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6694

Total database: 17430
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4518 (67.5%)
Target
3751 (56.0%)
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81 (1.2%)
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6694 (100.0%)

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Halaman 130 / 134
Vibegron Approved DB14895
small molecule | CAS: 1190389-15-1

Vibegron is a potent, selective beta-3 adrenergic receptor (?3) agonist that relaxes the detrusor smooth muscle of the bladder, thereby increasing bladder capacity.[L28305] Vibegron was first approved in Japan in September 2018 for the treatment of overactive…

Kategori:
Adrenergic AgonistsAdrenergic beta-3 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-3 adrenergic receptor
Waktu ParuhThe terminal plasma…
Vol. DistribusiThe mean apparent v…
KlirensThere is limited in…
Genetik -
Vibostolimab DB16420
biotech | CAS: 2231305-30-7

Vibostolimab is under investigation in clinical trial NCT04303169 (Substudy 02C: Safety and Efficacy of Pembrolizumab in Combination With Investigational Agents or Pembrolizumab Alone in Participants With Stage III Melanoma Who Are Candidates for Neoadjuvant …

Waktu Paruh-
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Genetik -
biotech | CAS: 1704499-30-8

_Vibrio cholerae_ CVD 103-HgR strain live antigen is a component of Vaxchora, an oral vaccine for immunization against _Vibrio cholerae_ serogroup O1.[L12801] Cholera is an acute bacterial disease of the small intestine caused by _Vibrio cholerae_, which is g…

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +3
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiPharmacokinetic inf…
KlirensPharmacokinetic inf…
Genetik -
Vidarabine Approved DB00194
small molecule | CAS: 24356-66-9

A nucleoside antibiotic isolated from Streptomyces antibioticus. It has some antineoplastic properties and has broad spectrum activity against DNA viruses in cell cultures and significant antiviral activity against infections caused by a variety of viruses su…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntimetabolites +17
Target Protein:
Adenosine receptor A2bDNA polymerase catalytic subunitThymidine kinase +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vidofludimus DB15446
small molecule | CAS: 717824-30-1

Vidofludimus is under investigation in clinical trial NCT03722576 (Vidofludimus Calcium for Primary Sclerosing Cholangitis).

Kategori:
Acids, AcyclicBenzene Derivatives
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VidPrevtyn Beta Approved DB16427
biotech

VidPrevtyn Beta is an adjuvanted, recombinant COVID-19 vaccine developed collaboratively by GlaxoSmithKline (GSK) and Sanofi Pasteur.[L49691] It comprises a recombinant SARS-CoV-2 spike protein (B.1.351 strain) - produced by recombinant DNA technology using a…

Kategori:
Biological ProductsComplex MixturesCOVID-19 Vaccines +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vidupiprant DB12272
small molecule | CAS: 1169483-24-2

Vidupiprant has been used in trials studying the treatment and basic science of Asthma.

Kategori:
Acids, CarbocyclicAmidesSulfones +1
Target Protein:
Prostaglandin D2 receptor 2Prostaglandin D2 receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vidutolimod DB17500
biotech | CAS: 147063-80-7

Vidutolimod is a Toll-like receptor 9 (TLR9) agonist. It is an investigational cancer vaccine.

Waktu Paruh-
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Genetik -
Vigabatrin Approved DB01080
small molecule | CAS: 68506-86-5

Vigabatrin is an analog of gamma-aminobutyric acid ([GABA]), the main inhibitory neurotransmitter in the central nervous system, used in the treatment of refractory seizures and infantile spasms.[L13616] It irreversibly inhibits the enzyme responsible for GAB…

Kategori:
Acids, AcyclicAminobutyratesAnti-epileptic Agent +15
Target Protein:
4-aminobutyrate aminotransferase, mitochondrial
Waktu ParuhThe terminal half-l…
Vol. DistribusiVigabatrin is widel…
KlirensThe oral clearance …
Genetik -
Vilamakitug DB18978
biotech | CAS: 2458202-06-5

Vilamakitug is under investigation in clinical trial NCT05201352 (Evaluation of Efficacy of Trifluridine/tipiracil Plus an Anti-il-1? True Human Antibody Versus Trifluridine/tipiracil Plus Placebo in Metastatic Colorectal Cancer Patients After Failure of Oxal…

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Genetik -
Vilanterol Approved DB09082
small molecule | CAS: 503068-34-6

Vilanterol is a selective long-acting ?2-adrenergic agonist (LABA) with inherent 24-hour activity for the once-daily treatment of COPD and asthma.[A7737] This is in response to the need for longer-acting ?2-adrenergic agonists to overcome poor patient complia…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +19
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhThe effective half-…
Vol. DistribusiFollowing intraveno…
KlirensFollowing intraveno…
Genetik -
Vilastobart DB19327
biotech | CAS: 2760549-50-4

Vilastobart is under investigation in clinical trial NCT04896697 (Vilastobart (XTX101) Monotherapy and Vilastobart and Atezolizumab Combination Therapy in Advanced Solid Tumors).

