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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 130 / 315
small molecule | CAS: 7698-93-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
small molecule | CAS: 172377-52-5

Deskripsi belum tersedia.

Kategori:
AmidesEstradiol CongenersEstranes +10
Target Protein:
Steryl-sulfatase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estradiol valerate Approved DB13956
small molecule | CAS: 979-32-8

Estradiol Valerate (also known as E2V) is a pro-drug ester of [DB00783], a naturally occurring hormone that circulates endogenously within the human body. Estradiol is the most potent form of all mammalian estrogenic steroids and acts as the major female sex …

Kategori:
Adrenal Cortex HormonesBCRP/ABCG2 InhibitorsContraceptive Agents, Female +38
Target Protein:
Estrogen receptorEstrogen receptor betaNuclear receptor subfamily 1 group I member 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estramustine Approved DB01196
small molecule | CAS: 2998-57-4

A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.

Kategori:
Alkylating ActivityAlkylating DrugsAntineoplastic Agents +18
Target Protein:
Estrogen receptor betaEstrogen receptorMicrotubule-associated protein 2 +1
Waktu Paruh20 hours
Vol. Distribusi-
Klirens-
Genetik -
Estramustine phosphate Approved DB14674
small molecule | CAS: 4891-15-0

A nitrogen mustard linked to estradiol, usually as phosphate; used to treat prostatic neoplasms; also has radiation protective properties.

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 5696-58-2

Estrane-3,17-dione is a potent inhibitor of isomerase.

Kategori:
Fused-Ring CompoundsSteroids
Target Protein:
Steroid Delta-isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estriol Approved DB04573
small molecule | CAS: 50-27-1

A hydroxylated metabolite of estradiol or estrone that has a hydroxyl group at C3-beta, 16-alpha, and 17-beta position. Estriol is a major urinary estrogen. During pregnancy, large amount of estriol is produced by the placenta. Isomers with inversion of the h…

Kategori:
Estradiol CongenersEstranesEstrenes +13
Target Protein:
Estrogen receptorEstrogen receptor betaSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 2236-31-9

Deskripsi belum tersedia.

Target Protein:
Estrogen receptorEstrogen receptor betaSex hormone-binding globulin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Estrone Approved DB00655
small molecule | CAS: 53-16-7

Estrone, one of the major mammalian estrogens, is an aromatized C18 steroid with a 3-hydroxyl group and a 17-ketone. It is produced in vivo from androstenedione or from testosterone via estradiol. It is produced primarily in the ovaries, placenta, and in peri…

Kategori:
17-KetosteroidsAdrenal Cortex HormonesBCRP/ABCG2 Inhibitors +28
Target Protein:
Estrogen receptorEstrogen receptor betaAndrogen receptor +2
Waktu Paruh19 hours
Vol. Distribusi-
Klirens-
Genetik -
Estrone sulfate Approved DB04574
small molecule | CAS: 481-97-0

Estrone sulfate (as estropipate) is a form of estrogen. It has several uses such as: alleviate symptoms of menopause as hormone replacement therapy, treatment some types of infertility, treatment of some conditions leading to underdevelopment of female sexual…

Kategori:
17-KetosteroidsAdrenal Cortex HormonesContraceptive Agents, Hormonal +31
Target Protein:
Estrogen receptorEstrogen receptor beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Esuberaprost DB18464
small molecule | CAS: 94132-88-4

Esuberaprost (GP-1681), a drug intended for participants with pulmonary arterial hypertension, was under investigation in clinical trial NCT03657095 to evaluate its efficacy and safety.

Target Protein:
Prostacyclin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eszopiclone Approved DB00402
small molecule | CAS: 138729-47-2

Eszopiclone, marketed by Sepracor under the brand-name Lunesta, is a nonbenzodiazepine hypnotic drug used to treat insomnia. It is the active stereoisomer of zopiclone, belonging to the class of drugs known as _cyclopyrrolones_.[A179638,L6850] Cyclopyrrolone …

Kategori:
Benzodiazepine hypnotics and sedativesCentral Nervous System AgentsCentral Nervous System Depressants +18
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Translocator proteinGABA(A) Receptor +3
Waktu ParuhThe half-life is 6.…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
ET-101 DB18255
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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ET140203 DB17196
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Etacrynic acid Approved DB00903
small molecule | CAS: 58-54-8

A compound that inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules. This pharmacological action results in excretion of these ions, increased urinary output, and reduction …

Kategori:
AcetatesAcids, AcyclicAgents that produce neuromuscular block (indirect) +16
Target Protein:
Solute carrier family 12 member 1Sodium/potassium-transporting ATPase subunit alpha-1Lymphoid enhancer-binding factor 1 +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etafedrine Approved DB11587
small molecule | CAS: 48141-64-6

Etafedrine (INN) or ethylephedrine is a long-acting bronchodilator and has been an ingredient combined with other drugs in the brand names Nethaprin [A32757] and Dalmacol [L2568]. It was previously available as both the free base and as the hydrochloride salt…

Kategori:
Adrenergic AgonistsAdrenergic beta-2 Receptor AgonistsAdrenergic beta-Agonists +10
Target Protein:
Beta-2 adrenergic receptor
Waktu ParuhIt has a plasma hal…
Vol. DistribusiSimilar to ephedrin…
Klirens-
Genetik -
Etafenone DB13845
small molecule | CAS: 90-54-0

Etafenone is a vasodilator.

