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12560

Total database: 17430
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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 131 / 252
IMMU-114 DB18458
biotech

IMMU-114 is antibody-drug conjugate consisting of humanized anti-HLA-DR IgG4 monoclonal antibody specific for alpha-chain linked to SN-38 via a CL2A linker.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
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biotech | CAS: 1807503-77-0

Deskripsi belum tersedia.

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Imolamine DB09284
small molecule | CAS: 318-23-0

Imolamine is a compound with a molecular weight of 260.33 g/mol with the formula diethyl[2-{5-imino-3-phenyl-4,5-dihydro-1,2,3-oxadiazol,-4-yl)ethyl]amine. It is developed under the brand name Coremax by Novartis consumer health SA.

Kategori:
Cardiac TherapyCardiovascular AgentsOxazoles +2
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Implitapide DB04852
small molecule | CAS: 177469-96-4

Implitapide is a microsomal triglyceride transfer protein (MTP)-inhibitor.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Microsomal triglyceride transfer protein large subunit
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Imrecoxib DB12354
small molecule | CAS: 395683-14-4

Imrecoxib has been used in trials studying the treatment of Knee Osteoarthritis.

Kategori:
AnionsElectrolytesHydrogen Sulfide +2
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
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Imsidolimab DB16658
biotech | CAS: 2102543-86-0

Imsidolimab is under investigation in clinical trial NCT03633396 (A Study to Evaluate the Efficacy and Safety of ANB019 in Subjects With Palmoplantar Pustulosis).

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IMT-288 DB19068
small molecule | CAS: 637771-94-9

IMT-288 is under investigation in clinical trial NCT01730638 (Immunotep for Patients With Medullary Thyroid Carcinoma.).

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
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IMT504 DB17792
biotech

IMT504, a non-CpG 24-mer oligodeoxynucleotide, is an immunomodulatory oligonucleotide currently being investigated as a rabies vaccine.[A259467]

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
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IN01 DB16434
biotech

The IN01 Vaccine, sponsored by the Instituto Oncologico Dr Rosell, IN3BIO, and PANGAEA, is a compound containing recombinant bacteria[L30543]. These cultures contain EGF-4-EGF with the cholera toxin B-subunit domain G33D sequence[L30543]. Administration of th…

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biotech

Developed by Sinopharm's Wuhan Institute of Biological Products co., this vaccine consists of the WIV04 strain of SARS-CoV-2. This strain was isolated from a patient in Wuhan, cultivated in a Vero cell line, and then subsequently inactivated using B-propiolac…

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biotech

The SARS-CoV-2 Inactivated Vaccine is a purified vaccine that contains multiple antigens from the virus and is inactivated in Vero Cells[A219758]. This vaccine specifically was developed in collaboration with the Chinese Academy of Medical Sciences, West Chin…

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Inalimarev DB17332
biotech | CAS: 685563-13-7

Deskripsi belum tersedia.

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Inarigivir DB15062
small molecule | CAS: 475650-36-3

Inarigivir is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

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small molecule | CAS: 942123-43-5

Inarigivir soproxil is under investigation in clinical trial NCT03434353 (Study to Evaluate the Antiviral Activity of Inarigivir (GS-9992) Plus Tenofovir Alafenamide (TAF) for 12 Weeks in Adults With Chronic Hepatitis B (CHB)).

Target Protein:
Nucleotide-binding oligomerization domain-containing protein 2
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biotech

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Inavolisib Approved DB15275
small molecule | CAS: 2060571-02-8

_PIK3CA_ is one of the most frequently mutated oncogenes, with the resulting mutated p110? protein it encodes playing a central role in tumor cell proliferation.[A264563] Chemotherapeutic agents targeting the PI3K p110? catalytic subunit have shown antitumor …

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2B6 InducersCytochrome P-450 CYP2B6 Inducers (strength unknown) +4
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
Waktu ParuhThe elimination hal…
Vol. DistribusiThe apparent volume…
KlirensThe total clearance…
Genetik -
Inbakicept DB16479
biotech | CAS: 2135939-52-3

Inbakicept is a dimeric human IL-15 receptor ? (IL-15R?) sushi domain/human IgG1 Fc fusion protein. It is one of the active ingredients in Anktiva, a combination product also containing [nogapendekin alfa], where a single inbakicept is complexed with two noga…

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsExperimental Unapproved Treatments for COVID-19 +4
Target Protein:
Interleukin-2 receptor subunit betaCytokine receptor common subunit gamma
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Incadronic acid DB06255
small molecule | CAS: 124351-85-5

Incadronate, or YM-175,[A202769] is a nitrogen containing bisphosphonate. Along with being investigated to treat hypercalcemia of malignancy,[A202862] it has also been investigated in the treatment of myeloma, leukemia, and other cancers.[A14426,A14431,A14427…

Kategori:
Antineoplastic AgentsBisphosphonatesBone Density Conservation Agents +2
Target Protein:
Farnesyl pyrophosphate synthaseCaspase-3Caspase-4 +1
Waktu ParuhIncadronate has a b…
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INCB-054329 DB16894
small molecule | CAS: 1628607-64-6

Deskripsi belum tersedia.

