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6694

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Halaman 131 / 134
Vofatamab DB14781
biotech | CAS: 1312305-12-6

Vofatamab is under investigation in clinical trial NCT02401542 (Dose Escalation, Expansion Study of Vofatamab (B-701) in Treatment of Locally Advanced or Metastatic Urothelial Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volanesorsen Approved DB15067
biotech | CAS: 915430-78-3

Volanesorsen is an antisense oligonucleotide that binds to apoC-III mRNA to prevent its translation.[L16621] It is indicated to treat familial chylomicronemia, a genetic condition that prevents breakdown of triglycerides and chylomicrons.[L16621] This drug is…

Kategori:
CarbohydratesGlycosidesLipid Modifying Agents +4
Target Protein:
Apolipoprotein C-III
Waktu ParuhVolanesorsen has a …
Vol. DistribusiThe volume of distr…
KlirensThe exact rate of c…
Genetik -
Volixibat DB13914
small molecule | CAS: 1025216-57-2

Volixibat, also known as SHP626 or LUM002, is an investigational drug that will potentially be used for the treatment of Non-Alcoholic Steatohepatitis (NASH). If approved for use, it will be the first available agent for the treatment of NASH. Volixibat is…

Kategori:
CarbohydratesHeterocyclic Compounds, Fused-RingLipid Regulating Agents +1
Target Protein:
Ileal sodium/bile acid cotransporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Volociximab DB06647
biotech | CAS: 558480-40-3

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2092457-20-8

Volrubigene ralaparvovec is under investigation in clinical trial NCT03223194 (Gene Transfer Clinical Study in Crigler-najjar Syndrome).

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Von Willebrand factor human Approved DB13133
biotech | CAS: 109319-16-6

The human von Willebrand factor (vWF) is a human plasma-derived vWF, an endogenous large multimeric plasma glycoprotein involved in hemostasis. It serves a dual role in hemostasis by mediating platelet adhesion and aggregation at the site of blood vessel inju…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood and Blood Forming Organs +8
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chainAsialoglycoprotein receptor 1 +1
Waktu ParuhIn patients with Ty…
Vol. DistribusiThe volume of distr…
KlirensIn patients with Ty…
Genetik -
Vonafexor DB18782
small molecule | CAS: 1192171-69-9

Deskripsi belum tersedia.

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vonicog alfa Approved DB12872
biotech

Vonicog alfa is a recombinant human von Willebrand factor (rVWF) produced from Chinese hamster ovary cells.[A264444] Used to treat von Willebrand Disease (vWD), it mimics the biological actions of endogenous VWF,[L51274] which is a critical plasma glycoprotei…

Kategori:
von Willebrand Factor
Target Protein:
Coagulation factor VIIICollagen alpha-1(I) chain
Waktu ParuhIn Study 071001, th…
Vol. Distribusi-
KlirensIn Study 071001, th…
Genetik -
Vonlerolizumab DB16352
biotech | CAS: 1638935-72-4

Vonlerolizumab is under investigation in clinical trial NCT03029832 (A Study of MOXR0916 in Combination With Atezolizumab Versus Atezolizumab Alone in Participants With Untreated Locally Advanced or Metastatic Urothelial Carcinoma Who Are Ineligible for Cispl…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vonoprazan Approved DB11739
small molecule | CAS: 881681-00-1

Vonoprazan is a potassium-competitive acid blocker (PCAB) that inhibits H<sup>+</sup>, K<sup>+</sup>-ATPase-mediated gastric acid secretion. PCABs represent an alternative to proton-pump inhibitors for the treatment of acid-related disorders. Unlike proton-pu…

Kategori:
Alimentary Tract and MetabolismAmidesCytochrome P-450 CYP2B6 Substrates +17
Target Protein:
Hydrogen potassium ATPase
Waktu ParuhVonoprazan has an e…
Vol. DistribusiVonoprazan has an a…
KlirensVonoprazan has an a…
Genetik -
Vorapaxar Approved DB09030
small molecule | CAS: 618385-01-6

Vorapaxar is a tricyclic himbacine-derived selective inhibitor of protease activated receptor (PAR-1) indicated for reducing the incidence of thrombotic cardiovascular events in patients with a history of myocardial infarction (MI) or with peripheral arterial…

Kategori:
AnticoagulantsAntiplatelet agentsBlood and Blood Forming Organs +11
Target Protein:
Proteinase-activated receptor 1
Waktu ParuhVorapaxar has an ef…
Vol. Distribusi424 L
Klirens-
Genetik -
Vorasidenib Approved DB17097
small molecule | CAS: 1644545-52-7

