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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
Referensi
11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 135 / 236
small molecule | CAS: 16610-63-2

Deskripsi belum tersedia.

Target Protein:
Farnesyl pyrophosphate synthaseGeranylgeranyl pyrophosphate synthase
Waktu Paruh-
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Genetik -
small molecule | CAS: 27836-64-2

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 683-10-3

Deskripsi belum tersedia.

Kategori:
AminesOnium CompoundsQuaternary Ammonium Compounds +1
Target Protein:
AppA protein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lavendustin A DB16768
small molecule | CAS: 125697-92-9

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesEnzyme InhibitorsTyrosine Kinase Inhibitors
Target Protein:
Epidermal growth factor receptorTyrosine-protein kinase Lck
Waktu Paruh-
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Lavendustin b DB16760
small molecule | CAS: 125697-91-8

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +5
Waktu Paruh-
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Lavoltidine DB12884
small molecule | CAS: 76956-02-0

Lavoltidine has been used in trials studying the diagnostic of Reflux, Gastroesophageal and Gastroesophageal Reflux Disease.

Kategori:
Gastric Acid Lowering AgentsHistamine AgentsHistamine Antagonists +2
Target Protein:
Histamine H2 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lawsone DB04744
small molecule | CAS: 83-72-7

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsColoring Agents +10
Waktu Paruh-
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Genetik -
LAX-101 DB05301
small molecule | CAS: 909712-41-0

LAX-101 treats hungtington’s disease, not just the symptoms but the disease itself. The active molecule in LAX-101 is Eicosapentaenoic Acid (EPA). All molecules of EPA are identical. The molecules of EPA found in LAX-101 are identical to the molecules of EPA …

Target Protein:
Phospholipase D1Caspase-1
Waktu Paruh-
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Genetik -
Lazertinib Approved DB16216
small molecule | CAS: 1903008-80-9

Lazertinib is an oral, third-generation, epidermal growth factor receptor (EGFR) tyrosine kinase inhibitor (TKI).[A264299, A264304] Lazertinib was first approved in South Korea on January 18, 2021, for the treatment of _EGFR_ T790M mutation-positive non-small…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Epidermal growth factor receptor
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Lazuvapagon DB19046
small molecule | CAS: 2379889-71-9

Lazuvapagon is under investigation in clinical trial NCT03116191 (Trial of SK-1404 for Nocturia Due to Nocturnal Polyuria in Japanese Subjects).

Waktu Paruh-
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LB-001 DB17685
biotech

LB-001 is a gene editing therapy designed to incorporate a functioning version of the faulty methylmalonyl-COA mutase (MUT) gene into the genome of patients with methylmalonic acidemia.

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LB-102 DB19214
small molecule | CAS: 2227154-23-4

LB-102 is under investigation in clinical trial NCT06179108 (Randomized, Double-blinded, Placebo-controlled, Evaluating the Treatment With LB-102 in Patients With Acute Schizophrenia).

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LCP-AtorFen DB05769
small molecule

LCP-AtorFen is a fixed-dose combination therapy for the treatment of high cholesterol levels combining atorvastatin (the active ingredient of Lipitor®) and the lowest dose of fenofibrate without food effect. LCP-AtorFen is designed to be a once daily tablet o…

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Lebrikizumab Approved DB11914
biotech | CAS: 953400-68-5

Lebrikizumab is a monoclonal antibody that binds to IL-13 with high affinity and slow off-rate.[L51374] It binds to a different epitope compared [tralokinumab].[A262874,A262879] On November 17, 2023, lebrikizumab was approved by the EMA under the brand nam…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAntibodies +10
Target Protein:
Interleukin-13
Waktu ParuhThe mean eliminatio…
Vol. DistribusiBased on a populati…
KlirensIn the population P…
Genetik -
Lecanemab Approved DB14580
biotech | CAS: 1260393-98-3

Lecanemab is a recombinant humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against aggregated soluble and insoluble forms of amyloid beta (A?), which are implicated in the pathophysiology of Alzheimer’s disease.[L44537] Lecanemab works to…

Kategori:
Alzheimer DiseaseAlzheimer Disease, drug therapyAmino Acids, Peptides, and Proteins +12
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe mean value (95%…
KlirensThe clearance of le…
Genetik -
small molecule | CAS: 8030-76-0

