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11778

Total database: 17430
Struktur (SMILES)
8554 (72.6%)
Target
6383 (54.2%)
Genomik
96 (0.8%)
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11778 (100.0%)

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Halaman 131 / 236
JNJ-75276617 DB17574
small molecule

JNJ-75276617 is under investigation in clinical trial NCT05453903 (A Study of JNJ-75276617 in Combination With Acute Myeloid Leukemia (AML) Directed Therapies).

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JNT-517 DB19305
small molecule | CAS: 2837993-05-0

Deskripsi belum tersedia.

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Jojoba oil Approved DB14252
biotech | CAS: 61789-91-1

Jojoba oil is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Kategori:
Biological ProductsCosmeticsLipids +3
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small molecule | CAS: 40922-77-8

Deskripsi belum tersedia.

Kategori:
Anti-Bacterial AgentsLactonesMacrolides +1
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JPC-3210 DB15609
small molecule | CAS: 1609655-35-7

JPC-3210 is a potent antimalarial agent. It is an erythrocytic schizonticide with potent in vitro antimalarial activity against multidrug-resistant _Plasmodium falciparum_ lines, low cytotoxicity, potent in vivo efficacy against murine malaria, and favourable…

Kategori:
AntimalarialsAntiviral AgentsBenzene Derivatives
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JQ1 DB17021
small molecule | CAS: 1268524-70-4

First-in-class potent and selective inhibitor of the BRD4 signaling pathway.[A252967]

Target Protein:
Bromodomain-containing protein 4Bromodomain testis-specific protein
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JS-K DB17257
small molecule | CAS: 205432-12-8

Deskripsi belum tersedia.

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JSM 6427 DB06139
small molecule

JSM 6427 is the first small molecule alpha5beta1 integrin receptor antagonist of its kind to be developed. It has been biologically validated for therapeutic use in the prevention and treatment of wet AMD, the leading cause of blindness in people over the age…

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small molecule | CAS: 244218-93-7

An antagonist of nociceptin receptor and analgesic agent, evaluated for its use in cancer treatment.[A253027]

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Nociceptin receptor
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JTT-251 DB18174
small molecule | CAS: 1627957-25-8

Deskripsi belum tersedia.

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Juglans californica pollen Approved DB10397
biotech

Juglans californica pollen is the pollen of the Juglans californica plant. Juglans californica pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Juniperus californica pollen Approved DB10473
biotech

Juniperus californica pollen is the pollen of the Juniperus californica plant. Juniperus californica pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Juniperus monosperma pollen Approved DB10727
biotech

Juniperus monosperma pollen is the pollen of the Juniperus monosperma plant. Juniperus monosperma pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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biotech

Juniperus occidentalis pollen is the pollen of the Juniperus occidentalis plant. Juniperus occidentalis pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Juniperus osteosperma pollen Approved DB10730
biotech

Juniperus osteosperma pollen is the pollen of the Juniperus osteosperma plant. Juniperus osteosperma pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Juniperus pinchotii pollen Approved DB10728
biotech

Juniperus pinchotii pollen is the pollen of the Juniperus pinchotii plant. Juniperus pinchotii pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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Juniperus scopulorum pollen Approved DB10729
biotech

Juniperus scopulorum pollen is the pollen of the Juniperus scopulorum plant. Juniperus scopulorum pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
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small molecule

JZP-386 is a deuterium-containing analog of sodium oxybate. Its safety, pharmacokinetics and pharmacodynamics were evaluated in clinical trial NCT02215499.

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K-00546 DB07664
small molecule | CAS: 443798-47-8

Deskripsi belum tersedia.

Target Protein:
Vascular endothelial growth factor receptor 1Cyclin-dependent kinase 1Cyclin-dependent kinase 2 +5
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K-252a DB02152
small molecule | CAS: 97161-97-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsEnzyme InhibitorsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
Dual specificity mitogen-activated protein kinase kinase 1Hepatocyte growth factor receptor
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K-777 DB17760
small molecule | CAS: 502960-90-9

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +5
Target Protein:
Cruzipain
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KAb201 DB17210
biotech

Deskripsi belum tersedia.

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KAHR-102 DB17427
biotech

KAHR-102 is a dual signaling protein fusing cytotoxic T-lymphocyte-associated protein 4 (CTLA-4) to the Fas-ligand (FasL).

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KAI-1678 DB16211
biotech | CAS: 1041004-14-1

KAI-1678 is under investigation in clinical trial NCT01106716 (Safety and Efficacy Study of KAI-1678 to Treat Pain in Subjects With Postherpetic Neuralgia).

