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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 139 / 282
GSBR-1290 DB18551
small molecule

GSBR-1290 is a small molecule agonist of the GLP-1 receptor.

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GSI-136 DB12819
small molecule | CAS: 443989-01-3

GSI-136 has been used in trials studying the treatment of Alzheimer Disease.

Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
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GSK-1004723 DB12806
small molecule | CAS: 955359-72-5

Gsk1004723 has been investigated for the treatment of Allergic Rhinitis and Rhinitis, Allergic, Seasonal.

Kategori:
Histamine AntagonistsHistamine H1 AntagonistsPyridazines
Target Protein:
Histamine H3 receptorHistamine H1 receptor
Waktu Paruh-
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GSK-1059615 DB11962
small molecule | CAS: 958852-01-2

GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.

Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 3-kinase catalytic subunit type 3
Waktu Paruh-
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GSK-1292263 DB12627
small molecule | CAS: 1032823-75-8

GSK1292263 has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.

Target Protein:
Glucose-dependent insulinotropic receptor
Waktu Paruh-
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GSK-1521498 DB12886
small molecule | CAS: 1007573-18-3

GSK1521498 has been used in trials studying the treatment of Obesity and Alcoholism.

Kategori:
IndenesReceptors, Opioid, mu
Target Protein:
Mu-type opioid receptor
Waktu Paruh-
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GSK-2018682 DB11987
small molecule | CAS: 1034688-30-6

GSK2018682 has been investigated for the treatment of Multiple Sclerosis, Relapsing-Remitting.

Kategori:
Heterocyclic Compounds, Fused-RingOxazoles
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
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GSK-239512 DB15120
small molecule | CAS: 720691-69-0

GSK-239512 is under investigation in clinical trial NCT00474513 (An Imaging Study to Investigate the Distribution of GSK239512 in the Brain.).

Kategori:
Heterocyclic Compounds, Fused-RingHistamine Antagonists
Target Protein:
Histamine H3 receptor
Waktu Paruh-
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GSK-256066 DB12137
small molecule | CAS: 801312-28-7

Gsk256066 has been used in trials studying the treatment and diagnostic of SAR, Asthma, Mild Asthma, Allergic Rhinitis, and Seasonal Allergic Rhinitis, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +3
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
Waktu Paruh-
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GSK-2636771 DB11795
small molecule | CAS: 1372540-25-4

GSK2636771 has been used in trials studying the treatment of CANCER, LYMPHOMA, Solid Neoplasm, Recurrent Solid Neoplasm, and Advanced Malignant Neoplasm, among others.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
Waktu Paruh-
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GSK-269962A DB17030
small molecule | CAS: 850664-21-0

GSK-269962A is a Rho kinase (ROCK) inhibitor with both ROCK1 and ROCK2 affinity.[A253012]

Kategori:
Oxazoles
Waktu Paruh-
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GSK-2879552 DB16895
small molecule | CAS: 1401966-69-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicBenzene DerivativesCycloparaffins
Target Protein:
Lysine-specific histone demethylase 1A
Waktu Paruh-
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GSK-2881078 DB16888
small molecule | CAS: 1539314-06-1

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsHeterocyclic Compounds, Fused-RingHormones +1
Waktu Paruh-
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GSK-2981278 DB16319
small molecule | CAS: 1474110-21-8

GSK-2981278 is under investigation in clinical trial NCT03004846 (A Study of GSK2981278 Ointment in Subjects With Plaque Psoriasis).

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Nuclear receptor ROR-gamma
Waktu Paruh-
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GSK-2982772 DB16875
small molecule | CAS: 1622848-92-3

Deskripsi belum tersedia.

Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
Waktu Paruh-
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GSK-3117391 DB15440
small molecule | CAS: 1018673-42-1

GSK-3117391 is under investigation in clinical trial NCT02965599 (Efficacy, Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of GSK3117391 in Subjects With Rheumatoid Arthritis).

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GSK-356278 DB12542
small molecule | CAS: 720704-34-7

Gsk356278 has been used in trials studying the treatment and basic science of Anxiety Disorders, Huntington Disease, Depressive Disorder, Huntingtons Disease, and Depressive Disorder, Major, among others.

Kategori:
OxazolesSulfur Compounds
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B
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GSK-376501 DB12654
small molecule | CAS: 1010412-80-2

GSK376501 has been used in trials studying the treatment and diagnostic of Type 2 Diabetes Mellitus.

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GSK-424887 DB12219
small molecule

Gsk424887 has been used in trials studying the basic science and treatment of Depressive Disorder and Anxiety Disorder.

Kategori:
AcetatesAcids, AcyclicAmides
Waktu Paruh-
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GSK-690693 DB12745
small molecule | CAS: 937174-76-0

GSK690693 has been used in trials studying the treatment of Tumor, CANCER, and Lymphoma.

Kategori:
Oxazoles
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
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GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
Waktu Paruh-
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GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
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GSK159797 DB05043
small molecule

GSK159797 ('797) is an inhaled, longer-acting Beta2 agonist developed for the treatment of respiratory disease such as asthma and COPD.

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GSK2245035 DB16076
small molecule | CAS: 1207629-49-9

GSK2245035 is under investigation in clinical trial NCT02833974 (Effect of the GSK2245035 on the Allergen-induced Asthmatic Response).

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Toll-like receptor 7
Waktu Paruh-
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GSK2256098 DB16106
small molecule | CAS: 1224887-10-8

GSK2256098 is under investigation in clinical trial NCT02523014 (Vismodegib and FAK Inhibitor GSK2256098 in Treating Patients With Progressive Meningiomas).

Kategori:
AminesHydroxy AcidsHydroxylamines +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
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GSK232802 DB16110
small molecule | CAS: 843661-24-5

GSK232802 is under investigation in clinical trial NCT00604825 (Treatment of Hot Flashes/flushes in Postmenopausal Women (WARM Study)).

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GSK2798745 DB16033
small molecule | CAS: 1419609-94-1

GSK2798745 is under investigation in clinical trial NCT03372603 (A Study to Assess the Effectiveness and Side Effects of GSK2798745 in Participants With Chronic Cough).

Kategori:
Heterocyclic Compounds, Fused-Ring
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GT 389-255 DB05894
small molecule

Peptimmune’s lead product GT 389-255, is a novel lipase inhibitor and fat binding hydrogel polymer conjugate for the treatment of obesity which has completed single and multiple ascending dose (SAD and MAD) Phase I trials. It is expected to block fat absorpti…

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GTA002 DB17187
biotech

Deskripsi belum tersedia.

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GTI 2040 DB05801
small molecule

GTI-2040 is a substance that is being studied as a treatment for cancer. It belongs to the family of drugs called antisense oligonucleotides.

Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
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GTI-2040 DB15030
biotech | CAS: 236391-66-5

GTI-2040 is under investigation in clinical trial NCT00084643 (GTI-2040, Oxaliplatin, and Capecitabine in Treating Patients With Locally Advanced or Metastatic Colorectal Cancer or Other Solid Tumors).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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GTI-2501 DB05406
small molecule

GTI-2501 is a novel antisense drug which has shown a favorable safety profile in preclinical studies, and in a phase I clinical trial. The drug is in a phase II clinical trial in combination with docetaxel for the treatment of hormone refractory prostate canc…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
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GTP-506 DB17682
biotech

GTP-506 is a gene therapy formed by two vectors, a nuclease vector targeting gene editing in the well-characterized PCSK9 gene locus and a therapeutic donor vector that inserts the OTC gene to provide the desired genetic correction.

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GTS-21 DB05708
small molecule | CAS: 148372-04-7

GTS-21 (also known as DMBX-A), is a novel, small-molecule, orally active and selective alpha-7 nicotinic acetylcholine (nACh) receptor agonist that has demonstrated memory and cognition enhancement activity in human clinical trials. Athenagen licensed the exc…

Kategori:
Benzene DerivativesCholinergic AgentsCholinergic Agonists +5
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
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GTX-102 DB16981
biotech

GTX-102 is an antisense oligonucleotide designed to target and inhibit the expression of UBE3A-AS. It is being investigated for the treatment of Angelman Syndrome.[L46772]

Kategori:
Antisense Oligonucleotide Specific to the Antisense Transcript of UBE3A
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GTX-758 DB14969
small molecule | CAS: 938067-78-8

GTX-758 is under investigation in clinical trial NCT01420861 (GTx-758 on Serum Prostate-specific Antigen (PSA) in Men With Castrate Resistant Prostate Cancer).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Guacetisal DB13538
small molecule | CAS: 55482-89-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Waktu Paruh-
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Guadecitabine DB11918
small molecule | CAS: 929901-49-5

Guadecitabine is under investigation for the treatment of Previously Treated Metastatic Colorectal Cancer.

