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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 134 / 272
GSK-3117391 DB15440
small molecule | CAS: 1018673-42-1

GSK-3117391 is under investigation in clinical trial NCT02965599 (Efficacy, Safety, Tolerability, Pharmacokinetics and Pharmacodynamics of GSK3117391 in Subjects With Rheumatoid Arthritis).

Waktu Paruh-
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GSK-356278 DB12542
small molecule | CAS: 720704-34-7

Gsk356278 has been used in trials studying the treatment and basic science of Anxiety Disorders, Huntington Disease, Depressive Disorder, Huntingtons Disease, and Depressive Disorder, Major, among others.

Kategori:
OxazolesSulfur Compounds
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A3',5'-cyclic-AMP phosphodiesterase 4D3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
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GSK-364735 DB13119
small molecule | CAS: 863434-13-3

GSK-364735 (Naphthyridinone) has been used in trials studying the treatment of HIV-1 Infection and Infection, Human Immunodeficiency Virus.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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GSK-376501 DB12654
small molecule | CAS: 1010412-80-2

GSK376501 has been used in trials studying the treatment and diagnostic of Type 2 Diabetes Mellitus.

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GSK-690693 DB12745
small molecule | CAS: 937174-76-0

GSK690693 has been used in trials studying the treatment of Tumor, CANCER, and Lymphoma.

Kategori:
Oxazoles
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
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GSK-923295 DB06097
small molecule

GSK-923295 is a small-molecule inhibitor of the mitotic kinesin centromere-associated protein E (CENP-E), and the third novel drug candidate to arise from Cytokinetics' broad strategic alliance with GlaxoSmithKline (GSK). GSK-923295 demonstrated a broad spect…

Target Protein:
Centromere-associated protein E
Waktu Paruh-
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GSK-945237 DB15345
small molecule | CAS: 944406-54-6

GSK-945237 is under investigation in clinical trial NCT01039610 (A Single Center Four Part Study in Healthy Adult Subjects to Evaluate: the Safety, Tolerability and Pharmacokinetics of a Single Oral Dose and Repeat Escalating Oral Doses of GSK945237; the Effe…

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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GSK159797 DB05043
small molecule

GSK159797 ('797) is an inhaled, longer-acting Beta2 agonist developed for the treatment of respiratory disease such as asthma and COPD.

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GSK2245035 DB16076
small molecule | CAS: 1207629-49-9

GSK2245035 is under investigation in clinical trial NCT02833974 (Effect of the GSK2245035 on the Allergen-induced Asthmatic Response).

Kategori:
Heterocyclic Compounds, Fused-RingPurines
Target Protein:
Toll-like receptor 7
Waktu Paruh-
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GSK2256098 DB16106
small molecule | CAS: 1224887-10-8

GSK2256098 is under investigation in clinical trial NCT02523014 (Vismodegib and FAK Inhibitor GSK2256098 in Treating Patients With Progressive Meningiomas).

Kategori:
AminesHydroxy AcidsHydroxylamines +1
Target Protein:
Focal adhesion kinase 1
Waktu Paruh-
Vol. Distribusi-
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GSK232802 DB16110
small molecule | CAS: 843661-24-5

GSK232802 is under investigation in clinical trial NCT00604825 (Treatment of Hot Flashes/flushes in Postmenopausal Women (WARM Study)).

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GSK2798745 DB16033
small molecule | CAS: 1419609-94-1

GSK2798745 is under investigation in clinical trial NCT03372603 (A Study to Assess the Effectiveness and Side Effects of GSK2798745 in Participants With Chronic Cough).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
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GT 389-255 DB05894
small molecule

Peptimmune’s lead product GT 389-255, is a novel lipase inhibitor and fat binding hydrogel polymer conjugate for the treatment of obesity which has completed single and multiple ascending dose (SAD and MAD) Phase I trials. It is expected to block fat absorpti…

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GT-AS DB17883
biotech

GT-AS recombinant adeno-associated virus serotype 9 vector containing the transgene UBE3A encoding for ubiquitin protein ligase E3A/E6-AP.

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GTA002 DB17187
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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GTB-3550 DB18494
biotech

GTB-3550 is a single-chain, tri-specific scFv recombinant fusion protein conjugate composed of the variable regions of the heavy and light chains of anti-CD16 and anti-CD33 antibodies and a modified form of Interleukin 15 (IL-15).