Vorasidenib is a first-in-class dual isocitrate dehydrogenase-1 (IDH1) and isocitrate dehydrogenase-2 (IDH2) inhibitor.[A264209] It works by suppressing the levels of D-2-hydroxyglutarate (2-HG), an oncometabolite produced by mutant IDH1 and IDH2 isoforms.[L5…

Kategori:
AminesBCRP/ABCG2 InhibitorsCytochrome P-450 CYP1A2 Substrates +26
Target Protein:
Isocitrate dehydrogenase [NAD] subunit alpha, mitochondrialIsocitrate dehydrogenase [NAD] subunit beta, mitochondrialIsocitrate dehydrogenase [NAD] subunit gamma, mitochondrial +2
Waktu ParuhThe mean (CV%) stea…
Vol. DistribusiThe mean (CV%) volu…
KlirensThe mean (CV%) stea…
Genetik -
Voretigene neparvovec Approved DB13932
biotech | CAS: 1646819-03-5

Voretigene Neparvovec-rzyl (VN-rzyl) is an adeno-associated virus vector-based gene therapy.[L1094] An adeno-associated virus is a small virus that infects humans and other primates. It is not pathogenic and it causes a very mild immune response. This type of…

Kategori:
Adeno-associated Viral Vector TherapiesOphthalmologicalsSensory Organs
Target Protein:
Retinoid isomerohydrolase
Waktu ParuhBased on the pharma…
Vol. DistribusiVN-rzyl was shown t…
KlirensAccording to the ki…
Genetik -
Vorinostat Approved DB02546
small molecule | CAS: 149647-78-9

Vorinostat (rINN) or suberoylanilide hydroxamic acid (SAHA), is a drug currently under investigation for the treatment of cutaneous T cell lymphoma (CTCL), a type of skin cancer, to be used when the disease persists, gets worse, or comes back during or after …

Kategori:
AmidesAminesAnilides +15
Target Protein:
Histone deacetylase 1Histone deacetylase 2Histone deacetylase 3 +4
Waktu Paruh2 hours
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1165741-01-4

Vorsetuzumab mafodotin is under investigation in clinical trial NCT01677390 (A Phase 1b Study of SGN-75 in Combination With Everolimus in Patients With Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vortioxetine Approved DB09068
small molecule | CAS: 508233-74-7

Vortioxetine is an antidepressant medication indicated for the treatment of major depressive disorder (MDD). It is classified as a serotonin modulator and stimulator (SMS) as it has a multimodal mechanism of action towards the serotonin neurotransmitter syste…

Kategori:
Agents that produce hypertensionAnti-Anxiety AgentsAntidepressive Agents +30
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 3A5-hydroxytryptamine receptor 7 +4
Waktu ParuhMean terminal half­…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
Voruciclib DB15157
small molecule | CAS: 1000023-04-0

Voruciclib is under investigation in clinical trial NCT03547115 (A Phase 1 Study of Voruciclib in Subjects With B-Cell Malignancies or AML).

Kategori:
Antineoplastic AgentsCarbohydratesEnzyme Inhibitors +6
Target Protein:
Cyclin-dependent kinase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vosoritide Approved DB11928
biotech | CAS: 1480724-61-5

Achondroplasia is an autosomal dominant genetic disease and the most common cause of dwarfism in humans.[A242277] It results from a gain-of-function missense mutation in _FGFR3_ that results in a dramatic suppression of bone growth, both in volume and in leng…

Kategori:
Amino Acids, Peptides, and ProteinsC-type Natriuretic Peptide AnalogDrugs Affecting Bone Structure and Mineralization +7
Target Protein:
Atrial natriuretic peptide receptor 2
Waktu ParuhThe mean half-life …
Vol. DistribusiThe mean apparent v…
KlirensThe mean apparent c…
Genetik -
Voxelotor Approved DB14975
small molecule | CAS: 1446321-46-5

Voxelotor is a novel hemoglobin S polymerization inhibitor for the treatment of sickle cell disease. This is a genetically inherited condition most prevalent in the Middle East, Africa, and certain parts of India. Sickle cell disease can lead to excruciating …

Kategori:
AldehydesBlood and Blood Forming OrgansCytochrome P-450 CYP2B6 Substrates +7
Target Protein:
Hemoglobin subunit alpha
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
KlirensThe apparent oral c…
Genetik -
Voxilaprevir Approved DB12026
small molecule | CAS: 1535212-07-7

