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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Halaman 139 / 236
Lomvastomig DB19060
biotech | CAS: 2648840-52-0

Lomvastomig is under investigation in clinical trial NCT04785820 (A Study of Lomvastomig (RO7121661) and Tobemstomig (RO7247669) Compared With Nivolumab in Participants With Advanced or Metastatic Squamous Cell Carcinoma of the Esophagus).

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Lonafarnib Approved DB06448
small molecule | CAS: 193275-84-2

Hutchinson-Gilford progeria syndrome (HGPS) is a rare autosomal dominant disorder estimated to affect approximately one in 20 million individuals resulting in adverse symptoms associated with premature ageing: skeletal dysplasia, joint contractures, atheroscl…

Kategori:
Alimentary Tract and MetabolismBCRP/ABCG2 InhibitorsBenzocycloheptenes +30
Target Protein:
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta
Waktu ParuhLonafarnib has a me…
Vol. DistribusiIn healthy patients…
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Genetik -
Lonapegsomatropin Approved DB16220
biotech | CAS: 1934255-39-6

Lonapegsomatropin, also known as TransCon hGH or ACP 001, is a methoxypegylated prodrug of human growth hormone ([somatropin]) indicated for the treatment of children 1 year and older, weighing at least 11.5 kg, with growth failure due to insufficient growth …

Kategori:
Amino Acids, Peptides, and ProteinsAnterior Pituitary Lobe Hormones and AnaloguesCytochrome P-450 CYP1A2 Inducers +18
Target Protein:
Growth hormone receptorProlactin receptor
Waktu ParuhThe half life of lo…
Vol. DistribusiLonapegsomatropin-t…
KlirensIn pediatric patien…
Genetik -
Lonaprisan DB16221
small molecule | CAS: 211254-73-8

Lonaprisan is under investigation in clinical trial NCT00555919 (ZK 230211 in Postmenopausal Woman With Metastatic Breast Cancer).

Kategori:
EstranesFused-Ring CompoundsHydrocarbons, Fluorinated +2
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor
Waktu Paruh-
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Loncastuximab tesirine Approved DB16222
biotech | CAS: 1879918-31-6

Relapsed and refractory B-cell acute lymphoblastic leukemia (B-ALL) are a therapeutic challenge for patients who have undergone prior systemic therapies with limited success.[A234439] Prognosis is poor and more effective therapies are needed to treat relapsed…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
B-lymphocyte antigen CD19
Waktu ParuhThe half-life of lo…
Vol. DistribusiIn clinical studies…
KlirensIn pharmacokinetic …
Genetik -
Londamocitinib DB19190
small molecule | CAS: 2241039-81-4

Londamocitinib is under investigation in clinical trial NCT06020014 (Phase 2a Study to Assess the Efficacy and Safety of AZD4604 in Adult Patients With Moderate-to-severe Asthma Uncontrolled on Medium-high Dose ICS-LABA).

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Lonigutamab DB18940
biotech | CAS: 2362015-67-4

Lonigutamab is under investigation in clinical trial NCT05683496 (Efficacy and Safety of Lonigutamab in Subjects With Thyroid Eye Disease (TED)).

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Loperamide Approved DB00836
small molecule | CAS: 53179-11-6

Loperamide is an anti-diarrheal agent that is available as an over-the-counter product for treating diarrhea.[L42785] The drug was first synthesized in 1969 and used medically in 1976.[A251610] It is a highly lipophilic synthetic phenylpiperidine opioid that …

Kategori:
Agents causing hyperkalemiaAlimentary Tract and MetabolismAntiarrhythmic agents +20
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +4
Waktu ParuhThe apparent elimin…
Vol. DistribusiLoperamide has a la…
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Lopinavir Approved DB01601
small molecule | CAS: 192725-17-0

Lopinavir is an antiretroviral protease inhibitor used in combination with other antiretrovirals in the treatment of HIV-1 infection.[L11163] Lopinavir is marketed and administered exclusively in combination with [ritonavir] - this combination, first marketed…

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +42
Target Protein:
Pol polyprotein
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe estimated appar…
Genetik -
Loprazolam DB13643
small molecule | CAS: 61197-73-7

Loprazolam is an imidazobenzodiazepine with anxiolytic, anticonvulsant, hypnotic, sedative and skeletal muscle relaxant properties. It is indicated for the short-term treatment of insomnia including difficulty in falling asleep and/or frequent nocturnal awake…

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepine hypnotics and sedatives +9
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
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Loracarbef Approved DB00447
small molecule | CAS: 76470-66-1

Loracarbef is a carbacephem antibiotic sometimes grouped together with the second-generation cephalosporin antibiotics. It is marketed under the trade name Lorabid.

