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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 137 / 236
LFA703 DB03932
small molecule

Deskripsi belum tersedia.

Target Protein:
Integrin alpha-L
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LFF-571 DB13013
small molecule | CAS: 1160959-55-6

LFF571 has been used in trials studying the treatment of Moderate Clostridium Difficile Infection.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +2
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LG-100268 DB01941
small molecule | CAS: 153559-76-3

LG-100268 is a retinoid X receptor (RXR) selective compound.

Kategori:
LigandsNaphthalenesPyridines
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor RXR-beta
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LGD-1550 DB05785
small molecule | CAS: 178600-20-9

LGD-1550 is an orally-active synthetic aromatic retinoic acid agent with potential antineoplastic and chemopreventive activities.

Kategori:
AlkenesBiological FactorsCarotenoids +8
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +1
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LGD-2226 DB08089
small molecule | CAS: 328947-93-9

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
Target Protein:
Androgen receptor
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LGD-3303 DB13937
small molecule | CAS: 917891-35-1

An androgen receptor modulator.

Kategori:
Heterocyclic Compounds, Fused-RingQuinolines
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LGD-6972 DB14779
small molecule | CAS: 1207989-09-0

LGD-6972 is under investigation in clinical trial NCT01919684 (Study to Evaluate Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of LGD-6972 in Healthy Subjects and Subjects With Type 2 Diabetes Mellitus).

Kategori:
Acids, CarbocyclicAlkanesAlkanesulfonic Acids +7
Target Protein:
Glucagon receptor
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LGH-447 DB14943
small molecule | CAS: 1210608-43-7

LGH-447 is under investigation in clinical trial NCT02160951 (Dose Escalation Study of LGH447 in Japanese Patients With Relapsed and/or Refractory Hematologic Malignancies).

Target Protein:
Serine/threonine-protein kinase pim-2
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LH-708 DB17636
small molecule | CAS: 1616758-14-5

Deskripsi belum tersedia.

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Liafensine DB14878
small molecule | CAS: 1198790-53-2

Liafensine is under investigation in clinical trial NCT00892840 (Multiple-Ascending Dose Study).

Kategori:
Heterocyclic Compounds, Fused-Ring
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Liarozole DB13066
small molecule | CAS: 115575-11-6

Liarozole has been used in trials studying the treatment of Ichthyosis, Lamellar.

Kategori:
Antineoplastic AgentsAntineoplastic Agents, HormonalDermatologicals +3
Target Protein:
Cytochrome P450 26A1Aromatase
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Libivirumab DB17748
biotech | CAS: 569658-79-3

Libivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

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LIC-477 DB05363
small molecule

LIC-477is indicated to be suitable for the treatment of psychosomatic disturbances, epilepsy, trigeminal neuralgia and cerebral spasticity.

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Licaminlimab DB18936
biotech | CAS: 1688648-13-6

Licaminlimab is under investigation in clinical trial NCT05896670 (Safety and Efficacy of Licaminlimab Ophthalmic Suspension for the Treatment of Dry Eye Disease).

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Licochalcone A DB19281
small molecule | CAS: 58749-22-7

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesFabaceae +5
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
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Licofelone DB04725
small molecule | CAS: 156897-06-2

Developed by the German pharmaceutical company, Merckle GmbH, together with EuroAlliance partners Alfa Wassermann and Lacer, licofelone (ML3000) is a dual COX/LOX inhibitor and the first member of this new class of analgesic and anti-inflammatory drugs. It is…

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +15
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenaseProstaglandin G/H synthase 2Group IIE secretory phospholipase A2
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Licogliflozin DB15048
small molecule | CAS: 1291094-73-9

Licogliflozin is under investigation in clinical trial NCT03320941 (A Dose-finding Study to Evaluate the Change in Weight After Treatment With LIK066 in Japanese Patients With Obesity).

