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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

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Hasil Pencarian (13591)

Halaman 133 / 272
Golexanolone DB18200
small molecule | CAS: 2089238-18-4

Deskripsi belum tersedia.

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Golidocitinib DB18057
small molecule | CAS: 2091134-68-6

Deskripsi belum tersedia.

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Golodirsen Approved DB15593
biotech | CAS: 1422959-91-8

Golodirsen is a morpholino antisense oligomer designed to treat about 8% of patients with Duchenne Muscular Dystrophy (DMD). This is an X-linked condition leading to progressive muscle degeneration that begins in early childhood, rendering many patients wheel…

Kategori:
Antisense Elements (Genetics)Antisense OligonucleotidesCompounds used in a research, industrial, or household setting +10
Target Protein:
Dystrophin
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe volume of distr…
KlirensThis drug is rapidl…
Genetik -
Golotimod DB05475
small molecule | CAS: 229305-39-9

SCV-07 (g -D-glutamyl-L-tryptophan) is a novel synthetic dipeptide that acts broadly on the Toll-like receptor pathway. It has been shown to stimulate T-lymphocyte differentiation, macrocytic phagocytosis, and specific immune responses, and enhance IL-2 and …

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Signal transducer and activator of transcription 3Toll-like receptor 2Toll-like receptor 4 +2
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Golvatinib DB11977
small molecule | CAS: 928037-13-2

Golvatinib has been investigated for the treatment of Platinum-Resistant Squamous Cell Carcinoma of the Head and Neck.

Kategori:
AminesPyridinesVascular Endothelial Growth Factor Receptor-2, antagonists & inhibitors
Target Protein:
Vascular endothelial growth factor receptor 2Hepatocyte growth factor receptor
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Gonadorelin Approved DB00644
biotech | CAS: 33515-09-2

Gonadorelin is another name for gonadotropin-releasing hormone (GnRH). It is a synthetic decapeptide prepared using solid phase peptide synthesis. GnRH is responsible for the release of follicle stimulating hormone and leutinizing hormone from the anterior pi…

Kategori:
Adrenal Cortex HormonesAmino Acids, Peptides, and ProteinsDiagnostic Agents +18
Target Protein:
Gonadotropin-releasing hormone receptorPutative gonadotropin-releasing hormone II receptor
Waktu ParuhVery short, initial…
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Gondoic acid DB14073
small molecule | CAS: 5561-99-9

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, UnsaturatedLipids
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Gontivimab DB16179
biotech | CAS: 1257358-38-5

Gontivimab is under investigation in clinical trial NCT03468829 (Efficacy and Safety of ALX-0171 in Adult Hematopoietic Stem Cell Transplant (HSCT) Recipients Who Present With Respiratory Syncytial Virus (RSV) Infection).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAntiviral Agents +11
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Gonyautoxin II DB19186
small molecule | CAS: 60508-89-6

Gonyautoxin II is under investigation in clinical trial NCT04799041 (Gonyautoxin 2/3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study).

Kategori:
Amino Acids, Peptides, and ProteinsBacterial ToxinsBiological Factors +9
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Gonyautoxin III DB19187
small molecule | CAS: 60537-65-7

Gonyautoxin III is currently under investigation in clinical trial (Gonyautoxin 2/?3 in the Treatment of Acute Back Pain: A Clinical Proof-of-concept Study) for the treatment of Acute Back Pain.

Kategori:
Bacterial ToxinsBiological FactorsComplex Mixtures +7
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Gosogliptin DB08382
small molecule | CAS: 869490-23-3

Gosogliptin has been used in trials studying the treatment of Renal Insufficiency, Chronic.

Kategori:
Agents causing angioedemaBlood Glucose Lowering AgentsDiabetes Mellitus, Type 2, drug therapy +1
Target Protein:
Dipeptidyl peptidase 4
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Gossypol DB13044
small molecule | CAS: 303-45-7

Gossypol has been used in trials studying the treatment of Non-small Cell Lung Cancer.

Kategori:
Adrenal Cortex HormonesContraceptive Agents, MaleHormonal Contraceptives for Systemic Use +3
Target Protein:
Apoptosis regulator Bcl-2Bcl-2-like protein 1
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Gosuranemab DB15376
biotech | CAS: 1788032-39-2

Gosuranemab is under investigation in clinical trial NCT02460094 (Multiple Ascending Dose Study of Intravenously Administered BMS-986168 (BIIB092) in Patients With Progressive Supranuclear Palsy).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
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Gotistobart DB19100
biotech | CAS: 2226344-78-9

Gotistobart is under investigation in clinical trial NCT05671510 (ONC-392 Versus Docetaxel in Metastatic NSCLC That Progressed on PD-1/PD-L1 Inhibitors).

