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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 138 / 236
Liothyronine Approved DB00279
small molecule | CAS: 6893-02-3

Liothyronine is a thyroidal hormone T3 which is normally produced by the thyroid gland in a ratio 4:1 when compared with T4: T3. Liothyronine is the active form of thyroxine which is composed in a basic chemical structure by a tyrosine with bound iodine.[T457…

Kategori:
Agents used to treat hypothyroidismDrugs that are Mainly Renally ExcretedHormones +12
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor betaProliferating cell nuclear antigen
Waktu ParuhThe half-life of li…
Vol. DistribusiThe reported volume…
KlirensThere are no report…
Genetik -
Lipegfilgrastim Approved DB13200
biotech | CAS: 1117844-87-7

Lipegfilgrastim, previously known as XM22, is a pegylated, recombinant granulocyte colony-stimulating factor (G-CSF) that was synthetized using a highly site-specific glycoPEGylation technology [A32665]. It is used as an alternate to [DB00019] for prophylacti…

Kategori:
Adjuvants, ImmunologicAlcoholsAmino Acids, Peptides, and Proteins +17
Target Protein:
Granulocyte colony-stimulating factor receptor
Waktu ParuhThe average termina…
Vol. DistribusiLipegfilgrastim has…
KlirensIn a phase 1, multi…
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lipotecan DB17385
small molecule | CAS: 1432468-79-5

Deskripsi belum tersedia.

Kategori:
Alkaloids
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 118731-97-8

Deskripsi belum tersedia.

Waktu Paruh-
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Lirafugratinib DB18300
small molecule | CAS: 2549174-42-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Liraglutide Approved DB06655
biotech | CAS: 204656-20-2

Victoza contains liraglutide, a synthetic analog of human glucagon-like peptide-1(GLP-1) and acts as a GLP-1 receptor agonist.[Label,A6932] Liraglutide is 97% similar to native human GLP-1, differing primarily by substituting arginine for lysine at position 3…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +17
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhTerminal half life …
Vol. Distribusi13L[Label].
Klirens1.2L/h[Label].
Genetik -
Lirentelimab DB16728
biotech | CAS: 2283348-97-8

Lirentelimab is under investigation in clinical trial NCT04856891 (A Study of Lirentelimab (AK002) in Patients With Active Eosinophilic Duodenitis).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lirilumab DB11754
biotech | CAS: 1000676-41-4

Lirilumab has been used in trials studying the treatment of Leukemia, CANCER,NOS, Multiple Myeloma, Lymphocytic Leukemia, and Acute Myeloid Leukemia, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisaftoclax DB18054
small molecule | CAS: 2180923-05-9

Lisaftoclax is a novel, orally active, selective and potent BCL-2 inhibitor

Kategori:
Benzene DerivativesNitro Compounds
Target Protein:
Apoptosis regulator Bcl-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lisdexamfetamine Approved DB01255
small molecule | CAS: 608137-32-2

Lisdexamfetamine is a prodrug of [dextroamphetamine], a central nervous system stimulant known as d-amphetamine,[A40246] covalently attached to the naturally occurring amino acid L-lysine.[A2230] Lisdexamfetamine is the first chemically formulated prodrug sti…

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAmines +17
Target Protein:
Trace amine-associated receptor 1
Waktu ParuhPlasma concentratio…
Vol. DistribusiDextroamphetamine, …
Klirens-
Genetik -
Lisinopril Approved DB00722
small molecule | CAS: 76547-98-3

Lisinopril is an angiotensin converting enzyme inhibitor (ACEI) used to treat hypertension, heart failure, and myocardial infarction.[L8384,L8387,L8390] Lisinopril and [captopril] are the only ACEIs that are not prodrugs.[A184853] It functions by inhibition o…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +20
Target Protein:
Angiotensin-converting enzymeRenin
Waktu ParuhLisinopril has an e…
Vol. DistribusiThe apparent volume…
KlirensA 30kg child has a …
Genetik -
biotech

Deskripsi belum tersedia.

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Genetik -
Lithium carbonate Approved DB14509
small molecule | CAS: 554-13-2

Lithium has been used to treat manic episodes since the 19th century[A176642]. Though it is widely used, its mechanism of action is still unknown[FDA Label][A14585,A176642,A176651,L5843]. Lithium carbonate has a narrow therapeutic range and so careful monitor…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +26
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu ParuhThe half life of li…
Vol. DistribusiApparent volume of …
KlirensClearance is genera…
Genetik -
Lithium cation DB01356
small molecule | CAS: 7439-93-2

Lithium was used during the 19th century to treat gout. Lithium salts such as lithium carbonate (Li2CO3), lithium citrate, and lithium orotate are mood stabilizers. They are used in the treatment of bipolar disorder, since unlike most other mood altering drug…