Kategori:
Cardiac TherapyCardiovascular AgentsKetones +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etalocib DB12850
small molecule | CAS: 161172-51-6

Etalocib has been used in trials studying the treatment of Pancreatic Cancer, Carcinoma, Non-Small-Cell Lung, and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
Acids, CarbocyclicBenzene Derivatives
Target Protein:
Leukotriene B4 receptor 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamicastat DB15288
small molecule | CAS: 760173-05-5

Etamicastat is under investigation in clinical trial NCT02840565 (Tolerability, Pharmacokinetics and Pharmacodynamics of Six Multiple Rising Dose Regimens of BIA 5-453).

Kategori:
Heterocyclic Compounds, Fused-RingPyrans
Target Protein:
Dopamine beta-hydroxylase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamiphylline DB13592
small molecule | CAS: 314-35-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnti-Asthmatic AgentsAutonomic Agents +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etamivan DB08989
small molecule | CAS: 304-84-7

Etamivan (INN) or ethamivan (USAN) is marketed under the name Analepticon. Etamvin is a respiratory stimulant drug similar to nikethamide. It is no longer used in the United States.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +2
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Etamsylate DB13483
small molecule | CAS: 2624-44-4

Deskripsi belum tersedia.

Kategori:
ArylsulfonatesArylsulfonic AcidsBenzene Derivatives +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etanautine DB13636
small molecule | CAS: 857401-00-4

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAnti-Parkinson DrugsAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etanercept Approved DB00005
biotech | CAS: 185243-69-0

Dimeric fusion protein consisting of the extracellular ligand-binding portion of the human 75 kilodalton (p75) tumor necrosis factor receptor (TNFR) linked to the Fc portion of human IgG1.[L14862,A216522] The Fc component of etanercept contains the CH2 domain…

Kategori:
Agents reducing cytokine levelsAmino Acids, Peptides, and ProteinsAnti-Inflammatory Agents +18
Target Protein:
Tumor necrosis factorLymphotoxin-alphaHigh affinity immunoglobulin gamma Fc receptor I +6
Waktu ParuhEtanercept has a me…
Vol. DistribusiPopulation pharmaco…
KlirensEtanercept has a me…
Genetik -
Etanidazole DB12736
small molecule | CAS: 22668-01-5

Etanidazole has been used in trials studying the diagnostic of Adult Ependymoma, Malignant Ascites, Adult Gliosarcoma, Adult Mixed Glioma, and Adult Glioblastoma, among others.

Kategori:
Antineoplastic AgentsImidazolesNitro Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etaracizumab DB12213
biotech | CAS: 892553-42-3

Etaracizumab has been investigated for the treatment of Psoriasis, Renal Cell Carcinoma, Stage IV Renal Cell Cancer, Recurrent Renal Cell Cancer, and Stage III Renal Cell Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etarfolatide DB11810
small molecule | CAS: 479578-27-3

Etarfolatide has been used in trials studying the treatment and diagnostic of Breast Neoplasms, Non Small Cell Lung Cancer, and Adenocarcinoma of the Lung.

Waktu Paruh-
Vol. Distribusi-
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Etavopivat DB18176
small molecule | CAS: 2245053-57-8

Etavopivat is a small molecule activator of erythrocyte pyruvate kinase (PKR) under investigation for the treatment of sickle cell disease.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Etazolate DB05881
small molecule

EHT 0202 is developed to treat neurodegenerative disorders by ExonHit Therapeutics.

Kategori:
Antipsychotic AgentsCentral Nervous System AgentsCentral Nervous System Depressants +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ETBX-011 DB17464
biotech

ETBX-011 is a cancer vaccine used to treat patients with cancers that express carcinoembryonic antigen (CEA).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
ETBX-021 DB17528
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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Genetik -
ETBX-041 DB17182
biotech

Deskripsi belum tersedia.

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ETBX-051 DB17529
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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ETBX-061 DB17530
biotech

Deskripsi belum tersedia.

Waktu Paruh-
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ETC-1001 DB05866
small molecule

ETC-1001 is Pfizer’s lead oral small molecule product candidate which is intended to be a chronic treatment for individuals with lipid disorders.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Etelcalcetide Approved DB12865
small molecule | CAS: 1262780-97-1

Etelcalcetide is a calcimimetic drug for the treatment of secondary hyperparathyroidism in patients undergoing hemodialysis. Etelcalcetide was approved (trade name Parsabiv) for the treatment of secondary hyperparathyroidism (HPT) in adult patients with chron…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Parathyroid AgentsCalcium Homeostasis +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh3 to 4 days
Vol. Distribusi796 L
Klirens7.66 L/hr
Genetik -
Eteplirsen Approved DB06014
biotech | CAS: 1173755-55-9

Eteplirsen is a synthetic antisense oligonucleotide and a phosphorodiamidate morpholino oligomer. It consists of a six-membered morpholino ring replacing the five-membered ribofuranosyl rings found in natural DNA and RNA.[L40015] Duchenne muscular dystrop…

Kategori:
Antisense OligonucleotidesMorpholinesMusculo-Skeletal System +5
Target Protein:
DMD-001 gene (exon 51 target site)
Waktu ParuhThe elimination hal…
Vol. DistribusiFollowing weekly in…
KlirensThe total clearance…
Genetik -
Etesevimab DB15897
biotech | CAS: 2423948-94-9

Etesevimab (LY-CoV016, also known as JS016) is a fully human and recombinant monoclonal antibody that targets the SARS-CoV-2 surface spike protein receptor binding domain.[L16651,L16661] