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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (14063)

Halaman 138 / 282
Go-6976 DB17029
small molecule | CAS: 136194-77-9

An inhibitor of calcium-dependent isoforms of protein kinase C.[A253002,A253007]

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
Waktu Paruh-
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Goat milk Approved DB10542
biotech

Goat milk allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Goflikicept DB16396
biotech | CAS: 2416984-26-2

Goflikicept is under investigation in clinical trial NCT04380519 (Study of the Efficacy and Safety of a Single Administration of Olokizumab and RPH-104 With Standard Therapy in Patients With Severe Severe Acute Respiratory Syndrome Coronavirus 2 (Sars-cov-2) …

Kategori:
Experimental Unapproved Treatments for COVID-19
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Golcadomide DB18115
small molecule | CAS: 2379572-34-4

Deskripsi belum tersedia.

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Gold Au-198 DB13427
small molecule | CAS: 10043-49-9

Deskripsi belum tersedia.

Kategori:
Anti-Inflammatory AgentsElementsGold Isotopes +6
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small molecule | CAS: 20681-14-5

Deskripsi belum tersedia.

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small molecule | CAS: 15283-45-1

Deskripsi belum tersedia.

Kategori:
Antirheumatic AgentsGold CompoundsSodium Compounds +5
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Golexanolone DB18200
small molecule | CAS: 2089238-18-4

Deskripsi belum tersedia.

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Golidocitinib DB18057
small molecule | CAS: 2091134-68-6

Deskripsi belum tersedia.

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biotech | CAS: 957472-14-9

Deskripsi belum tersedia.

Kategori:
Gene Transfer TechniquesNucleic AcidsNucleic Acids, Nucleotides, and Nucleosides
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Golodirsen Approved DB15593
biotech | CAS: 1422959-91-8

Golodirsen is a morpholino antisense oligomer designed to treat about 8% of patients with Duchenne Muscular Dystrophy (DMD). This is an X-linked condition leading to progressive muscle degeneration that begins in early childhood, rendering many patients wheel…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesCompounds used in a research, industrial, or household setting +10
Target Protein:
Dystrophin
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe volume of distr…
KlirensThis drug is rapidl…
Genetik -
Golotimod DB05475
small molecule | CAS: 229305-39-9

SCV-07 (g -D-glutamyl-L-tryptophan) is a novel synthetic dipeptide that acts broadly on the Toll-like receptor pathway. It has been shown to stimulate T-lymphocyte differentiation, macrocytic phagocytosis, and specific immune responses, and enhance IL-2 and …

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Signal transducer and activator of transcription 3Toll-like receptor 2Toll-like receptor 4 +2
Waktu Paruh-
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Golvatinib DB11977
small molecule | CAS: 928037-13-2

Golvatinib has been investigated for the treatment of Platinum-Resistant Squamous Cell Carcinoma of the Head and Neck.

Kategori:
AminesPyridinesVascular Endothelial Growth Factor Receptor-2, antagonists & inhibitors
Target Protein:
Vascular endothelial growth factor receptor 2Hepatocyte growth factor receptor
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Gonadorelin Approved DB00644
biotech | CAS: 33515-09-2

Gonadorelin is another name for gonadotropin-releasing hormone (GnRH). It is a synthetic decapeptide prepared using solid phase peptide synthesis. GnRH is responsible for the release of follicle stimulating hormone and leutinizing hormone from the anterior pi…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsDiagnostic Agents +18
Target Protein:
Gonadotropin-releasing hormone receptorPutative gonadotropin-releasing hormone II receptor
Waktu ParuhVery short, initial…
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Gontivimab DB16179
biotech | CAS: 1257358-38-5

Gontivimab is under investigation in clinical trial NCT03468829 (Efficacy and Safety of ALX-0171 in Adult Hematopoietic Stem Cell Transplant (HSCT) Recipients Who Present With Respiratory Syncytial Virus (RSV) Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +11
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Gonyautoxin II DB19186
small molecule | CAS: 60508-89-6

Gonyautoxin II is under investigation in clinical trial NCT04799041 (Gonyautoxin 2/3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study).

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ToxinsBiological Factors +9
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Gonyautoxin III DB19187
small molecule | CAS: 60537-65-7

Gonyautoxin III is currently under investigation in clinical trial (Gonyautoxin 2/?3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study) for the treatment of Acute Back Pain.

