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14361

Total database: 17430
Struktur (SMILES)
9916 (69.0%)
Target
7893 (55.0%)
Genomik
112 (0.8%)
Referensi
14361 (100.0%)

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Hasil Pencarian (14361)

Halaman 133 / 288
Gantacurium DB05710
small molecule | CAS: 758669-50-0

Gantacurium chloride is a new, investigational, non-depolarizing ultra-short acting neuromuscular blocker. It is being developed by Avera Pharmaceuticals.

Kategori:
Anticholinergic AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +3
Target Protein:
Neuronal acetylcholine receptor subunit alpha-3
Waktu Paruh3.09±0.21 minutes
Vol. Distribusi-
Klirens-
Genetik -
Gantenerumab DB12034
biotech | CAS: 1043556-46-2

Alzheimer's disease (AD) is the most common cause of dementia in elderly patients, with classical histopathological hallmarks including extracellular amyloid-beta (A?) plaques and intraneuronal neurofibrillary tangles (NFTs). As the classical view of AD patho…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Target Protein:
Amyloid-beta precursor protein
Waktu ParuhGantenerumab admini…
Vol. Distribusi-
Klirens-
Genetik -
Garadacimab DB15629
biotech | CAS: 2162134-62-3

Garadacimab is under investigation in clinical trial NCT04281524 (A Clinical Study to Test the Efficacy and Safety of CSL312 on Catheter-associated Blood Clot Formation in Subjects With Cancer Who Receive Chemotherapy Through a PICC Line).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Garcinia gummi-gutta fruit is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Garden snail mucin is an animal extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garenoxacin DB06160
small molecule | CAS: 194804-75-6

Garenoxacin, a quinolone antibiotic, is being investigated for the treatment of gram-positive and gram-negative bacterial infections.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +15
Target Protein:
DNA topoisomerase 2-alphaDNA topoisomerase 2-beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Garetosmab DB16379
biotech | CAS: 2097125-54-5

Fibrodysplasia ossificans progressiva (FOP) is a rare autosomal dominant disorder of episodic, progressive heterotropic ossification. FOP is characterized by episodic inflammatory episodes, which may be precipitated by trauma, including immunizations and mino…

Target Protein:
Inhibin beta A chain
Waktu Paruh-
Vol. DistribusiGaretosmab had a st…
KlirensWhen administered a…
Genetik -
Garlic oil DB15989
biotech | CAS: 8000-78-0

Deskripsi belum tersedia.

Kategori:
AlkenesAnionsAnticarcinogenic Agents +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gartisertib DB18770
small molecule | CAS: 1613191-99-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 100040-31-1

Gastric inhibitory polypeptide is under investigation in clinical trial NCT03081676 (The Effect of GIP and GLP-1 on Insulin and Glucagon Secretion in Patients With HNF1A-diabetes Treated With or Without Sulphonylurea).

Kategori:
Amino Acids, Peptides, and ProteinsBlood Glucose Lowering AgentsGastrointestinal Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gastric intrinsic factor Approved DB09349
biotech

Intrinsic factor (IF), also known as gastric intrinsic factor (GIF), is a glycoprotein produced by the parietal cells of the stomach that is necessary for the absorption of vitamin B12 (cobalamin) later on in the small intestine. When vitamin B12 is provided …

Kategori:
Amino Acids, Peptides, and ProteinsCarbohydratesGlycoconjugates +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gatifloxacin Approved DB01044
small molecule | CAS: 112811-59-3

Gatifloxacin is an antibiotic agent and a member of the fourth-generation fluoroquinolone family. It works by inhibiting the bacterial enzymes DNA gyrase and topoisomerase IV. It was first introduced by Bristol-Myers Squibb in 1999 under the brand name Tequin…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +3
Waktu Paruh7-14 hours
Vol. Distribusi-
Klirens-
Genetik -
Gatipotuzumab DB18861
biotech | CAS: 1264737-26-9

Gatipotuzumab is under investigation in clinical trial NCT01899599 (Pankomab-gex™ Versus Placebo as Maintenance Therapy in Advanced Ovarian Cancer).

