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12560

Total database: 17430
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9109 (72.5%)
Target
6912 (55.0%)
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109 (0.9%)
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12560 (100.0%)

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Halaman 130 / 252
IGN301 DB05117
biotech

IGN301 is a cancer vaccine based on an anti-idiotypic antibody which provokes an immune response to Lewis Y. Lewis Y is a carbohydrate molecule expressed on the surface of tumor cells of epithelial origin (e.g. lung, intestinal, breast, prostate or ovarian ca…

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IL-2 pDNA DB05935
small molecule

Vical incorporated has initiated a human Phase 1 study of an investigational method of delivering interleukin-2 (IL-2), a potent immune system stimulant, for patients with recurrent metastatic melanoma.

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IL15-NK Cell DB15725
biotech

Natural killer (NK) cells can be incubated with ‘feeder cells’ expressing certain cytokines prior to maturation to enhance their activity. In particular, incubation with IL-15 allows NK cells to lyse a broad range of fresh and cultured tumor targets that the …

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Ilacirnon DB16066
small molecule | CAS: 1100318-47-5

Ilacirnon (CCX-140) is under investigation in clinical trial NCT01440257 (A Study to Evaluate the Effect of CCX140-B on Urinary Albumin Excretion in Subjects With Type 2 Diabetes and Albuminuria).

Target Protein:
C-C chemokine receptor type 2
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Ilaprazole DB11964
small molecule | CAS: 172152-36-2

Ilaprazole has been investigated in Helicobacter Infections.

Kategori:
Anti-Ulcer AgentsBenzimidazolesGastric Acid Lowering Agents +5
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Ilepcimide DB16942
small molecule | CAS: 82857-82-7

Deskripsi belum tersedia.

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Ilginatinib DB12784
small molecule | CAS: 1239358-86-1

NS-018 has been used in trials studying the treatment of Primary Myelofibrosis, Post-Polycythemia Vera Myelofibrosis, and Post-Essential Thrombocythemia Myelofibrosis.

Target Protein:
Tyrosine-protein kinase JAK2
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Ilodecakin DB06449
small molecule | CAS: 149824-15-7

Deskripsi belum tersedia.

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Ilomastat DB02255
small molecule | CAS: 142880-36-2

Ilomastat is a broad-spectrum matrix metalloproteinase inhibitor.

Kategori:
AminesAmino Acids, Peptides, and ProteinsEnzyme Inhibitors +7
Target Protein:
Interstitial collagenaseMatrix metalloproteinase-14Neutrophil collagenase +8
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Iloperidone Approved DB04946
small molecule | CAS: 133454-47-4

Iloperidone is a benzisoxazole [A263557] and an atypical antipsychotic agent that was first approved by the FDA on May 6, 2009.[A3024] It is considered to be a second-generation antipsychotic drug [A263552] with multiple receptor binding profile, although it …

Kategori:
Adrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-AntagonistsAdrenergic Antagonists +31
Target Protein:
5-hydroxytryptamine receptor 2AD(2) dopamine receptor5-hydroxytryptamine receptor 1A +14
Waktu ParuhThe observed mean e…
Vol. DistribusiThe apparent volume…
KlirensIloperidone has an …
Genetik -
Iloprost Approved DB01088
small molecule | CAS: 78919-13-8

Iloprost is an analog of prostacyclin (PGI2; epoprostenol), an endogenous prostanoid mainly produced in the vascular endothelium. It is more stable than prostacyclin, which is short-lived.[A263326] Iloprost consists of a mixture of the 4R and 4S diastereoisom…

Kategori:
Agents Causing Muscle ToxicityAntiplatelet agentsAutacoids +16
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP2 subtypeProstaglandin E2 receptor EP1 subtype +6
Waktu ParuhThe half-life of il…
Vol. DistribusiFollowing intraveno…
KlirensClearance in normal…
Genetik -
ILS-920 DB15422
small molecule | CAS: 892494-07-4

ILS-920 is under investigation in clinical trial NCT00827190 (Study Evaluating Single Ascending Doses Of ILS-920).

