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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 136 / 252
Inobrodib DB17514
small molecule | CAS: 2222941-37-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Inolimomab DB15628
biotech | CAS: 152981-31-2

Inolimomab is under investigation as an agent to treat steroid-resistant graft vs host disease. It has thus far offered similar efficacy to other monoclonal antibody options, though it may carry a higher risk of infections.[A241385]

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +9
Target Protein:
Interleukin-2 receptor subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inosine DB04335
small molecule | CAS: 58-63-9

A purine nucleoside that has hypoxanthine linked by the N9 nitrogen to the C1 carbon of ribose. It is an intermediate in the degradation of purines and purine nucleosides to uric acid and in pathways of purine salvage. It also occurs in the anticodon of certa…

Kategori:
DermatologicalsGenito Urinary System and Sex HormonesGynecological Antiinfectives and Antiseptics +8
Target Protein:
Purine nucleoside phosphorylaseIAG-nucleoside hydrolasePurine nucleoside phosphorylase DeoD-type
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 70023-32-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Inosine pranobex Approved DB13156
small molecule | CAS: 36703-88-5

Inosine pranobex (Isoprinosine or Methisoprinol) is a combination of inosine, acetamidobenzoic acid, and dimethylaminoisopropanol used as an antiviral drug.

Kategori:
AcetanilidesAdjuvants, ImmunologicAmides +14
Waktu Paruh50 min
Vol. Distribusi-
Klirens-
Genetik -
Inosinic Acid DB04566
small molecule | CAS: 131-99-7

Inosine 5'-Monophosphate. A purine nucleotide which has hypoxanthine as the base and one phosphate group esterified to the sugar moiety.

Kategori:
Heterocyclic Compounds, Fused-RingInosine NucleotidesNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Hypoxanthine-guanine-xanthine phosphoribosyltransferaseAdenylosuccinate synthetase +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inositol Approved DB13178
small molecule | CAS: 87-89-8

Inositol is a collection of nine different stereoisomers but the name is usually used to describe only the most common type of inositol, myo-inositol. Myo-inositol is the cis-1,2,3,5-trans-4,6-cyclohexanehexol and it is prepared from an aqueous extract of cor…

Kategori:
AlcoholsAlimentary Tract and MetabolismCarbohydrates +6
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe pharmacokinetic…
KlirensThe pharmacokinetic…
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesSugar Alcohols +1
Target Protein:
RAC-alpha serine/threonine-protein kinaseTyrosine-protein kinase BTKInositol-trisphosphate 3-kinase A +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 91840-07-2

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydratesSugar Alcohols +1
Target Protein:
1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase delta-1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inositol nicotinate Approved DB08949
small molecule | CAS: 6556-11-2

Inositol nicotinate, also known as Inositol hexaniacinate/hexanicotinate or "no-flush niacin", is a niacin ester and vasodilator. It is used in food supplements as a source of niacin (vitamin B3), where hydrolysis of 1 g (1.23 mmol) inositol hexanicotinate yi…

Kategori:
Cardiovascular AgentsNicotinic Acid and DerivativesOther Nutritional Agents +5
Target Protein:
Hydroxycarboxylic acid receptor 3Hydroxycarboxylic acid receptor 2
Waktu ParuhMean elimination ha…
Vol. DistribusiMean Vd following i…
KlirensMean clearance rate…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Cytohesin-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inotersen Approved DB14713
biotech | CAS: 1492984-65-2

Inotersen is a transthyretin-directed antisense oligonucleotide for the treatment of the polyneuropathy caused by hereditary transthyretin-mediated amyloidosis in adults. It was FDA approved in October 2018.[L11761] Inotersen has been shown to improve the cou…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesDecreased RNA Integrity +15
Target Protein:
TransthyretinTransthyretin mRNA
Waktu ParuhThe terminal elimin…
Vol. DistribusiBased on animal stu…
KlirensInotersen is mainly…
Genetik -
Inotuzumab ozogamicin Approved DB05889
biotech | CAS: 635715-01-4

Inotuzumab ozogamicin is an antibody-drug conjugate consisting of a humanized IgG4 kappa CD22-targeting monoclonal antibody covalently attached to calicheamicin derivative, N-acetyl-gamma-calicheamicin dimethylhydrazide.[A20352] The antibody portion of the dr…

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntibodies +33
Target Protein:
B-cell receptor CD22
Waktu ParuhIn patients with re…
Vol. DistribusiIn humans, the tota…
KlirensThe pharmacokinetic…
Genetik -
INS 316 DB05390
small molecule

INS316 belongs to the family of drugs called nucleoside triphosphates.It is studied in the diagnosis of lung diseases, including lung cancer. It is selective P2y2 receptor antagonists claimed to be useful as anti-inflammatory agents.