Waktu Paruh-
Vol. Distribusi-
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Gatralimab DB16528
biotech | CAS: 1826020-80-7

Gatralimab is under investigation in clinical trial NCT02389452 (Study of Safety and Efficacy of 6 Ml Synvisc-one (Hylan G-F 20) in Indian Patients With Symptomatic Osteoarthritis of Knee(s) After Initial and Repeat Treatment).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavestinel DB06741
small molecule | CAS: 153436-22-7

Highly potent and selective non-competitive antagonist acting at the strychnine-insensitive glycine binding site of the NMDA receptor-channel complex (Kd = 0.8 nM). Gavestinel displays > 1000-fold selectivity over NMDA, AMPA and kainate binding sites and is o…

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsGlycine Agents +5
Target Protein:
Glycine receptor subunit alpha-1Glycine receptor subunit alpha-2Glycine receptor subunit alpha-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Gavocabtagene autoleucel is a novel cell therapy consisting of autologous genetically engineered T cells expressing a single-domain antibody that recognizes human Mesothelin, fused to the CD3-epsilon subunit which, upon expression, is incorporated into the en…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gavorestat DB16707
small molecule | CAS: 2170729-29-8

Gavorestat is under investigation in clinical trial NCT04902781 (Clinical Benefit, Safety, PK and PD Study of AT-007 in Pediatric Subjects With Classic Galactosemia).

Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB-115 DB19204
small molecule | CAS: 678996-63-9

GB-115 is under investigation in clinical trial NCT05586789 (A Study of the Efficacy and Safety of Ranquilon Tablets in Patients With Anxiety in Neurasthenia and Adjustment Disorders).

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GB-13 DB18387
biotech

GB-13 is a genetically engineered recombinant protein consisting of an IL13Ra2-targeted genetically engineered mutant of IL-13 and PE4E, a derivative of Pseudomonas exotoxin A.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GBR-12783 DB17027
small molecule | CAS: 145428-33-7

A selective inhibitor of dopamine uptake.[A252997]

Kategori:
Dopamine AgentsDopamine AgonistsDopamine Uptake Inhibitors +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GBR-12879 DB17028
small molecule | CAS: 67469-43-6

Deskripsi belum tersedia.

Kategori:
Piperazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GC-373 DB15797
small molecule

GC-373 is a peptide aldehyde which is metabolized from the bisulfide adduct, [GC-376 free acid][A219031,A219036]. It is an inhibitor of M<sup>pro</sup> (otherwise known as 3CL<sup>pro</sup>), a viral encoded protease that cleaves and activates functional prot…

Kategori:
AmidesAmino AcidsAmino Acids, Branched-Chain +3
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1417031-79-8

GC-376 is a 3C-like protease (3CL<sup>pro</sup> or M<sup>pro</sup>) inhibitor that stops the cleavage and activation of functional viral proteins required for replication and transcription in host cells[A219036]. The compound is known as a direct acting antiv…

Kategori:
AcidsAcids, NoncarboxylicAlkalies +15
Target Protein:
Replicase polyprotein 1abReplicase polyprotein 1aReplicase polyprotein 1ab +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GCS-100 DB17566
biotech

Deskripsi belum tersedia.

Kategori:
Carbohydrates
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0134 DB17079
small molecule | CAS: 1637394-01-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0349 DB13072
small molecule | CAS: 1207360-89-1

GDC-0349 has been used in trials studying the treatment of Non-Hodgkin's Lymphoma, Solid Tumor.

Kategori:
AmidesBenzene Derivatives
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0425 DB14791
small molecule | CAS: 1627539-18-7

GDC-0425 is under investigation in clinical trial NCT01359696 (A Study Evaluating the Safety, Tolerability, and Pharmacokinetics of GDC-0425 Administered With and Without Gemcitabine in Patients With Refractory Solid Tumors or Lymphoma).

