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11778

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11778 (100.0%)

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Halaman 134 / 236
biotech | CAS: 1939139-26-0

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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Genetik -
Lanadelumab Approved DB14597
biotech | CAS: 1426055-14-2

Lanadelumab, also known as DX-2930, is a human IgG1 monoclonal antibody designed for subcutaneous self-injection.[L4538] It is a fully human immunoglobulin, k-light-chain made in recombinant Chinese Hamster Ovary cells.[L4537] It has been granted priority rev…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Plasma kallikrein
Waktu ParuhLanadelumab has a h…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Lanatoside C DB13467
small molecule | CAS: 17575-22-3

Deskripsi belum tersedia.

Kategori:
CarbohydratesCardanolidesCardenolides +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Landipirdine DB16214
small molecule | CAS: 1000308-25-7

Landipirdine is under investigation in clinical trial NCT02258152 (SYN120 Study to Evaluate Its Safety, Tolerability and Efficacy in Parkinson's Disease Dementia (SYNAPSE)).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT2 Receptor Antagonists +3
Target Protein:
5-hydroxytryptamine receptor 65-hydroxytryptamine receptor 2A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Landogrozumab DB11862
biotech | CAS: 1391726-30-9

Landogrozumab has been used in trials studying the treatment of Advanced Cancer, Muscular Atrophy, and Pancreatic Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanifibranor DB14801
small molecule | CAS: 927961-18-0

Lanifibranor is under investigation in clinical trial NCT03008070 (Phase 2b Study in NASH to Assess IVA337).

Kategori:
AmidesHeterocyclic Compounds, Fused-RingSulfones +2
Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor deltaPeroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanimostim DB06559
small molecule | CAS: 117276-75-2

Deskripsi belum tersedia.

Waktu Paruh-
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Laninamivir DB12791
small molecule | CAS: 203120-17-6

Laninamivir has been used in trials studying the treatment of Influenza.

Kategori:
Acids, AcyclicAmidinesAmino Sugars +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laniquidar DB12799
small molecule | CAS: 197509-46-9

Laniquidar has been used in trials studying the treatment of Breast Cancer.

Kategori:
Carbon RadioisotopesDrug Resistance, MultipleHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Phosphatidylcholine translocator ABCB4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanolin Approved DB11112
small molecule | CAS: 8006-54-0

Lanolin is a yellow fat obtained from sheep's wool. It is used as an emollient, cosmetic, and pharmaceutic aid [L2580]. The US federal code of regulations states that lanolin in the concentration range of 12-50% may be included in over the counter skin ointme…

Kategori:
Basic Ointments and ProtectantsCompounds used in a research, industrial, or household settingCosmetics +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lanolin alcohols Approved DB14181
small molecule | CAS: 8027-33-6

Lanolin alcohols are a complex combination of organic alcohols obtained by the hydrolysis of lanolin. It is administered as an ointment base with topical insulin and has shown to be antagonistic to wound healing. It is commonly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
Waktu Paruh-
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Lanopepden DB11912
small molecule | CAS: 1152107-25-9

Lanopepden has been used in trials studying the treatment of Pneumonia, Infections, Bacterial, Skin Diseases, Infectious, and Skin Infections, Bacterial.

Kategori:
AminesAnti-Bacterial AgentsEnzyme Inhibitors +2
Target Protein:
Peptide deformylase
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lanosterol DB03696
small molecule | CAS: 79-63-0

Deskripsi belum tersedia.

Kategori:
CholestadienesCholestadienolsCholestanes +9
Target Protein:
Lanosterol synthase
Waktu Paruh-
Vol. Distribusi-
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Lanoteplase DB06245
biotech | CAS: 171870-23-8

Deskripsi belum tersedia.

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsBiological Factors +10
Target Protein:
Urokinase plasminogen activator surface receptorFibrinogen alpha chainKallikrein-1 +14
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lanraplenib DB14770
small molecule | CAS: 1800046-95-0

Lanraplenib is under investigation in clinical trial NCT03285711 (Safety and Efficacy of Filgotinib and Lanraplenib in Adults With Lupus Membranous Nephropathy (LMN)).

Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Lanreotide Approved DB06791
small molecule | CAS: 108736-35-2

Lanreotide is a drug employed in the management of acromegaly (a hormonal condition caused by excess growth hormone) in addition to symptoms caused by neuroendocrine tumors, especially carcinoid syndrome. This drug is a long-acting analog of the drug somatost…

Kategori:
AcromegalyAmino Acids, Peptides, and ProteinsAntineoplastic Agents +22
Target Protein:
Somatostatin receptor type 2Somatostatin receptor type 5
Waktu ParuhHalf-life is approx…
Vol. DistribusiEstimated Volume of…
KlirensEstimated Clearance…
Genetik -
Lansoprazole Approved DB00448
small molecule | CAS: 103577-45-3

Lansoprazole marketed under the brand Prevacid, is a proton pump inhibitor (PPI) and is structurally classified as a substituted benzimidazole.[A177065] It reduces gastric acid secretion by targeting gastric H,K-ATPase pumps and is thus effective at promoting…

Kategori:
Acid ReducersAlimentary Tract and MetabolismAnti-Ulcer Agents +39
Target Protein:
Potassium-transporting ATPase alpha chain 1Microtubule-associated protein tau
Gen Terkait:
CYP2C19 CYP2C19 ABCB1
Waktu ParuhOne source reports …
Vol. DistribusiThe apparent volume…
KlirensThe reported cleara…
Genetik 3 Varian
small molecule | CAS: 131926-99-3

Deskripsi belum tersedia.

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesBenzimidazolesHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lanthanum carbonate Approved DB06792
small molecule | CAS: 587-26-8

Lanthanum carbonate is a phosphate binder marketed under the trade name _Fosrenol_ by Shire Pharmaceuticals. It is a large pill that requires thorough chewing to avoid choking and other gastrointestinal adverse effects. It is used to treat elevated phosphate …

Kategori:
Drugs for Treatment of Hyperkalemia and HyperphosphatemiaElementsKidney Failure, Chronic +6
Target Protein:
Phosphate
Waktu ParuhThe elimination hal…
Vol. Distribusi-
KlirensIn healthy voluntee…
Genetik -
small molecule | CAS: 16096-89-2

Deskripsi belum tersedia.

Kategori:
Metal cationsPhosphate BinderPhosphate Chelating Activity
Waktu Paruh-
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Lapachone DB11948
small molecule | CAS: 4707-32-8

Lapachone has been used in trials studying the treatment of Cancer, Carcinoma, Advanced Solid Tumors, Head and Neck Neoplasms, and Carcinoma, Squamous Cell.

Kategori:
Anti-Infective AgentsAnti-Retroviral AgentsAntiviral Agents +6
Target Protein:
DNA topoisomerase 1Retinol-binding protein 3
Waktu Paruh-
Vol. Distribusi-
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Lapaquistat DB16215
small molecule | CAS: 189059-71-0

Lapaquistat is under investigation in clinical trial NCT00256178 (Efficacy of Lapaquistat Acetate and Simvastatin in Subjects With Primary Dyslipidemia.).

Kategori:
AzepinesFarnesyl-Diphosphate Farnesyltransferase, antagonists & inhibitors
Waktu Paruh-
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Genetik -
Lapatinib Approved DB01259
small molecule | CAS: 231277-92-2

Lapatinib is an anti-cancer drug developed by GlaxoSmithKline (GSK) as a treatment for solid tumours such as breast and lung cancer. It was approved by the FDA on March 13, 2007, for use in patients with advanced metastatic breast cancer in conjunction with t…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +22
Target Protein:
Epidermal growth factor receptorEukaryotic elongation factor 2 kinaseReceptor tyrosine-protein kinase erbB-2
Gen Terkait:
HLA-DQA1 HLA-DRB1 HLA-DQB1 +1
Waktu ParuhSingle-dose termina…
Vol. Distribusi-
Klirens-
Genetik 4 Varian
Lapuleucel-t DB19117
biotech | CAS: 845680-07-1

Deskripsi belum tersedia.