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Penicillin-binding protein 3Penicillin-binding protein 1A
Waktu Paruh1 hour. In subjects…
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Lorajmine DB13651
small molecule | CAS: 47562-08-3

Deskripsi belum tersedia.

Kategori:
AlkaloidsAntiarrhythmic agentsAntiarrhythmics, Class I +11
Waktu Paruh-
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Loratadine Approved DB00455
small molecule | CAS: 79794-75-5

Loratadine is a second generation antihistamine used to manage symptoms of allergic rhinitis.[A176435] A lack of sedative and CNS adverse effects make loratadine, along with other second generation antihistamines, preferable over their 1st generation counterp…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseAntipruritics +34
Target Protein:
Histamine H1 receptorVoltage-gated inwardly rectifying potassium channel KCNH2
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of lo…
Genetik -
Lorazepam Approved DB00186
small molecule | CAS: 846-49-1

Lorazepam is a short-acting and rapidly cleared benzodiazepine used commonly as a sedative and anxiolytic.[A957] It was developed by DJ Richards, presented and marketed initially by Wyeth Pharmaceuticals in the USA in 1977. The first historic FDA label approv…

Kategori:
Anti-Anxiety AgentsAnticonvulsantsAntiemetics +21
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhWhen administered p…
Vol. DistribusiThe reported volume…
Klirens_In vivo_ studies w…
Genetik -
Lorcainide DB13653
small molecule | CAS: 59729-31-6

Deskripsi belum tersedia.

Kategori:
AcetamidesAmidesAntiarrhythmic agents +7
Waktu Paruh-
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Lorcaserin Approved DB04871
small molecule | CAS: 616202-92-7

Lorcaserin (previously APD-356), a highly selective 5HT2C receptor agonist, is used for the treatment of obesity. It has been shown to reduce body weight and food intake in animal models of obesity, and it is thought that targeting the 5HT2C receptor may alte…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiobesity Preparations, Excl. Diet Products +22
Target Protein:
5-hydroxytryptamine receptor 2C
Waktu ParuhThe plasma half lif…
Vol. DistribusiThe volume of distr…
KlirensThe clearance value…
Genetik -
Lorecivivint DB14883
small molecule | CAS: 1467093-03-3

Lorecivivint is under investigation in clinical trial NCT03246399 (A Study of the Safety, Tolerability, and Pharmacokinetics of SM04690 Injectable Suspension Following Single Intradiscal Injection in Subjects With Degenerative Disc Disease).

Kategori:
Anti-Inflammatory AgentsHeterocyclic Compounds, Fused-RingPyrazoles
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Lorigerlimab DB18942
biotech | CAS: 2416595-46-3

Lorigerlimab is under investigation in clinical trial NCT05848011 (A Study of Lorigerlimab With Docetaxel or Docetaxel Alone in Participants With Metastatic Castration-resistant Prostate Cancer).

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Lormetazepam Approved DB13872
small molecule | CAS: 848-75-9

Lormatazepam is an orally available benzodiazepine used in the UK for the treatment of short-term insomnia [L927]. It is marketed by Auden Mckenzie (Pharma Division) in 0.5 and 1 mg tablet formulations.

Kategori:
BenzazepinesBenzodiazepines and benzodiazepine derivativesBenzodiazepinones +6
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhThe terminal phase …
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Lornoxicam Approved DB06725
small molecule | CAS: 70374-39-9

Lornoxicam (chlortenoxicam) is a new nonsteroidal anti-inflammatory drug (NSAID) of the oxicam class with analgesic, anti-inflammatory and antipyretic properties. Lornoxicam differs from other oxicam compounds in its potent inhibition of prostaglandin biosynt…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +17
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh3-5 hours
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Lorpiprazole Approved DB09195
small molecule | CAS: 108785-69-9

Lorpiprazole is a serotonin antagonist and reuptake inhibitor used for the treatment of major depressive disorder.[A31634] It is a piperazinyl-triazole derivative.[T83]

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2D6 Substrates +10
Target Protein:
5-hydroxytryptamine receptor 2A5-hydroxytryptamine receptor 2CAlpha-1 adrenergic receptors +3
Waktu ParuhThe estimated half-…
Vol. DistribusiThe serotonin antag…
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Lortalamine DB09187
small molecule | CAS: 70384-91-7

Lortalamine (LM-1404) is a selective norepinephrine reuptake inhibitor developed in the 1980s. This drug never made it past clinical trials, likely due to ocular toxicity in animals, but has been used in positron emission tomography studies to label norepinep…

Kategori:
Adrenergic Uptake InhibitorsAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
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Lorukafusp alfa DB15443
biotech | CAS: 2131168-99-3

Lorukafusp alfa is under investigation in clinical trial NCT01334515 (Biological Therapy, Sargramostim, and Isotretinoin in Treating Patients With Relapsed or Refractory Neuroblastoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBiological Factors +11
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Lorundrostat DB18957
small molecule | CAS: 1820940-17-7

Lorundrostat is under investigation in clinical trial NCT06153693 (Efficacy and Safety of Lorundrostat in Subjects With Uncontrolled and Resistant Hypertension).

