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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 135 / 282
Geldanamycin DB02424
small molecule | CAS: 30562-34-6

Deskripsi belum tersedia.

Kategori:
AmidesAnti-Infective AgentsAntibiotics, Antineoplastic +7
Target Protein:
Heat shock protein HSP 90-alphaEndoplasminHeat shock protein HSP 90-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GEM-231 DB05798
biotech | CAS: 255810-66-3

GEM231 is a second-generation antisense oligonucleotide targeting the mRNA of the R1alpha regulatory subunit of cAMP dependent protein kinase. A monoclonal antibody combined with a toxic substance that is used treat certain types of acute myeloid leukemia in …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
cAMP-dependent protein kinase type II-alpha regulatory subunitcAMP-dependent protein kinase type I-alpha regulatory subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcabene DB05123
small molecule | CAS: 183293-82-5

Gemcabene is a new drug that lowers low-density lipoprotein cholesterol (LDL-C), decreases triglycerides, and raises high-density lipoprotein cholesterol (HDL-C).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcitabine Approved DB00441
small molecule | CAS: 95058-81-4

Gemcitabine is a nucleoside analog and a chemotherapeutic agent. It was originally investigated for its antiviral effects, but it is now used as an anticancer therapy for various cancers.[A233135] Gemcitabine is a cytidine analog with two fluorine atoms repla…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +23
Target Protein:
DNARibonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit +2
Gen Terkait:
RRM1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn patients with va…
KlirensFollowing intraveno…
Genetik 1 Varian
small molecule | CAS: 210829-30-4

Gemcitabine elaidate has been used in trials studying the treatment of Solid Tumor, Lung Cancer, Non-small-cell Lung Cancer, and Metastatic Pancreatic Adenocarcinoma.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemeprost Approved DB08964
small molecule | CAS: 64318-79-2

Gemeprost is a prostaglandin E1 (PGE1) analog and antiprogestogen used for preoperative dilation of the cervix before surgical abortion. It is available as vaginal suppositories and also used in combination with the antiprogestin and mifepristone for terminat…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAutacoids +14
Target Protein:
Prostaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemfibrozil Approved DB01241
small molecule | CAS: 25812-30-0

Gemfibrozil is a fibric acid agent, similar to [clofibrate], used to treat Type IIb, IV, and V hyperlipidemias.[A185777,L8525] Gemfibrozil is not a first line treatment and is prescribed to patients who have not responded adequately to weight loss, diet, exer…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +53
Target Protein:
Peroxisome proliferator-activated receptor alphaLipoprotein lipaseSolute carrier organic anion transporter family member 1B1 +3
Waktu ParuhGemfibrozil has a p…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ge…
Genetik -
Gemigliptin DB12412
small molecule | CAS: 911637-19-9

Gemigliptin is under investigation in Type 2 Diabetes Mellitus. Gemigliptin has been investigated for the treatment of Cancer and Cisplatin Adverse Reaction.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemlapodect DB18769
small molecule | CAS: 1380329-87-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech

Gemogenovatucel-T is a bi-shRNA furin/Granulocyte Macrophage Colony Stimulating Factor (GMCSF) Augmented autologous tumour cell vaccine. Furin is a convertase involved in the activation of TGF?-1 and TGF?-2.[A255163] Gemogenovatucel-T is being investigated in…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemtuzumab ozogamicin Approved DB00056
biotech | CAS: 220578-59-6

Gemtuzumab ozogamicin is a recombinant humanized IgG4 kappa antibody which is conjugated with calicheamicin derivative, a cytotoxic antitumor antibiotic isolated from fermentation of Micromonospora echinospora ssp. calichensis. Gemtuzumab ozogamicin has appro…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +28
Target Protein:
Myeloid cell surface antigen CD33Low affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +1
Waktu ParuhIn pediatric patien…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Geneticin DB04263
small molecule | CAS: 49863-47-0

Geneticin (also known as G418) is an aminoglycoside antibiotic similar in structure to gentamicin B1, produced by Micromonospora rhodorangea. Geneticin blocks polypeptide synthesis by inhibiting the elongation step in both prokaryotic and eukaryotic cells and…

Kategori:
Agents that produce neuromuscular block (indirect)AmebicidesAminoglycoside Antibacterials +8
Target Protein:
Ornithine decarboxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Genipin DB19124
small molecule | CAS: 6902-77-8

Genipin is under investigation in clinical trial NCT05755750 (Intratendinous Genipin Injection in Horses With Tendon Injuries).

