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12560

Total database: 17430
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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 138 / 252
Ipafricept DB15045
biotech | CAS: 1391727-24-4

Ipafricept is under investigation in clinical trial NCT01608867 (A Dose Escalation Study of OMP-54F28 in Subjects With Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +10
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Ipamorelin DB12370
small molecule | CAS: 170851-70-4

Ipamorelin has been investigated for the treatment of Ileus.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Growth hormone secretagogue receptor type 1
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Ipecac Approved DB13293
small molecule | CAS: 8012-96-2

Ipecac is obtained from the plant _Cephaelis ipecacuanha_ and contains a number of emetic alkaloids including emetine and cephaeline.[L2753] Ipecac was approved by Health Canada as an OTC but all those products are now discontinued.[L1113] The FDA does not ha…

Kategori:
Agents Causing Muscle ToxicityAntidotesAutonomic Agents +15
Waktu ParuhThe effect of ipeca…
Vol. DistribusiThe volume of distr…
KlirensThe urinary excreti…
Genetik -
IPH 1101 DB05754
small molecule

IPH 1101 is a chemically-synthesized structural analog of non-conventional bacterial phosphoantigens which specifically activate the V?9V?2 T cell subset. IPH 1101 is the most advanced drug candidate of the ?? T cell platform

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IPH 2101 DB06049
biotech | CAS: 1000676-42-5

IPH-2101 (NN-1975), a fully human monoclonal antibody developed for patients with acute myeloid leukemia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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IPI-549 DB16296
small molecule | CAS: 1693758-51-8

IPI-549 is under investigation in clinical trial NCT03795610 (Window of Opportunity Study of IPI-549 in Patients With Locally Advanced HPV+ and HPV- Head and Neck Squamous Cell Carcinoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
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Ipilimumab Approved DB06186
biotech | CAS: 477202-00-9

Ipilimumab is a fully humanized IgG1 monoclonal antibody that blocks cytotoxic T lymphocyte antigen-4 (CTLA-4).[L12126] Blocking CTLA-4 removes an inhibitory signal from reducing the activity of T lymphocytes.[A35065,A35080,L12126] Ipilimumab was developed by…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntibodies +21
Target Protein:
Cytotoxic T-lymphocyte protein 4
Waktu ParuhIpilimumab has a ha…
Vol. DistribusiThe volume of distr…
KlirensIpilimumab has a cl…
Genetik -
IPL-344 DB16958
small molecule | CAS: 877120-59-7

Deskripsi belum tersedia.

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Ipratropium Approved DB00332
small molecule | CAS: 60205-81-4

Ipratropium is a quaternary ammonium derivative of [atropine][A176957] that acts as an anticholinergic agent.[A176939] It is commonly administered through inhalation which allows producing a local effect without presenting a significant systemic absorption.[A…

Kategori:
Adrenergics, InhalantsAgents producing tachycardiaAgents to Treat Airway Disease +19
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2
Waktu ParuhIpratropium present…
Vol. DistribusiIpratropium has a v…
KlirensThe average clearan…
Genetik -
Iprazochrome DB13541
small molecule | CAS: 7248-21-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAntidepressive AgentsAntimigraine Preparations +10
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Ipriflavone DB13618
small molecule | CAS: 35212-22-7

Deskripsi belum tersedia.

Kategori:
BenzopyransBone RemodelingChromones +6
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Iprindole DB13496
small molecule | CAS: 5560-72-5

Deskripsi belum tersedia.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +14
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Iproclozide DB09247
small molecule | CAS: 3544-35-2

Iproclozide is an irreversible and selective hydrazine class based monoamine oxidase inhibitor (MAOI). Although it was employed as an antidepressant for a time, the fact that the agent is capable of causing fulminant hepatitis and that its use has been docume…

Kategori:
AcetatesAcids, AcyclicAntidepressive Agents +4
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Iproniazid DB04818
small molecule | CAS: 54-92-2

Withdrawn from the Canadian market in July 1964 due to interactions with food products containing tyrosine.

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +18
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
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Iptacopan Approved DB16200
small molecule | CAS: 1644670-37-0

Iptacopan is a small-molecule factor B inhibitor previously investigated as a potential treatment for the rare blood disease paroxysmal nocturnal hemoglobinuria (PNH) by inhibiting the complement factor B.[A262566] Factor B is a positive regulator of the alte…

Kategori:
Acids, CarbocyclicAntineoplastic and Immunomodulating AgentsBenzene Derivatives +8
Target Protein:
Complement factor B
Waktu ParuhThe half-life (t<su…
Vol. DistribusiAfter administratio…
KlirensThe clearance of ip…
Genetik -
IQP-0528 DB14888
small molecule | CAS: 301297-45-0

IQP-0528 is under investigation in clinical trial NCT03082690 (ImQuest (IQP) DuoGel Phase 1 Pharmacokinetic Study).

Kategori:
Anti-HIV AgentsPyrimidines
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IR-901 DB17932
biotech | CAS: 146446-23-3

Deskripsi belum tersedia.