Kategori:
Biological ProductsComplex MixturesVaccines
Waktu Paruh-
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Lapyrium Approved DB09376
small molecule | CAS: 109260-82-4

Lapyrium is a quaternary ammonium cation used as a surfactant, antistatic agent, and biocide in various cosmetic products [A19426]. It is commonly found formulated as lapyrium chloride.

Kategori:
Pyridines
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Laquinimod DB06685
small molecule | CAS: 248281-84-7

Laquinimod is an immunomodulator developed by Active Biotech and produced by Teva Pharmaceutical Industries. It is currently under development in phase III trials for treatment of multiple sclerosis as an oral therapy, like fingolimod. It has been shown to re…

Kategori:
Cytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 SubstratesCytochrome P-450 Substrates +3
Target Protein:
Transcription factor RelBNuclear factor NF-kappa-B p105 subunitNuclear factor NF-kappa-B p100 subunit +3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Larazotide DB05645
small molecule | CAS: 258818-34-7

An octapeptide inhibitor of paracellular permeability whose structure is derived from a protein (zonula occludens toxin) secreted by Vibrio cholerae for treatment of Coeliac disease.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Target Protein:
Haptoglobin
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Larcaviximab DB17775
biotech | CAS: 1792982-56-9

Deskripsi belum tersedia.

Waktu Paruh-
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Largemouth bass Approved DB10976
biotech

Largemouth bass allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
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Laromustine DB05817
small molecule | CAS: 173424-77-6

VNP40101M is a novel alkylating agent that has been used in trials studying the treatment of Leukemia, Lymphoma, Lung Cancer, Small Intestine Cancer, and Myelodysplastic Syndromes, among others.

Kategori:
AmidesSulfonesSulfur Compounds
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Laropiprant Approved DB11629
small molecule | CAS: 571170-77-9

Laropiprant is an ingredient in the EMA-withdrawn product Pelzont.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Prostaglandin E2 receptor EP2 subtype3-hydroxy-3-methylglutaryl-coenzyme A reductaseThromboxane A2 receptor +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Larotrectinib Approved DB14723
small molecule | CAS: 1223403-58-4

Larotrectinib is an orally administered inhibitor of tropomyosin receptor kinase (Trk), a receptor tyrosine kinase activated by neurotrophins which is mutated in a variety of cancer cell types and plays an important role in tumor cell growth and survival.[L49…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +8
Target Protein:
High affinity nerve growth factor receptorBDNF/NT-3 growth factors receptorNT-3 growth factor receptor
Waktu ParuhIn healthy subjects…
Vol. DistribusiFollowing intraveno…
KlirensThe mean clearance …
Genetik -
Larsucosterol DB18079
small molecule | CAS: 884905-07-1

Deskripsi belum tersedia.

Kategori:
CholestanesCholestenesFused-Ring Compounds +5
Waktu Paruh-
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Lartesertib DB19045
small molecule | CAS: 2495096-26-7

Lartesertib is under investigation in clinical trial NCT06433219 (Tuvusertib Combined With Niraparib or Lartesertib in Participants With Epithelial Ovarian Cancer (Ddriver EOC 302)).

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biotech | CAS: 2425817-08-7

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
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LAS-191954 DB17816
small molecule | CAS: 1403947-26-1

Deskripsi belum tersedia.

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Lasmiditan Approved DB11732
small molecule | CAS: 439239-90-4

Lasmiditan is an oral medication used in the termination of migraine headaches that was first approved for use in the United States in October 2019.[L9338,L9356] It was also approved by the European Commission on August 17, 2022.[L43997] Traditionally, the…

Kategori:
AmidesAnalgesicsAntidepressive Agents +17
Target Protein:
5-hydroxytryptamine receptor 1F
Waktu ParuhThe mean eliminatio…
Vol. DistribusiLasmiditan has been…
Klirens-
Genetik -
Lasofoxifene Approved DB06202
small molecule | CAS: 180916-16-9

Lasofoxifene is a non-steroidal 3rd generation selective estrogen receptor modulator (SERM) that selectively binds to both ER? and ER? with high affinity. It is a naphthalene derivative marketed for prevention and treatment of osteoporosis and for the treatme…