Kategori:
Bacterial ToxinsBiological FactorsComplex Mixtures +7
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Goserelin Approved DB00014
small molecule | CAS: 65807-02-5

Goserelin is a synthetic hormone. In men, it stops the production of the hormone testosterone, which may stimulate the growth of cancer cells. In women, goserelin decreases the production of the hormone estradiol (which may stimulate the growth of cancer cell…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Lutropin-choriogonadotropic hormone receptorProgonadoliberin-1Gonadotropin-releasing hormone receptor
Waktu Paruh4-5 hours
Vol. Distribusi* 44.1 ± 13.6 L [su…
Klirens* 121 +/- 42.4 mL/m…
Genetik -
Gosogliptin DB08382
small molecule | CAS: 869490-23-3

Gosogliptin has been used in trials studying the treatment of Renal Insufficiency, Chronic.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDiabetes Mellitus, Type 2, drug therapy +1
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
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Gosuranemab DB15376
biotech | CAS: 1788032-39-2

Gosuranemab is under investigation in clinical trial NCT02460094 (Multiple Ascending Dose Study of Intravenously Administered BMS-986168 (BIIB092) in Patients With Progressive Supranuclear Palsy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Gotistobart DB19100
biotech | CAS: 2226344-78-9

Gotistobart is under investigation in clinical trial NCT05671510 (ONC-392 Versus Docetaxel in Metastatic NSCLC That Progressed on PD-1/PD-L1 Inhibitors).

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GP-100 antigen DB14800
biotech

GP-100 antigen is under investigation in clinical trial NCT00006385 (Vaccine Therapy With or Without Biological Therapy in Treating Patients With Metastatic Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +5
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GP2 peptide DB16180
biotech | CAS: 160790-21-6

GP2 peptide is under investigation in clinical trial NCT00524277 (Vaccine Therapy in Treating Patients With Breast Cancer).

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Genetik -
biotech

The gp209-2M antigen is derived from gp209, and has potential immunomodulatory and antineoplastic activities.

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GPI-0100 DB05929
small molecule

GPI-0100 is Avantogen’s lead adjuvanat-immunopotentiator, a key component of vaccines for boosting the immune response. The GPI-0100 adjuvant, which has been shown to significantly enhance the immune response with a variety of vaccines, has been shown to hav…

Kategori:
CarbohydratesGlycosides
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GPI-1485 DB05814
small molecule | CAS: 186268-78-0

GPI 1485 is a product candidate that belongs to a class of small molecule compounds called neuroimmunophilin ligands. In preclinical experiments, neuroimmunophilin ligands have been shown to repair and regenerate damaged nerves without affecting normal, heal…

Kategori:
Cytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 InhibitorsCytochrome P-450 CYP3A4 Inhibitors (strength unknown) +2
Target Protein:
Peptidyl-prolyl cis-trans isomerase FKBP1A
Waktu Paruh-
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GR270773 DB06427
small molecule

GR270773, was investigated in two clinical trials for its potential to treat sepsis: NCT00158769 (completed, comparing the effects of infusion between healthy adults and those with damaged livers) and NCT00089986 (completed with results, treatment of suspecte…

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GRAd-COV2 DB16428
biotech

GRAd-COV2 is a COVID-19 vaccine candidate being developed by ReiThera[L30420, L30423]. This therapy is based on a novel replication-incompetent simian adenoviral vector that encodes the full-length SARS-CoV-2 spike protein (GRAd-COV2)[L30420, L30423]. Preclin…

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Gramicidin D Approved DB00027
small molecule | CAS: 1405-97-6

Gramcidin D is a heterogeneous mixture of three antibiotic compounds, gramicidins A, B and C, making up 80%, 6%, and 14% respectively all of which are obtained from the soil bacterial species Bacillus brevis and called collectively gramicidin D. Gramcidins ar…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Dihydropteroate synthase
Waktu Paruh-
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Granaticin B DB17273
small molecule | CAS: 19879-03-9

Deskripsi belum tersedia.

Kategori:
BenzopyransBenzoquinonesChromans +5
Waktu Paruh-
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Granotapide DB12934
small molecule | CAS: 594842-13-4

Granotapide has been used in trials studying the treatment of Type II Diabetes Mellitus.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +3
Target Protein:
Microsomal triglyceride transfer protein large subunit
Waktu Paruh-
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Grape seed oil DB14323
biotech | CAS: 8016-21-5

Grape seed oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Grapefruit oil DB15663
biotech | CAS: 8016-20-4

Deskripsi belum tersedia.

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Graphite Approved DB18717
small molecule | CAS: 7782-42-5

Deskripsi belum tersedia.