Waktu Paruh-
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Vilazodone Approved DB06684
small molecule | CAS: 163521-12-8

Vilazodone is a novel compound with combined high affinity and selectivity for the 5-hydroxytryptamine (5-HT) transporter and 5-HT(1A) receptors[Label,A177622]. Vilazodone may also be associated with less sexual dysfunction and weight gain[A6947]. Vilazodone …

Kategori:
Agents that produce hypertensionAntidepressive AgentsAntidepressive Agents Indicated for Depression +26
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1A
Waktu Paruh25 hours[Label,A384…
Vol. DistribusiVilazodone's volume…
KlirensClearance of vilazo…
Genetik -
Vildagliptin Approved DB04876
small molecule | CAS: 274901-16-5

Vildagliptin (LAF237) is an orally active antihyperglycemic agent that selectively inhibits the dipeptidyl peptidase-4 (DPP-4) enzyme. It is used to manage type II diabetes mellitus, where GLP-1 secretion and insulinotropic effects are impaired.[A232488] By i…

Kategori:
Agents causing angioedemaAlimentary Tract and MetabolismBlood Glucose Lowering Agents +11
Target Protein:
Dipeptidyl peptidase 4
Waktu ParuhThe mean eliminatio…
Vol. DistribusiThe mean volume of …
KlirensAfter intravenous a…
Genetik -
Vilobelimab DB16416
biotech | CAS: 2250440-41-4

Vilobelimab is a chimeric monoclonal immunoglobulin G4 (IgG4) antibody that binds to the soluble form of human C5a with high affinity. It consists of mouse anti-human complement factor 5a (C5a) monoclonal binding sites (variable regions of heavy and light cha…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Complement C5
Waktu ParuhThe elimination hal…
Vol. DistribusiNo information is a…
KlirensNo information is a…
Genetik -
Viloxazine Approved DB09185
small molecule | CAS: 46817-91-8

Viloxazine is a selective norepinephrine reuptake inhibitor.[L41685] For decades, an immediate-release formulation of viloxazine has been used in Europe as an antidepressant. It was first approved in the UK in 1974; however, the immediate-release formulation …

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +46
Target Protein:
Sodium-dependent noradrenaline transporter5-hydroxytryptamine receptor 2B5-hydroxytryptamine receptor 2C +10
Waktu ParuhThe mean (± SD) hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance rate …
Genetik -
Viltolarsen Approved DB15005
biotech | CAS: 2055732-84-6

Duchenne muscular dystrophy (DMD) is an X-linked recessive allelic disorder characterized by a lack of functional dystrophin protein, which leads to progressive ambulatory, pulmonary, and cardiac function and is invariably fatal. A related, albeit a less seve…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD gene (exon 53 viltolarsen target site)
Waktu ParuhViltolarsen has a r…
Vol. DistribusiViltolarsen has a s…
KlirensViltolarsen has a r…
Genetik -
Vincristine Approved DB00541
small molecule | CAS: 57-22-7

Vincristine is an antitumor vinca alkaloid isolated from Vinca Rosea. It is marketed under several brand names, many of which have different formulations such as Marqibo (liposomal injection) and Vincasar. Vincristine is indicated for the treatment of acute l…

Kategori:
Agents Causing Muscle ToxicityAlkaloidsAntimitotic Agents +33
Target Protein:
Tubulin beta chainTubulin alpha-4A chain
Waktu ParuhWhen intravenously …
Vol. DistribusiWithin 15 to 30 min…
Klirens-
Genetik -
Vindesine Approved DB00309
small molecule | CAS: 53643-48-4

Vinblastine derivative with antineoplastic activity against cancer. Major side effects are myelosuppression and neurotoxicity. Vindesine is used extensively in chemotherapy protocols (antineoplastic combined chemotherapy protocols).