Voxilaprevir is a Direct-Acting Antiviral (DAA) medication used as part of combination therapy to treat chronic Hepatitis C, an infectious liver disease caused by infection with Hepatitis C Virus (HCV). HCV is a single-stranded RNA virus that is categorized i…

Kategori:
Acids, AcyclicAmidesAmino Acids +36
Target Protein:
Genome polyproteinGenome polyprotein
Waktu Paruh33 hr [FDA Label]
Vol. Distribusi-
Klirens-
Genetik -
VP025 DB05133
small molecule

VP025, a novel drug formulation based on phospholipid microparticles incorporating phosphatidylglycerol, can inhibit neuroinflammation. VP025 may inhibit immune system activation and protect motoneurons from injury. It also shows the ability to reduce inflamm…

Target Protein:
Interleukin-1 beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VPM1002 DB15801
biotech

The bacille Calmette-Guérin (BCG) vaccine protects against severe extrapulmonary forms of tuberculosis (TB) but does not adequately protect against pulmonary TB -- the most prevalent form of TB. This recombinant BCG, VPM1002, has been created in response and …

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VPM4001 DB05089
biotech

VPM4001 is an allogeneic vaccine for treatment of prostate carcinoma. It consists of irradiated human LNCaP cells that have been genetically modified to permanently secrete interferon-? and interleukin-2 (LNCaP/IL-2/IFN-?). Interferon-? enhances presentation …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VPO-227 DB18004
small molecule | CAS: 1314873-02-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VTP-27999 DB12416
small molecule | CAS: 942142-51-0

VTP-27999 has been used in trials studying the basic science of Renal Function.

Kategori:
Acids, AcyclicAgents Acting on the Renin-Angiotensin SystemRenin Inhibitors
Target Protein:
Renin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VTX-801 DB17646
biotech

VTX-801 is a replication-deficient recombinant adeno-associated viral vector (rAAV) consisting of an AAV liver tropic capsid containing a single-stranded DNA genome carrying a shortened version of the ATP7B gene (ATP7B-minigene). It is being investigated in W…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vudalimab DB18833
biotech | CAS: 2329669-72-7

Vudalimab is under investigation in clinical trial NCT05005728 (Xmab®20717 (Vudalimab) Alone or in Combination With Chemotherapy or Targeted Therapy in Patients With Metastatic Castration-resistant Prostate Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vutrisiran Approved DB16699
biotech | CAS: 1867157-35-4

Vutrisiran is a double-stranded small interfering ribonucleic acid (siRNA) that targets wild-type and mutant transthyretin (TTR) messenger RNA (mRNA).[L42065] This siRNA therapeutic is indicated for the treatment of neuropathies associated with hereditary tra…

Kategori:
Antisense OligonucleotidesNervous SystemNucleic Acids, Nucleotides, and Nucleosides +4
Target Protein:
Transthyretin mRNA
Waktu ParuhThe median half-lif…
Vol. DistribusiBased on a populati…
KlirensThe apparent cleara…
Genetik -
VX-148 DB06103
small molecule

VX-148 is a second-generation, orally administered inhibitor of inosine monophosphate dehydrogenase (IMPDH). The IMPDH enzyme plays a key role in regulating immune response and proliferation of specific cell types, including lymphocytes. VX-148 is a developed…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Inosine-5'-monophosphate dehydrogenase 1Inosine-5'-monophosphate dehydrogenase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VX-702 DB05470
small molecule | CAS: 745833-23-2

VX-702 is a small molecule investigational oral anti-cytokine therapy for treatment of inflammatory diseases, specifically rheumatoid arthritis (RA). It acts as a p38 MAP kinase inhibitor. In the future, VX-702 may be investigated for combination with methotr…

Kategori:
AmidesBenzene Derivatives
Target Protein:
Mitogen-activated protein kinase 14Tumor necrosis factorInterleukin-1 beta +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VXA-CoV2-1 DB16433
biotech

VXA-CoV2-1 is a non-replicating adenoviral vector-based oral tableted vaccine candidate that expresses a SARS-CoV-2 antigen and dsRNA adjuvant[L30493]. This oral vaccine aims to induce immunogenicity through induction of potent serum neutralizing antibodies t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VXM01 DB17420
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VY-HTT01 DB16999
biotech

VY-HTT01 is a gene therapy designed to reduce the expression of huntingtin, thereby altering disease progression. VY-HTT01 is comprised of an adeno-associated virus capsid (AAV1) and a proprietary transgene that harnesses the canonical RNA interference pathwa…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Warfarin Approved DB00682
small molecule | CAS: 81-81-2

