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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

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Hasil Pencarian (6694)

Halaman 133 / 134
Zileuton Approved DB00744
small molecule | CAS: 111406-87-2

Leukotrienes are substances that induce numerous biological effects including augmentation of neutrophil and eosinophil migration, neutrophil and monocyte aggregation, leukocyte adhesion, increased capillary permeability, and smooth muscle contraction. These …

Kategori:
Agents to Treat Airway DiseaseAmidesAnalgesics +19
Target Protein:
Polyunsaturated fatty acid 5-lipoxygenase
Waktu Paruh2.5 hours
Vol. Distribusi* 1.2 L/kg
Klirens* Apparent oral cl=…
Genetik -
Zilovertamab DB18403
biotech | CAS: 2485779-13-1

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2376463-48-6

Zilovertamab vedotin is an Antibody-drug conjugate (ADC) comprising an anti-ROR1 monoclonal antibody (UC-961), a proteolytically cleavable maleimidocaproyl-valine-citrulline-para-aminobenzoate linker (mc-vc-PAB), and a monomethyl auristatin E (MMAE) cytotoxin.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ziltivekimab DB18836
biotech | CAS: 2226654-05-1

Ziltivekimab is under investigation in clinical trial NCT06200207 (A Research Study Looking Into How Ziltivekimab Works Compared to Placebo in Participants With Heart Failure and Inflammation).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zilucoplan Approved DB15636
small molecule | CAS: 1841136-73-9

Zilucoplan is a 15 amino-acid, synthetic macrocyclic peptide. It is a complement inhibitor that works to prevent the activation of C5, which is a complement protein involved in the innate immune system to initiate inflammatory responses.[A261841] On October 1…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsBlood Proteins +5
Target Protein:
Complement C5
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe mean volume of …
KlirensNo information is a…
Genetik -
Zimelidine Approved DB04832
small molecule | CAS: 56775-88-3

Zimelidine has been banned worldwide due to serious, sometimes fatal, cases of central and/or peripheral neuropathy known as Guillain-Barré syndrome and due to a peculiar hypersensitivity reaction involving many organs including skin exanthema, flu-like sympt…

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsCytochrome P-450 CYP3A Inhibitors +16
Target Protein:
Sodium-dependent serotonin transporterAmine oxidase [flavin-containing] BAmine oxidase [flavin-containing] A
Waktu Paruh8.4 +/- 2.0 hours f…
Vol. Distribusi-
Klirens-
Genetik -
Zinc Approved DB01593
small molecule | CAS: 7440-66-6

A metallic element of atomic number 30 and atomic weight 65.38. It is a necessary trace element in the diet, forming an essential part of many enzymes, and playing an important role in protein synthesis and in cell division. Zinc deficiency is associated with…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseDiet, Food, and NutritionElements +12
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc acetate Approved DB14487
small molecule | CAS: 557-34-6

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +7
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +121
Waktu ParuhThe half-life of zi…
Vol. DistribusiA pharmacokinetic s…
KlirensIn one study of hea…
Genetik -
Zinc ascorbate Approved DB14485
small molecule | CAS: 331242-75-2

Deskripsi belum tersedia.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc chloride Approved DB14533
small molecule | CAS: 7646-85-7

Zinc chloride is a solution of ions indicated for use in total parenteral nutrition to maintain zinc levels and prevent deficiency syndromes.[L14189] Zinc chloride was granted FDA approval before 26 June 1986.[L14189]

Kategori:
AcidsAcids, NoncarboxylicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical Use +20
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +94
Waktu ParuhUsing a two compart…
Vol. Distribusi-
KlirensIn one study of hea…
Genetik -
Zinc citrate DB11154
small molecule | CAS: 546-46-3

Zinc citrate is a zinc salt of citric acid. It is available as dietary supplements as a treatment of zinc deficiency and source of zinc, which is an essential trace element. Zinc citrate demonstrates effective absorption following oral administration [A27280].

Kategori:
Metal cationsMetal divalent cationsZinc Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc gluconate Approved DB11248
small molecule | CAS: 4468-02-4

Zinc gluconate is a zinc salt of gluconic acid comprised of two gluconic acid molecules for each zinc cation (2+). Zinc gluconate is a generally recognized as safe (GRAS) substance by FDA [L2081]. It is available as a trace mineral supplement and over the cou…

Kategori:
Acids, AcyclicAgents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and Metabolism +8
Waktu Paruh280 days [L2091]
Vol. DistribusiStored primarily in…
KlirensPlease refer to Dru…
Genetik -
Zinc glycinate DB14493
small molecule | CAS: 14281-83-5

Glycoprotein marker of gastrointestinal cancer.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsAntigens +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 955009-96-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 14354-67-7

Deskripsi belum tersedia.

Kategori:
Biological FactorsCoordination ComplexesHeterocyclic Compounds, Fused-Ring +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc oxide Approved DB09321
small molecule | CAS: 1314-13-2

Zinc oxide is an inorganic compound used in a number of manufacturing processes. It can be found in rubbers, plastics, ceramics, glass, cement, lubricants, paints, ointments, adhesives, sealants, pigments, foods, batteries, ferrites, fire retardants, and firs…

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseBasic Ointments and ProtectantsBasic Powders and Demulcents +12
Waktu ParuhIntended for local …
Vol. DistribusiIntended for local …
KlirensIntended for local …
Genetik -
Zinc phenolsulfonate Approved DB15793
small molecule | CAS: 127-82-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc picolinate DB11175
small molecule | CAS: 17949-65-4

Zinc picolinate is a zinc salt of picolinic acid. It is available as OTC dietary supplements as a source of zinc to treat and prevent zinc deficiency. The absorption of zinc after oral administration of zinc picolinate is shown to be effective.

Kategori:
Compounds used in a research, industrial, or household settingMetal cationsMetal divalent cations +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zinc sulfate Approved DB09322
small molecule | CAS: 7733-02-0

Zinc sulfate is the inorganic compound with the formula ZnSO4 and historically known as "white vitriol". It is on the World Health Organization's List of Essential Medicines, a list of the most important medication needed in a basic health system.

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseAlimentary Tract and MetabolismAstringents +17
Waktu Paruh3 hours
Vol. DistribusiAfter absorption zi…
Klirens-
Genetik -
small molecule

Zinc sulfate is a common zinc supplement in parenteral nutrition.[A216916,L12888]

Kategori:
Agents for Treatment of Hemorrhoids and Anal Fissures for Topical UseMetal cationsMetal divalent cations +2
Target Protein:
B1 bradykinin receptorMethylated-DNA--protein-cysteine methyltransferaseFructose-bisphosphate aldolase A +94
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1387453-03-3

Zinpentraxin alfa is a recombinant form of PTX-2, a naturally circulating human protein. It is under investigation in clinical trial NCT01981850 (A Phase 2 Study Of PRM-151 In Subjects With Myelofibrosis).

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsAmyloid +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ziprasidone Approved DB00246
small molecule | CAS: 146939-27-7

Disorders such as schizophrenia and bipolar disorder can significantly impair mood, cognition, and behavior.[A190525] These mental illnesses can often be accompanied by comorbidities such as depression and substance abuse, and can significantly impact the qua…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +45
Target Protein:
D(2) dopamine receptorNeuronal acetylcholine receptor subunit alpha-75-hydroxytryptamine receptor 2A +24
Waktu ParuhThe half life of zi…
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent s…
Genetik -
biotech

Zirconium panitumumab Zr-89 is under investigation in clinical trial NCT05423197 (Study Evaluating Zr-panitumumab for Assessment of Suspected Metastatic Lesions on 18F-FDG-PET/CT in Head and Neck Squamous Cell Carcinoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ZK-93423 DB17063
small molecule | CAS: 83910-44-5

ZK-93423 is a beta-carboline with muscle relaxant activity with agonistic properties at the benzodiazepine receptor.[A253172]

Kategori:
Anti-Anxiety AgentsAnticonvulsantsCentral Nervous System Agents +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit gamma-2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zoalene DB11480
small molecule | CAS: 148-01-6

Dinitolmide is a fodder additive for prophylaxis against coccidiosis infections in poultry.