Kategori:
Antidepressive AgentsAntimanic AgentsAntipsychotic Agents +11
Target Protein:
Glycogen synthase kinase-3 betaInositol monophosphatase 1Inositol monophosphatase 2 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 7447-41-8

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntimanic AgentsCentral Nervous System Agents +8
Target Protein:
Glycogen synthase kinase-3 alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lithium citrate Approved DB14507
small molecule | CAS: 919-16-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntidepressive AgentsAntimanic Agents +12
Target Protein:
Inositol monophosphatase 2Inositol monophosphatase 1Glycogen synthase kinase-3 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Litifilimab DB18864
biotech | CAS: 2407378-48-5

Litifilimab is under investigation in clinical trial NCT05531565 (A Study to Assess the Efficacy and Safety of BIIB059 (Litifilimab) in Participants With Active Subacute Cutaneous Lupus Erythematosus (SCLE) And/or Chronic Cutaneous Lupus Erythematosus (CCLE) …

Waktu Paruh-
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Litoxetine DB15038
small molecule | CAS: 86811-09-8

Litoxetine is under investigation in clinical trial NCT03397771 (DBPC Trial to Evaluate the Safety, Tolerability and Efficacy of Oral Litoxetine in Subjects With Urinary Incontinence).

Target Protein:
Sodium-dependent serotonin transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lividomycin A DB04728
small molecule | CAS: 36441-41-5

Deskripsi belum tersedia.

Target Protein:
Telomerase reverse transcriptase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Livmoniplimab DB18939
biotech | CAS: 2412004-88-5

Livmoniplimab is under investigation in clinical trial NCT06109272 (A Study to Assess the Dose, Adverse Events, and Change in Disease Activity of Livmoniplimab as an Intravenous (IV) Solution in Combination With Budigalimab as an IV Solution in Adult Particip…

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Livoletide DB15188
small molecule | CAS: 1088543-62-7

Livoletide is under investigation in clinical trial NCT03790865 (Effects of Livoletide (AZP-531) on Food-related Behaviors in Patients With Prader-Willi Syndrome).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsHormones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lixadesiran DB17295
biotech | CAS: 1152798-49-6

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
Lixisenatide Approved DB09265
biotech | CAS: 320367-13-3

Lixisenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist used in the treatment of type II diabetes mellitus (T2DM). It is sold by Sanofi-Aventis under the brand name Adlyxin in the US[L763] and Lyxumia in the EU.[L764] Adlyxin recieved FDA approval …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +11
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhFollowing the admin…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent c…
Genetik -
Lixivaptan DB06666
small molecule | CAS: 168079-32-1

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzazepines +3
Target Protein:
Histidine decarboxylaseVasopressin V2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lixudebart DB19244
biotech | CAS: 2749515-10-2

Lixudebart, an investigational first-in-class monoclonal antibody, aims to reverse fibrosis.[L50833]

Waktu Paruh-
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Genetik -
Lixumistat DB18748
small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

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Genetik -
LJ-2698 DB18018
small molecule | CAS: 945457-84-1

Deskripsi belum tersedia.

Kategori:
Adenosine A3 Receptor AntagonistsNeurotransmitter AgentsNucleic Acids, Nucleotides, and Nucleosides +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LJP-538 DB17810
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
LJP-539 DB17811
biotech

Deskripsi belum tersedia.

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Vol. Distribusi-
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Genetik -
LL-37 DB16532
biotech

LL-37 is a human cathelicidin that inhibits viral replication and while also playing a role in host defense against infection.

Waktu Paruh-
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LLL-3348 DB05771
biotech

The botanical drug product LLL-3348 is a once-daily oral formulation for treatment of chronic stable plaque type psoriasis.

Kategori:
Biological ProductsComplex MixturesPharmaceutical Preparations +1
Target Protein:
Interleukin-10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
LM-030 DB18283
small molecule | CAS: 1122484-55-2

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
LM-609 DB05787
biotech

LM-609 (Vitaxin) is an artificial antibody that targets a protein on the surface of newly forming blood vessels, as well as on certain tumors. In addition to cancer, the protein has been implicated in bone destruction in rheumatoid arthritis and the inflammat…

Target Protein:
Integrin beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

LNP-nCoVsaRNA is a purified, synthetic mRNA vaccine candidate encoding the S glycoprotein of SARS-CoV-2, which is used primarily by the virus to attach to and invade human cells. The vaccine was developed in and tested by the Medical Research Council Clinical…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lobeglitazone DB09198
small molecule | CAS: 607723-33-1

Lobeglitazone is an antidiabetic medication from the thiazolidinedione class of drugs. It primarily functions as an insulin sensitizer by binding and activating Peroxisome Proliferator-Activated Receptors (PPAR) gamma within fat cells. By activating PPAR-gamm…

