicitabine DB14808
small molecule | CAS: 1445385-02-3

Lumicitabine is under investigation in clinical trial NCT03010059 (A Study to Assess the Relative Bioavailability of JNJ64041575 Administered as 2 Different New Concept Formulations (Oral Suspension and Tablet) Compared to Their Respective Current Formulation…

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiflavin DB04726
small molecule | CAS: 1088-56-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoenzymesEnzymes and Coenzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiliximab DB06162
biotech | CAS: 357613-86-6

Lumiliximab is a chimeric monoclonal antibody which is used as an immunosuppressive drug. It is a primatized anti-CD23 macaque/human chimeric antibody that inhibits the production of the IgE antibody, for the potential treatment of allergic conditions. Lumili…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Low affinity immunoglobulin epsilon Fc receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lumiracoxib Approved DB01283
small molecule | CAS: 220991-20-8

Lumiracoxib is a COX-2 selective non-steroidal anti-inflammatory drug (NSAID). On August 11, 2007, Australia's Therapeutic Goods Administration (TGA, the Australian equivalent of the FDA) cancelled the registration of lumiracoxib in Australia due to concerns …

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +21
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhTerminal half-life …
Vol. Distribusi-
Klirens-
Genetik -
Lumretuzumab DB12683
biotech | CAS: 1448327-63-6

Lumretuzumab has been used in trials studying the treatment of Neoplasms, Breast Cancer, Squamous Non-Small Cell Lung Cancer, and Non-Squamous Non-Small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lunasine DB16223
small molecule | CAS: 6901-22-0

Lunasine is under investigation in clinical trial NCT02709330 (ALS Reversals - Lunasin Regimen).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lunresertib DB19241
small molecule | CAS: 2719793-90-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lunsekimig DB19009
biotech | CAS: 2770858-49-4

Lunsekimig is under investigation in clinical trial NCT06102005 (Dose Ranging Study of Lunsekimig Compared With Placebo-control in Adult Participants With Moderate-to-severe Asthma).

Waktu Paruh-
Vol. Distribusi-
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Lupeol DB12622
small molecule | CAS: 545-47-1

Lupeol has been investigated for the treatment of Acne.

Kategori:
Anti-Inflammatory AgentsPentacyclic TriterpenesTerpenes +1
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaNeutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luprostiol DB11425
small molecule | CAS: 67110-79-6

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lurasidone Approved DB08815
small molecule | CAS: 367514-87-2

Lurasidone is an atypical antipsychotic developed by Dainippon Sumitomo Pharma. It was approved by the U.S. Food and Drug Administration (FDA) for treatment of schizophrenia on October 29, 2010 and is currently pending approval for the treatment of bipolar di…

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +34
Target Protein:
D(2) dopamine receptor5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 7 +3
Waktu Paruh40 mg dose= 18 hour…
Vol. Distribusi6173 L
Klirens3902 mL/min
Genetik -
Lurbinectedin Approved DB12674
small molecule | CAS: 497871-47-3

Lurbinectedin is a DNA alkylating agent that has been investigated in the treatment of a variety of cancers, including mesothelioma,[A214325] chronic lymphocytic leukemia (CLL),[A214328] breast cancer,[A214322] and small-cell lung cancer (SCLC).[A214310] It i…

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +12
Target Protein:
DNA
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe steady-state vo…
KlirensThe total plasma cl…
Genetik -
Lusacomfar Alfa DB18526
biotech | CAS: 2640087-71-2

Lusacomfar Alfa is a recombinant complement factor H

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luseogliflozin DB12214
small molecule | CAS: 898537-18-3

Luseogliflozin has been used in trials studying the treatment of Diabetes Melltius, Type 2.

Kategori:
AlcoholsAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luspatercept Approved DB12281
biotech | CAS: 1373715-00-4

Luspatercept is a recombinant fusion protein comprised of a modified extracellular domain of activin receptor type IIB fused to the FC domain of human IgG1.[A187829,L42455] It was first approved for use in the United States in November 2019 under the brand na…

Kategori:
Activin ReceptorsAmino Acids, Peptides, and ProteinsAntianemia Drugs +25
Waktu ParuhThe average half-li…
Vol. DistribusiThe average apparen…
KlirensThe total apparent …
Genetik -
Lusutrombopag Approved DB13125
small molecule | CAS: 1110766-97-6

Lusutrombopag is an orally bioavailable thrombopoietin receptor (TPOR) agonist developed by Shionogi & Company (Osaka, Japan). TPOR is a regulatory target site for endogenous thrombopoietin, which acts as a primary cytokine to promote megakaryocyte proliferat…

Kategori:
Acids, CarbocyclicBCRP/ABCG2 SubstratesBlood and Blood Forming Organs +4
Target Protein:
Thrombopoietin receptor
Waktu ParuhIn healthy adult su…
Vol. DistribusiThe mean (%CV) lusu…
KlirensThe approximate mea…
Genetik -
Lusvertikimab DB18778
biotech | CAS: 2375835-91-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lutein Approved DB00137
small molecule | CAS: 127-40-2

Lutein is an xanthophyll and one of 600 known naturally occurring carotenoids. Lutein is synthesized only by plants and like other xanthophylls is found in high quantities in green leafy vegetables such as spinach, kale and yellow carrots. In green plants, xa…

Kategori:
AlkenesBiological FactorsCarotenoids +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luteinizing hormone Approved DB14741
biotech | CAS: 9002-67-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsGonadotropinsGonadotropins, Pituitary +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Luteolin DB15584
small molecule | CAS: 491-70-3

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFlavones +3
Target Protein:
Signal transducer and activator of transcription 3Lysophosphatidylcholine acyltransferase 2Lysophosphatidylcholine acyltransferase 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lutetium Lu 177 dotatate Approved DB13985
small molecule | CAS: 437608-50-9

A 177Lu-labeled somatostatin analog peptide, Lutetium Lu 177 dotatate belongs to an emerging form of treatments called Peptide Receptor Radionuclide Therapy (PRRT), which involves targeting tumours with molecules carrying radioactive particles that bind to sp…

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +8
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 1Somatostatin receptor type 3 +2
Waktu ParuhThe mean (± standar…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
Lutetium Lu-177 Approved DB13982
small molecule | CAS: 14265-75-9

Deskripsi belum tersedia.