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IR208 DB05106
biotech

IR208 is a synthetic T-Cell receptor peptide vaccine developed by Immune Response Corporation. It contains three peptides (BV5S2, BV6S5 and BV13S1) expressed by T-Cells in over 90% of MS patients. IR208 is currently undergoing Phase II studies in a 200-p…

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IR501 DB06464
biotech

IR501 (Ravax) is a potential first-in-class vaccine for the treatment of Rheumatoid Arthritis. It specifically targets autoreactive T-cells, reducing their activity. It was last known to be in phase III clinical trials.

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IR502 DB06463
biotech

IR502 (Zorcell) is a potential treatment for psoriasis.

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Iratumumab DB05550
biotech | CAS: 640735-09-7

Immunoglobulin G1, anti-(human CD30 (antigen)) (human monoclonal MDX-060 heavy chain), disulfide with human monoclonal MDX-060 light chain, dimer. Molecular weight is approximately 170,000 daltons. In phase I/II clinical trials for treatment of CD30+ lymphoma…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 8
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Irbesartan Approved DB01029
small molecule | CAS: 138402-11-6

Irbesartan is an angiotensin receptor blocker (ARB) indicated to treat hypertension or diabetic nephropathy.[L7456,L7459] It can also be used as part of a combination product with [hydrochlorothiazide] for patients not well controlled or not expected to be we…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +24
Target Protein:
Type-1 angiotensin II receptorTranscription factor Jun
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensTotal plasma cleara…
Genetik -
Irdabisant DB12900
small molecule | CAS: 1005402-19-6

Irdabisant has been used in trials studying Cognitive Impairment.

Kategori:
Receptors, Histamine H3
Target Protein:
Histamine H3 receptor
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Irinotecan Approved DB00762
small molecule | CAS: 97682-44-5

Irinotecan is a topoisomerase inhibitor used for chemotherapy. It is a water-soluble analogue of [camptothecin], which is extracted from the Chinese tree _Camptotheca acuminate_.[A263376] The bis-piperidine side chain in the structure of irinotecan bestows en…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +29
Target Protein:
DNA topoisomerase I, mitochondrialDNA topoisomerase 1
Gen Terkait:
SLCO1B1 UGT1A1 UGT1A7 +2
Waktu ParuhAfter intravenous i…
Vol. DistribusiFollowing intraveno…
KlirensThe mean (± standar…
Genetik 5 Varian
IRL-1620 DB06138
small molecule | CAS: 142569-99-1

SPI-1620 is an endothelin B receptor agonist. In animal models SPI-1620 selectively and transiently increases tumor blood flow allowing increased delivery of anticancer agents to the tumor. It is being developed as an adjunct to chemotherapy.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Target Protein:
Endothelin receptor type B
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Irofulven DB05786
small molecule | CAS: 158440-71-2

A novel anti-cancer compound synthesized by scientists at the University of California, San Diego more than a decade ago from toxins of the poisonous jack-o-lantern mushroom, has been granted “fast track” status by the U.S. Food and Drug Administration (FDA) …

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +4
Target Protein:
Serine/threonine-protein kinase Chk2Far upstream element-binding protein 1
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Iron Approved DB01592
small molecule | CAS: 7439-89-6

A metallic element found in certain minerals, in nearly all soils, and in mineral waters. It is an essential constituent of hemoglobin, cytochrome, and other components of respiratory enzyme systems. Its chief functions are in the transport of oxygen to tissu…

Kategori:
Alimentary Tract and MetabolismAntianemia DrugsAntianemic Preparations +14
Target Protein:
Hemoglobin subunit alphaTransferrin receptor protein 1Egl nine homolog 1 +10
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small molecule | CAS: 764-65-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsOAT3/SLC22A8 Inhibitors
Target Protein:
Organic anion transporter 3
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Iron isomaltoside 1000 Approved DB12208
small molecule | CAS: 1370654-58-2

Iron isomaltoside 1000 is under investigation in Iron Deficiency Anaemia. Iron isomaltoside 1000 has been investigated for the treatment and basic science of Anemia, Gastric Cancer, Esophageal Cancer, Chronic Kidney Disease, and Anemia, Iron-Deficiency, among…

Kategori:
CarbohydratesHematinicsHematologic Agents +3
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small molecule | CAS: 53858-86-9

Deskripsi belum tersedia.

Kategori:
HematinicsHematologic AgentsIron Compounds +1
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Iron protein succinylate Approved DB11209
small molecule | CAS: 250705-13-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmino Acids, Peptides, and ProteinsAntianemic Preparations +8
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Irosustat DB02292
small molecule | CAS: 288628-05-7

Irosustat has been investigated for the treatment of Metastatic Breast Cancer and Locally Advanced Breast Cancer.