A complex mixture of phospholipids; glycolipids; and triglycerides; with substantial amounts of phosphatidylcholines; phosphatidylethanolamines; and phosphatidylinositols, which are sometimes loosely termed as 1,2-diacyl-3-phosphocholines. Lecithin is a compo…

Waktu Paruh-
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Ledipasvir Approved DB09027
small molecule | CAS: 1256388-51-8

Ledipasvir is a direct acting antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized int…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +10
Target Protein:
Genome polyproteinNonstructural protein 5A
Waktu ParuhThe median terminal…
Vol. Distribusi-
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Lefamulin Approved DB12825
small molecule | CAS: 1061337-51-6

Lefamulin is a pleuromutilin antibiotic used for the treatment of bacterial community-acquired pneumonia. A pleuromotilin is a more recently developed type of antibiotic that is derived from the fungus, Pleurotus mutilus.[A183206] Lefamulin is available in in…

Kategori:
AcetatesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
50S ribosomal protein L22
Waktu ParuhThe average elimina…
Vol. DistribusiThe average volume …
KlirensThe total body clea…
Genetik -
Lefitolimod DB15061
biotech | CAS: 1548439-51-5

Lefitolimod is under investigation in clinical trial NCT03837756 (Combining TLR9 Agonist With bNAbs for Reservoir Reduction and Immunological Control of HIV).

Kategori:
Nucleic AcidsNucleic Acids, Nucleotides, and Nucleosides
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Leflunomide Approved DB01097
small molecule | CAS: 75706-12-6

Leflunomide is a pyrimidine synthesis inhibitor belonging to the DMARD (disease-modifying antirheumatic drug) class of drugs, which are chemically and pharmacologically very heterogeneous. Leflunomide was approved by FDA and in many other countries (e.g., Can…

Kategori:
AdjuvantsAgents Causing Muscle ToxicityAntineoplastic and Immunomodulating Agents +16
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialDihydroorotate dehydrogenase (quinone), mitochondrialAryl hydrocarbon receptor +1
Gen Terkait:
CYP1A2
Waktu Paruh2 weeks
Vol. Distribusi* 0.13 L/kg
Klirens-
Genetik 1 Varian
Leflutrozole DB19047
small molecule | CAS: 143030-47-1

Leflutrozole is under investigation in clinical trial NCT02908074 (A 6 Month Safety Extension Study of MBGS205).

Kategori:
Aromatase Inhibitors
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Lefradafiban DB04863
small molecule | CAS: 149503-79-7

Lefradafiban is an oral platelet glycoprotein IIb/IIIa receptor antagonist being investigated in the treatment of angina.

Kategori:
Antianginal AgentsBenzene DerivativesPlatelet Glycoprotein GPIIb-IIIa Complex, antagonists & inhibitors +1
Target Protein:
Integrin alpha-IIbIntegrin beta-3
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Lemborexant Approved DB11951
small molecule | CAS: 1369764-02-2

Lemborexant is a novel dual orexin receptor antagonist used in the treatment of insomnia characterized by difficulties with sleep onset and/or sleep maintenance.[L10863] Recent research in the field of sleep disorders has revealed that insomnia is likely driv…

Kategori:
Central Nervous System AgentsCentral Nervous System DepressantsCytochrome P-450 CYP2B6 Inducers +17
Target Protein:
Orexin/Hypocretin receptor type 1Orexin receptor type 2
Waktu ParuhThe half-life for l…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Lemzoparlimab DB17572
biotech | CAS: 2377483-71-9

Lemzoparlimab is under investigation in clinical trial NCT04912063 (Study to Evaluate Adverse Events and Movement of Lemzoparlimab in Body When Used Intravenously (IV) With Azacitidine Subcutaneously or IV and Venetoclax Orally in Participants With Acute Myel…

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Lenabasum DB12193
small molecule | CAS: 137945-48-3

Ajulemic acid has been used in trials studying the treatment of Cystic Fibrosis, Dermatomyositis, and Diffuse Cutaneous Systemic Sclerosis.

