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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 140 / 282
Guanosine DB02857
small molecule | CAS: 118-00-3

Guanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a ?-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP (guanosine diphosphate) and G…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunitPurine nucleoside phosphorylase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenylosuccinate synthetaseBifunctional (p)ppGpp synthase/hydrolase RelA
Waktu Paruh-
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Genetik -
small molecule | CAS: 33503-72-9

Guanosine tetraphosphate is a guanine nucleotide containing four phosphate groups. Two phosphate groups are esterified to the sugar moiety in the 5' position and the other two in the 2' or 3' position. This nucleotide serves as a messenger to turn off the syn…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferaseGTPase Obg
Waktu Paruh-
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Genetik -
small molecule | CAS: 38557-85-6

Deskripsi belum tersedia.

Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
small molecule | CAS: 130-50-7

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP-ribosylation factor 1
Waktu Paruh-
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Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 4,6 dehydratase
Waktu Paruh-
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Genetik -
small molecule | CAS: 85-32-5

Guanosine 5'-monophosphate. A guanine nucleotide containing one phosphate group esterified to the sugar moiety and found widely in nature. [PubChem]

Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseDNA polymerase catalytic subunitDNA polymerase catalytic subunit +14
Waktu Paruh-
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Genetik -
Guanoxabenz DB13410
small molecule | CAS: 24047-25-4

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
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Genetik -
Guanoxan Approved DB13211
small molecule | CAS: 2165-19-7

Guanoxan is an antihypertensive agent similar in its mechanism of action to guanethidine; may cause liver damage. Guanoxan was approved in the UK but was withdrawn from the market due to hepatotoxicity.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
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Gunagratinib DB18191
small molecule | CAS: 2211082-53-8

Deskripsi belum tersedia.

Waktu Paruh-
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Gusacitinib DB15670
small molecule | CAS: 1425381-60-7

Gusacitinib is under investigation in clinical trial NCT02550678 (A Study of the Efficacy and Safety of ASN-002 in Adult Patients With Low-risk Nodular Basal Cell Carcinoma).

Kategori:
Nitriles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
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Guselkumab Approved DB11834
biotech | CAS: 1350289-85-8

Guselkumab is a human immunoglobulin G1 lambda (IgG1?) monoclonal antibody that selectively blocks interleukin-23. IL-23 is an inflammatory cytokine that activates the CD4+ T-helper (Th17) cell pathway to mediate the inflammatory cascade that induces psoriati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhMean half-life of g…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Gusperimus DB12692
small molecule | CAS: 98629-43-7

Gusperimus has been used in trials studying the treatment of Lupus Nephritis, Wegeners Granulomatosis, and Wegener's Granulomatosis.

Kategori:
AmidinesAntibiotics, AntineoplasticAntineoplastic Agents +7
Waktu Paruh-
Vol. Distribusi-
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GVAX DB17276
biotech

GVAX is a granulocyte-macrophage colony-stimulating factor (GM-CSF) gene-transfected tumor cell vaccine.

Waktu Paruh-
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GW 468816 DB05417
small molecule

GW 468816 is glycine receptor antagonist. It is designed to aid abstinence in people who have just quit smoking, delaying the time to relapse. It was undergoing phase II trials since December 2003.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glycine receptor subunit alpha-1
Waktu Paruh-
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Genetik -
GW-274150 DB12237
small molecule | CAS: 210354-22-6

GW274150 has been used in trials studying the treatment and prevention of Asthma, Migraine, Migraine Disorders, and Arthritis, Rheumatoid.

Kategori:
AnionsElectrolytesHydrogen Sulfide +3
Target Protein:
Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-406381 DB12009
small molecule | CAS: 221148-46-5

GW-406381 has been used in trials studying the treatment of Pain, Trauma, Neurodynia, Dental Pain, and Hyperalgesia, among others.

Target Protein:
Prostaglandin G/H synthase 2
Waktu Paruh-
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GW-468816 DB15099
small molecule | CAS: 476689-77-7

GW-468816 is under investigation in clinical trial NCT00218465 (Effectiveness of GW468816, an NMDA Glycine Site Antagonist, for Prevention of Relapse to Smoking).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Waktu Paruh-
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GW-493838 DB12760
small molecule | CAS: 253124-46-8

GW493838 has been used in trials studying the treatment of Neuropathic Pain.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-559090 DB06508
small molecule | CAS: 278598-52-0

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Integrin alpha-5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
GW-590735 DB07215
small molecule | CAS: 343321-96-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Nuclear receptor coactivator 1Peroxisome proliferator-activated receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-813893 DB07278
small molecule | CAS: 478644-12-1

Deskripsi belum tersedia.

Kategori:
AmidesAnticoagulantsAntithrombins +8
Target Protein:
Coagulation factor XProthrombin
Waktu Paruh-
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GW-870086 DB12322
small molecule | CAS: 827319-43-7

GW870086X has been investigated for the treatment of ASTHMA.

Kategori:
Fused-Ring Compounds
Waktu Paruh-
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GW810781 DB16032
small molecule | CAS: 280571-30-4

GW810781 is under investigation in clinical trial NCT00046332 (A Study Comparing 4 Doses of GW810781 Versus Placebo in Hiv-infected Patients).

Kategori:
Anti-HIV Agents
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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GW842166 DB11903
small molecule | CAS: 666260-75-9

GW842166X has been used in trials studying the treatment of Pain, Analgesia, Inflammation, Osteoarthritis, and Pain, Inflammatory, among others.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +1
Target Protein:
Cannabinoid receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GX-19 Vaccine DB15891
biotech

The GX-19 vaccine is a DNA vaccine created by Genexine, Inc. Company in Gyeonggi, Korea[A219758]. As of June 2020, the vaccine candidate is undergoing Phase I and Phase IIa trials to determine dose levels for safety and efficacy[A219758,L16488].