Kategori:
Antineoplastic Agents
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INCB-057643 DB16054
small molecule | CAS: 1820889-23-3

INCB-057643 is under investigation in clinical trial NCT02959437 (Azacitidine Combined With Pembrolizumab and Epacadostat in Subjects With Advanced Solid Tumors (ECHO-206)).

Kategori:
AcidsAcids, NoncarboxylicAntineoplastic Agents +1
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INCB-086550 DB18901
small molecule | CAS: 2230911-59-6

INCB-086550 is under investigation in clinical trial NCT04629339 (Study of INCB086550 in Select Solid Tumors).

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INCB-9471 DB12960
small molecule | CAS: 869769-98-2

INCB-9471 is a novel, orally available CCR5 antagonist that is part of a new class of drugs to treat HIV/AIDS. It is a potent, selective inhibitor of the HIV-1 virus.

Kategori:
Receptors, CCR4, antagonists & inhibitors
Target Protein:
C-C chemokine receptor type 5
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INCB052793 DB17567
small molecule

Deskripsi belum tersedia.

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INCB13739 DB05064
small molecule

INCB13739 is developed as a new treatment for type 2 diabetes. It is an orally available small molecule inhibitor of 11beta-HSD1 (11-beta hydroxysteroid dehydrogenase type 1). 11beta-HSD1 is an enzyme that appears to be critical to the development of type 2…

Kategori:
11-beta-Hydroxysteroid Dehydrogenase Type 1, antagonists & inhibitorsAmidesSulfones +1
Target Protein:
11-beta-hydroxysteroid dehydrogenase 1
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INCB3284 DB05130
small molecule

INCB3284 is a CCR2 antagonist for Inflammation-driven Diseases.

Kategori:
Acids, CarbocyclicAmidesAmino Acids +3
Target Protein:
C-C chemokine receptor type 2
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INCB7839 DB05033
small molecule

INCB7839 is a novel, orally available ADAM metalloprotease inhibitor that is designed to block activation of the epidermal growth factor (EGFR) pathways. It represents a potentially important new class of targeted breast cancer therapy. It has shown promising…

Target Protein:
Disintegrin and metalloproteinase domain-containing protein 9
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Inclacumab DB12246
biotech | CAS: 1256258-86-2

Inclacumab has been used in trials studying the treatment and prevention of Myocardial Infarction, Peripheral Arterial Disease (PAD), and Coronary Heart Disease, Graft Occlusion, Vascular.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
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Inclisiran Approved DB14901
biotech | CAS: 1639324-58-5

Inclisiran is a long-acting, synthetic small interfering RNA (siRNA) directed against proprotein convertase subtilisin-kexin type 9 (PCSK9), which is a serine protease that regulates plasma low-density lipoprotein cholesterol (LDL-C) levels. By binding to PCS…

Kategori:
Antisense Elements (Genetics)Compounds used in a research, industrial, or household settingDiagnostic Uses of Chemicals +16
Target Protein:
Proprotein convertase subtilisin/kexin type 9
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe apparent volume…
KlirensThere is limited in…
Genetik -
biotech

Deskripsi belum tersedia.

Kategori:
Adjuvants, ImmunologicAlcoholsCarbohydrates +7
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Incyclinide DB11647
small molecule | CAS: 15866-90-7

Incyclinide has been used in trials studying the treatment of HIV Infection, AIDS-related Kaposi Sarcoma, Brain and Central Nervous System Tumors, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Naphthacenes
Target Protein:
72 kDa type IV collagenase
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Indacaterol Approved DB05039
small molecule | CAS: 312753-06-3

Indacaterol is a novel, ultra-long-acting, rapid onset ?(2)-adrenoceptor agonist developed for Novartis for the once-daily management of asthma and chronic obstructive pulmonary disease. It was approved by the European Medicines Agency (EMA) on 30 November 20…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +17
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIndacaterol serum c…
Vol. DistribusiAfter intravenous i…
KlirensRenal clearance of …
Genetik -
Indalpine DB08953
small molecule | CAS: 63758-79-2

Indalpine was one of the first selective serotonin reuptake inhibitors to reach the American market. It was initially marketed by Pharmuka. However, after the emergence of widespread concern regarding adverse effects caused by SSRIs, and reported hematologica…

Kategori:
Antidepressive AgentsCentral Nervous System AgentsCentral Nervous System Depressants +16
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Indanazoline DB13827
small molecule | CAS: 40507-78-6

Deskripsi belum tersedia.

Kategori:
Nasal PreparationsSympathomimetics, Plain
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small molecule

Deskripsi belum tersedia.