Kategori:
AlcoholsBlood Glucose Lowering AgentsCarbohydrates +2
Target Protein:
Sodium/glucose cotransporter 1Sodium/glucose cotransporter 2
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Licorice Approved DB10675
biotech

Licorice allergenic extract is used in allergenic testing.

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Lidocaine Approved DB00281
small molecule | CAS: 137-58-6

Ever since its discovery and availability for sale and use in the late 1940s, lidocaine has become an exceptionally commonly used medication [T583]. In particular, lidocaine's principal mode of action in acting as a local anesthetic that numbs the sensations …

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAgents that reduce seizure thresholdAmides +49
Target Protein:
Sodium channel protein type 11 subunit alphaSodium channel protein type 10 subunit alphaSodium channel protein type 9 subunit alpha +5
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe mean systemic c…
Genetik -
Lidoflazine Approved DB13766
small molecule | CAS: 3416-26-0

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAntiarrhythmic agentsBradycardia-Causing Agents +13
Target Protein:
Sodium channel protein type 3 subunit alphaEquilibrative nucleoside transporter 1
Waktu Paruh-
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Lidorestat DB07063
small molecule | CAS: 245116-90-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsHeterocyclic Compounds, Fused-RingIndoles +1
Target Protein:
Aldo-keto reductase family 1 member B1
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biotech | CAS: 1401812-88-1

Lifastuzumab vedotin is under investigation in clinical trial NCT01363947 (Safety and Pharmacokinetics of Escalating Doses of DNIB0600A in Participants With Non-Small Cell Lung Cancer (NSCLC) and Platinum Resistant Ovarian Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Lifileucel Approved DB17107
biotech | CAS: 2306267-74-1

Lifileucel is a tumour-derived autologous T cell immunotherapy composed of a suspension of tumour-derived T cells from the patient [L50171] which undergo isolation, ex vivo expansion, and activation[A263341] Lifileucel was granted accelerated approval by the …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsAntineoplastic cell and gene therapy +3
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Lifirafenib DB14773
small molecule | CAS: 1446090-79-4

Lifirafenib is under investigation in clinical trial NCT03641586 (The Study of BGB-283 in Chinese Subjects With Local Advanced or Metastatic Malignant Solid Tumor).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase B-raf
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Lifitegrast Approved DB11611
small molecule | CAS: 1025967-78-5

Lifitegrast is a FDA approved drug for the treatment of keratoconjunctivitis sicca (dry eye syndrome). It is a tetrahydroisoquinoline derivative and lymphocyte function-associated antigen-1 ( LFA-1) antagonist that was discovered through the rational design p…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +18
Target Protein:
Intercellular adhesion molecule 1Integrin alpha-L
Waktu ParuhNot possible to cal…
Vol. Distribusi-
KlirensNot possible to cal…
Genetik -
Ligelizumab DB11856
biotech | CAS: 1322627-61-1

Ligelizumab is a humanized IgG1k monoclonal antibody targeted against immunoglobulin E (IgE). Similar in mechanism to [omalizumab], another IgE-directed monoclonal antibody, ligelizumab has a distinct binding epitope as compared to its peer (with a small degr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Immunoglobulin heavy constant epsilon
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Light mineral oil Approved DB11579
small molecule | CAS: 92062-35-6

Deskripsi belum tersedia.

Kategori:
Basic Ointments and Protectants
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Ligufalimab DB17542
biotech | CAS: 2428381-55-7

Ligufalimab is a humanized immunoglobulin G4 (IgG4) monoclonal antibody targeting leukocyte surface antigen CD47. It is under investigation in clinical trial NCT04900350 (A Trial of AK117 (Anti-cd47) in Patients With Myelodysplastic Syndrome).

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Ligustrazine DB19074
small molecule | CAS: 1124-11-4

Ligustrazine is under investigation in clinical trial NCT05942352 (Clinical Study of Ligustrazine in Treating Alcohol Addiction).