Kategori:
AdhesivesCholagogues and CholereticsCycloparaffins +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Genistein DB01645
small molecule | CAS: 446-72-0

An isoflavonoid derived from soy products. It inhibits protein-tyrosine kinase and topoisomerase-II (DNA topoisomerases, type II) activity and is used as an antineoplastic and antitumor agent. Experimentally, it has been shown to induce G2 phase arrest in hum…

Kategori:
Anticarcinogenic AgentsAntineoplastic AgentsBCRP/ABCG2 Inhibitors +31
Target Protein:
Estrogen receptor betaNuclear receptor coactivator 1Estrogen receptor +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentamicin Approved DB00798
small molecule | CAS: 1403-66-3

Gentamicin is a bactericidal aminoglycoside that was discovered and isolated from _Micromonospora purpurea_ in 1963.[A234349] It is one of the most frequently prescribed aminoglycosides due to its spectrum of activity, low cost, and availability.[A234339,A234…

Kategori:
Agents that produce neuromuscular block (indirect)alpha-Galactosidase, antagonists & inhibitorsAminoglycoside Antibacterials +21
Target Protein:
30S ribosomal protein S1216S ribosomal RNA23S ribosomal RNA +4
Waktu ParuhOne study assessing…
Vol. Distribusi-
KlirensThe renal clearance…
Genetik -
Gentamicin C1a DB04729
small molecule | CAS: 26098-04-4

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +6
Target Protein:
30S ribosomal protein S1216S ribosomal RNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentamicin C2 DB17884
small molecule | CAS: 25876-11-3

Deskripsi belum tersedia.

Kategori:
Aminoglycoside AntibacterialsAnti-Bacterial AgentsCarbohydrates +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gentian violet cation Approved DB00406
small molecule | CAS: 7438-46-2

A dye that is a mixture of violet rosanilinis with antibacterial, antifungal, and anthelmintic properties.

Kategori:
AminesAniline CompoundsAnti-Infective Agents +7
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Genz-10850 DB04289
small molecule

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Enoyl-[acyl-carrier-protein] reductase [NADH]
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gepirone Approved DB12184
small molecule | CAS: 83928-76-1

Gepirone, an azapirone, is a pharmacologic analog of [buspirone] that acts selectively on the pre- and post-synaptic 5HT<sub>1A</sub> receptors. Although earlier clinical trials showed promising results for gepirone, its formulation as an immediate-release ta…

Kategori:
Anti-Anxiety AgentsAntidepressive AgentsCentral Nervous System Agents +12
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe apparent volume…
KlirensAfter the administr…
Genetik -
Gepotidacin DB12134
small molecule | CAS: 1075236-89-3

Gepotidacin has been used in trials studying the treatment of Gonorrhea, Infections, Bacterial, and Infections, Respiratory Tract.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +2
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Geptanolimab DB16417
biotech | CAS: 2348469-43-0

Geptanolimab is under investigation in clinical trial NCT03502629 (Clinical Trial in Chinese Patients of Relapsed and Refractory Peripheral T Cell Lymphoma (GB226)).

Target Protein:
Programmed cell death protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Geraniol Approved DB14183
small molecule | CAS: 106-24-1

Geraniol is a monoterpene that is found within many essential oils of fruits, vegetables, and herbs including rose oil, citronella, lemongrass, lavender, and other aromatic plants. It is emitted from the flowers of many species of plant and is commonly used b…

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseMonoterpenes +2
Target Protein:
Transient receptor potential cation channel subfamily M member 8
Waktu ParuhIn vitro measuremen…
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAnions +8
Target Protein:
Farnesyl pyrophosphate synthase2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthasePrenyltransferase +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gestodene DB06730
small molecule | CAS: 60282-87-3

Gestodene is a progestogen hormonal contraceptive. Products containing gestoden include Meliane, which contains 20 mcg of ethinylestradiol and 75 mcg of gestodene; and Gynera, which contains 30 mcg of ethinylestradiol and 75 mcg of gestodene.

Kategori:
Adrenal Cortex HormonesCombination Contraceptives (with Estrogen and derivatives)Contraceptive Agents, Female +30
Target Protein:
Progesterone receptor
Waktu Paruh16 to 18 hrs.
Vol. Distribusi-
Klirens-
Genetik -
Gestonorone DB13230
small molecule | CAS: 2137-18-0

Gestonorone is often mistaken for gestonorone capproate which has a different chemical structure.

Kategori:
Adrenal Cortex HormonesAntineoplastic and Immunomodulating AgentsEndocrine Therapy +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gestonorone caproate Approved DB14677
small molecule | CAS: 1253-28-7

Deskripsi belum tersedia.

Kategori:
Fused-Ring CompoundsNorpregnanesNorpregnenes +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gestrinone Approved DB11619
small molecule | CAS: 16320-04-0

Gestrinone, also known as ethylnorgestrienone, is a synthetic steroid of the 19-nortestosterone group that is marketed in Europe, Australia, and Latin America, though not the United States or Canada, and is used primarily in the treatment of endometriosis. …

Kategori:
Adrenal Cortex HormonesAntigonadotropins and Similar AgentsContraceptive Agents, Female +19
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor +3
Waktu ParuhPlasma half-life is…
Vol. Distribusi67 L [L1700]
KlirensRenal Excretion acc…
Genetik -
GET-73 DB12928
small molecule | CAS: 202402-01-5

Get 73 has been investigated for the treatment of Alcohol Dependence.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gevokizumab DB12119
biotech | CAS: 1129435-60-4

Gevokizumab has been used in trials studying the treatment of Acne Vulgaris, Osteoarthritis, Behcet's Uveitis, Pyoderma Gangrenosum, and Behcet's Disease Uveitis, among others. Gevokizumab acts as a modulator of cytokine imbalance in IL-1 mediated disease sta…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Interleukin-1 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GFH-925 DB17481
small molecule

GFH-925 is an irreversibly covalent inhibitor of KRAS G12C.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ghavamiol DB02492
small molecule

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmmonium Compounds +10
Target Protein:
Alpha-mannosidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI heptapeptide DB15070
biotech

GI heptapeptide is under investigation in clinical trial NCT01391208 (Esophageal Protocol for Detection of Neoplasia in the Digestive Tract).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-101 DB17243
biotech

GI-101 is a bi-specific fragment crystallizable region (Fc) fusion protein containing a cluster of differentiation 80 ectodomain as an N-terminal moiety and interleukin-2 variant as a C-terminal moiety conjugated with human immunoglobulin G4 Fc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-181771X DB12309
small molecule | CAS: 305366-98-7

Gski181771 X is under investigation in clinical trial NCT00600743 (Effect of a CCK-1R Agonist on Food Intake in Humans).

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-RingReceptor, Cholecystokinin A, agonists
Target Protein:
Cholecystokinin receptor type A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-4000 DB05698
biotech

A vaccine containing a heat-killed recombinant <em>Saccharomyces cerevisiae</em> yeast transfected with mutated forms of Ras, an oncogene frequently found in solid tumors, with potential immunostimulant and antitumor activity. [L112]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-5005 DB05942
biotech | CAS: 1001913-27-4

GI-5005 is GlobeImmune's lead infectious disease product from its proprietary Tarmogen active immunotherapy platform for the treatment of chronic hepatitis C infection. GI-5005 is whole, heat-killed recombinant yeast genetically modified to express HCV-specif…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensBiological Factors +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GI-6207 DB17532
biotech

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gibberellin A4 DB07815
small molecule | CAS: 468-44-0

Deskripsi belum tersedia.

