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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 135 / 321
Emylcamate DB13572
small molecule | CAS: 78-28-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAnti-Anxiety AgentsCarbamates +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
EMZ702 DB05021
small molecule

EMZ702, a non-toxic agent that has strong anti-viral synergy with interferon, is an ideal candidate for combination with current standard hepatitis C treatments. EMZ702 has an excellent safety profile and the combination of EMZ702 with interferon and ribaviri…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ENA-001 DB18153
small molecule | CAS: 1380341-99-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enadenotucirev DB14873
biotech | CAS: 1402042-02-7

Enadenotucirev is under investigation in clinical trial NCT02636036 (Phase I Study of Enadenotucirev and PD-1 Inhibitor in Subjects With Metastatic or Advanced Epithelial Tumors).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enadoline DB16967
small molecule | CAS: 124378-77-4

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsCardiovascular AgentsCentral Nervous System Agents +4
Target Protein:
Kappa-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enalapril Approved DB00584
small molecule | CAS: 75847-73-3

Enalapril is a prodrug belonging to the angiotensin-converting enzyme (ACE) inhibitor drug class that works on the renin-angiotensin-aldosterone system, which is responsible for the regulation of blood pressure and fluid and electrolyte homeostasis. Enalapril…

Kategori:
ACE Inhibitors and Calcium Channel BlockersACE Inhibitors and DiureticsAgents Acting on the Renin-Angiotensin System +21
Target Protein:
Angiotensin-converting enzyme
Waktu ParuhThe average termina…
Vol. DistribusiThe volume of distr…
KlirensFollowing oral admi…
Genetik -
Enalaprilat Approved DB09477
small molecule | CAS: 76420-72-9

Enalaprilat is the active metabolite of the orally available pro-drug, [enalapril]. Used in the treatment of hypertension, enalapril is an ACE inhibitor that prevents Angiotensin Converting Enzyme (ACE) from transforming angiotensin I into angiotensin II. As …

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing angioedemaAgents causing hyperkalemia +15
Target Protein:
Angiotensin-converting enzymeB1 bradykinin receptor
Waktu Paruh11 hr
Vol. Distribusi-
KlirensThe disposition of …
Genetik -
Enalkiren DB03395
small molecule | CAS: 113082-98-7

Deskripsi belum tersedia.

Kategori:
Agents Acting on the Renin-Angiotensin SystemAmino Acids, Peptides, and ProteinsEnzyme Inhibitors +4
Target Protein:
Renin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1912424-97-5

Enapotamab vedotin is under investigation in clinical trial NCT02988817 (Enapotamab Vedotin (Humax-axl-adc) Safety Study in Patients With Solid Tumors).

Kategori:
Antibody-drug Conjugates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enarodustat DB14985
small molecule | CAS: 1262132-81-9

Enarodustat is under investigation in clinical trial NCT02581124 (Study to Evaluate Effect of Lapatinib on Pharmacokinetics of JTZ-951 in Subjects With End-stage Renal Disease).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsPeptides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enasidenib Approved DB13874
small molecule | CAS: 1446502-11-9

Enasidenib is an orally available treatment for the treatment of adult patients with relapsed or refractory acute myeloid leukemia (AML) with specific mutations in the isocitrate dehydrogenase 2 (IDH2) gene, which is a recurrent mutation detected in 12-20% of…

Kategori:
AminesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +62
Target Protein:
Isocitrate dehydrogenase [NADP] cytoplasmicIsocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrial +2
Waktu ParuhEnasidenib has a te…
Vol. DistribusiThe mean volume of …
KlirensEnasidenib has a me…
Genetik -
Enavogliflozin DB18970
small molecule | CAS: 1415472-28-4

Enavogliflozin is under investigation in clinical trial NCT06399835 (Enavogliflozin vs. Pioglitazone on Glucose and Atherosclerosis).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
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Genetik -
ENB-003 DB17340
small molecule

ENB-003 is a selective and potent inhibitor of the endothelin B receptor (ETBR) being investigated for cancer.