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Losartan Approved DB00678
small molecule | CAS: 114798-26-4

Losartan is an angiotensin II receptor blocker (ARB) used to treat hypertension.[L7423] Angiotensin-converting enzyme (ACE) inhibitors are used for a similar indication but are associated with a cough.[L7423] When patients with ACE inhibitor associated coughs…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +39
Target Protein:
Erythropoietin receptorType-1 angiotensin II receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensLosartan has a tota…
Genetik -
Losmapimod DB12270
small molecule | CAS: 585543-15-3

Losmapimod has been investigated for the prevention of Chronic Obstructive Pulmonary Disease.

Kategori:
Cycloparaffinsp38 Mitogen-Activated Protein KinasesProtein Kinase Inhibitors
Target Protein:
Mitogen-activated protein kinase 14
Waktu Paruh-
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Loteprednol Approved DB00873
small molecule | CAS: 129260-79-3

Deskripsi belum tersedia.

Kategori:
Adrenal Cortex HormonesAndrostadienesAndrostanes +9
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Lotilaner Approved DB17992
small molecule | CAS: 1369852-71-0

Lotilaner is an ectoparasiticide that is a member of the isoxazoline family of compounds.[L47546] Lotilaner has largely been used for veterinary uses as an antiparasitic agent to treat flea and tick infestations in animals.[A260746, L47556] Lotilaner consists…

Kategori:
Antiparasitic AgentsEctoparasiticideEctoparasiticides, Incl. Scabicides +2
Target Protein:
Gaba-gated chloride channel, putative
Waktu ParuhThe effective half-…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Lovastatin Approved DB00227
small molecule | CAS: 75330-75-5

Lovastatin, also known as the brand name product Mevacor, is a lipid-lowering drug and fungal metabolite derived synthetically from a fermentation product of _Aspergillus terreus_.[A174550] Originally named Mevinolin, lovastatin belongs to the statin class of…

Kategori:
Agents Causing Muscle ToxicityAnticholesteremic AgentsBSEP/ABCB11 Substrates +21
Target Protein:
3-hydroxy-3-methylglutaryl-coenzyme A reductaseIntegrin alpha-LHistone deacetylase 2
Waktu ParuhLovastatin half-lif…
Vol. DistribusiLovastatin is able …
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Lovotibeglogene autotemcel Approved DB18680
biotech

Lovotibeglogene autotemcel consists of autologous hematopoietic stem and progenitor cells transduced with the BB305 lentiviral vector encoding a modified ?-globin gene. Specifically, lovotibeglogene autotemcel provides a functional copy of a modified beta-glo…

Kategori:
Autologous Cultured CellAutologous Hematopoietic Stem Cell-Based Gene TherapyGenetic Therapy
Target Protein:
Hemoglobin subunit beta
Waktu ParuhLovotibeglogene aut…
Vol. DistribusiLovotibeglogene aut…
KlirensLovotibeglogene aut…
Genetik -
Loxapine Approved DB00408
small molecule | CAS: 1977-10-2

An antipsychotic agent used in schizophrenia. [PubChem]

Kategori:
Antidepressive AgentsAntipsychotic AgentsAntipsychotic Agents (First Generation [Typical]) +24
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 2C +30
Waktu ParuhOral-4 hours
Vol. Distribusi-
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Loxicodegol DB14146
small molecule | CAS: 1211231-76-3

Loxicodegol was developed by Nektar Therapeutics as an opioid analgesic with low abuse potential for the treatment of chronic pain [L3263]. The lack of abuse potential is believed to be due to the drug's slow rate of entry into brain, a unique characteristic …

Kategori:
AlkaloidsHeterocyclic Compounds, Fused-RingOpiate Alkaloids +1
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor
Waktu ParuhLoxicodegol has a h…
Vol. DistribusiLoxicodegol has a s…
KlirensLoxicodegol has a c…
Genetik -
Loxoprofen Approved DB09212
small molecule | CAS: 68767-14-6

Loxoprofen is a propionic acid derivative non-steroidal anti-inflammatory drug. It is marketed under the trade name Loxonin in Brazil, Mexico and Japan by Sankyo, as Loxomac in India, and as Oxeno in Argentina. A transdermal preparation was approved for use i…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +13
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhThe elimination hal…
Vol. DistribusiLoxoprofen has a vo…
KlirensMost of the drug as…
Genetik -
Loxoribine DB17589
small molecule | CAS: 121288-39-9

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Toll-like receptor 7
Waktu Paruh-
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LP-184 DB18215
small molecule | CAS: 924835-67-6

Deskripsi belum tersedia.