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +19
Target Protein:
Tubulin beta-1 chain
Waktu Paruh24 hours.
Vol. Distribusi-
Klirens-
Genetik -
Vinflunine Approved DB11641
small molecule | CAS: 162652-95-1

Vinflunine is a third-generation member of the vinca alkaloid family with anti-tumour actions. It was first described in 1998 at the Pierre Fabre research center in France. Like other vinca agents, vinflunine is an anti-mitotic agent that induces a cell cycle…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +14
Target Protein:
Tubulin beta chain
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe terminal volume…
KlirensThe total blood cle…
Genetik -
Vinorelbine Approved DB00361
small molecule | CAS: 71486-22-1

Vinorelbine is an anti-mitotic chemotherapy drug that is used in the treatment of several types of malignancies, including breast cancer and non-small cell lung cancer (NSCLC) [L1998]. It was initially approved in the USA in 1990's for the treatment of NSCLC…

Kategori:
AlkaloidsAntimitotic AgentsAntineoplastic Agents +23
Target Protein:
Tubulin beta chain
Waktu ParuhThe terminal phase …
Vol. DistribusiThe volume of distr…
KlirensThe plasma clearanc…
Genetik -
Vinylglycine DB03214
small molecule | CAS: 70982-53-5

Vinylglycine is an irreversible inhibitor of aspartate aminotransferase.

Kategori:
Amino AcidsAmino Acids, Peptides, and Proteins
Target Protein:
L-amino-acid oxidase1-aminocyclopropane-1-carboxylate synthase-like protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1184-84-5

Deskripsi belum tersedia.

Kategori:
AcidsAcids, NoncarboxylicAlkenes +4
Target Protein:
Phosphonoacetaldehyde hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viomycin Approved DB06827
small molecule | CAS: 32988-50-4

Viomycin is a tuberactinomycin antibiotic that was used to treat Mycobacterium tuberculosis until it was replaced by the less toxic capreomycin. These drugs bind RNA in bacterial ribosomes and inhibit protein synthesis. Viomycin was derived from the actinomyc…

Kategori:
Agents that produce neuromuscular block (indirect)Amino Acids, Peptides, and ProteinsAnti-Bacterial Agents +8
Target Protein:
16S/23S rRNA (cytidine-2'-O)-methyltransferase TlyA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vipoglanstat DB18126
small molecule | CAS: 1360622-01-0

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
VIR201 DB05110
biotech

is an experimental therapeutic vaccine currently in clinical trial. The aim of therapeutic vaccines is to augment the body's immune response to HIV and to delay or prevent progression to AIDS.

Target Protein:
Interferon gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Viral macrophage inflammatory protein-II (vMIP) is a highly basic protein and human chemokine analog encoded by human herpesvirus-8. The structure of vMIP consists of 71 residues and is a monomer under most conditions. It helps its virus evade the host immune…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Viralym-C DB17975
biotech

Viralym-C is an investigational T-cell immunotherapy developed by ViraCyte. It consists of Human Leukocyte Antigen (HLA)-matched cytomegalovirus (CMV)-specific T lymphocytes. It was granted FDA orphan designation in January 2017 and investigated for the treat…

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Virginiamycin DB11476
small molecule | CAS: 11006-76-1

Virginiamycin is a streptogramin antibiotic similar to pristinamycin and quinupristin/dalfopristin. It is a combination of pristinamycin IIA and virginiamycin S1. Virginiamycin is used in the fuel ethanol industry to prevent microbial contamination and in liv…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 21411-53-0

Pristinamycin IIA is a macrolide antibiotic, a member of the streptogramin A group of antibiotics, and one component of pristinamycin. It is produced by Streptomyces graminofaciens and other bacteria.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +4
Target Protein:
Streptogramin A acetyltransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 23152-29-6

One of the components of virginiamycin, a cyclic polypeptide antibiotic complex from streptomyces virginiae, s. Loidensis, s. Mitakaensis, s. Pristina-spiralis, s. Ostreogriseus, and others. It is used to treat infections with gram-positive organisms and as a…

Kategori:
Amino Acids, Peptides, and ProteinsPeptidesPeptides, Cyclic +1
Target Protein:
Large ribosomal subunit protein eL37
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Virus Specific T-Cells (VSTs) are a target therapy that are generated for specific viral antigens. These products are generated from virus-naive or virus-experienced autologous or allogenic sources. Antigens identified as an immune target are presented by ant…

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Vismodegib Approved DB08828
small molecule | CAS: 879085-55-9

Vismodegib is an orally active small molecule that inhibits the hedgehog signaling pathway by binding to and inhibiting the transmembrane protein smoothened homologue (SMO).[A258613,A258618,L45803] It was discovered by high-throughput screening of a library o…