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Serine/threonine-protein kinase Chk1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0917 DB12336
small molecule | CAS: 1446182-94-0

CUDC-427 has been used in trials studying the treatment of LYMPHOMA and Solid Cancers.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDC-0927 DB14934
small molecule | CAS: 2100830-77-9

GDC-0927 is under investigation in clinical trial NCT02316509 (A Study of GDC-0927 in Postmenopausal Women With Locally Advanced or Metastatic Estrogen Receptor Positive Breast Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GDP-mannose 6-dehydrogenase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
GDP-L-fucose DB18689
small molecule | CAS: 15839-70-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gebasaxturev DB17296
biotech | CAS: 2122169-83-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gedatolisib DB11896
small molecule | CAS: 1197160-78-3

Gedatolisib has been used in trials studying the basic science and treatment of Neoplasm, Ovary Cancer, Breast Cancer, Advanced Cancer, and Endometrial Cancer, among others.

Kategori:
Enzyme InhibitorsOxazinesProtein Kinase Inhibitors
Target Protein:
Serine/threonine-protein kinase mTORPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gedivumab DB15277
biotech | CAS: 1807954-17-1

Gedivumab is under investigation in clinical trial NCT01877785 (A Study of MHAA4549A to Assess Safety And Pharmacokinetics in Healthy Volunteers).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gefapixant Approved DB15097
small molecule | CAS: 1015787-98-0

It has been estimated that 5-10% of adults globally suffer from chronic cough, which is defined as a cough lasting longer than eight weeks.[L48601] A subset of these patients remain symptomatic despite thorough investigation and treatment, termed refractory c…

Kategori:
AmidesBCRP/ABCG2 SubstratesBenzene Derivatives +8
Target Protein:
P2X purinoceptor 3P2X purinoceptor 2
Waktu ParuhThe terminal half-l…
Vol. DistribusiBased on population…
KlirensPopulation pharmaco…
Genetik -
Gefarnate DB12079
small molecule | CAS: 51-77-4

Gefarnate has been investigated for the treatment and prevention of Stomach Ulcer, Duodenal Ulcer, and Cardio-cerebrovascular Disease.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsDrugs for Acid Related Disorders +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gefitinib Approved DB00317
small molecule | CAS: 184475-35-2

Gefitinib (originally coded ZD1839) is a drug used in the treatment of certain types of cancer. Acting in a similar manner to erlotinib (marketed as Tarceva), gefitinib selectively targets the mutant proteins in malignant cells. It is marketed by AstraZeneca …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Inhibitors +25
Target Protein:
Epidermal growth factor receptor
Gen Terkait:
EGFR EGFR EGFR +1
Waktu Paruh48 hours [IV admini…
Vol. Distribusi* 1400 L [IV admini…
Klirens* 595 mL/min [IV ad…
Genetik 4 Varian
Gefurulimab DB18928
biotech | CAS: 2456407-94-4

Gefurulimab is under investigation in clinical trial NCT05556096 (Safety and Efficacy of ALXN1720 in Adults With Generalized Myasthenia Gravis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gelatin Approved DB11242
small molecule | CAS: 9000-70-8

Gelatin is a multifunctional ingredient that is used in foods, pharmaceuticals, cosmetics, and photographic films as a gelling agent, stabilizer, thickener, emulsifier, as well as film former.[A32432] As a thermoreversible hydrocolloid with a small gap bet…

Kategori:
Amino Acids, Peptides, and ProteinsBlood and Blood Forming OrgansBlood and Related Products +4
Waktu ParuhHalf-life is about …
Vol. Distribusi-
KlirensA large percentage …
Genetik -
GEM-231 DB05798
biotech | CAS: 255810-66-3

GEM231 is a second-generation antisense oligonucleotide targeting the mRNA of the R1alpha regulatory subunit of cAMP dependent protein kinase. A monoclonal antibody combined with a toxic substance that is used treat certain types of acute myeloid leukemia in …

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Target Protein:
cAMP-dependent protein kinase type II-alpha regulatory subunitcAMP-dependent protein kinase type I-alpha regulatory subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcabene DB05123
small molecule | CAS: 183293-82-5