Kategori:
Acids, CarbocyclicAmidesAnti-Infective Agents +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zolazepam DB11555
small molecule | CAS: 31352-82-6

Zolazepam is a pyrazolodiazepinone derivative used as an anaesthetic in veterinary medicine. Zolazepam is typically used in combination with the NMDA antagonist tiletamine or the ?2 adrenoceptor agonist xylazine. It is around four times the potency of diazepa…

Kategori:
Anti-Anxiety AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zoledronic acid Approved DB00399
small molecule | CAS: 118072-93-8

Zoledronic acid, or CGP 42'446,[A203120] is a third generation, nitrogen containing bisphosphonate similar to [ibandronic acid], [minodronic acid], and [risedronic acid].[A203111] Zoledronic acid is used to treat and prevent multiple forms of osteoporosis, hy…

Kategori:
BisphosphonatesBone Density Conservation AgentsDrugs Affecting Bone Structure and Mineralization +5
Target Protein:
Geranylgeranyl pyrophosphate synthaseHydroxylapatiteFarnesyl pyrophosphate synthase
Waktu ParuhZoledronic acid has…
Vol. Distribusi-
KlirensZoledronic acid has…
Genetik -
Zoliflodacin DB12817
small molecule | CAS: 1620458-09-4

Zoliflodacin has been used in trials studying the basic science and treatment of Gonorrhoea.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +5
Target Protein:
DNA gyrase subunit ADNA gyrase subunit B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zolmitriptan Approved DB00315
small molecule | CAS: 139264-17-8

Zolmitriptan is a member of the triptan class of 5-hydroxytryptamine(5-HT)<sub>1B/1D/(1F)</sub> receptor agonists used to treat acute migraine.[A462, L12978] [Sumatriptan] was the first triptan to be developed, but had poor oral bioavailability and lipophilic…

Kategori:
Agents that produce hypertensionAminesAnalgesics +24
Target Protein:
5-hydroxytryptamine receptor 1B5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 1F +5
Gen Terkait:
GNB3
Waktu ParuhZolmitriptan has a …
Vol. DistribusiZolmitriptan has a …
KlirensZolmitriptan has a …
Genetik 1 Varian
Zomepirac DB04828
small molecule | CAS: 33369-31-2

Zomepirac, formerly marketed as Zomax tablets, was associated with fatal and near-fatal anaphylactoid reactions. The manufacturer voluntarily removed Zomax tablets from the Canadian, US, and UK markets in March 1983.

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +15
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zonisamide Approved DB00909
small molecule | CAS: 68291-97-4

Zonisamide is a sulfonamide anticonvulsant used as an adjunctive therapy in adults with partial-onset seizures.[L42530,L42535] Zonisamide may act by blocking repetitive firing of voltage-gated sodium channels, leading to a reduction of T-type calcium channel…

Kategori:
Agents causing hyperkalemiaAmidesAnti-epileptic Agent +32
Target Protein:
Sodium channel protein type 1 subunit alphaSodium channel protein type 2 subunit alphaSodium channel protein type 3 subunit alpha +29
Waktu ParuhIn plasma, the elim…
Vol. DistribusiFollowing a 400 mg …
KlirensIn patients not tak…
Genetik -
small molecule | CAS: 139570-93-7

Zoptarelin doxorubicin has been used in trials studying the treatment of Breast Cancer, Ovarian Cancer, Prostate Cancer, Endometrial Cancer, and Urothelial Carcinoma, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAnthracyclinesCarbohydrates +12
Target Protein:
Gonadotropin-releasing hormone receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zorubicin DB11618
small molecule | CAS: 54083-22-6

Zorubicin is a drug of the anthracycline class - a class of medications that have historically demonstrated effective chemotherapy for a variety of cancer types.