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GTI-2040 DB15030
biotech | CAS: 236391-66-5

GTI-2040 is under investigation in clinical trial NCT00084643 (GTI-2040, Oxaliplatin, and Capecitabine in Treating Patients With Locally Advanced or Metastatic Colorectal Cancer or Other Solid Tumors).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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GTS-21 DB05708
small molecule | CAS: 148372-04-7

GTS-21 (also known as DMBX-A), is a novel, small-molecule, orally active and selective alpha-7 nicotinic acetylcholine (nACh) receptor agonist that has demonstrated memory and cognition enhancement activity in human clinical trials. Athenagen licensed the exc…

Kategori:
Benzene DerivativesCholinergic AgentsCholinergic Agonists +5
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
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GTX-102 DB16981
biotech

GTX-102 is an antisense oligonucleotide designed to target and inhibit the expression of UBE3A-AS. It is being investigated for the treatment of Angelman Syndrome.[L46772]

Kategori:
Antisense Oligonucleotide Specific to the Antisense Transcript of UBE3A
Waktu Paruh-
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GTX-758 DB14969
small molecule | CAS: 938067-78-8

GTX-758 is under investigation in clinical trial NCT01420861 (GTx-758 on Serum Prostate-specific Antigen (PSA) in Men With Castrate Resistant Prostate Cancer).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Guacetisal DB13538
small molecule | CAS: 55482-89-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +18
Waktu Paruh-
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Guaiacol Approved DB11359
small molecule | CAS: 90-05-1

Guaiacol is an agent thought to have disinfectant properties and used as an expectorant. Guaiacol is a phenolic natural product first isolated from Guaiac resin and the oxidation of lignin. Guaiacol is also present in wood smoke, as a product of pyrolysis of …

Kategori:
Benzene DerivativesCatecholsEthers +4
Target Protein:
Albumin
Waktu Paruh-
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Guaiazulen DB13329
small molecule | CAS: 489-84-9

Deskripsi belum tersedia.

Kategori:
CycloheptanesCycloparaffinsOphthalmologicals +5
Waktu Paruh-
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Guaifenesin Approved DB00874
small molecule | CAS: 93-14-1

Guaifenesin possesses a storied history, having been originally formally approved by the US FDA in 1952 and continues to be one of very few - if not perhaps the only drug that is readily available and used as an expectorant [F4525]. Since that time the agent …

Kategori:
Benzene DerivativesCatecholsCough and Cold Preparations +6
Target Protein:
NMDA receptor
Waktu ParuhThe half-life in pl…
Vol. DistribusiThe geometric mean …
KlirensThe mean clearance …
Genetik -
Guanazodine DB13604
small molecule | CAS: 32059-15-7

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
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Guanfacine Approved DB01018
small molecule | CAS: 29110-47-2

Guanfacine, or BS 100-141,[A189838,A189841] is a selective alpha-A2 adrenergic receptor agonist initially indicated for the treatment of hypertension[L11274] but is now indicated as an extended release tablet for the treatment of ADHD.[L11277] Guanfacine was …

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-2 Receptor Agonists +26
Target Protein:
Alpha-2A adrenergic receptorAlpha-2B adrenergic receptor
Waktu ParuhGuanfacine has a ha…
Vol. DistribusiGuanfacine has a vo…
KlirensGuanfacine has a to…
Genetik -
Guanidine Approved DB00536
small molecule | CAS: 113-00-8

A strong organic base existing primarily as guanidium ions at physiological pH. It is found in the urine as a normal product of protein metabolism. It is also used in laboratory research as a protein denaturant. (From Martindale, the Extra Pharmacopoeia, 30th…

Kategori:
Acetylcholine Releasing AgentAmidinesGuanidines +7
Target Protein:
Aldehyde dehydrogenase, mitochondrialRibonuclease pancreaticDNA +4
Waktu Paruh7-8 hours
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Trypsin-3
Waktu Paruh-
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Guanine DB02377
small molecule | CAS: 73-40-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-RingPurinesPurinones +1
Target Protein:
GTP cyclohydrolase 1Purine nucleoside phosphorylasePurine nucleoside phosphorylase 2 +2
Waktu Paruh-
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Guanoclor DB13779
small molecule | CAS: 5001-32-1

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
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Genetik -
Guanosine DB02857
small molecule | CAS: 118-00-3

Guanosine is a nucleoside comprising guanine attached to a ribose (ribofuranose) ring via a ?-N9-glycosidic bond. Guanosine can be phosphorylated to become GMP (guanosine monophosphate), cGMP (cyclic guanosine monophosphate), GDP (guanosine diphosphate) and G…