Kategori:
ElementsIsotopesLanthanoid Series Elements +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1703749-62-5

Lutetium Lu-177 vipivotide tetraxetan is a radioligand therapeutic agent. It consists of a radionuclide, [lutetium Lu-177], linked to a moiety that binds to PSMA, a transmembrane protein that is expressed in prostate cancer.[L41280] Lutetium Lu-177 vipivot…

Kategori:
Compounds used in a research, industrial, or household settingDiagnostic Uses of ChemicalsRadioactive Therapeutic Agent +6
Target Protein:
Prostate-specific antigen
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 321835-55-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsCompounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lutikizumab DB16224
biotech | CAS: 1791411-57-8

Lutikizumab is under investigation in clinical trial NCT02087904 (A Study Evaluating the Safety, Efficacy, and Pharmacodynamic Effects of ABT-981 in Patients With Knee Osteoarthritis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lutropin alfa Approved DB00044
biotech | CAS: 152923-57-4

Lutropin alfa is a recombinant human luteinizing hormone produced in yeast with 2 subunits, alpha = 92 residues, beta = 121 residues. It is a heterodimeric glycoprotein made up of monomeric units. Lutropin alfa was the first and only recombinant human form of…

Kategori:
Genito Urinary System and Sex HormonesGonadotropinsGonadotropins and Antigonadotropins +1
Target Protein:
Lutropin-choriogonadotropic hormone receptor
Waktu ParuhBiphasic; terminal …
Vol. DistribusiThe steady state vo…
Klirens* 2 – 3 L/h [health…
Genetik -
Luvadaxistat DB16067
small molecule | CAS: 1425511-32-5

Luvadaxistat is under investigation in clinical trial NCT03214588 (Efficacy, Tolerability, and Pharmacokinetics of Multiple Doses of Oral TAK-831 in Adults With Friedreich Ataxia).

Kategori:
D-Amino Acid Oxidase Inhibitor
Target Protein:
D-amino-acid oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Luveltamab tazevibulin, formerly known as STRO-002, is novel homogeneous folate receptor alpha (FolR?) targeting antibody-drug conjugate.[A257414] It is under investigation in clinical trial NCT05200364 (A Study of STRO-002, an Anti-folate Receptor Alpha Anti…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Luvixasertib DB19200
small molecule | CAS: 1610759-22-2

Luvixasertib is under investigation in clinical trial NCT05251714 (CFI-402257, a Potent and Selective TTK Inhibitor, in Solid Tumors and With Fulvestrant in Breast Cancer).

Waktu Paruh-
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Klirens-
Genetik -
Luxeptinib DB19179
small molecule | CAS: 1616428-23-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LV-FAH DB17686
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LV305 DB17288
biotech

LV305 is a lentiviral vector encoding NY-ESO-1 gene. LV305 is an active component of CMB305 along with [G305].[L47346]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX-1004 DB18272
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX-2931 DB06297
small molecule | CAS: 948840-25-3

Deskripsi belum tersedia.

Kategori:
AminesHydroxylamines
Target Protein:
Sphingosine-1-phosphate lyase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX-7101 DB16009
small molecule | CAS: 1192189-69-7

LX-7101 is under investigation in clinical trial NCT01528111 (Study to Evaluate the Safety, Tolerability, and Efficacy of LX7101 in Subjects With Primary Open-angle Glaucoma or Ocular Hypertension).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX2006 DB18273
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LX6171 DB05180
small molecule

LX6171 is an oral drug candidate that was generated by Lexicon medicinal chemists and is being developed to treat disorders characterized by cognitive impairment, such as Alzheimer's disease, schizophrenia or vascular dementia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2183240 DB17035
small molecule | CAS: 874902-19-9

LY-2183240 is an inhibitor of endocannabinoid reuptake/breakdown.[A253037]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2300559 DB13016
small molecule | CAS: 889116-06-7

Ly2300559 has been used in trials studying the prevention of Migraine Headache.

Kategori:
Acids, CarbocyclicBenzene DerivativesKetones
Target Protein:
Metabotropic glutamate receptor 2Cysteinyl leukotriene receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2334737 DB12906
small molecule | CAS: 892128-60-8

LY2334737 has been used in trials studying the treatment of Solid Tumor, Metastatic Tumor, and Malignant Solid Tumor.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2452473 DB12573
small molecule | CAS: 1029692-15-6

Ly2452473 is under investigation for the supportive care of Prostate Cancer. Ly2452473 has been investigated for the treatment of Erectile Dysfunction.

Kategori:
Acids, Acyclic
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LY-2584702 DB12690
small molecule | CAS: 1082949-67-4

LY2584702 has been used in trials studying the treatment of Cancer, Advanced Cancer, Renal Cell Carcinoma, Metastases, Neoplasm, and Neuroendocrine Tumors, among others.

Kategori:
Ribosomal Protein S6 Kinases, 70-kDa, antagonists & inhibitors
Waktu Paruh-
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Genetik -
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