Gemcabene is a new drug that lowers low-density lipoprotein cholesterol (LDL-C), decreases triglycerides, and raises high-density lipoprotein cholesterol (HDL-C).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemcitabine Approved DB00441
small molecule | CAS: 95058-81-4

Gemcitabine is a nucleoside analog and a chemotherapeutic agent. It was originally investigated for its antiviral effects, but it is now used as an anticancer therapy for various cancers.[A233135] Gemcitabine is a cytidine analog with two fluorine atoms repla…

Kategori:
AntimetabolitesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +23
Target Protein:
DNARibonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit +2
Gen Terkait:
RRM1
Waktu ParuhFollowing intraveno…
Vol. DistribusiIn patients with va…
KlirensFollowing intraveno…
Genetik 1 Varian
small molecule | CAS: 210829-30-4

Gemcitabine elaidate has been used in trials studying the treatment of Solid Tumor, Lung Cancer, Non-small-cell Lung Cancer, and Metastatic Pancreatic Adenocarcinoma.

Kategori:
DeoxyribonucleosidesNucleic Acids, Nucleotides, and NucleosidesNucleosides +2
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemeprost Approved DB08964
small molecule | CAS: 64318-79-2

Gemeprost is a prostaglandin E1 (PGE1) analog and antiprogestogen used for preoperative dilation of the cervix before surgical abortion. It is available as vaginal suppositories and also used in combination with the antiprogestin and mifepristone for terminat…

Kategori:
Abortifacient AgentsAbortifacient Agents, NonsteroidalAutacoids +14
Target Protein:
Prostaglandin E2 receptor EP3 subtypeProstaglandin E2 receptor EP2 subtype
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemfibrozil Approved DB01241
small molecule | CAS: 25812-30-0

Gemfibrozil is a fibric acid agent, similar to [clofibrate], used to treat Type IIb, IV, and V hyperlipidemias.[A185777,L8525] Gemfibrozil is not a first line treatment and is prescribed to patients who have not responded adequately to weight loss, diet, exer…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +53
Target Protein:
Peroxisome proliferator-activated receptor alphaLipoprotein lipaseSolute carrier organic anion transporter family member 1B1 +3
Waktu ParuhGemfibrozil has a p…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of ge…
Genetik -
Gemifloxacin Approved DB01155
small molecule | CAS: 175463-14-6

Gemifloxacin is a quinolone antibacterial agent with a broad-spectrum activity that is used in the treatment of acute bacterial exacerbation of chronic bronchitis and mild-to-moderate pneumonia. It is available in oral formulations. Gemifloxacin acts by inhib…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh7 (&plusmn; 2) hours
Vol. Distribusi* 1.66 to 12.12 L/kg
Klirens* renal cl=11.6+/- …
Genetik -
Gemigliptin DB12412
small molecule | CAS: 911637-19-9

Gemigliptin is under investigation in Type 2 Diabetes Mellitus. Gemigliptin has been investigated for the treatment of Cancer and Cisplatin Adverse Reaction.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +5
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemlapodect DB18769
small molecule | CAS: 1380329-87-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Gemogenovatucel-T is a bi-shRNA furin/Granulocyte Macrophage Colony Stimulating Factor (GMCSF) Augmented autologous tumour cell vaccine. Furin is a convertase involved in the activation of TGF?-1 and TGF?-2.[A255163] Gemogenovatucel-T is being investigated in…

Kategori:
Biological ProductsComplex MixturesVaccines +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Gemtuzumab ozogamicin Approved DB00056
biotech | CAS: 220578-59-6

Gemtuzumab ozogamicin is a recombinant humanized IgG4 kappa antibody which is conjugated with calicheamicin derivative, a cytotoxic antitumor antibiotic isolated from fermentation of Micromonospora echinospora ssp. calichensis. Gemtuzumab ozogamicin has appro…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +28
Target Protein:
Myeloid cell surface antigen CD33Low affinity immunoglobulin gamma Fc region receptor III-BLow affinity immunoglobulin gamma Fc region receptor III-A +1
Waktu ParuhIn pediatric patien…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Menampilkan 6601–6650 dari 14361
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