Kategori:
Genito Urinary System and Sex HormonesNaphthalenesSelective Estrogen Receptor Modulators +1
Target Protein:
Fusion glycoprotein F0Estrogen receptorEstrogen receptor beta +1
Waktu ParuhElimination half-li…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Latamoxef Approved DB04570
small molecule | CAS: 64952-97-2

Latamoxef is a broad- spectrum beta-lactam antibiotic similar in structure to the cephalosporins except for the substitution of an oxaazabicyclo moiety for the thiaazabicyclo moiety of certain cephalosporins. It has been proposed especially for the meningitid…

Kategori:
AmidesAnti-Bacterial AgentsAnti-Infective Agents +10
Target Protein:
Peptidoglycan synthase FtsIPenicillin-binding protein 3Penicillin-binding protein 1A +2
Waktu Paruh1.6 hours
Vol. Distribusi8.51 L
Klirens-
Genetik -
Latanoprost Approved DB00654
small molecule | CAS: 130209-82-4

Latanoprost is a prodrug analog of prostaglandin F2 alpha that is used to treat elevated intraocular pressure (IOP). It was initially approved by the FDA in 1998. Latanoprost is the first topical prostaglandin F2 alpha analog used for glaucoma treatment.[A184…

Kategori:
Antiglaucoma Preparations and MioticsAntihypertensive AgentsAutacoids +18
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe systemic cleara…
Genetik -
Latanoprost acid Approved DB19360
small molecule | CAS: 41639-83-2

Deskripsi belum tersedia.

Kategori:
AutacoidsBiological FactorsEicosanoids +6
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Latanoprostene bunod Approved DB11660
small molecule | CAS: 860005-21-6

Latanoprostene Bunod has been used in trials studying the treatment of Glaucoma, Ocular Hypertension, Open-Angle Glaucoma, Open Angle Glaucoma, and Intraocular Pressure. As of November 2, 2017 the FDA approved Bausch + Lomb's Vyzulta (latanoprostene bunod …

Kategori:
Antiglaucoma Preparations and MioticsAutacoidsBiological Factors +12
Target Protein:
Prostaglandin F2-alpha receptor
Waktu ParuhThe half-life after…
Vol. DistribusiUnfortunately there…
KlirensSince latanoprost a…
Genetik -
Latozinemab DB16978
biotech

Deskripsi belum tersedia.

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Latrepirdine DB11725
small molecule | CAS: 3613-73-8

Latrepirdine has been investigated for the treatment of Alzheimer's Disease and Huntington's Disease.

Kategori:
Alzheimer DiseaseHeterocyclic Compounds, Fused-Ring
Target Protein:
5-hydroxytryptamine receptor 6Histamine H1 receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Latrunculin A DB02621
small molecule | CAS: 76343-93-6

Latrunculin A is an actin binding macrolide purified from the red sea sponge Latrunculia magnifica. It is under investigation for the treatment of cancer. It disrupts actin polymerization, prevents mitotic spindle formation and thus cell replication.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleGelsolinIota toxin component Ia
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Latrunculin B DB08080
small molecule | CAS: 76343-94-7

Latrunculin B is a 14-membered macrolide attached to 2-thiazolidinone moiety, isolated from Red Sea sponge _Latrunculia magnifica_.

Kategori:
PoriferaSulfur CompoundsThiazoles
Target Protein:
Actin, alpha skeletal muscleMyocardin-related transcription factor AProtein spire homolog 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Lauric acid Approved DB03017
small molecule | CAS: 143-07-7

Lauric acid is an inexpensive, non-toxic and safe to handle compound often used in laboratory investigations of melting-point depression. Lauric acid is a solid at room temperature but melts easily in boiling water, so liquid lauric acid can be treated with v…

Kategori:
Fatty AcidsLipids
Target Protein:
Toll-like receptor 4LactotransferrinPhospholipase A2, membrane associated +18
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Laurocapram Approved DB17308
small molecule | CAS: 59227-89-3

Deskripsi belum tersedia.

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Genetik -
small molecule | CAS: 112-16-3

Deskripsi belum tersedia.

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Laurus nobilis Approved DB10670
biotech

Laurus nobilis allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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