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LP-2307 DB17470
biotech

LP-2307 is an investigational allogeneic large multivalent immunogen (LMI) vaccine developed by Avanir. It was investigated for melanoma.

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LP-284 DB18006
small molecule | CAS: 2412580-47-1

Deskripsi belum tersedia.

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LPT-99 DB17142
small molecule | CAS: 1263477-83-3

Deskripsi belum tersedia.

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LSALT Peptide DB16472
biotech

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
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LSTA1 DB17346
biotech | CAS: 1392278-76-0

Deskripsi belum tersedia.

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LSZ-102 DB15362
small molecule | CAS: 2135600-76-7

LSZ-102 is under investigation in clinical trial NCT02734615 (Phase I/Ib Trial of LSZ102 Single Agent or LSZ102 + LEE011 or LSZ102 + BYL719 in ER+ Breast Cancers).

Kategori:
Sulfur Compounds
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LTI-03 DB18491
biotech | CAS: 1504575-10-3

LTI-03 is a caveolin-1 Scaffolding Domain 7-Mer

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LTX-109 DB12711
small molecule | CAS: 1166254-80-3

LTX-109 has been investigated for the treatment of Atopic Dermatitis, Mild Eczema/Dermatoses, and Gram-positive, Skin Infections.

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptidomimetics
Waktu Paruh-
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LTX-315 DB12748
small molecule | CAS: 1345407-05-7

LTX-315 has been used in trials studying the treatment of Cancer, Lymphoma, Melanoma, Carcinoma, and Breast Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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Lubazodone DB09196
small molecule | CAS: 161178-07-0

Lubazodone (YM-992, YM-35,995) is an arylpiperazine antidepressant which was being developed as a treatment for depression and obsessive compulsive disorder, and reached phase II clinical trials, but was discontinued. It acts as a serotonin reuptake inhibitor…

Kategori:
Oxazines
Target Protein:
5-hydroxytryptamine receptor 2ASodium-dependent serotonin transporter
Waktu Paruh-
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Lubiprostone Approved DB01046
small molecule | CAS: 136790-76-6

Lubiprostone is a medication used in the management of idiopathic chronic constipation. A prostaglandin E1 derivative, lubiprostone is a bicyclic fatty acid that activates ClC-2 chloride channels located on the apical side of the gastrointestinal epithelial c…

Kategori:
Alimentary Tract and MetabolismChloride Channel AgonistsDrugs for Constipation +9
Target Protein:
Chloride channel protein 2
Waktu Paruh0.9 to 1.4 hours
Vol. Distribusi-
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Lucanthone DB04967
small molecule | CAS: 479-50-5

One of the schistosomicides, it has been replaced largely by hycanthone and more recently praziquantel. (From Martindale The Extrapharmacopoeia, 30th ed., p46). It is currently being tested as a radiation sensitizer.

Kategori:
AnthelminticsAnti-Infective AgentsAntiparasitic Agents +7
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-betaDNA repair nuclease/redox regulator APEX1 +2
Waktu Paruh-
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Lucerastat DB14872
small molecule | CAS: 141206-42-0

Lucerastat is under investigation in clinical trial NCT03425539 (Efficacy and Safety of Lucerastat Oral Monotherapy in Adult Subjects With Fabry Disease).

Kategori:
AlkaloidsCarbohydratesImines +3
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Lucinactant Approved DB04897
biotech | CAS: 825600-90-6

Lucinactant is a new synthetic peptide-containing surfactant for intratracheal use. It contains sinapultide, a novel, hydrophobic, 21-amino acid peptide (leucine and lysine repeating units, KL4 peptide) designed to mimic human surfactant protein-B (SB-P). Mor…

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBiological Factors +11
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Lucitanib DB11845
small molecule | CAS: 1058137-23-7

Lucitanib has been used in trials studying the treatment of ER+, MBC, SCLC, HER2+, and NSCLC, among others.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Vascular endothelial growth factor receptor 2 +5
Waktu Paruh-
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