Kategori:
Amino Acids, Peptides, and ProteinsProtein Kinase C-epsilon, antagonists & inhibitors
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Kallidinogenase DB13197
biotech | CAS: 9001-01-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +17
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Kanamycin Approved DB01172
small molecule | CAS: 59-01-8

Kanamycin (also known as kanamycin A) is an aminoglycoside bacteriocidal antibiotic, available in oral, intravenous, and intramuscular forms, and used to treat a wide variety of infections. Kanamycin is isolated from the bacterium Streptomyces kanamyceticus a…

Kategori:
Agents that produce neuromuscular block (indirect)Alimentary Tract and MetabolismAminoglycoside Antibacterials +16
Target Protein:
30S ribosomal protein S1216S ribosomal RNA
Waktu Paruh2.5 hours
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KAND567 DB16511
small molecule | CAS: 911715-90-7

KAND567, a small molecule, blocks the fractaline (CX3CL1) receptor, which mediates the immune system response to inflammation[L32908]. Because COVID-19 involves cytotoxic cells associated with this pathway, KAND567 is currently being tested as a treatment for…

Kategori:
Experimental Unapproved Treatments for COVID-19
Target Protein:
CX3C chemokine receptor 1
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Kaolin Approved DB01575
small molecule | CAS: 1332-58-7

Kaolin is a layered silicate mineral. Kaolin is used in ceramics, medicine, coated paper, as a food additive, in toothpaste, as a light diffusing material in white incandescent light bulbs, and in cosmetics. Until the early 1990s it was the active substance o…

Kategori:
Alimentary Tract and MetabolismAluminium CompoundsAluminum Silicates +11
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KB-141 DB03176
small molecule | CAS: 219691-94-8

An anticholesteremic agent.

Kategori:
Acids, CarbocyclicBenzene DerivativesEthers +2
Target Protein:
Thyroid hormone receptor alphaThyroid hormone receptor beta
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KB3305 DB06349
small molecule | CAS: 639520-46-0

KB3305 is an investigational liver selective antagonist for the glucocorticoid receptor, developed by Karo Bio for the treatment of Type 2 Diabetes.

Kategori:
17-KetosteroidsAdrenal Cortex HormonesBile Acids and Salts +11
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KB407 DB18223
biotech

Deskripsi belum tersedia.

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KBP-COVID-19 DB15858
biotech

The KBP-201 COVID-19 Vaccine was developed by British American Tobacco’s (BAT) U.S. biotech subsidiary, Kentucky BioProcessing (KBP). KBP cloned COVID-19’s genetic sequence, identified a potential antigen, and then inserted it into tobacco plants for reproduc…

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KC706 DB05157
small molecule

KC706 is a novel anti-inflammatory drug that works by inhibiting the activity of p38 MAP kinase. KC706 holds potential to treat inflammatory conditions such as rheumatoid arthritis, psoriasis, inflammatory bowel disease and cardiovascular disease.

Target Protein:
Mitogen-activated protein kinase 14Mitogen-activated protein kinase 11Mitogen-activated protein kinase 12 +1
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KD3010 DB05188
small molecule | CAS: 934760-90-4

KD3010 is a small molecule peroxisome proliferator-activator receptor delta (PPAR Delta) agonist for the treatment of metabolic disorders, including obesity.

Kategori:
AmidesPPAR delta, antagonists & inhibitorsSulfones +1
Target Protein:
Peroxisome proliferator-activated receptor delta
Waktu Paruh-
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KD7040 DB05214
small molecule

KD7040 is a topically-delivered inducible nitric oxide synthase (iNOS) inhibitor for the treatment of neuropathic pain. The KD7040 IND was filed in 4Q06, and a Phase Ib clinical trial began 2Q07. It is being developed by Kalypsys.

Target Protein:
Nitric oxide synthase, inducible
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KDT-3594 DB17085
small molecule

KDT-3594 is a non-ergot dopamine receptor agonist developed by Kissei Pharmaceutical.

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Kelatorphan DB08040
small molecule | CAS: 92175-57-0

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsCentral Nervous System Agents +4
Target Protein:
Aminopeptidase NGlutamyl aminopeptidaseLeukotriene A-4 hydrolase
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KER-047 DB19111
small molecule | CAS: 2248154-85-8

KER-047 is under investigation in clinical trial NCT05927012 (A Study to Evaluate the Safety and Preliminary Efficacy of a Response-guided Dose Titration of KER-047 in the Treatment of Functional IDA (Iron Deficiency Anemia).).