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Iltamiocel DB19059
biotech

Deskripsi belum tersedia.

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Iluzanebart DB18275
biotech | CAS: 2733621-19-5

Deskripsi belum tersedia.

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ILY101 DB05059
small molecule

ILY101 is a metal-free, non-absorbed polymeric drug designed for the selective binding and removal of phosphate anions from the gastrointestinal tract. ILY101 is being developed for the treatment of hyperphosphatemia in CKD patients on dialysis and works by …

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small molecule | CAS: 1422365-93-2

Deskripsi belum tersedia.

Kategori:
Amidines
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Imagabalin DB12105
small molecule | CAS: 610300-07-7

Imagabalin has been investigated in Generalized Anxiety Disorder.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Anxiety AgentsCentral Nervous System Depressants
Target Protein:
Voltage-dependent calcium channel subunit alpha-2/delta-1
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Imalumab DB15558
biotech | CAS: 1430205-07-4

Imalumab is under investigation in clinical trial NCT02540356 (Phase 1/2a Two-arm Dose-escalation Study of BAX69 in Subjects With Malignant Ascites of Ovarian Cancer).

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Imaradenant DB16192
small molecule | CAS: 1321514-06-0

Imaradenant is under investigation in clinical trial NCT03381274 (Oleclumab (MEDI9447) Egfrm NSCLC Novel Combination Study).

Target Protein:
Adenosine receptor A2a
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Imatinib Approved DB00619
small molecule | CAS: 152459-95-5

Imatinib is a small molecule kinase inhibitor that revolutionized the treatment of cancer, particularly chronic myeloid leukemia, in 2001.[A249305] It was deemed a "miracle drug" due to its clinical success, as oncologist Dr. Brian noted that "complete hemato…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +51
Target Protein:
Breakpoint cluster region proteinInduced myeloid leukemia cell differentiation protein Mcl-1Mast/stem cell growth factor receptor Kit +8
Waktu ParuhFollowing oral admi…
Vol. DistribusiPopulation pharmaco…
KlirensTypically, clearanc…
Genetik -
Imazaquin DB04582
small molecule

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingHerbicides +3
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biotech | CAS: 138660-99-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +6
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Imdevimab Approved DB15940
biotech | CAS: 2415933-40-1

Imdevimab is a monoclonal antibody combined with [casirivimab] in Regeneron's antibody cocktail known as REGEN-COV2 for the treatment of COVID-19.[L23539] This drug is a combination of antibodies derived from humanized VelocImmune® mice in addition to blood …

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Target Protein:
Spike glycoprotein
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Imdusiran DB19014
biotech | CAS: 2839476-19-4

Imdusiran is under investigation in clinical trial NCT06245291 (Study of Imdusiran (AB-729) in Combination With Intermittent Dosing of Durvalumab in Subjects With Chronic HBV Infection).

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Imeglimin DB12509
small molecule | CAS: 775351-65-0

Imeglimin has been used in trials studying the treatment of Type 2 Diabetes Mellitus.

Kategori:
Alimentary Tract and MetabolismBlood Glucose Lowering AgentsDrugs Used in Diabetes
Target Protein:
5'-AMP-activated protein kinase catalytic subunit alpha-15'-AMP-activated protein kinase subunit beta-15'-AMP-activated protein kinase subunit gamma-1
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Imelasomeran Approved DB17090
biotech | CAS: 2763208-92-8

Imelasomeran was first approved in Canada on September 1, 2022, as one-half of Moderna's Spikevax Bivalent COVID-19 mRNA vaccine.[L45320] It encodes for the viral spike protein of the Omicron BA.1 variant of SARS-CoV-2, a particularly infectious variant of co…

Kategori:
COVID-19 VaccinesmRNA VaccinesVaccines +1
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Imetelstat Approved DB14909
small molecule | CAS: 868169-64-6

Imetelstat is a first-in-class 18-amino acid oligonucleotide that directly and competitively inhibits human telomerase.[A263973] It is used to treat anemia in patients with myelodysplastic syndromes (MDS), a group of hematologic disorders characterized by ine…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsEnzyme Inhibitors +6
Target Protein:
Telomerase reverse transcriptaseHuman telomerase RNA component
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
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Imexon DB05003
small molecule | CAS: 59643-91-3