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GP-100 antigen DB14800
biotech

GP-100 antigen is under investigation in clinical trial NCT00006385 (Vaccine Therapy With or Without Biological Therapy in Treating Patients With Metastatic Melanoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Neoplasm +5
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GR270773 DB06427
small molecule

GR270773, was investigated in two clinical trials for its potential to treat sepsis: NCT00158769 (completed, comparing the effects of infusion between healthy adults and those with damaged livers) and NCT00089986 (completed with results, treatment of suspecte…

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GRAd-COV2 DB16428
biotech

GRAd-COV2 is a COVID-19 vaccine candidate being developed by ReiThera[L30420, L30423]. This therapy is based on a novel replication-incompetent simian adenoviral vector that encodes the full-length SARS-CoV-2 spike protein (GRAd-COV2)[L30420, L30423]. Preclin…

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Granaticin B DB17273
small molecule | CAS: 19879-03-9

Deskripsi belum tersedia.

Kategori:
BenzopyransBenzoquinonesChromans +5
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Granisetron Approved DB00889
small molecule | CAS: 109889-09-0

A serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic and antinauseant for cancer chemotherapy patients.

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +23
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh4-6 hours in health…
Vol. Distribusi-
Klirens* 0.52 L/h/kg [Canc…
Genetik -
Granotapide DB12934
small molecule | CAS: 594842-13-4

Granotapide has been used in trials studying the treatment of Type II Diabetes Mellitus.

Kategori:
Acids, AcyclicAcids, CarbocyclicAmides +3
Target Protein:
Microsomal triglyceride transfer protein large subunit
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Grape Approved DB10533
biotech

Grape allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Grape seed oil DB14323
biotech | CAS: 8016-21-5

Grape seed oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Grapefruit Approved DB10534
biotech

Grapefruit allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +4
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Grapefruit oil DB15663
biotech | CAS: 8016-20-4

Deskripsi belum tersedia.

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Grapiprant DB12836
small molecule | CAS: 415903-37-6

Grapiprant, also known as AT-001 and CJ-023, is a drug from the piprant class. These molecules were derived from acylsulfonamide and are characterized to be a novel series of para-N-acylaminomethylbenzoic acid known to be prostaglandin receptor antagonists.[A…

Kategori:
AmidesBenzene DerivativesP-glycoprotein substrates +3
Target Protein:
Prostaglandin E2 receptor EP4 subtype
Waktu ParuhThe reported elimin…
Vol. DistribusiThe reported volume…
KlirensThe reported cleara…
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Grazoprevir Approved DB11575
small molecule | CAS: 1350514-68-9

Grazoprevir is a direct acting antiviral medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized into nin…

Kategori:
Acids, AcyclicAmidesAnti-Infective Agents +24
Target Protein:
Genome polyprotein
Waktu ParuhThe geometric mean …
Vol. DistribusiGrazoprevir has an …
KlirensThe clearance of Gr…
Genetik -
Green tea leaf DB14307
biotech

Green tea leaf is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
BeveragesBiological ProductsComplex Mixtures +3
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Gremubamab DB15014
biotech | CAS: 1800381-36-5

Gremubamab is under investigation in clinical trial NCT02255760 (Phase 1 Randomized Double-blind Placebo Controlled Study to Evaluate Safety and PK of MEDI3902 in Healthy Adults).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Grepafloxacin Approved DB00365
small molecule | CAS: 119914-60-2

Grepafloxacin is an oral broad-spectrum quinoline antibacterial agent used to treat bacterial infections. Due to the QTc-prolonging potential, as indicated by the changes in the QT interval on the electrocardiogram, and the risk for cardiovascular adverse eve…

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +22
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +1
Waktu Paruh15 ± 3 hours
Vol. Distribusi-
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Gresonitamab DB18210
biotech | CAS: 2413817-97-5

Deskripsi belum tersedia.

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Grn163l DB05036
small molecule

GRN163L is a novel anti-cancer drug. It has been characterized preclinically and shown to inhibit telomerase in human tumor cells of many cancer types (including lung, breast, prostate, liver, and early stage of human breast cancer), in both cell culture syst…

Target Protein:
Telomerase-binding protein EST1AN-terminal kinase-like proteinProstaglandin E synthase 3 +1
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GRObeta DB18205
biotech

Deskripsi belum tersedia.

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small molecule | CAS: 141925-59-9

Growth hormone-releasing peptide 1 is under investigation in clinical trial NCT00381602 (A Phase II, Randomized, Cross-over, Vehicle-controlled, Double-blind, Multicenter Study of the Safety, Pharmacodynamics, and Preliminary Efficacy of GHRP-1/AG in Subjects…

Kategori:
Amino Acids, Peptides, and ProteinsGrowth Hormone-Releasing HormonePeptides
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GS 0573 DB08843
small molecule | CAS: 113852-41-8

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsHeterocyclic Compounds, Fused-RingImmunologic Factors +1
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GS-100 DB18337
biotech

GS-100 is an adeno-associated virus serotype 9 virus particle containing viral DNA that includes an expression cassette containing the human NGLY1 gene coding sequence

Kategori:
CyclohexanesCycloparaffinsLipids +3
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GS-441524 DB15686
small molecule | CAS: 1191237-69-0