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP1A2 Inhibitors +19
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gamma
Waktu ParuhFollowing an intrav…
Vol. DistribusiThe steady state vo…
KlirensIn rat studies, sys…
Genetik -
Lobeline DB05137
small molecule | CAS: 90-69-7

An alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has been proposed for a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation. …

Kategori:
AlkaloidsAutonomic AgentsCholinergic Agents +7
Target Protein:
Synaptic vesicular amine transporterNeuronal acetylcholine receptor subunit alpha-7Neuronal acetylcholine receptor subunit alpha-9 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lobucavir DB12531
small molecule | CAS: 127759-89-1

Lobucavir has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +10
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 398507-55-6

Lodenafil carbonate has been used in trials studying the treatment of Coronaropathy and Erectile Dysfunction.

Kategori:
AlkaliesAnionsCarbon Compounds, Inorganic +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lodoxamide Approved DB06794
small molecule | CAS: 53882-12-5

Lodoxamide is a mast-cell stabilizer for topical administration into the eye. Mast-cell stabilizers, first one approved being cromolyn sodium, are used in treatment of ocular hypersensitivity reactions such as vernal conjunctivitis. These conditions often req…

Kategori:
Acids, AldehydicAlcoholsAmino Acids +13
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
Lofentanil DB09174
small molecule | CAS: 61380-40-3

Lofentanil is an analog of fentanyl and is one of the most potent opioids available today. It displays most similarity to carfentanil (4-carbomethoxyfentanyl) and is considered to be slightly more potent than this drug.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +6
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lofepramine DB13411
small molecule | CAS: 23047-25-8

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lofexidine Approved DB04948
small molecule | CAS: 31036-80-3

Lofexidine is a non-opioid centrally acting alpha2-adrenergic receptor agonist that was first approved for the treatment of opioid withdrawal in the United Kingdom in 1992.[A33084] It was first studied for use as an antihypertensive in 1980, but its researche…

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +31
Target Protein:
Alpha-2A adrenergic receptorAlpha-1A adrenergic receptor5-hydroxytryptamine receptor 1A +3
Waktu ParuhThe reported elimin…
Vol. DistribusiLofexidine has a vo…
KlirensThe total eliminati…
Genetik -
Lomefloxacin Approved DB00978
small molecule | CAS: 98079-51-7

Lomefloxacin is a fluoroquinolone antibiotic, used to treat bacterial infections including bronchitis and urinary tract infections (UTIs). Additionally, it has been employed for the prophylaxis of UTIs prior to surgery as well.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA topoisomerase 2-betaDNA topoisomerase 4 subunit A +1
Waktu Paruh8 hours
Vol. Distribusi-
Klirens* 271 mL/min/1.73 m…
Genetik -
Lomerizine DB14065
small molecule | CAS: 101477-55-8

Lomerizine is a diphenylmethylpiperazine calcium channel blocker[A245378, A245383] with relatively selective central nervous system (CNS) effects.[A245383] This drug is used to prophylactically treat migraines[A245368, A245373] and is also being investigated…

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +8
Target Protein:
Sodium channel protein type 5 subunit alphaVoltage-dependent N-type calcium channel subunit alpha-1BATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lometrexol DB12769
small molecule | CAS: 106400-81-1

Lometrexol has been used in trials studying the treatment of Lung Cancer, Drug/Agent Toxicity by Tissue/Organ, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
AntimetabolitesAntineoplastic AgentsCoenzymes +9
Target Protein:
Dihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lomibuvir DB11954
small molecule | CAS: 1026785-55-6

Lomibuvir has been used in trials studying the treatment of Chronic Hepatitis C Virus and Chronic Hepatitis C Virus Infection.

Kategori:
AlcoholsCyclohexanesCycloparaffins +4
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lomifylline Approved DB18002
small molecule | CAS: 10226-54-7

Deskripsi belum tersedia.

Kategori:
AlkaloidsDrugs for Obstructive Airway DiseasesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lomitapide Approved DB08827
small molecule | CAS: 182431-12-5

Lomitapide is a microsomal triglyceride transfer protein (MTP) inhibitor used in homozygous familial hypercholesterolemia (HoFH) patients. It is marketed under the name Juxtapid (R).

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Inhibitors +17
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu ParuhLomitapide half-lif…
Vol. DistribusiThe steady state vo…
Klirens-
Genetik -
Lomustine Approved DB01206
small molecule | CAS: 13010-47-4

An alkylating agent of value against both hematologic malignancies and solid tumors.

Kategori:
Alkylating ActivityAlkylating DrugsAmides +17
Target Protein:
DNAStathmin-4
Waktu ParuhApproximately 94 mi…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6851–6900 dari 11778
Sebelumnya Halaman 138 / 236 Berikutnya