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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 133 / 315
Evacetrapib DB11655
small molecule | CAS: 1186486-62-3

Evacetrapib has been used in trials studying the basic science and treatment of Dyslipidemia, Hyperlipidemia, Hypercholesterolemia, Hepatic Insufficiency, and Cardiovascular Disease.

Kategori:
Anticholesteremic AgentsBenzazepinesCholesterol Ester Transfer Proteins, antagonists & inhibitors +3
Target Protein:
Cholesteryl ester transfer protein
Waktu Paruh-
Vol. Distribusi-
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Evalstotug DB19410
biotech | CAS: 2460399-39-5

Evalstotug is under investigation in clinical trial NCT05271604 (A Phase 2 Open Label Study of BA3021 in Patients With Recurrent or Metastatic Squamous Cell Carcinoma of the Head and Neck).

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Evans blue DB09361
small molecule | CAS: 314-13-6

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsAzo Compounds +7
Target Protein:
Albumin
Waktu Paruh-
Vol. Distribusi-
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Evatanepag DB12022
small molecule | CAS: 223488-57-1

Evatanepag has been used in trials studying the treatment of Tibial Fractures.

Target Protein:
Prostaglandin E2 receptor EP2 subtype
Waktu Paruh-
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Evenamide DB18775
small molecule | CAS: 1092977-61-1

Deskripsi belum tersedia.

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biotech | CAS: 308064-97-3

Evening primrose oil comes from the extraction from _Oenothera biennis_ seeds and it is commonly used as an alternative source for omega-6 essential fatty acids. In its composition it presents some fatty acids such as [DB00132] and [DB13854].[A33131] Evening …

Kategori:
Agents that reduce seizure thresholdAngiospermsAnti-Inflammatory Agents +26
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Evernia prunastri Approved DB14172
biotech

Evernia prunastri allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseStandardized Chemical Allergen
Waktu Paruh-
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Evernimicin DB06431
small molecule | CAS: 109545-84-8

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsCarbohydratesGlycosides
Waktu Paruh-
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Everolimus Approved DB01590
small molecule | CAS: 159351-69-6

Everolimus is a derivative of Rapamycin (sirolimus), and works similarly to Rapamycin as an mTOR (mammalian target of rapamycin) inhibitor. It is currently used as an immunosuppressant to prevent rejection of organ transplants. In a similar fashion to other m…

Kategori:
Anti-Bacterial AgentsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +32
Target Protein:
Serine/threonine-protein kinase mTOR
Waktu Paruh~30 hours.
Vol. DistribusiThe blood-to-plasma…
KlirensFollowing a 3 mg ra…
Genetik -
Evexomostat DB19140
small molecule | CAS: 2416263-67-5

Evexomostat is under investigation in clinical trial NCT05570253 (A Study of SDX-7320 in Combination With Eribulin for People With Breast Cancer).

Waktu Paruh-
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Evinacumab Approved DB15354
biotech | CAS: 1446419-85-7

Evinacumab is a recombinant human IgG4 monoclonal antibody targeted against angiopoietin-like protein 3 (ANGPTL3) and the first drug of its kind. The ANGPTL family of proteins serve a number of physiologic functions - including involvement in the regulation o…

Kategori:
Amino Acids, Peptides, and ProteinsAngiopoietin-like 3 InhibitorAngiopoietin-like 3 Inhibitors +8
Target Protein:
Angiopoietin-related protein 3
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
Klirens-
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Evobrutinib DB15170
small molecule | CAS: 1415823-73-2

Evobrutinib is under investigation in clinical trial NCT03934502 (Effect of Meal Composition and Timing on Evobrutinib Bioavailability).

Target Protein:
Tyrosine-protein kinase BTK
Waktu Paruh-
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Evocalcet DB12388
small molecule | CAS: 870964-67-3

Evocalcet has been used in trials studying the treatment of Hyperparathyroidism and Secondary Hyperparathyroidism.

Kategori:
Anti-Parathyroid AgentsCalcium HomeostasisSystemic Hormonal Preparations, Excl. Sex Hormones and Insulins
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Evodenoson DB12295
small molecule | CAS: 844873-47-8

Evodenoson has been used in trials studying the treatment of Open-angle Glaucoma and Ocular Hypertension.

Target Protein:
Adenosine receptor A2a
Waktu Paruh-
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Evofosfamide DB06091
small molecule | CAS: 918633-87-1

TH-302 is a novel cancer therapeutic specifically activated under the low oxygen or "hypoxic" conditions typical of solid tumor cancer cells. TH-302 is a nitroimidazole-linked prodrug of a brominated derivative of an isophosphoramide mustard previously used i…

Kategori:
Hydrocarbons, HalogenatedImidazolesMustard Compounds +4
Waktu Paruh-
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Evogliptin DB12625
small molecule | CAS: 1222102-29-5

Evogliptin has been used in trials studying the treatment and screening of Osteoporosis, Renal Impairment, Type 2 Diabetes Mellitus, Diabetes Mellitis Type 2, and Diabetes Mellitus, Type 2.

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +4
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
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Evolocumab Approved DB09303
biotech | CAS: 1256937-27-5

Evolocumab is a monoclonal antibody designed for the treatment of hyperlipidemia by Amgen. It is a subcutaneous injection approved by the FDA for individuals on maximum statin therapy who still require additional LDL-cholesterol lowering. It is approved for b…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +18
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu Paruh-
Vol. Distribusi-
KlirensEvolocumab showed n…
Genetik -
Evorpacept DB17573
biotech | CAS: 2484949-51-9

evorpacept is under investigation in clinical trial NCT04755244 (A Study of Evorpacept (ALX148) With Venetoclax and Azacitidine for Acute Myeloid Leukemia (ASPEN-05)).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +8
Waktu Paruh-
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EVT 201 DB05721
small molecule | CAS: 308239-86-3

EVT 201 is a novel partial positive allosteric modulator of the GABAA receptor complex which is being developed as a treatment for insomnia. It is being developed by Evotec Inc.

Kategori:
BenzazepinesHeterocyclic Compounds, Fused-Ring
Target Protein:
Gamma-aminobutyric acid receptor subunit gamma-3Gamma-aminobutyric acid receptor subunit alpha-1
Waktu Paruh-
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EVT-101 DB05956
small molecule | CAS: 1189088-41-2

Deskripsi belum tersedia.

Target Protein:
Glutamate receptor ionotropic, NMDA 2BRetinoic acid receptor RXR-alpha
Waktu Paruh-
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EW-A-401 DB05525
biotech

EW-A-401 is a circle of genetic material (plasmid DNA) that instructs the body to produce a genetically-engineered transcription factor, a protein that regulates expression of genes. This specific transcription factor has been shown in animal studies to incre…

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Genetik -
biotech

Holoclar (_ex vivo_ expanded autologous human corneal epithelial cells containing stem cells) is a stem cell therapy used to treat limbal stem cell deficiencies.[L48375]

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Exagamglogene autotemcel Approved DB15572
biotech

Sickle cell disease (SCD) is a genetic disorder characterized by the production of abnormal sickle-shaped red blood cells (called hemoglobin S, HbS) that initiate a pathophysiology resulting in severe pain, progressive multi-organ damage, and premature death.…

Kategori:
Autologous Cultured CellBlood and Blood Forming Organs
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Exaluren DB17631
small molecule | CAS: 1375073-93-0

Deskripsi belum tersedia.

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Exametazime Approved DB11179
small molecule | CAS: 105613-48-7

Exametazime is a diagnostic radiopharmaceutical agent commonly used for the preparation of Tc99m Exametazime injection. It acts as a chelating agent for the radioisotope technetium-99m to form a cationic complex. It is used in the detection of altered regiona…

Kategori:
Ketones
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Exarafenib DB17582
small molecule | CAS: 2639957-39-2

Deskripsi belum tersedia.

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Exatecan DB12185
small molecule | CAS: 171335-80-1

Exatecan has been used in trials studying the treatment of Sarcoma, Leukemia, Lymphoma, Lung Cancer, and Liver Cancer, among others.

Kategori:
AlkaloidsAntineoplastic AgentsEnzyme Inhibitors +2
Target Protein:
DNA topoisomerase 1
Waktu Paruh-
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Exbivirumab DB17747
biotech | CAS: 569658-80-6

Exbivirumab is an investigational monoclonal antibody. It is one of the active ingredients in HepeX-B, a drug product containing two human monoclonal antibodies to the hepatitis B virus (HBV) surface antigen.[A259202]

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Excindogen DB18754
small molecule

Excindogen is an investigational immunotherapy.

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Exebacase DB16161
biotech | CAS: 1404122-92-4

Exebacase is under investigation in clinical trial NCT03163446 (Safety, Efficacy and Pharmacokinetics of CF-301 vs. Placebo in Addition to Antibacterial Therapy for Treatment of S. Aureus Bacteremia).