GS-441524 is an adenosine nucleotide analog antiviral, similar to [remdesivir].[A203057,L13239] This molecule was patented in 2009.[L13775] _In vitro_ studies of GS-441524 have determined it has a higher EC<sub>50</sub> than remdesivir against a number of vir…

Kategori:
Adenine NucleotidesAnti-Infective AgentsAntiviral Agents +10
Target Protein:
Replicase polyprotein 1abRNA-directed RNA polymerase L
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GS-6620 DB15222
small molecule | CAS: 1350735-70-4

GS-6620 is under investigation in clinical trial NCT01316237 (A Study Evaluating the Safety, Tolerability, Pharmacokinetics and Antiviral Activity of GS-6620 in Treatment Naïve Subjects With Chronic Hepatitis C Virus Infection).

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsHeterocyclic Compounds, Fused-Ring +5
Target Protein:
Genome polyprotein
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GS030-DP DB17847
biotech

GS030-DP is an optogenetic gene therapy being investigated for the treatment of retinitis pigmentosa. It targets retinal ganglion cells that encodes a light-sensitive channelrhodopsin, ChrimsonR-tdTomato (ChR-tdT), delivered by an AAV2.7m8 vector. It is a com…

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GSI-136 DB12819
small molecule | CAS: 443989-01-3

GSI-136 has been used in trials studying the treatment of Alzheimer Disease.

Target Protein:
Gamma-secretase subunit APH-1BNicastrinGamma-secretase subunit APH-1A +2
Waktu Paruh-
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GSK-1004723 DB12806
small molecule | CAS: 955359-72-5

Gsk1004723 has been investigated for the treatment of Allergic Rhinitis and Rhinitis, Allergic, Seasonal.

Kategori:
Histamine AntagonistsHistamine H1 AntagonistsPyridazines
Target Protein:
Histamine H3 receptorHistamine H1 receptor
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GSK-1292263 DB12627
small molecule | CAS: 1032823-75-8

GSK1292263 has been investigated for the treatment of DIABETES MELLITUS, TYPE 2.

Target Protein:
Glucose-dependent insulinotropic receptor
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GSK-1521498 DB12886
small molecule | CAS: 1007573-18-3

GSK1521498 has been used in trials studying the treatment of Obesity and Alcoholism.

Kategori:
IndenesReceptors, Opioid, mu
Target Protein:
Mu-type opioid receptor
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GSK-2018682 DB11987
small molecule | CAS: 1034688-30-6

GSK2018682 has been investigated for the treatment of Multiple Sclerosis, Relapsing-Remitting.

Kategori:
Heterocyclic Compounds, Fused-RingOxazoles
Target Protein:
Sphingosine 1-phosphate receptor 1
Waktu Paruh-
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GSK-239512 DB15120
small molecule | CAS: 720691-69-0

GSK-239512 is under investigation in clinical trial NCT00474513 (An Imaging Study to Investigate the Distribution of GSK239512 in the Brain.).

Kategori:
Heterocyclic Compounds, Fused-RingHistamine Antagonists
Target Protein:
Histamine H3 receptor
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GSK-256066 DB12137
small molecule | CAS: 801312-28-7

Gsk256066 has been used in trials studying the treatment and diagnostic of SAR, Asthma, Mild Asthma, Allergic Rhinitis, and Seasonal Allergic Rhinitis, among others.

Kategori:
Enzyme InhibitorsHeterocyclic Compounds, Fused-RingPhosphodiesterase 4 Inhibitors +3
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4A
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GSK-2636771 DB11795
small molecule | CAS: 1372540-25-4

GSK2636771 has been used in trials studying the treatment of CANCER, LYMPHOMA, Solid Neoplasm, Recurrent Solid Neoplasm, and Advanced Malignant Neoplasm, among others.

Kategori:
Antineoplastic AgentsEnzyme InhibitorsOxazines +1
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
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GSK-269962A DB17030
small molecule | CAS: 850664-21-0

GSK-269962A is a Rho kinase (ROCK) inhibitor with both ROCK1 and ROCK2 affinity.[A253012]

Kategori:
Oxazoles
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GSK-2881078 DB16888
small molecule | CAS: 1539314-06-1

Deskripsi belum tersedia.

Kategori:
Anabolic AgentsHeterocyclic Compounds, Fused-RingHormones +1
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GSK-2981278 DB16319
small molecule | CAS: 1474110-21-8

GSK-2981278 is under investigation in clinical trial NCT03004846 (A Study of GSK2981278 Ointment in Subjects With Plaque Psoriasis).

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Nuclear receptor ROR-gamma
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GSK-2982772 DB16875
small molecule | CAS: 1622848-92-3

Deskripsi belum tersedia.

Target Protein:
Receptor-interacting serine/threonine-protein kinase 1
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Menampilkan 6601–6650 dari 13591
Sebelumnya Halaman 133 / 272 Berikutnya