Imexon is currently being studied for the treatment of pancreatic, lung, breast, prostate, melanoma, and multiple myeloma cancers. It belongs to the family of drugs called cyanoaziridine derivatives. Also called Amplimexon. Imexon is a cyanoaziridine derivati…

Kategori:
Ketones
Target Protein:
Ribonucleoside-diphosphate reductase subunit M2Ribonucleoside-diphosphate reductase large subunit
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IMG-7289 DB15126
small molecule | CAS: 1990504-34-1

IMG-7289 is under investigation in clinical trial NCT03136185 (IMG-7289 in Patients With Myelofibrosis).

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Target Protein:
Lysine-specific histone demethylase 1A
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Imgatuzumab DB14884
biotech | CAS: 959963-46-3

Imgatuzumab is under investigation in clinical trial NCT01326000 (A Study of RO5083945 in Combination With FOLFIRI Versus FOLFIRI Plus Cetuximab or FOLFIRI Alone as Second Line Treatment in Patients With Metastatic Colorectal Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
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IMGN632 DB17337
biotech

Deskripsi belum tersedia.

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Imidacloprid DB11421
small molecule | CAS: 105827-78-9

Imidacloprid is a neonicotinoid, which is a class of neuro-active insecticides modeled after nicotine. Imidacloprid is a patented chemical, Imidacloprid is manufactured by Bayer Cropscience (part of Bayer AG) and sold under trade names Kohinor, Admire, Advant…

Kategori:
AgrochemicalsCholinergic AgentsCompounds used in a research, industrial, or household setting +4
Target Protein:
CHRNA7-FAM7A fusion protein
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Imidafenacin DB09262
small molecule | CAS: 170105-16-5

Imidafenacin is an antispasmodic agent with anticholinergic effects. It antagonizes muscarinic receptors in the bladder to reduce the frequency of urination in the treatment of overactive bladder. It is marketed in Japan under the tradenames Staybla by Ono Ph…

Kategori:
Agents producing tachycardiaAnticholinergic AgentsCytochrome P-450 CYP3A Substrates +8
Target Protein:
Muscarinic acetylcholine receptor M1Muscarinic acetylcholine receptor M2Muscarinic acetylcholine receptor M3
Waktu ParuhThe half life of el…
Vol. DistribusiThe estimated volum…
KlirensThe estimated clear…
Genetik -
small molecule | CAS: 36364-49-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +16
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small molecule | CAS: 1072-84-0

Imidazole-4-carboxylic acid is under investigation in clinical trial NCT00583895 (Safety and Efficacy Study of Imcooh Cream in Patients Suffering From Moderate Atopic Dermatitis).

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small molecule

Deskripsi belum tersedia.

Target Protein:
Serine/threonine-protein kinase pim-1
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small molecule

Deskripsi belum tersedia.

Target Protein:
Methionine aminopeptidase
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Imidocarb DB11521
small molecule | CAS: 27885-92-3

Imidocarb is a urea derivative used in veterinary medicine as an antiprotozoal agent for the treatment of infection with Babesia and other parasites.

Kategori:
AmidesAminesAnilides +7
Target Protein:
Acetylcholinesterase
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Imidurea Approved DB14075
small molecule | CAS: 39236-46-9

Imidurea is an antimicrobial preservative used in cosmetics. It acts as a formaldehyde releaser.

