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14494

Total database: 17430
Struktur (SMILES)
9687 (66.8%)
Target
7525 (51.9%)
Genomik
112 (0.8%)
Referensi
14494 (100.0%)

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Hasil Pencarian (14494)

Halaman 139 / 290
Guanabenz Approved DB00629
small molecule | CAS: 5051-62-7

An alpha-2 selective adrenergic agonist used as an antihypertensive agent. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +11
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu Paruh6 hours.
Vol. Distribusi-
Klirens-
Genetik -
Guanadrel Approved DB00226
small molecule | CAS: 40580-59-4

Guanadrel is an antihypertensive agent and postganglionic adrenergic blocking agent.

Kategori:
Adrenergic AntagonistsAmidinesAntihypertensive Agents +1
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh10 hours
Vol. Distribusi-
Klirens-
Genetik -
Guanethidine Approved DB01170
small molecule | CAS: 55-65-2

An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sym…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmidines +16
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh1.5 days
Vol. Distribusi-
Klirens* Renal cl=56 ml/min
Genetik -
Guanfacine Approved DB01018
small molecule | CAS: 29110-47-2

Guanfacine, or BS 100-141,[A189838,A189841] is a selective alpha-A2 adrenergic receptor agonist initially indicated for the treatment of hypertension[L11274] but is now indicated as an extended release tablet for the treatment of ADHD.[L11277] Guanfacine was …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +26
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu ParuhGuanfacine has a ha…
Vol. DistribusiGuanfacine has a vo…
KlirensGuanfacine has a to…
Genetik -
Guanidine Approved DB00536
small molecule | CAS: 113-00-8

A strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of protein metabolism. It is also used in laboratory research as a protein denaturant. (From Martindale, the Extra Pharmacopoeia, 30th…

Kategori:
Acetylcholine Releasing AgentAmidinesGuanidines +7
Target Protein:
Aldehyde dehydrogenase, mitochondrialRibonuclease pancreaticDNA +4
Waktu Paruh7-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77482-44-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
Carboxypeptidase D
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoclor DB13779
small molecule | CAS: 5001-32-1

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanosine DB02857
small molecule | CAS: 118-00-3

Guanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a ?-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP (guanosine diphosphate) and G…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunitPurine nucleoside phosphorylase +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 117-68-0

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
RibonucleaseBifunctional protein PyrR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenylosuccinate synthetaseBifunctional (p)ppGpp synthase/hydrolase RelA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 33503-72-9

Guanosine tetraphosphate is a guanine nucleotide containing four phosphate groups. Two phosphate groups are esterified to the sugar moiety in the 5' position and the other two in the 2' or 3' position. This nucleotide serves as a messenger to turn off the syn…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferaseGTPase Obg
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 38557-85-6

Deskripsi belum tersedia.

Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 130-50-7

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 146-91-8

A guanine nucleotide containing two phosphate groups esterified to the sugar moiety. [PubChem]

Target Protein:
Protein-glutamine gamma-glutamyltransferase 2Elongation factor 1-alphaAdenylosuccinate synthetase +49
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 85-32-5

Guanosine 5'-monophosphate. A guanine nucleotide containing one phosphate group esterified to the sugar moiety and found widely in nature. [PubChem]

Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseDNA polymerase catalytic subunitDNA polymerase catalytic subunit +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 86-01-1

Guanosine 5'-(tetrahydrogen triphosphate). A guanine nucleotide containing three phosphate groups esterified to the sugar moiety. [PubChem]

Target Protein:
GTP cyclohydrolase 1Genome polyproteinRNA-directed RNA polymerase +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guanoxan Approved DB13211
small molecule | CAS: 2165-19-7

Guanoxan is an antihypertensive agent similar in its mechanism of action to guanethidine; may cause liver damage. Guanoxan was approved in the UK but was withdrawn from the market due to hepatotoxicity.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gunagratinib DB18191
small molecule | CAS: 2211082-53-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gusacitinib DB15670
small molecule | CAS: 1425381-60-7

Gusacitinib is under investigation in clinical trial NCT02550678 (A Study of the Efficacy and Safety of ASN-002 in Adult Patients With Low-risk Nodular Basal Cell Carcinoma).

Kategori:
Nitriles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Guselkumab Approved DB11834
biotech | CAS: 1350289-85-8

Guselkumab is a human immunoglobulin G1 lambda (IgG1?) monoclonal antibody that selectively blocks interleukin-23. IL-23 is an inflammatory cytokine that activates the CD4+ T-helper (Th17) cell pathway to mediate the inflammatory cascade that induces psoriati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhMean half-life of g…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Guvacine DB08848
small molecule | CAS: 498-96-4

Guvacine is a pyridine alkaloid found in the Areca nut (also known as the Betel nut). It is an experimental drug with no approved indication. Experimental studies are still being investigated to determine all of the physiological effects and mechanisms of act…

Kategori:
Pyridines
Target Protein:
Sodium- and chloride-dependent GABA transporter 2Sodium- and chloride-dependent GABA transporter 1Sodium- and chloride-dependent GABA transporter 3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GVAX DB17276
biotech

GVAX is a granulocyte-macrophage colony-stimulating factor (GM-CSF) gene-transfected tumor cell vaccine.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW 468816 DB05417
small molecule

GW 468816 is glycine receptor antagonist. It is designed to aid abstinence in people who have just quit smoking, delaying the time to relapse. It was undergoing phase II trials since December 2003.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glycine receptor subunit alpha-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW 597599 DB05418
small molecule

GW 597599, a neurokinin-1 (NK1) receptor antagonist is currently in phase II trials for chemotherapy-induced vomiting; functional dyspepsia; depression and anxiety.

Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-3965 DB03791
small molecule | CAS: 405911-09-3

GW-3965 is a liver X receptor ligand.

Kategori:
Acids, CarbocyclicAminesBenzene Derivatives +2
Target Protein:
Oxysterols receptor LXR-betaOxysterols receptor LXR-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-468816 DB15099
small molecule | CAS: 476689-77-7

GW-468816 is under investigation in clinical trial NCT00218465 (Effectiveness of GW468816, an NMDA Glycine Site Antagonist, for Prevention of Relapse to Smoking).

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW-493838 DB12760
small molecule | CAS: 253124-46-8

GW493838 has been used in trials studying the treatment of Neuropathic Pain.

Target Protein:
Adenosine receptor A1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GW810781 DB16032
small molecule | CAS: 280571-30-4

GW810781 is under investigation in clinical trial NCT00046332 (A Study Comparing 4 Doses of GW810781 Versus Placebo in Hiv-infected Patients).

Kategori:
Anti-HIV Agents
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GX-19 Vaccine DB15891
biotech

The GX-19 vaccine is a DNA vaccine created by Genexine, Inc. Company in Gyeonggi, Korea[A219758]. As of June 2020, the vaccine candidate is undergoing Phase I and Phase IIa trials to determine dose levels for safety and efficacy[A219758,L16488].

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GX-G8 DB18196
biotech

GX-G8 is a long-acting glucagon-like peptide 2 (GLP-2) being investigated for the treatment of short bowel syndrome.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GXC-301 DB18831
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GYM329 DB18590
biotech

GYM329 is a recombinant humanized IgG1-based monoclonal antibody which binds to human latent myostatin in a pH-dependent manner

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GZ-389988 DB16056
small molecule | CAS: 1788906-96-6

GZ-389988 is under investigation in clinical trial NCT02845271 (Proof-of-concept Study to Assess the Efficacy, Tolerability and Safety of a Single Intraarticular Dose of GZ389988 Versus Placebo in Patients With Painful Osteoarthritis of the Knee).

Target Protein:
NT-3 growth factor receptorHigh affinity nerve growth factor receptorBDNF/NT-3 growth factors receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Histo-blood group ABO system transferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H-89 DB07995
small molecule | CAS: 127243-85-0

Deskripsi belum tersedia.

Kategori:
AmidesEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
cAMP-dependent protein kinase catalytic subunit alphacAMP-dependent protein kinase inhibitor alphaSerine/threonine-protein kinase haspin +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H3B-6527 DB15169
small molecule | CAS: 1702259-66-2

H3B-6527 is under investigation in clinical trial NCT03424577 (A Study to Evaluate the Food-Effect of H3B-6527).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
H3B-8800 DB14017
small molecule | CAS: 1825302-42-8

H3B-8800 is a novel spliceosome inhibitor developed by H3 Biomedicine [L2551]. It offers the benefit of preferentially killing spliceosome-mutant cancer cells whereas other splicesome inhibitors, such as the pladienolide analogue E7107, show no such preferent…

Target Protein:
Splicing factor 3B subunit 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hachimycin DB13302
small molecule | CAS: 1394-02-1

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungals for Dermatological UseAntifungals for Topical Use +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hadacidin DB02109
small molecule | CAS: 689-13-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntibiotics, Antineoplastic +4
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Adenylosuccinate synthetaseAdenylosuccinate synthetase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Haddock Approved DB10615
biotech

Haddock allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Haematonectria haematococca Approved DB10934
biotech

Haematonectria haematococca is a fungus which can provoke allergic reactions. Haematonectria haematococca extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Haemophilus influenzae type b capsular polysaccharide meningococcal outer membrane protein conjugate antigen is a vaccine containing outer membrane antigen extracted from *Haemophilus influenzae*.

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Haemophilus influenzae type b strain 1482 capsular polysaccharide tetanus toxoid conjugate antigen is a vaccine for intramuscular injection used in the prevention of invasive disease caused by *Haemophilus influenzae* type b. *H. influenzae* is a Gram-negativ…

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Haemophilus influenzae type b strain 20752 capsular polysaccharide tetanus toxoid conjugate antigen is an active immunization as a booster dose given intramuscularly to pediatric patients who have received a primary series with a Haemophilus b Conjugate Vacci…

Kategori:
Actively Acquired ImmunityHaemophilus VaccinesInactivated Haemophilus Influenzae B Vaccine +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Hafnium oxide DB17508
small molecule | CAS: 12055-23-1

Deskripsi belum tersedia.

Kategori:
AnionsElectrolytesElements +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Halazepam Approved DB00801
small molecule | CAS: 23092-17-3

Halazepam is a _benzodiazepine_ derivative drug exerting anxiolytic, anticonvulsant, sedative, a muscle relaxing effects.[A1212, A178114] It has been shown to be less toxic than chlordiazepoxide or diazepam.[A1212] This drug is no longer marketed in the Unite…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +7
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Halcinonide Approved DB06786
small molecule | CAS: 3093-35-4

Halcinonide is a corticosteroid indicated for the relief of the inflammatory and pruritic manifestations of corticosteroid-responsive dermatoses, and is distributed as a cream and ointment. Halcinonide is marketed under the brand name Halog® by Ranbaxy Labora…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +13
Target Protein:
Steroid hormone receptor ERR1Steroid hormone receptor ERR2Estrogen-related receptor gamma +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Halicin DB15624
small molecule | CAS: 40045-50-9

Deskripsi belum tersedia.

Kategori:
Sulfur CompoundsThiazoles
Target Protein:
c-Jun N-terminal kinases
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6901–6950 dari 14494
Sebelumnya Halaman 139 / 290 Berikutnya