Target Protein:
P2Y purinoceptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
INS018_055 DB18083
small molecule

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Insulin argine DB11564
biotech | CAS: 68859-20-1

Deskripsi belum tersedia.

Kategori:
Blood Glucose Lowering AgentsCytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown) +2
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Insulin aspart Approved DB01306
biotech | CAS: 116094-23-6

Insulin aspart is a rapid-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insulin…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +14
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens1.2 L/h/kg
Genetik -
Insulin beef Approved DB09456
biotech | CAS: 11070-73-8

Insulin beef has been discontinued in the US and Canada since 2017.[L10827]

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsCytochrome P-450 CYP1A2 Inducers +6
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Insulin degludec Approved DB09564
biotech | CAS: 844439-96-9

Insulin degludec is an ultra-long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A18561,A18562,A18563,A18564,A174934] Insulin is typically prescribed for the management of diabetes mellitus to mimic the ac…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
InsulinInsulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUsing a one-compart…
KlirensThe mean apparent c…
Genetik -
Insulin detemir Approved DB01307
biotech | CAS: 169148-63-4

Insulin detemir is a long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes.[A2358, A2359, A2360, A44] Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenou…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiInsulin detemir has…
KlirensThe apparent cleara…
Genetik -
biotech | CAS: 2131038-11-2

Insulin efsitora alfa is under investigation in clinical trial NCT05662332 (A Study of Insulin Efsitora Alfa (LY3209590) Compared to Glargine in Adult Participants With Type 2 Diabetes Who Are Starting Basal Insulin for the First Time (QWINT-1)).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Insulin glargine Approved DB00047
biotech | CAS: 160337-95-1

Insulin glargine is a long-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insuli…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAntimetabolites +18
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Insulin glulisine Approved DB01309
biotech | CAS: 207748-29-6

Insulin glulisine is a short-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is typically prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insu…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +15
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhElimination half li…
Vol. Distribusi13 L
Klirens-
Genetik -
Insulin human Approved DB00030
biotech | CAS: 11061-68-0

Human Insulin, also known as Regular Insulin, is a short-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Human insulin is produced by recombinant DNA technology and is identical to endogenously produced ins…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +14
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptorCarboxypeptidase E +3
Waktu ParuhSystemic insulin di…
Vol. Distribusi-
Klirens-
Genetik -
Insulin icodec Approved DB16693
biotech | CAS: 1188379-43-2

Insulin icodec is an ultra long-acting basal insulin analogue. It is a re-engineered version of the ultra long-acting oral basal insulin OI338, with several modifications introduced to significantly extend the half-life.[A264093] These modifications - which c…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +10
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhThe mean half-life …
Vol. DistribusiAccording to popula…
KlirensAccording to popula…
Genetik -
Insulin lispro Approved DB00046
biotech | CAS: 133107-64-9

Insulin lispro is a rapid-acting form of insulin used for the treatment of hyperglycemia caused by Type 1 and Type 2 Diabetes. Insulin is prescribed for the management of diabetes mellitus to mimic the activity of endogenously produced human insulin, a peptid…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +14
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu ParuhAfter subcutaneous …
Vol. DistribusiWhen administered i…
KlirensWhen administered i…
Genetik -
biotech | CAS: 1200440-65-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +16
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Insulin pork Approved DB00071
biotech | CAS: 12584-58-6

Insulin isolated from pig pancreas. Composed of alpha and beta chains, processed from pro-insulin. Forms a hexameric structure.

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +13
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 874442-57-6

Deskripsi belum tersedia.

Kategori:
Blood Glucose Lowering AgentsCytochrome P-450 CYP1A2 InducersCytochrome P-450 CYP1A2 Inducers (strength unknown) +3
Target Protein:
Insulin receptorInsulin-like growth factor 1 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
INT41 DB17935
biotech

INT41 (also known as rAAV6-INT41) is a recombinant adeno-associated virus vector containing DNA encoding INT41 intrabody.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Interferon alfa DB05258
biotech

Natural interferon alpha or Multiferon is obtained from the leukocyte fraction of human blood following induction with Sendai virus. Interferon alfa contains several naturally occurring IFN-? subtypes and is purified by affinity chromatography. Interferon alp…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +14
Target Protein:
Interferon alpha/beta receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntineoplastic Agents +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Interferon alfa-2a Approved DB00034
biotech | CAS: 76543-88-9

Interferon a (human leukocyte protein moiety reduced). A type I interferon consisting of 165 amino acid residues with lysine in position 23. This protein is produced by recombinant DNA technology and resembles interferon secreted by leukocytes. It is used ext…