Kategori:
Agents producing tachycardiaCannabinoid Receptor AgonistsCannabinoids and similars +5
Target Protein:
Tumor necrosis factor
Waktu Paruh-
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Lenacapavir Approved DB15673
small molecule | CAS: 2189684-44-2

HIV/AIDS remains an area of concern despite the introduction of numerous successful therapies, mainly due to the emergence of multidrug resistance and patient difficulty in adhering to treatment regimens.[A244170, A244175] Lenacapavir is a first-in-class caps…

Kategori:
AcetatesAcids, AcyclicAmides +17
Target Protein:
Gag-Pol polyprotein
Waktu ParuhThe median half-lif…
Vol. DistribusiThe steady state vo…
KlirensLenacapavir clearan…
Genetik -
biotech | CAS: 1640969-63-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lenalidomide Approved DB00480
small molecule | CAS: 191732-72-6

Lenalidomide (previously referred to as CC-5013) is an immunomodulatory drug with potent antineoplastic, anti-angiogenic, and anti-inflammatory properties.[A228553] It is a 4-amino-glutamyl analogue of [thalidomide] [A228543] and like thalidomide, lenalidomid…

Kategori:
Acids, CarbocyclicAngiogenesis InhibitorsAngiogenesis Modulating Agents +18
Target Protein:
Tumor necrosis factorProtein cereblonTumor necrosis factor ligand superfamily member 11 +2
Waktu ParuhIn healthy subjects…
Vol. DistribusiIn healthy male sub…
KlirensThe renal clearance…
Genetik -
Leniolisib Approved DB16217
small molecule | CAS: 1354690-24-6

Leniolisib is a potent and selective inhibitor of phosphoinositide 3-kinase ? (PI3K?). The FDA approved leniolisib on March 24, 2023, making it the first treatment for activated phosphoinositide 3-kinase delta syndrome (APDS).[L45758] APDS is a primary immuno…

Kategori:
Adjuvants, ImmunologicAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +14
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe effective half-…
Vol. DistribusiThe systemic decay …
KlirensIn one study, healt…
Genetik -
Lenomorelin DB11895
biotech | CAS: 258279-04-8

Lenomorelin has been investigated for the treatment and basic science of Cancer, Alcoholism, Metabolism, Hypopituitarism, and Frailty Syndrome, among others.

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lentinan DB13480
small molecule | CAS: 37339-90-5

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lenvatinib Approved DB09078
small molecule | CAS: 417716-92-8

Lenvatinib is a receptor tyrosine kinase (RTK) inhibitor that inhibits the kinase activities of vascular endothelial growth factor (VEGF) receptors VEGFR1 (FLT1), VEGFR2 (KDR), and VEGFR3 (FLT4). Lenvatinib also inhibits other RTKs that have been implicated i…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +41
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3 +7
Waktu ParuhThe terminal elimin…
Vol. Distribusi-
Klirens-
Genetik -
Lenvervimab DB17814
biotech | CAS: 2055006-79-4

Deskripsi belum tersedia.

Waktu Paruh-
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Lenzilumab DB15148
biotech | CAS: 1229575-09-0

Lenzilumab is under investigation in clinical trial NCT02546284 (Study of Lenzilumab in Previously Treated Patients With Chronic Myelomonocytic Leukemia (CMML)).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Inflammatory AgentsAntibodies +7
Waktu Paruh-
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Lepirudin Approved DB00001
biotech | CAS: 138068-37-8

Lepirudin is a recombinant hirudin formed by 65 amino acids that acts as a highly specific and direct thrombin inhibitor.[L41539,L41569] Natural hirudin is an endogenous anticoagulant found in _Hirudo medicinalis_ leeches.[L41539] Lepirudin is produced in yea…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Target Protein:
Prothrombin
Waktu ParuhLepirudin has an in…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of le…
Genetik -
Lepunafusp alfa DB19011
biotech | CAS: 2396411-71-3

Lepunafusp alfa is under investigation in clinical trial NCT04453085 (An Extension Study of JR-171-101 Study in Patients With MPS I).