Kategori:
CarbonElementsGraphite +1
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Grapiprant DB12836
small molecule | CAS: 415903-37-6

Grapiprant, also known as AT-001 and CJ-023, is a drug from the piprant class. These molecules were derived from acylsulfonamide and are characterized to be a novel series of para-N-acylaminomethylbenzoic acid known to be prostaglandin receptor antagonists.[A…

Kategori:
AmidesBenzene DerivativesP-glycoprotein substrates +3
Target Protein:
Prostaglandin E2 receptor EP4 subtype
Waktu ParuhThe reported elimin…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
Genetik -
Grazoprevir Approved DB11575
small molecule | CAS: 1350514-68-9

Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nin…

Kategori:
Acids, AcyclicAmidesAnti-Infective Agents +24
Target Protein:
Genome polyprotein
Waktu ParuhThe geometric mean …
Vol. DistribusiGrazoprevir has an …
KlirensThe clearance of Gr…
Genetik -
Gremubamab DB15014
biotech | CAS: 1800381-36-5

Gremubamab is under investigation in clinical trial NCT02255760 (Phase 1 Randomized Double-blind Placebo Controlled Study to Evaluate Safety and PK of MEDI3902 in Healthy Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Grepafloxacin Approved DB00365
small molecule | CAS: 119914-60-2

Grepafloxacin is an oral broad-spectrum quinoline antibacterial agent used to treat bacterial infections. Due to the QTc-prolonging potential, as indicated by the changes in the QT interval on the electrocardiogram, and the risk for cardiovascular adverse eve…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh15 ± 3 hours
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Gresonitamab DB18210
biotech | CAS: 2413817-97-5

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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Griseofulvin Approved DB00400
small molecule | CAS: 126-07-8

An antifungal antibiotic. Griseofulvin may be given by mouth in the treatment of tinea infections.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +14
Target Protein:
Tubulin beta chainKeratin, type I cytoskeletal 12
Waktu Paruh9-21 hours
Vol. Distribusi-
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GRObeta DB18205
biotech

Deskripsi belum tersedia.

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small molecule | CAS: 141925-59-9

Growth hormone-releasing peptide 1 is under investigation in clinical trial NCT00381602 (A Phase II, Randomized, Cross-over, Vehicle-controlled, Double-blind, Multicenter Study of the Safety, Pharmacodynamics, and Preliminary Efficacy of GHRP-1/AG in Subjects…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth Hormone-Releasing HormonePeptides
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GS 0573 DB08843
small molecule | CAS: 113852-41-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsHeterocyclic Compounds, Fused-RingImmunologic Factors +1
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GS-441524 DB15686
small molecule | CAS: 1191237-69-0

GS-441524 is an adenosine nucleotide analog antiviral, similar to [remdesivir].[A203057,L13239] This molecule was patented in 2009.[L13775] _In vitro_ studies of GS-441524 have determined it has a higher EC<sub>50</sub> than remdesivir against a number of vir…

Kategori:
Adenine NucleotidesAnti-Infective AgentsAntiviral Agents +10
Target Protein:
Replicase polyprotein 1abRNA-directed RNA polymerase L
Waktu Paruh-
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GS-5745 DB12296
biotech | CAS: 1518996-49-0

GS-5745 has been used in trials studying the treatment of Tumors, Breast Cancer, Crohn's Disease, Colorectal Cancer, and Pancreatic Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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GS-6620 DB15222
small molecule | CAS: 1350735-70-4

GS-6620 is under investigation in clinical trial NCT01316237 (A Study Evaluating the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of GS-6620 in Treatment Naïve Subjects With Chronic Hepatitis C Virus Infection).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Genome polyprotein
Waktu Paruh-
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GS-9191 DB15084
small molecule | CAS: 859209-84-0

GS-9191 is under investigation in clinical trial NCT00499967 (Safety and Effectiveness Study of an Experimental Topical Ointment (GS-9191) for the Treatment of Genital Warts).

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
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GS-9256 DB12876
small molecule | CAS: 1001094-46-7

GS-9256 has been used in trials studying the treatment of HCV Infection and Chronic Hepatitis C Infection.

Kategori:
AcidsAcids, NoncarboxylicAmino Acids, Peptides, and Proteins +4
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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GS030-DP DB17847
biotech

GS030-DP is an optogenetic gene therapy being investigated for the treatment of retinitis pigmentosa. It targets retinal ganglion cells that encodes a light-sensitive channelrhodopsin, ChrimsonR-tdTomato (ChR-tdT), delivered by an AAV2.7m8 vector. It is a com…

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