Kategori:
AcidsAcids, NoncarboxylicSteryl-Sulfatase, antagonists & inhibitors +2
Target Protein:
Steryl-sulfataseCarbonic anhydrase 2
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Iroxanadine DB05444
small molecule | CAS: 276690-58-5

BRX-235 (iroxanadine) is a a novel small molecule synthesized by Biorex, Hungary that acts as a cardioprotective agent. It induces phosphorylation of p38 SAPK, which plays an important role in EC homeostasis. endothelial cell (EC). EC function plays a central…

Target Protein:
Heat shock 70 kDa protein 1AHeat shock 70 kDa protein 1B
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Irpagratinib DB18732
small molecule | CAS: 2230974-62-4

Irpagratinib (ABSK011) is a highly selective inhibitor of fibroblast growth factor receptor (FGFR) 4.

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Irsenontrine DB19044
small molecule | CAS: 1429509-82-9

Irsenontrine is under investigation in clinical trial NCT03467152 (Study to Evaluate the Efficacy, Safety and Tolerability of E2027 (Hereinafter Referred to as Irsenontrine) in Participants With Dementia With Lewy Bodies).

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Irsogladine DB13056
small molecule | CAS: 57381-26-7

Irsogladine is under investigation in clinical trial NCT02581696 (The Drug-drug Interaction and Safety of Lafutidine and Irsogladine Maleate in Healthy Adult Volunteers).

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAnticarcinogenic Agents +6
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Iruplinalkib DB17494
small molecule | CAS: 1854943-32-0

Deskripsi belum tersedia.

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IRX-2 DB05643
biotech | CAS: 951209-71-5

IRX-2 contains a human leukocyte-derived cytokine mixture. It is being investigated to promote or enhance an anti-cancer immune response.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
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IRX-5183 DB05653
small molecule | CAS: 367273-07-2

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
Retinoic acid receptor alpha
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Genetik -
biotech | CAS: 2378601-29-5

Isaralgagene civaparvovec, formerly known as ST-920, is liver-tropic rAAV 2/6 vector carrying the cDNA for human alpha-galactosidase A (?-Gal A) enzyme. It is developed by Sangamo Therapeutics and investigated in Fabry Disease.

Kategori:
Adeno-associated Viral Vector Therapies
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Isatin DB02095
small molecule | CAS: 91-56-5

Isatin is an indole derivative first obtained by Erdman and Laurent in 1841 as an oxidation product of Indigo dye with nitric acid and chromic acids. The compound is found in many plants and Schiff bases of Isatin are have been investigated for pharmaceutical…

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Amine oxidase [flavin-containing] B
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small molecule | CAS: 118-48-9

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsAnti-Infective Agentsbeta-Lactamase Inhibitors +1
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Isatoribine DB04860
small molecule | CAS: 122970-40-5

Isatoribine is a selective agonist of TLR7.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Toll-like receptor 7
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Isatuximab Approved DB14811
biotech | CAS: 1461640-62-9

Isatuximab (formerly SAR650984) is a humanized, IgG1-derived monoclonal antibody (mAb) produced from a Chinese hamster ovary (CHO) cell line.[L12099,A191799] Structurally, isatuximab is comprised of two identical immunoglobulin kappa light chains and two iden…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. DistribusiThe predicted volum…
KlirensTotal clearance dec…
Genetik -
Isavuconazole Approved DB11633
small molecule | CAS: 241479-67-4

Isavuconazole is an triazole antifungal with broad spectrum of activity and good safety profile [A32026]. It is approved by the FDA and EMA for the treatment of invasive aspergillosis and mucormycosis. It works by inhibiting fungal cell membrane synthesis. In…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiinfectives for Systemic Use +38
Target Protein:
Lanosterol 14-alpha demethylaseVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-dependent L-type calcium channel subunit alpha-1C +7
Waktu ParuhBased on a populati…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance (CL) …
Genetik -
Isavuconazonium Approved DB06636
small molecule | CAS: 742049-41-8

Isavuconazonium is a second-generation triazole antifungal approved on March 6, 2015 by the FDA and July 2015 by the EMA for the treatment of adults with invasive aspergillosis and invasive mucormycosis, marketed by Astellas under the brand Cresemba.[A38834] …

Kategori:
Anti-Infective AgentsAntifungal AgentsAzole Antifungals +31
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhBased on a populati…
Vol. DistribusiIsavuconazole is ex…
KlirensIn healthy subjects…
Genetik -
ISB 1342 DB17251
biotech

ISB 1342 is a bispecific antibody simultaneously targeting CD38 and CD3.

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ISB 1442 DB18475
biotech

ISB 1442 is a bispecific, biparatopic antibody targeting CD38 and CD47

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ISB 2001 DB18570
biotech

ISB 2001 is a T cell-engaging antibody that targets BCMA, CD38, and CD3.

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Iscalimab DB15260
biotech | CAS: 2031153-61-2

Iscalimab is under investigation in clinical trial NCT03905525 (Study of Safety and Efficacy of Multiple Doses of CFZ533 in Two Distinct Populations of Patients With Sjögren's Syndrome).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Menampilkan 6851–6900 dari 12560
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