Target Protein:
Carbonic anhydrase 2Carbonic anhydrase 14Carbonic anhydrase 12 +1
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Indapamide Approved DB00808
small molecule | CAS: 26807-65-8

The most significant modifiable risk factor for cardiovascular disease and the most prominent contributor to all-cause mortality is hypertension.[A204155] Characterized by an office blood pressure of ?140/90, hypertension is pervasive and impacts an estimated…

Kategori:
AmidesAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +26
Target Protein:
Solute carrier family 12 member 3Potassium voltage-gated channel subfamily KQT member 1
Waktu ParuhIndapamide is chara…
Vol. DistribusiSome sources report…
KlirensIndapamide's renal …
Genetik -
Indatraline DB17032
small molecule | CAS: 86939-10-8

Indatraline is a nonselective monoamine reuptake inhibitor.[A253022]

Kategori:
AminesIndenes
Target Protein:
Sodium-dependent dopamine transporter
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biotech | CAS: 1238517-16-2

Indatuximab ravtansine is under investigation in clinical trial NCT01001442 (Safety and Dose Determining Multi-dose Study of BT062 in Patients With Relapsed or Refractory Multiple Myeloma).

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAntibodies +10
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Indecainide Approved DB00192
small molecule | CAS: 74517-78-5

Indecainide is a rarely used antidysrhythmic. Indecainide has local anesthetic activity and belongs to the membrane stabilizing (Class 1) group of antiarrhythmic agents; it has electrophysiologic effects characteristic of the IC class of antiarrhythmics.

Target Protein:
Sodium channel protein type 5 subunit alpha
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Indeglitazar DB07724
small molecule | CAS: 835619-41-5

Deskripsi belum tersedia.

Target Protein:
Peroxisome proliferator-activated receptor alphaPeroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor delta +1
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Indenolol DB08952
small molecule | CAS: 60607-68-3

Indenolol is a drug of the beta-adrenergic blocker class.

Kategori:
Adrenergic AgentsAdrenergic AntagonistsAdrenergic beta-Antagonists +15
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Indian frankincense Approved DB14275
biotech

Indian frankincense is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

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Indibulin DB06169
small molecule | CAS: 204205-90-3

Deskripsi belum tersedia.

Kategori:
AcetatesAcids, AcyclicAmides +1
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Indigotindisulfonic acid Approved DB11577
small molecule | CAS: 483-20-5

Indigotindisulfonic acid is a blue-colored dye with a variety of uses.[A32490,A32491,A32492,L2222] Its salt form, indigotindisulfonate sodium, is also known as indigo carmine, indigotine or FD&C Blue #2. This compound is an acid-base indicator and is used in …

Kategori:
Coloring AgentsCompounds used in a research, industrial, or household settingDiagnostic Agents +5
Target Protein:
Alpha adrenergic receptor
Waktu ParuhIn healthy adults g…
Vol. DistribusiThe volume of distr…
KlirensIn healthy adults g…
Genetik -
Indinavir Approved DB00224
small molecule | CAS: 150378-17-9

A potent and specific HIV protease inhibitor that appears to have good oral bioavailability. [PubChem]

Kategori:
Agents Causing Muscle ToxicityAnti-HIV AgentsAnti-Infective Agents +33
Target Protein:
Gag-Pol polyproteinPol polyprotein
Waktu Paruh1.8 (± 0.4) …
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Indiplon DB12590
small molecule | CAS: 325715-02-4

Indiplon has been used in trials studying the treatment of Insomnia and Depression.

Kategori:
BenzazepinesCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1
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Indirubin DB12379
small molecule | CAS: 479-41-4

Indirubin is under investigation in clinical trial NCT01735864 (Dosage Determination Trial for Indigo Naturalis Extract in Oil Ointment).

Kategori:
Antibiotics, AntineoplasticAntineoplastic AgentsColoring Agents +4
Target Protein:
Cytochrome P450 1A1Aryl hydrocarbon receptor
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small molecule

Deskripsi belum tersedia.

Kategori:
AminesHeterocyclic Compounds, Fused-RingHydroxylamines
Target Protein:
Cyclin-dependent kinase 5 activator 1Cyclin-dependent kinase 2Aryl hydrocarbon receptor +3
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small molecule | CAS: 244021-67-8

Deskripsi belum tersedia.

Target Protein:
Glycogen phosphorylase, muscle formCell division control protein 2 homolog
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Indisulam DB06370
small molecule | CAS: 165668-41-7

Deskripsi belum tersedia.

Kategori:
AmidesAntineoplastic AgentsCarbonic Anhydrase Inhibitors +15
Target Protein:
Carbonic anhydrase 9
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Indium DB11659
small molecule | CAS: 7440-74-6

Indium has been used in trials studying the basic science of Clear Cell Renal Cell Carcinoma.

Kategori:
AnionsElectrolytesElements +5
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