Warfarin is an anticoagulant drug normally used to prevent blood clot formation as well as migration. Although originally marketed as a pesticide (d-Con, Rodex, among others), Warfarin has since become the most frequently prescribed oral anticoagulant in Nort…

Kategori:
4-HydroxycoumarinsAgrochemicalsAnticoagulants +38
Target Protein:
Vitamin K epoxide reductase complex subunit 1Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
CYP2C9 VKORC1 CYP4F2 +2
Waktu ParuhR-warfarin is clear…
Vol. DistribusiVd of 0.14 L/kg.[la…
KlirensClearance of warfar…
Genetik 5 Varian
biotech

Fecal microbiota transplantation (FMT) is effective in enhancing the gut microbiota of patients experiencing a high range of disease states, including Clostridioides difficile (C. diff) infection, Crohn’s disease, and ulcerative colitis. Washed microbiota pre…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Wheat Approved DB10579
biotech

Wheat allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Willardiine DB04129
small molecule | CAS: 21416-43-3

Willardiine is a compound isolated from seeds of _Acacia willariana_.

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsPyrimidines +1
Target Protein:
Glutamate receptor 1Glutamate receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Willow bark Approved DB14691
biotech

Deskripsi belum tersedia.

Kategori:
AngiospermsBiological ProductsComplex Mixtures +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WL-1002 DB05346
small molecule

WL-1002 is developed by Winston Laboratories which is a topical cream formulation of 075% zucapaicin (also known as civamide), for the treatment of pain due to osteoarthritis.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WNT-974 DB12561
small molecule | CAS: 1243244-14-5

WNT974 has been used in trials studying the treatment of Metastatic Colorectal Cancer and Squamous Cell Carcinoma, Head And Neck.

Kategori:
Enzyme Inhibitors
Target Protein:
Protein-serine O-palmitoleoyltransferase porcupine
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Wormwood Approved DB14291
biotech

Wormwood is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
LipidsOils
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Wortmannin DB08059
small molecule | CAS: 19545-26-7

Wortmannin is a steroid metabolite of _Penicillium funiculosum_ and _Talaromyces wortmannii_ fungi. This drug acts as a nonspecific, covalent inhibitor of phosphoinositide 3-kinase enzymes (PI3Ks).

Kategori:
AndrostadienesAndrostanesAndrostenes +16
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformSerine/threonine-protein kinase PLK1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WP-1122 DB17192
small molecule

WP-1122 is a prodrug of 2-deoxy-D-glucose (2-DG). It was granted FDA orphan designation for the treatment of glioblastoma multiforme.[L47361]

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WP-1301 DB17702
biotech | CAS: 1609460-62-9

WP1301 is a synthetic peptide derived from hFVIII. It binds to an MHC class II molecule and is recognized by a Factor VIII-specific T cell.[L46138]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WT-1 A1 DB17352
small molecule | CAS: 852243-39-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WU-CART-007 DB18617
biotech

WU-CART-007 consists of allogeneic, fratricide-resistant genetically modified T cells transduced with a 2nd generation 4-1BB-CD3z chimeric antigen receptor targeting human CD7.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
WX-UK1 DB05476
small molecule | CAS: 255374-84-6

WX-UK1 is a 3-amidinophenylalanine-based non-cytotoxic small molecule that belongs to a new class of drugs. In animal models, WX-UK1 blocks tumor cell invasion, metastasis and primary tumor growth by inhibiting serine proteases and the urokinase Plasminogen A…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +1
Target Protein:
Urokinase plasminogen activator surface receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xaluritamig DB18137
biotech

Xaluritamig is a novel humanized bispecific T cell recruiting antibody cross-reactive to human and nonhuman primate STEAP1 and CD3.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Xanomeline Approved DB15357
small molecule | CAS: 131986-45-3

Schizophrenia is a complex disease involving a number of different neurotransmitters, including serotonin, dopamine, and acetylcholine.[A264509] Positive symptoms (e.g. hallucinations, delusions) have traditionally been attributed to increased dopaminergic ac…

Kategori:
Autonomic AgentsCentral Nervous System AgentsCholinergic Agents +18
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M2 +2
Waktu ParuhThe half-life of xa…
Vol. DistribusiThe apparent volume…
KlirensThe apparent cleara…
Genetik -
Xanthan gum Approved DB11253
small molecule | CAS: 11138-66-2

Xanthan gum is a polysaccharide gum derived from* Xanthomonas campestris* by a pure-culture fermentation process and purified by recovery with isopropyl alcohol. The major constituents include D-glucose, D-mannose, and D-glucuronic acid. Xanthan gum is a dire…

Kategori:
AntigensAntigens, BacterialBiological Factors +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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