Waktu Paruh-
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Enbucrilate DB12358
small molecule | CAS: 6606-65-1

Enbucrilate is under investigation in clinical trial NCT02468206 (Secondary Prophylaxis of Gastric Variceal Bleed).

Kategori:
Acids, AcyclicAcrylatesCompounds used in a research, industrial, or household setting +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encainide Approved DB01228
small molecule | CAS: 66778-36-7

All drug products containing encainide hydrochloride. Encainide hydrochloride, formerly marketed as Enkaid capsules, was associated with increased death rates in patients who had asymptomatic heart rhythm abnormalities after a recent heart attack. The manufac…

Kategori:
AmidesAminesAnilides +13
Target Protein:
Sodium channel protein type 5 subunit alpha
Waktu Paruh1-2 hours
Vol. Distribusi-
Klirens-
Genetik -
Encaleret DB18096
small molecule | CAS: 787583-71-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmines +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encenicline DB11726
small molecule | CAS: 550999-75-2

Encenicline has been investigated for the treatment of Cognition, Schizophrenia, Alzheimer's Disease, Cardiac Repolarization, and Central Nervous System Diseases.

Kategori:
Nicotinic AgonistsSulfur Compounds
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enclomiphene DB06735
small molecule | CAS: 15690-57-0

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsClomiphene +11
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encorafenib Approved DB11718
small molecule | CAS: 1269440-17-6

Encorafenib, also known as _BRAFTOVI_, is a kinase inhibitor. Encorafenib inhibits BRAF gene, which encodes for B-raf protein, which is a proto-oncogene involved in various genetic mutations.[L12216] This protein plays a role in regulating the MAP kinase/E…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +47
Target Protein:
Serine/threonine-protein kinase B-rafG1/S-specific cyclin-D1RAF proto-oncogene serine/threonine-protein kinase +7
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent cleara…
Genetik -
Endostar DB11727
biotech

Endostar is under investigation for the treatment of Nasopharyngeal Carcinoma. Endostar has been investigated for the treatment of Non-small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endostatin DB06423
biotech | CAS: 187888-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
72 kDa type IV collagenaseMatrix metalloproteinase-9Collagenase 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endothelin-1 DB12652
biotech | CAS: 117399-94-7

Endothelin 1 is under investigation in clinical trial NCT00745693 (The Effects of Diesel Exhaust Inhalation on Vascular Function - the Role of Endothelin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsEndothelin-1, antagonists & inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endralazine DB13435
small molecule | CAS: 39715-02-1

Deskripsi belum tersedia.

Kategori:
Antihypertensive AgentsArteriolar Smooth Muscle, Agents Acting OnCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eneboparatide DB18207
biotech | CAS: 1349298-00-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enecadin DB13032
small molecule | CAS: 259525-01-4

Enecadin has been investigated for the treatment of Stroke.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Enflurane Approved DB00228
small molecule | CAS: 13838-16-9

Enflurane is a halogenated inhalational anesthetic initially approved by the FDA in 1972. Since this date, it has been withdrawn from the US market.[L13646,L13649] Unlike its other inhalational anesthetic counterparts including [isoflurane] and [halothane], e…

Kategori:
Agents that reduce seizure thresholdAnestheticsAnesthetics, General +8
Target Protein:
GABA(A) ReceptorVoltage-dependent calcium channelGlycine receptor subunit alpha-1 +4
Waktu Paruh-
Vol. DistribusiEnflurane distribut…
Klirens-
Genetik -
Enfortumab vedotin Approved DB13007
biotech | CAS: 1346452-25-2

Enfortumab vedotin is an antibody-drug conjugate used in the treatment of patients with advanced, treatment-resistant urothelial cancers.[L10836] It is comprised of a fully human monoclonal antibody targeted against Nectin-4 and a microtubule-disrupting chemo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Nectin-4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimated stead…
KlirensThe mean clearance …
Genetik -
Enfuvirtide Approved DB00109
biotech | CAS: 159519-65-0

Enfuvirtide is a 36 amino acid biomimetic peptide that is structurally similar to the HIV proteins that are responsible for the fusion of the virus to cell membranes and subsequent intracellular uptake. The first agent in the novel class of antiretroviral dru…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +31
Target Protein:
Envelope glycoprotein
Waktu Paruh3.8 +/- 0.6 hrs
Vol. Distribusi* 5.5 ± 1.1 L
Klirens* 24.8 +/- 4.1 mL/h…
Genetik -
biotech | CAS: 2567881-77-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Englitazone DB14035
small molecule | CAS: 109229-58-5

Englitazone is a hypoglycemic agent.