Kategori:
Antiplatelet agentsCardiovascular AgentsVasodilating Agents
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Lilotomab DB19076
biotech | CAS: 1453362-55-4

Lilotomab is under investigation in clinical trial NCT01796171 (A Phase 1/2 Study of Betalutin for Treatment of Relapsed Non-hodgkin Lymphoma).

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Limaprost DB09211
small molecule | CAS: 74397-12-9

Limaprost (as Limaprost alfadex; CAS number 88852-12-4) is an oral prostaglandin E1 analog. Prostaglandins act on a variety of cells such as vascular smooth muscle cells causing constriction or dilation, on platelets causing aggregation or disaggregation and …

Kategori:
AnticoagulantsAutacoidsBiological Factors +11
Target Protein:
Prostaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtypeProstaglandin E2 receptor EP3 subtype +1
Waktu ParuhThe mean half life …
Vol. Distribusi-
KlirensMean total clearanc…
Genetik -
Linaclotide Approved DB08890
small molecule | CAS: 851199-59-2

Linaclotide is a synthetic 14-amino acid cyclic peptide [A260271] and first-in-class guanylate cyclase-C (G-CC) agonist.[A260271, L47211] Linaclotide is structurally related to human guanylin and uroguanylin, paracrine peptide hormones that are endogenous act…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsDrugs for Constipation +7
Target Protein:
Guanylyl cyclase C
Waktu ParuhThere is no availab…
Vol. DistribusiGiven that linaclot…
KlirensNo information is a…
Genetik -
Linagliptin Approved DB08882
small molecule | CAS: 668270-12-0

Linagliptin is a DPP-4 inhibitor developed by Boehringer Ingelheim for the treatment of type II diabetes [L9557]. Linagliptin differs from other DPP-4 inhibitors in that it has a non-linear pharmacokinetic profile, is not primarily eliminated by the renal sys…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +24
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe terminal half l…
Vol. DistribusiA single intravenou…
KlirensTotal clearance of …
Genetik -
Lincomycin Approved DB01627
small molecule | CAS: 154-21-2

Lincomycin is a lincosamide antibiotic first isolated from the soil bacterium _Streptomyces lincolnensis_ in Lincoln, Nebraska.[A190621] Clinical use of lincomycin has largely been superseded by its semisynthetic derivative [clindamycin] due to its higher eff…

Kategori:
Agents that produce neuromuscular block (indirect)Anti-Bacterial AgentsAnti-Infective Agents +11
Target Protein:
23S ribosomal RNA
Waktu ParuhLincomycin has a bi…
Vol. DistribusiLincomycin administ…
KlirensLincomycin administ…
Genetik -
Linerixibat DB11729
small molecule | CAS: 1345982-69-5

GSK2330672 has been investigated for the treatment of Diabetes Mellitus, Type 2.

Kategori:
AminesAzepinesSulfur Compounds +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
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Linezolid Approved DB00601
small molecule | CAS: 165800-03-3

Linezolid is a synthetic antibiotic which is used for the treatment of infections caused by aerobic Gram-positive bacteria. Its effects are bacteriostatic against both enterococci and staphylococci and bactericidal against most isolates of streptococci.[L3296…

Kategori:
AcetamidesAcetatesAcids, Acyclic +22
Target Protein:
23S ribosomal RNA
Waktu ParuhThe elimination hal…
Vol. DistribusiAt steady-state, th…
KlirensTotal clearance of …
Genetik -
Linifanib DB06080
small molecule | CAS: 796967-16-3

Linifanib (ABT-869) is a small molecule vascular endothelial growth factor (VEGF) receptor-based kinase inhibitor that is designed to suppress tumor growth by preventing the formation of new blood vessels that supply the tumor with oxygen and nutrients and by…

Kategori:
AmidesBenzene DerivativesHeterocyclic Compounds, Fused-Ring +2
Target Protein:
Vascular endothelial growth factor receptor 3Receptor-type tyrosine-protein kinase FLT3Vascular endothelial growth factor receptor 1 +3
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Linopirdine DB13806
small molecule | CAS: 105431-72-9

Deskripsi belum tersedia.