Kategori:
AnthracyclinesAnthracyclines and Related SubstancesAntibiotics, Antineoplastic +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zotatifin DB16408
small molecule | CAS: 2098191-53-6

Zotatifin is under investigation in clinical trial NCT04092673 (Study of Eft226 in Subjects With Selected Advanced Solid Tumor Malignancies).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zotiraciclib DB16656
small molecule | CAS: 1204918-72-8

Zotiraciclib is under investigation in clinical trial NCT02942264 (Zotiraciclib (TG02) Plus Dose-dense or Metronomic Temozolomide Followed by Randomized Phase II Trial of Zotiraciclib (TG02) Plus Temozolomide Versus Temozolomide Alone in Adults With Recurrent…

Kategori:
Cyclin-Dependent Kinases, antagonists & inhibitorsHeterocyclic Compounds, Fused-Ring
Target Protein:
Cyclin-dependent kinase 2Cyclin-dependent kinase 9Tyrosine-protein kinase Fyn +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zotizalkib DB19238
small molecule | CAS: 2648641-36-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Zucapsaicin Approved DB09120
small molecule | CAS: 25775-90-0

Zucapsaicin, the cis-isomer of capsaicin, is a topical analgesic used to treat osteoarthritis of the knee and other neuropathic pain. It is a modulator of transient receptor potential cation channel subfamily V member 1 (TRPV-1), also known as the vanilloid o…

Kategori:
AlkaloidsAlkenesAlkynes +25
Target Protein:
Transient receptor potential cation channel subfamily V member 1
Waktu ParuhIn rats, the elimin…
Vol. Distribusi-
Klirens-
Genetik -
Zuclopenthixol Approved DB01624
small molecule | CAS: 53772-83-1

Zuclopenthixol, also known as Zuclopentixol or Zuclopenthixolum, is an antipsychotic agent. Zuclopenthixol is a thioxanthene-based neuroleptic with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine rece…

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +34
Target Protein:
D(1A) dopamine receptorD(1B) dopamine receptorD(2) dopamine receptor +4
Waktu Paruh20 hours (range 12-…
Vol. Distribusi20 L/kg.
Klirensapproximately 0.9 L…
Genetik -
ZVS101e DB18424
biotech

ZVS101e is a recombinant adeno-associated virus vector carrying human CYP4V2 gene.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ZYC300 DB04986
biotech

ZYC300 is a plasmid DNA of CYP1B1 encapsulated in biodegradable poly-DL-lactide-coglycolide microparticles. It is designed as a vaccine, intended to increase immune system sensitivity to CYP1B1, an enzyme highly prevalent in tumor cells.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ZYCOV-D DB15892
biotech

The ZYCOV-D vaccine candidate was developed by Cadila Healthcare Ltd. based in India[A219758]. The vaccine was developed using a DNA vaccine platform with a non-replicating and non-integrating plasmid carrying the gene of interest[L16503]. Once the plasmid D…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Zytron Approved DB11768
small molecule | CAS: 299-85-4

Zytron (DMPA) is under investigation for the treatment and health services research of HIV, Lactation, Contraception, Postpartum Depression, and Immune Cells (Mucosal and Systemic). DMPA has been investigated for the prevention, treatment, and basic science o…

Kategori:
AminesOrganophosphorus CompoundsSulfur Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Chymase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase TEM
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Beta-lactamase TEMBeta-lactamase TEMBeta-lactamase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Carboxylesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
GTPase KRasProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaProtein farnesyltransferase subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Type I polyketide synthase PikAIV
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6601–6650 dari 6694
Sebelumnya Halaman 133 / 134 Berikutnya