Waktu Paruh-
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LErafAON DB04973
biotech

NeoPharm is developing liposome-encapsulated, c-Raf antisense oligodeoxynucleotides (LErafAON) for the potential treatment of various solid tumors, including those that have become resistant to radiation or chemotherapy. Phase I/II trials commenced in March 2…

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu ParuhIn monkeys, the ter…
Vol. Distribusi-
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Lerapolturev DB17217
biotech | CAS: 2430048-02-3

Deskripsi belum tersedia.

Waktu Paruh-
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Lercanidipine Approved DB00528
small molecule | CAS: 100427-26-7

Lercanidipine is a calcium channel blocker of the dihydropyridine class. It is sold under various commercial names including Zanidip.

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAgents Causing Muscle Toxicity +25
Target Protein:
Voltage-dependent calcium channel gamma-1 subunitVoltage-dependent calcium channel subunit alpha-2/delta-1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lerdelimumab DB06557
biotech | CAS: 285985-06-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leridistim DB15095
biotech | CAS: 193700-51-5

Leridistim is under investigation in clinical trial NCT00004215 (Leridistim Compared With Filgrastim in Treating Older Patients With Acute Myeloid Leukemia).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCarbohydrates +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Leriglitazone DB15021
small molecule | CAS: 146062-44-4

Leriglitazone is under investigation in clinical trial NCT03917225 (A Clinical Study to Evaluate the Effect of MIN-102 on the Progression of Friedreich's Ataxia in Male and Female Patients).

Kategori:
Alimentary Tract and MetabolismSulfur CompoundsThiazoles +1
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lerisetron DB12964
small molecule | CAS: 143257-98-1

Lerisetron has been used in trials studying the supportive care of Nausea and Vomiting and Testicular Germ Cell Tumor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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Lerociclib DB16218
small molecule | CAS: 1628256-23-4

Lerociclib is under investigation in clinical trial NCT02983071 (G1T38, a CDK 4/6 Inhibitor, in Combination With Fulvestrant in Hormone Receptor-positive, Her2-negative Locally Advanced or Metastatic Breast Cancer).

Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lerodalcibep DB19071
biotech | CAS: 2250073-78-8

Lerodalcibep is under investigation in clinical trial NCT05004675 (Trial to Evaluate Efficacy and Safety of LIB003 and Inclisiran in High-risk CVD Patients).

Waktu Paruh-
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Leronlimab DB05941
biotech | CAS: 674782-26-4

Leronlimab, or PRO-140, is a human monoclonal antibody developed by CytoDyn.[L12684] It was first described in the literature in 2001.[A3922] This antibody binds to CCR5, which may be useful in treating HIV, cancers, and severely ill COVID-19 patients.[A19284…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +17
Target Protein:
C-C chemokine receptor type 5
Waktu ParuhThe half life of a …
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Lersivirine DB11649
small molecule | CAS: 473921-12-9

Lersivirine has been used in trials studying the treatment of HIV-1.

Kategori:
RNA-Directed DNA Polymerase
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lesinidase alfa DB15267
biotech | CAS: 1522433-40-4

Lesinidase alfa is under investigation in clinical trial NCT02324049 (Safety, Pharmacokinetics, and Pharmacodynamics/Efficacy of SBC-103 in Mucopolysaccharidosis III, Type B (MPS IIIB)).

Waktu Paruh-
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Lesinurad Approved DB11560
small molecule | CAS: 878672-00-5

Lesinurad is an oral uric acid transporter 1 (URAT1) inhibitor indicated for the treatment of hyperuricemia associated with gout. It reduces serum uric acid concentration through the inhibition of URAT1, an enzyme responsible for reuptake of uric acid from th…

Kategori:
AcetatesAcids, AcyclicAntigout Preparations +15
Target Protein:
Solute carrier family 22 member 12Solute carrier family 22 member 11
Waktu Paruh-
Vol. DistribusiThe mean steady sta…
Klirens-
Genetik -
Lesogaberan DB11920
small molecule | CAS: 344413-67-8

Lesogaberan has been used in trials studying the treatment and basic science of GERD, Reflux, Heartburn, Regurgitation, and Reflux Disease, among others.

Kategori:
AcidsAcids, NoncarboxylicAmines +8
Target Protein:
Gamma-aminobutyric acid type B receptor subunit 1Gamma-aminobutyric acid type B receptor subunit 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6701–6750 dari 11778
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