Kategori:
Blood Glucose Lowering AgentsHeterocyclic Compounds, Fused-RingPyrans +2
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2417199-08-5

Englumafusp alfa is under investigation in clinical trial NCT04077723 (A Study to Evaluate the Safety, Pharmacokinetics and Preliminary Anti-tumor Activity of Englumafusp Alfa in Combination With Obinutuzumab and in Combination With Glofitamab Following a Pre…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibomal DB13229
small molecule | CAS: 125-55-3

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, GeneralNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eniluracil DB03516
small molecule | CAS: 59989-18-3

Eniluracil, which was previously under development by GlaxoSmithKline (GSK), is being developed by Adherex to enhance the therapeutic value and effectiveness of 5-fluorouracil (5-FU), one of the world’s most widely-used oncology agents. 5-FU is widely used i…

Kategori:
Enzyme InhibitorsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Aldehyde oxidaseXanthine dehydrogenase/oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-1198 DB05959
small molecule | CAS: 864668-87-1

Deskripsi belum tersedia.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Hypoxia-inducible factor 1-alphaTumor necrosis factor receptor superfamily member 11ASignal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-981693 DB16891
small molecule | CAS: 934353-76-1

Deskripsi belum tersedia.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoblituzumab DB15017
biotech | CAS: 1353485-38-7

Enoblituzumab is under investigation in clinical trial NCT02982941 (Enoblituzumab (MGA271) in Children With B7-H3-expressing Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enobosarm DB12078
small molecule | CAS: 841205-47-8

Enobosarm has been used in trials studying the treatment of Stress Urinary Incontinence and Triple Negative Breast Cancer.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enokizumab DB05555
biotech | CAS: 909875-08-7

A humanized immunoglobulin G1k anti-interleukin-9 mAb.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enoxacin Approved DB00467
small molecule | CAS: 74011-58-8

A broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Enoximone Approved DB04880
small molecule | CAS: 77671-31-9

Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the …

Kategori:
Cardiac Stimulants Excl. Cardiac GlycosidesCardiac TherapyCardiotonic Agents +10
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu Paruh4-10 hours
Vol. Distribusi-
Klirens-
Genetik -
Enoxolone DB13089
small molecule | CAS: 471-53-4

Enoxolone (glycyrrhetic acid) has been investigated for the basic science of Apparent Mineralocorticoid Excess (AME).

Kategori:
Anti-Inflammatory AgentsCicatrizantsDermatologicals +4
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enpatoran DB16501
small molecule | CAS: 2101938-42-3

Enpatoran (M5049) was under investigation in clinical trials for various conditions. It was investigated for systemic lupus erythematosus and cutaneous lupus erythematosus in completed trials (NCT04647708 and NCT05162586) and in a recruiting trial (NCT0554032…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enprofylline Approved DB00824
small molecule | CAS: 41078-02-8

Enprofylline is a derivative of theophylline which shares bronchodilator properties. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of cerebrovascular insufficiency, sickle cell disease, and diabetic neuropathy. L…

Kategori:
Adenosine A2 Receptor AntagonistsAlkaloidsAnti-Asthmatic Agents +11
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidaseAdenosine receptor A2b +4
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
Enprostil DB13824
small molecule | CAS: 73121-56-9

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAutacoids +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enrasentan DB06460
small molecule | CAS: 167256-08-8

Deskripsi belum tersedia.

Kategori:
Endothelin Receptor AntagonistsIndenes
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6701–6750 dari 16004
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