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +1
Waktu Paruh-
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Exemestane Approved DB00990
small molecule | CAS: 107868-30-4

Exemestane is an oral steroidal aromatase inhibitor used in the adjuvant treatment of hormonally-responsive (also called hormone-receptor-positive, estrogen-responsive) breast cancer in postmenopausal women. It irreversibly binds to the active site of the enz…

Kategori:
AndrostanesAndrostenesAntineoplastic Agents +14
Target Protein:
Aromatase
Waktu Paruh24 hours
Vol. Distribusi-
Klirens-
Genetik -
Exenatide Approved DB01276
biotech | CAS: 141758-74-9

Exenatide is a glucagon-like peptide-1 (GLP-1) analog[L42690]. It activates the GLP-1 receptor and increases insulin secretion, decreases glucagon secretion, and slows gastric emptying to improve glycemic control[L42690]. Exenatide was given FDA approval on A…

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsAnti-Obesity Agents +16
Target Protein:
Glucagon-like peptide 1 receptor
Waktu Paruh2.4 hours[Label]
Vol. Distribusi28.3L[Label].
Klirens9.1 L/hour[Label].
Genetik -
Exicorilant DB16162
small molecule | CAS: 1781244-77-6

Exicorilant is under investigation in clinical trial NCT03437941 (Study to Evaluate CORT125281 in Combination With Enzalutamide in Patients With Mcrpc).

Target Protein:
Glucocorticoid receptor
Waktu Paruh-
Vol. Distribusi-
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Exidavnemab DB19452
biotech | CAS: 2438229-02-6

Exidavnemab is under investigation in clinical trial NCT06671938 (Safety, Tolerability, and Pharmacokinetics of Exidavnemab in Patients With Parkinson's Disease).

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Exisulind DB06246
small molecule | CAS: 59973-80-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAnti-Inflammatory Agents +10
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesteraseGlutathione S-transferase PAldo-keto reductase family 1 member B1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Exlinkibart DB17474
biotech | CAS: 2642171-64-8

Deskripsi belum tersedia.

Waktu Paruh-
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EXOB-001 DB18257
biotech

EXOB-001 consists of extracellular vesicles derived from cultured human umbilical cord mesenchymal stromal cells.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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biotech

Deskripsi belum tersedia.

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EXT608 DB18453
biotech

EXT608 is a long-acting PTH derivative under investigation for the treatment of hyperparathyroidism.[L48270]

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Ezabenlimab DB17483
biotech | CAS: 2249882-54-8

Deskripsi belum tersedia.

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biotech | CAS: 2226647-27-2

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Ezatiostat DB05460
small molecule | CAS: 168682-53-9

Ezatiostat is investigated in clinical trials for treating myelodysplastic syndrome. This compound belongs to the peptides. These are compounds containing an amide derived from two or more amino carboxylic acid molecules (the same or different) by formation o…

Kategori:
Amino Acids, Peptides, and ProteinsOligopeptidesPeptides
Target Protein:
Glutathione S-transferase P
Waktu Paruh-
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Ezeprogind DB16954
small molecule | CAS: 615539-20-3

Deskripsi belum tersedia.

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Ezetimibe Approved DB00973
small molecule | CAS: 163222-33-1

Ezetimibe is a lipid-lowering compound that inhibits intestinal cholesterol and phytosterol absorption. The discovery and research of this drug began in the early 1990s, after the intravenous administration of radiolabelled ezetimibe in rats revealed that it …

Kategori:
Anticholesteremic AgentsAzetinesBCRP/ABCG2 Substrates +20
Target Protein:
NPC1-like intracellular cholesterol transporter 1Sterol O-acyltransferase 1Aminopeptidase N
Waktu ParuhBoth ezetimibe and …
Vol. DistribusiThe relative volume…
KlirensThere are no pharma…
Genetik -
Ezogabine Approved DB04953
small molecule | CAS: 150812-12-7

Ezogabine (D23129) is a close structural analog of the centrally acting analgesic flupitrine. It is a neuronal potassium channel opener being developed as a first-in-class antiepileptic drug (AED) and is currently being studied in Phase 3 trials as an adjunct…

Kategori:
Acids, AcyclicAminesAniline Compounds +15
Target Protein:
Potassium voltage-gated channel subfamily KQT member 3Potassium voltage-gated channel subfamily KQT member 2Potassium voltage-gated channel subfamily KQT member 4 +1
Waktu ParuhTerminal half-life …
Vol. Distribusi8.7 L/kg
Klirens0.58 - 0.76 L/h·kg.…
Genetik -
Ezurpimtrostat DB16458
small molecule | CAS: 1914148-72-3

Deskripsi belum tersedia.

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
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Ezutromid DB12888
small molecule | CAS: 945531-77-1

Ezutromid has been investigated for the treatment of Muscular Dystrophy, Duchenne.

Kategori:
Heterocyclic Compounds, Fused-RingMuscular Dystrophy, Duchenne
Target Protein:
Utrophin
Waktu Paruh-
Vol. Distribusi-
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