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAmino Acids, Peptides, and Proteins +20
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Waktu ParuhThe IM half-life of…
Vol. Distribusi* 0.223 to 0.748 L/…
Klirens* 2.14 - 3.62 mL/mi…
Genetik -
Interferon alfa-2b Approved DB00105
biotech | CAS: 98530-12-2

Interferon alpha 2b (human leukocyte clone hif-sn 206 protein moiety reduced). A type I interferon consisting of 165 amino acid residues with arginine in position 23. This protein is produced by recombinant DNA technology and resembles interferon secreted by …

Kategori:
Adjuvants, ImmunologicAlfa InterferonsAmino Acids, Peptides, and Proteins +24
Target Protein:
Interferon alpha/beta receptor 2Interferon alpha-2Interferon alpha/beta receptor 1
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 142192-09-4

Interferon alfa-2c is under investigation in clinical trial NCT00485563 (A Phase II Study of EC17 (Folate-hapten Conjugate) in Patients With Progressive Metastatic Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytochrome P-450 CYP1A2 Inhibitors +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Interferon beta-1a Approved DB00060
biotech | CAS: 145258-61-3

Human interferon beta (166 residues), glycosylated, MW=22.5kD. It is produced by mammalian cells (Chinese Hamster Ovary cells) into which the human interferon beta gene has been introduced. The amino acid sequence is identical to that of natural human interfe…

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAnti-Infective Agents +16
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Waktu Paruh10 hrs
Vol. Distribusi-
Klirens* 33-55 L/hour [Hea…
Genetik -
Interferon beta-1b Approved DB00068
biotech | CAS: 145155-23-3

Human interferon beta (165 residues), cysteine 17 is substituted with serine. Produced in E. coli, no carbohydrates, MW=18.5kD

Kategori:
Adjuvants, ImmunologicAmino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating Agents +15
Target Protein:
Interferon alpha/beta receptor 1Interferon alpha/beta receptor 2
Waktu Paruh-
Vol. Distribusi* 0.25 to 2,88 L/kg
Klirens* 9.4 – 28.9 mL/min…
Genetik -
biotech

Interferon gamma is a Type 1 inflammatory cytokine and the only type II interferon. It has antitumor properties, antiviral activities, and important immunoregulatory functions. The interferon is primarily produced by activated T lymphocytes and natural killer…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsInterferons
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Interferon gamma-1b Approved DB00033
biotech | CAS: 98059-61-1

Human Interferon gamma-1b (140 residues), produced from E. coli. Production of Actimmune is achieved by fermentation of a genetically engineered Escherichia coli bacterium containing the DNA which encodes for the human protein. Purification of the product is …

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytochrome P-450 CYP1A2 Inhibitors +12
Target Protein:
Interferon gamma receptor 1Interferon gamma receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Interferon kappa is a subclass of type I interferon mediating host defence which consists of 207 amino acids and has 30% homology with others of the same class as it consists of a series of cysteine and a 27-amino acid signal peptide conserved in type I inter…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Interleukin-7 DB11997
biotech | CAS: 858376-81-5

Interleukin 7 has been used in trials studying the treatment of Metastatic Breast Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Intermedine DB17612
biotech | CAS: 581-05-5

Deskripsi belum tersedia.

Kategori:
AlkaloidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Intetumumab DB12701
biotech | CAS: 725735-28-4

Intetumumab has been used in trials studying the treatment of Melanoma.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Intoplicine DB12868
small molecule | CAS: 125974-72-3

Intoplicine has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inula helenium root Approved DB14350
biotech

Inula helenium root is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Inulin Approved DB00638
biotech | CAS: 9005-80-5

A starch found in the tubers and roots of many plants. Since it is hydrolyzable to fructose, it is classified as a fructosan. It has been used in physiologic investigation for determination of the rate of glomerular function.

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +9
Target Protein:
InsulinCycloinulo-oligosaccharide fructanotransferase
Waktu Paruh2-4 hours
Vol. Distribusi-
Klirens-
Genetik -
Inupadenant DB19129
small molecule | CAS: 2246607-08-7

Inupadenant is under investigation in clinical trial NCT05060432 (Study of EOS-448 With Standard of Care And/or Investigational Therapies in Participants With Advanced Solid Tumors).

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
INVAC-1 DB16196
biotech | CAS: 1708137-44-3

INVAC-1 is under investigation in clinical trial NCT03265717 (DNA Plasmid Encoding a Modified Human Telomerase Reverse Transcriptase (Htert), Invac-1 in Chronic Lymphocytic Leukemia).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IO-202 DB17548
biotech

IO-202 is a first-in-class antibody targeting the Leukocyte Immunoglobulin-Like Receptor subfamily B (LILRB) member 4 (LILRB4).[A257276] It is being investigated in cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6751–6800 dari 12560
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