Kategori:
Cardiovascular AgentsCentral Nervous System AgentsCompounds used in a research, industrial, or household setting +8
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3
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Linopristin DB19296
small molecule | CAS: 325965-23-9

Linopristin is an antibiotic of the streptogramin B class. It is one part of the combination product NXL 103, along with [Virginiamycin M1]. The combination product was under investigation in clinical trials NCT00653172 and NCT00949130 for treatment of variou…

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Linperlisib DB17235
small molecule | CAS: 1702816-75-8

Deskripsi belum tersedia.

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Linrodostat DB14986
small molecule | CAS: 1923833-60-6

Linrodostat is under investigation in clinical trial NCT03247283 (Pharmacokinetics and Metabolism Study in Healthy Male Participants).

Kategori:
AcetatesAcids, AcyclicAmides +2
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Linseed oil DB11357
biotech | CAS: 66071-03-2

Linseed oil is a rich source of ?-Linolenic acid extracted from the dried, ripened seeds of the flax plant *Linum usitatissimum*. Other fatty acids contained in linseed oil include palmitic acid, stearic acid, oleic acid and linolenic acid. Linseed oil is par…

Kategori:
Biological ProductsComplex MixturesFats +5
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Linsidomine DB13400
small molecule | CAS: 33876-97-0

Deskripsi belum tersedia.

Kategori:
Antihypertensive AgentsAntiplatelet agentsCardiac Therapy +12
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Linsitinib DB06075
small molecule | CAS: 867160-71-2

An orally bioavailable small molecule inhibitor of the insulin-like growth factor 1 receptor (IGF-1R) with potential antineoplastic activity. IGF-1R inhibitor OSI-906 selectively inhibits IGF-1R, which may result in the inhibition of tumor cell proliferation …

Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
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Lintitript DB04867
small molecule | CAS: 136381-85-6

Lintitript is a new, highly specific and potent CCK-A receptor antagonist.

Kategori:
Heterocyclic Compounds, Fused-RingHormone AntagonistsHormones, Hormone Substitutes, and Hormone Antagonists +2
Target Protein:
Cholecystokinin receptor type A
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Lintuzumab DB14877
biotech | CAS: 166089-32-3

Lintuzumab is under investigation in clinical trial NCT00016159 (Chemotherapy Plus Monoclonal Antibody in Treating Patients With Acute Promyelocytic Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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biotech | CAS: 2209911-94-2

Lintuzumab actinium Ac-225 is under investigation in clinical trial NCT00672165 (Targeted Atomic Nano-Generators (Actinium-225-Labeled Humanized Anti-CD33 Monoclonal Antibody HuM195) in Patients With Advanced Myeloid Malignancies).

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Linvoseltamab DB17447
biotech

Linvoseltamab is an investigational bispecific antibody. It promotes the interaction of B-cell maturation antigen (BCMA) on multiple myeloma cells with CD3-expressing T cells.

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Linzagolix Approved DB17083
small molecule | CAS: 935283-04-8

Linzagolix is a non-peptide, selective antagonist of the gonadotropin-releasing hormone (GnRH) receptor. It has been studied for the treatment of estrogen-dependent conditions such as uterine fibroids and endometriosis.[A253642,A253647] It is similar to other…

Kategori:
Anti-Gonadotropin-Releasing HormonesBCRP/ABCG2 SubstratesCytochrome P-450 CYP2C8 Inhibitors +18
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu ParuhThe half-life of li…
Vol. DistribusiAfter seven days of…
KlirensThe geometric mean …
Genetik -
LioCyx-M004 DB17368
biotech

LioCyx-M004 are autologous T cells transduced with a retroviral vector encoding a hepatitis B virus antigen-specific T cell receptor.

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