Waktu Paruh-
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GX-G8 DB18196
biotech

GX-G8 is a long-acting glucagon-like peptide 2 (GLP-2) being investigated for the treatment of short bowel syndrome.

Waktu Paruh-
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GYM329 DB18590
biotech

GYM329 is a recombinant humanized IgG1-based monoclonal antibody which binds to human latent myostatin in a pH-dependent manner

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GZ-389988 DB16056
small molecule | CAS: 1788906-96-6

GZ-389988 is under investigation in clinical trial NCT02845271 (Proof-of-concept Study to Assess the Efficacy, Tolerability and Safety of a Single Intraarticular Dose of GZ389988 Versus Placebo in Patients With Painful Osteoarthritis of the Knee).

Target Protein:
NT-3 growth factor receptorHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H-89 DB07995
small molecule | CAS: 127243-85-0

Deskripsi belum tersedia.

Kategori:
AmidesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
cAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alphaSerine/threonine-protein kinase haspin +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H3B-6527 DB15169
small molecule | CAS: 1702259-66-2

H3B-6527 is under investigation in clinical trial NCT03424577 (A Study to Evaluate the Food-Effect of H3B-6527).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H3B-8800 DB14017
small molecule | CAS: 1825302-42-8

H3B-8800 is a novel spliceosome inhibitor developed by H3 Biomedicine [L2551]. It offers the benefit of preferentially killing spliceosome-mutant cancer cells whereas other splicesome inhibitors, such as the pladienolide analogue E7107, show no such preferent…

Target Protein:
Splicing factor 3B subunit 1
Waktu Paruh-
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Hachimycin DB13302
small molecule | CAS: 1394-02-1

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungals for Dermatological UseAntifungals for Topical Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hadacidin DB02109
small molecule | CAS: 689-13-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntibiotics, Antineoplastic +4
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Adenylosuccinate synthetaseAdenylosuccinate synthetase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Haemagglutinin-strain B Approved DB15482
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
biotech

Haemophilus influenzae type b capsular polysaccharide meningococcal outer membrane protein conjugate antigen is a vaccine containing outer membrane antigen extracted from *Haemophilus influenzae*.

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine
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Genetik -
biotech

Haemophilus influenzae type b strain 1482 capsular polysaccharide tetanus toxoid conjugate antigen is a vaccine for intramuscular injection used in the prevention of invasive disease caused by *Haemophilus influenzae* type b. *H. influenzae* is a Gram-negativ…

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Haemophilus influenzae type b strain 20752 capsular polysaccharide tetanus toxoid conjugate antigen is an active immunization as a booster dose given intramuscularly to pediatric patients who have received a primary series with a Haemophilus b Conjugate Vacci…

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Hafnium oxide DB17508
small molecule | CAS: 12055-23-1

Deskripsi belum tersedia.

Kategori:
AnionsElectrolytesElements +5
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Halazepam Approved DB00801
small molecule | CAS: 23092-17-3

Halazepam is a _benzodiazepine_ derivative drug exerting anxiolytic, anticonvulsant, sedative, a muscle relaxing effects.[A1212, A178114] It has been shown to be less toxic than chlordiazepoxide or diazepam.[A1212] This drug is no longer marketed in the Unite…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
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Genetik -
Halcinonide Approved DB06786
small molecule | CAS: 3093-35-4

Halcinonide is a corticosteroid indicated for the relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses, and is distributed as a cream and ointment. Halcinonide is marketed under the brand name Halog® by Ranbaxy Labora…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +13
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
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Haletazole DB15942
small molecule | CAS: 15599-36-7

Deskripsi belum tersedia.

Waktu Paruh-
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Halicin DB15624
small molecule | CAS: 40045-50-9

Deskripsi belum tersedia.

Kategori:
Sulfur CompoundsThiazoles
Target Protein:
c-Jun N-terminal kinases
Waktu Paruh-
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Halofantrine Approved DB01218
small molecule | CAS: 69756-53-2

Halofantrine is an antimalarial. It belongs to the phenanthrene class of compounds that includes quinine and lumefantrine. It appears to inhibit polymerisation of heme molecules (by the parasite enzyme "heme polymerase"), resulting in the parasite being poiso…

Kategori:
Agents that reduce seizure thresholdAnti-Infective AgentsAntimalarials +13
Target Protein:
Fe(II)-protoporphyrin IXCalmodulin-1Calmodulin-3 +3
Waktu Paruh6-10 days
Vol. Distribusi-
Klirens-
Genetik -
Halofuginone DB04866
small molecule | CAS: 55837-20-2

Halofuginone is a low molecular weight quinazolinone alkaloid, and a potent inhibitor of collagen alpha1(I) and matrix metalloproteinase 2 (MMP-2) gene expression. Halofuginone also effectively suppresses tumor progression and metastasis in mice. Collgard Bio…

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAnti-Infective Agents +10
Target Protein:
Collagen alpha-1(I) chain72 kDa type IV collagenase
Waktu Paruh23.8 to 72.1 hours
Vol. Distribusi-
Klirens-
Genetik -
Halometasone DB13728
small molecule | CAS: 50629-82-8

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroids +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6951–7000 dari 14063
Sebelumnya Halaman 140 / 282 Berikutnya