Kategori:
AlkaloidsDiterpene AlkaloidsDiterpenes +2
Target Protein:
Arylacetamide deacetylase-like 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gildeuretinol DB18468
small molecule | CAS: 118139-36-9

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Giloralimab DB18862
biotech | CAS: 2226292-20-0

Giloralimab is under investigation in clinical trial NCT04807972 (Study to Evaluate Adverse Events and Change in Disease Activity When Intravenous (IV) Infusion of ABBV-927 Is Administered in Combination With IV Modified FOLFIRINOX (Mffx) With or Without IV B…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gilteritinib Approved DB12141
small molecule | CAS: 1254053-43-4

Gilteritinib, also known as ASP2215, is a small molecule part of the FLT3 tyrosine kinase inhibitors that presented a greater selectivity and potency when compared with other agents from this group.[A40036] It is a pyrazinecarboxamide derivative that showed h…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +16
Target Protein:
Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase receptor UFOALK tyrosine kinase receptor +1
Waktu ParuhThe reported median…
Vol. DistribusiThe estimated appar…
KlirensThe estimated clear…
Genetik -
Gimatecan DB06721
small molecule | CAS: 292618-32-7

Gimatecan is an orally available 7-t-butoxyiminomethyl-substituted lipophilic camptothecin derivative.

Kategori:
AlkaloidsOATP1B1/SLCO1B1 Substrates
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gimeracil Approved DB09257
small molecule | CAS: 103766-25-2

Gimeracil is an adjunct to antineoplastic therapy, used to increase the concentration and effect of the main active componets within chemotherapy regimens. Approved by the European Medicines Agency (EMA) in March 2011, Gimeracil is available in combination wi…

Kategori:
Drugs that are Mainly Renally Excreted
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]
Waktu ParuhFollowing a single …
Vol. DistribusiAlthough no intrave…
Klirens-
Genetik -
Gimsilumab DB15280
biotech | CAS: 1648796-29-5

Gimsilumab is under investigation in clinical trial NCT01357759 (Safety and Tolerability of MORAb-022 in Healthy and Rheumatoid Arthritis Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnti-Inflammatory Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gingerol DB19255
small molecule | CAS: 23513-14-6

Gingerol is under investigation in clinical trial NCT05882864 (Efficacy of Ginger Muco-bioadhesive Gel in Management of Oral Lichen Planus With Immunohistochemical Analysis).

Kategori:
AlcoholsBenzene DerivativesLipids +2
Target Protein:
Transient receptor potential cation channel subfamily A member 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginisortamab DB18863
biotech | CAS: 2390147-17-6

Ginisortamab is under investigation in clinical trial NCT04393298 (A Study to Assess the Safety, Pharmacokinetics and Anti Tumor Activity of UCB6114 Administered Intravenously to Participants With Advanced Solid Tumors).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginkgo biloba Approved DB01381
biotech | CAS: 90045-36-6

_Ginkgo biloba_ extract contains a group of terpene lactones (notably, ginkgolides and diterpenes) and ginkgo flavone glycosides (notably, ginkgetin, bilobetin, and sciadopitysin) that have antioxidant and vasoactive properties.[A232389] Most of the studies t…

Kategori:
Anti-Dementia DrugsBiological ProductsBlood Circulation +27
Target Protein:
Sodium-dependent noradrenaline transporterPhospholipase A2, membrane associatedGlycine receptor subunit alpha-1 +5
Waktu ParuhUnpublished human d…
Vol. DistribusiNo data available.
KlirensNo data available.
Genetik -
biotech

Ginkgo biloba leaf oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ginkgolide A DB06743
small molecule | CAS: 15291-75-5

Ginkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inflammatory and immunological disorders.

Kategori:
DiterpenesTerpenes
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6701–6750 dari 14063
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