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
DNA polymerase catalytic subunitDNA polymerase catalytic subunitPurine nucleoside phosphorylase +2
Waktu Paruh-
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small molecule | CAS: 117-68-0

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
RibonucleaseBifunctional protein PyrR
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenylosuccinate synthetaseBifunctional (p)ppGpp synthase/hydrolase RelA
Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 33503-72-9

Guanosine tetraphosphate is a guanine nucleotide containing four phosphate groups. Two phosphate groups are esterified to the sugar moiety in the 5' position and the other two in the 2' or 3' position. This nucleotide serves as a messenger to turn off the syn…

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseXanthine phosphoribosyltransferaseGTPase Obg
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 38557-85-6

Deskripsi belum tersedia.

Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
small molecule | CAS: 130-50-7

Deskripsi belum tersedia.

Kategori:
Guanine NucleotidesHeterocyclic Compounds, Fused-RingIsomerism +5
Target Protein:
Guanyl-specific ribonuclease Sa
Waktu Paruh-
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Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
ADP-ribosylation factor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
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small molecule | CAS: 146-91-8

A guanine nucleotide containing two phosphate groups esterified to the sugar moiety. [PubChem]

Target Protein:
Protein-glutamine gamma-glutamyltransferase 2Elongation factor 1-alphaAdenylosuccinate synthetase +49
Waktu Paruh-
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Genetik -
small molecule | CAS: 85-32-5

Guanosine 5'-monophosphate. A guanine nucleotide containing one phosphate group esterified to the sugar moiety and found widely in nature. [PubChem]

Target Protein:
Hypoxanthine-guanine-xanthine phosphoribosyltransferaseDNA polymerase catalytic subunitDNA polymerase catalytic subunit +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 86-01-1

Guanosine 5'-(tetrahydrogen triphosphate). A guanine nucleotide containing three phosphate groups esterified to the sugar moiety. [PubChem]

Target Protein:
GTP cyclohydrolase 1Genome polyproteinRNA-directed RNA polymerase +18
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Guanoxabenz DB13410
small molecule | CAS: 24047-25-4

Deskripsi belum tersedia.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +2
Waktu Paruh-
Vol. Distribusi-
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Guanoxan Approved DB13211
small molecule | CAS: 2165-19-7

Guanoxan is an antihypertensive agent similar in its mechanism of action to guanethidine; may cause liver damage. Guanoxan was approved in the UK but was withdrawn from the market due to hepatotoxicity.

Kategori:
AmidinesAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +1
Waktu Paruh-
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Guar gum DB13446
small molecule | CAS: 9000-30-0

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBiological ProductsBiopolymers +10
Waktu Paruh-
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Gunagratinib DB18191
small molecule | CAS: 2211082-53-8

Deskripsi belum tersedia.

Waktu Paruh-
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Gusacitinib DB15670
small molecule | CAS: 1425381-60-7

Gusacitinib is under investigation in clinical trial NCT02550678 (A Study of the Efficacy and Safety of ASN-002 in Adult Patients With Low-risk Nodular Basal Cell Carcinoma).

Kategori:
Nitriles
Target Protein:
Tyrosine-protein kinase SYK
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Guselkumab Approved DB11834
biotech | CAS: 1350289-85-8

Guselkumab is a human immunoglobulin G1 lambda (IgG1?) monoclonal antibody that selectively blocks interleukin-23. IL-23 is an inflammatory cytokine that activates the CD4+ T-helper (Th17) cell pathway to mediate the inflammatory cascade that induces psoriati…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +12
Target Protein:
Interleukin-23 subunit alpha
Waktu ParuhMean half-life of g…
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Gusperimus DB12692
small molecule | CAS: 98629-43-7

Gusperimus has been used in trials studying the treatment of Lupus Nephritis, Wegeners Granulomatosis, and Wegener's Granulomatosis.

Kategori:
AmidinesAntibiotics, AntineoplasticAntineoplastic Agents +7
Waktu Paruh-
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GW 468816 DB05417
small molecule

GW 468816 is glycine receptor antagonist. It is designed to aid abstinence in people who have just quit smoking, delaying the time to relapse. It was undergoing phase II trials since December 2003.

Kategori:
Heterocyclic Compounds, Fused-RingReceptors, N-Methyl-D-Aspartate, antagonists & inhibitors
Target Protein:
Glycine receptor subunit alpha-1
Waktu Paruh-
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Genetik -
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