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Ketamine Approved DB01221
small molecule | CAS: 6740-88-1

Ketamine is an NMDA receptor antagonist with a potent anesthetic effect.[A31869] It was developed in 1963 as a replacement for phencyclidine (PCP) by Calvin Stevens at Parke Davis Laboratories. It started being used for veterinary purposes in Belgium and in 1…

Kategori:
Agents producing tachycardiaAmino AcidsAmino Acids, Acidic +35
Target Protein:
Glutamate receptor ionotropic, NMDA 3A5-hydroxytryptamine receptor 3ANeuronal acetylcholine receptor subunit alpha-7 +11
Waktu ParuhThe reported half-l…
Vol. DistribusiThe apparent volume…
KlirensThe clearance rate …
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Ketanserin DB12465
small molecule | CAS: 74050-98-9

Ketanserin has been investigated for the treatment of Septic Shock, Severe Sepsis, and Diabetic Foot Ulcer.

Kategori:
Antidepressive AgentsAntihypertensive AgentsAntiplatelet agents +11
Target Protein:
5-hydroxytryptamine receptor 2A
Waktu Paruh-
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Ketazolam Approved DB01587
small molecule | CAS: 27223-35-4

Ketazolam is a benzodiazepine derivative with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant activity. Ketazolam is not approved in Canada or America.

Kategori:
Anti-Anxiety AgentsBenzazepinesBenzodiazepines and benzodiazepine derivatives +16
Target Protein:
GABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu Paruh26-200 hours
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Ketobemidone DB06738
small molecule | CAS: 469-79-4

Ketobemidone is a powerful opioid analgesic. It also has some NMDA-antagonist properties. This makes it useful for some types of pain that don't respond well to other opioids. The most commonly cited equalisation ratio for analgesic doses is 25 mg of ketobemi…

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +20
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhPlasma half-life: 2…
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Ketoconazole Approved DB01026
small molecule | CAS: 65277-42-1

Ketoconazole is an imidazole antifungal agent used in the prevention and treatment of a variety of fungal infections.[FDA Label] It functions by preventing the synthesis of ergosterol, the fungal equivalent of cholesterol, thereby increasing membrane fluidity…

Kategori:
14-alpha Demethylase InhibitorsAgents causing hyperkalemiaAnti-Infective Agents +55
Target Protein:
Lanosterol 14-alpha demethylaseLanosterol 14-alpha demethylaseSteroid 17-alpha-hydroxylase/17,20 lyase +5
Waktu ParuhKetoconazole experi…
Vol. DistribusiKetoconazole has an…
KlirensKetoconazole has an…
Genetik -
small molecule | CAS: 1297537-33-7

Ketodarolutamide, a nonsteroidal antiandrogen (NSAA), is the major active metabolite of [darolutamide].

Kategori:
AntiandrogensAntiandrogens, non-steroidal
Target Protein:
Androgen receptor
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Ketoprofen Approved DB01009
small molecule | CAS: 22071-15-4

Ketoprofen, a propionic acid derivative, is a nonsteroidal anti-inflammatory agent (NSAIA) with analgesic and antipyretic properties.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +38
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1C-X-C chemokine receptor type 1
Waktu ParuhConventional capsul…
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Klirens* Oral-dose cl=6.9 …
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Ketorolac Approved DB00465
small molecule | CAS: 74103-06-3

Ketorolac is a Non-steroidal anti-inflammatory drug (NSAID) and is commercially available as an oral tablet, injectable, nasal spray and as an ophthalmic solution.[L6358][L6508][L11055][L3674][L11070] It's analgesic properties make it a useful pain manage…

Kategori:
Acetic Acid Derivatives and Related SubstancesAgents causing hyperkalemiaAgents that produce hypertension +26
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1
Waktu ParuhKetorolac trometham…
Vol. DistribusiThe apparent volume…
KlirensThe plasma clearanc…
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Ketotifen Approved DB00920
small molecule | CAS: 34580-13-7

Ketotifen is a benzocycloheptathiophene derivative[A231204] with potent antihistaminic and mast cell stabilizing properties. It has a similar structure to some other first-generation antihistamines such as [cyproheptadine] and [azatadine].[A231204] Ketotif…

Kategori:
Anti-Allergic AgentsAnti-Asthmatic AgentsAntihistamine Drugs +15
Target Protein:
Histamine H1 receptor6-phosphogluconate dehydrogenase, decarboxylating
Waktu ParuhKetotifen clearance…
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KF-0210 DB17476
small molecule

KF-0210 is a small molecule developed by Keythera Pharmaceuticals. It is being investigated for cancers.

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KF-1601 DB18297
small molecule | CAS: 2699634-21-2

Deskripsi belum tersedia.

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KH064 DB04287
small molecule | CAS: 393569-31-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +2
Target Protein:
Phospholipase A2, membrane associated
Waktu Paruh-
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