Kategori:
Antineoplastic AgentsAza CompoundsImmunologic Factors +5
Target Protein:
DNA (cytosine-5)-methyltransferase 1
Waktu Paruh-
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Guaiacol Approved DB11359
small molecule | CAS: 90-05-1

Guaiacol is an agent thought to have disinfectant properties and used as an expectorant. Guaiacol is a phenolic natural product first isolated from Guaiac resin and the oxidation of lignin. Guaiacol is also present in wood smoke, as a product of pyrolysis of …

Kategori:
Benzene DerivativesCatecholsEthers +4
Target Protein:
Albumin
Waktu Paruh-
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Guaiazulen DB13329
small molecule | CAS: 489-84-9

Deskripsi belum tersedia.

Kategori:
CycloheptanesCycloparaffinsOphthalmologicals +5
Waktu Paruh-
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Guaifenesin Approved DB00874
small molecule | CAS: 93-14-1

Guaifenesin possesses a storied history, having been originally formally approved by the US FDA in 1952 and continues to be one of very few - if not perhaps the only drug that is readily available and used as an expectorant [F4525]. Since that time the agent …

Kategori:
Benzene DerivativesCatecholsCough and Cold Preparations +6
Target Protein:
NMDA receptor
Waktu ParuhThe half-life in pl…
Vol. DistribusiThe geometric mean …
KlirensThe mean clearance …
Genetik -
Guanabenz Approved DB00629
small molecule | CAS: 5051-62-7

An alpha-2 selective adrenergic agonist used as an antihypertensive agent. [PubChem]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +11
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu Paruh6 hours.
Vol. Distribusi-
Klirens-
Genetik -
Guanadrel Approved DB00226
small molecule | CAS: 40580-59-4

Guanadrel is an antihypertensive agent and postganglionic adrenergic blocking agent.

Kategori:
Adrenergic AntagonistsAmidinesAntihypertensive Agents +1
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh10 hours
Vol. Distribusi-
Klirens-
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Guanazodine DB13604
small molecule | CAS: 32059-15-7

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
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Guanethidine Approved DB01170
small molecule | CAS: 55-65-2

An antihypertensive agent that acts by inhibiting selectively transmission in post-ganglionic adrenergic nerves. It is believed to act mainly by preventing the release of norepinephrine at nerve endings and causes depletion of norepinephrine in peripheral sym…

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAmidines +16
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh1.5 days
Vol. Distribusi-
Klirens* Renal cl=56 ml/min
Genetik -
Guanfacine Approved DB01018
small molecule | CAS: 29110-47-2

Guanfacine, or BS 100-141,[A189838,A189841] is a selective alpha-A2 adrenergic receptor agonist initially indicated for the treatment of hypertension[L11274] but is now indicated as an extended release tablet for the treatment of ADHD.[L11277] Guanfacine was …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +26
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu ParuhGuanfacine has a ha…
Vol. DistribusiGuanfacine has a vo…
KlirensGuanfacine has a to…
Genetik -
Guanidine Approved DB00536
small molecule | CAS: 113-00-8

A strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of protein metabolism. It is also used in laboratory research as a protein denaturant. (From Martindale, the Extra Pharmacopoeia, 30th…

Kategori:
Acetylcholine Releasing AgentAmidinesGuanidines +7
Target Protein:
Aldehyde dehydrogenase, mitochondrialRibonuclease pancreaticDNA +4
Waktu Paruh7-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77482-44-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic Acids
Target Protein:
Carboxypeptidase D
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Guanine DB02377
small molecule | CAS: 73-40-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPurinesPurinones +1
Target Protein:
GTP cyclohydrolase 1Purine nucleoside phosphorylasePurine nucleoside phosphorylase 2 +2
Waktu Paruh-
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Genetik -
Guanoclor DB13779
small molecule | CAS: 5001-32-1

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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