Kategori:
AmidesCell-mediated ImmunityIncreased Histamine Release +2
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Imiglitazar DB12511
small molecule | CAS: 250601-04-8

Imiglitazar has been used in trials studying the treatment of Diabetes Mellitus.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Peroxisome proliferator-activated receptor gammaPeroxisome proliferator-activated receptor alpha
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Imiglucerase Approved DB00053
biotech | CAS: 154248-97-2

Human Beta-glucocerebrosidase or Beta-D-glucosyl-N-acylsphingosine glucohydrolase E.C. 3.2.1.45. 497 residue protein with N-linked carbohydrates, MW=59.3 kD. Alglucerase is prepared by modification of the oligosaccharide chains of human Beta-glucocerebrosidas…

Kategori:
Alimentary Tract and MetabolismEnzyme Replacement TherapyEnzymes +6
Target Protein:
Glucocerebroside
Waktu Paruh3.6-10.4 min
Vol. Distribusi* 0.09 to 0.15 L/kg
Klirens* 14.5 +/- 4.0 mL/m…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Serine protease 1
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Imipenem Approved DB01598
small molecule | CAS: 64221-86-9

Imipenem is a semisynthetic thienamycin that has a wide spectrum of antibacterial activity against gram-negative and gram-positive aerobic and anaerobic bacteria, including many multiresistant strains.[label] It is stable to many beta-lactamases. Similar comp…

Kategori:
Agents that reduce seizure thresholdAmidesAnti-Bacterial Agents +12
Target Protein:
Penicillin-binding protein 2Penicillin-binding protein 1BPenicillin-binding protein 1A +3
Waktu ParuhWhen given via IV i…
Vol. DistribusiThe reported volume…
KlirensThe total clearance…
Genetik -
Imipramine Approved DB00458
small molecule | CAS: 50-49-7

Imipramine, the prototypical tricyclic antidepressant (TCA), is a dibenzazepine-derivative TCA. TCAs are structurally similar to phenothiazines. They contain a tricyclic ring system with an alkyl amine substituent on the central ring. In non-depressed individ…

Kategori:
Adrenergic AgentsAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +70
Target Protein:
Sodium-dependent noradrenaline transporterSodium-dependent serotonin transporter5-hydroxytryptamine receptor 2A +21
Gen Terkait:
CYP2D6 CYP2D6 CYP2D6 +6
Waktu ParuhImipramine has a me…
Vol. DistribusiImipramine has a hi…
KlirensImipramine has a me…
Genetik 9 Varian
Imiquimod Approved DB00724
small molecule | CAS: 99011-02-6

Imiquimod is an immune response modifier that acts as a toll-like receptor 7 agonist. Imiquimod is commonly used topically to treat warts on the skin of the genital and anal areas. Imiquimod does not cure warts, and new warts may appear during treatment. Imiq…

Kategori:
Adjuvants, ImmunologicAminoquinolinesAntineoplastic Agents +17
Target Protein:
Toll-like receptor 7Toll-like receptor 8
Waktu Paruh20 hours (topical d…
Vol. Distribusi-
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Imlifidase Approved DB15258
biotech | CAS: 1947415-68-0

Chronic kidney disease (CKD) is a progressive and irreversible disease that represents a significant burden for both the individual and healthcare system at large.[A225916] Currently available treatments for end-stage renal disease are limited to dialysis and…

Kategori:
Antineoplastic and Immunomodulating AgentsEndopeptidasesImmunosuppressive Agents +2
Target Protein:
IgG heavy chain
Waktu ParuhThe mean distributi…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Imlunestrant DB19043
small molecule | CAS: 2408840-26-4

Imlunestrant is under investigation in clinical trial NCT05514054 (A Study of Imlunestrant Versus Standard Endocrine Therapy in Participants With Early Breast Cancer).

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Estrogen receptor
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IMM-0306 DB19309
biotech

IMM-0306 (bispecific antibody-trap selectively targeting cd47 and cd20) is under investigation in clinical trial NCT05805943 (Study of IMM0306 in Patients With Relapsed or Refractory Cd20-positive B-cell Non-hodgkin's Lymphoma).

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IMM-101 DB15850
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma[A220013,A220018,A220023]. Studies with …

Kategori:
Biological ProductsComplex MixturesMelanoma, therapy +1
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IMM101 DB15851
biotech

IMM-101 is a heat-inactivated immune-activating mycobacterial product. It has shown to be safe and well tolerated to complement conventional cancer therapy for patients with melanoma and pancreatic ductal adenocarcinoma [PMID: 21930686; PMID: 30107850; PMID: …

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