Kategori:
AmidesAminesAniline Compounds +18
Target Protein:
Protein smoothened
Waktu ParuhThe half-life of vi…
Vol. DistribusiThe volume of distr…
Klirens-
Genetik -
Vistusertib DB11925
small molecule | CAS: 1009298-59-2

Vistusertib is under investigation for the treatment of Advanced Gastric Adenocarcinoma.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +3
Target Protein:
Target of rapamycin complex 2 subunit MAPKAP1Serine/threonine-protein kinase mTOR
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Aspartate aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vitamin D Approved DB11094
small molecule | CAS: 1406-16-2

Vitamin D ultimately comprises a group of lipid-soluble secosteroids responsible for a variety of biological effects, some of which include increasing the intestinal absorption of calcium, magnesium, and phosphate. With reference to human use, there are 2 mai…

Kategori:
Bone Density Conservation AgentsCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Vitamin D3 receptorVitamin D-binding protein
Waktu ParuhAlthough certain st…
Vol. Distribusi-
KlirensSome studies propos…
Genetik -
Vitamin E Approved DB00163
small molecule | CAS: 59-02-9

In 1922, vitamin E was demonstrated to be an essential nutrient[A32448]. Vitamin E is a term used to describe 8 different fat soluble tocopherols and tocotrienols, alpha-tocopherol being the most biologically active[A176104]. Vitamin E acts as an antioxidant,…

Kategori:
AntioxidantsBasic Ointments and ProtectantsBenzopyrans +23
Target Protein:
SEC14-like protein 4SEC14-like protein 3SEC14-like protein 2 +7
Waktu Paruh44 hours in prematu…
Vol. Distribusi0.41L/kg in prematu…
Klirens6.5mL/hr/kg in prem…
Genetik -
Vitespen DB06400
biotech | CAS: 492448-75-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological ProductsComplex Mixtures +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Vitex agnus-castus fruit extract is obtained from dry fruits of Vitex agnus-castus. The fruits contain mixture of iridoids, flavonoids and compounds in leaves and flowers that structurally resemble sex hormones. Clinical studies demonstrates effectiveness of …

Kategori:
AngiospermsBiological ProductsComplex Mixtures +12
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Vixarelimab DB16350
biotech | CAS: 2243320-83-2

Vixarelimab is under investigation in clinical trial NCT03816891 (A Study to Assess the Efficacy, Safety, and Tolerability of KPL-716 in Reducing Pruritus in Prurigo Nodularis).

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Vol. Distribusi-
Klirens-
Genetik -
VK-0214 DB17670
small molecule | CAS: 852949-30-5

Deskripsi belum tersedia.

Target Protein:
Thyroid hormone receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VMD-928 DB18052
small molecule | CAS: 1802770-18-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
VO659 DB18160
biotech | CAS: 1479142-52-3

VO659 is an antisense oligonucleotide being investigated for the treatment of Huntington's disease.

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Vol. Distribusi-
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Genetik -
biotech | CAS: 2490556-51-7

Vobramitamab duocarmazine is under investigation in clinical trial NCT05551117 (A Study of Vobramitamab Duocarmazine in Participants With Metastatic Castration Resistant Prostate Cancer and Other Solid Tumors).

Waktu Paruh-
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Genetik -
Vocacapsaicin DB17071
small molecule | CAS: 1931116-86-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 1300724-82-6

Vocimagene amiretrorepvec is under investigation in clinical trial NCT02576665 (A Study of Toca 511, a Retroviral Replicating Vector, Combined With Toca FC in Patients With Solid Tumors or Lymphoma (Toca 6)).

Kategori:
Amino Acids, Peptides, and ProteinsAminohydrolasesEnzymes +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Voclosporin Approved DB11693
small molecule | CAS: 515814-01-4

Lupus nephritis (LN) is a type of glomerulonephritis occurring in patients with systemic lupus erythematosus (SLE). LN is a significant cause of renal failure, morbidity, and death in patients with SLE. Within 10 years of being diagnosed with SLE, 5-20% of …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic and Immunomodulating AgentsCalcineurin Inhibitor Immunosuppressant +16
Target Protein:
Guided entry of tail-anchored proteins factor CAMLGProtein phosphatase 3 catalytic subunit alphaCalcineurin subunit B type 1 +1
Waktu ParuhThe average termina…
Vol. DistribusiThe apparent volume…
KlirensThe mean apparent s…
Genetik -
Vodobatinib DB17141
small molecule | CAS: 1388803-90-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Vodudeutentan DB17410
small molecule | CAS: 2364365-83-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6451–6500 dari 6694
Sebelumnya Halaman 130 / 134 Berikutnya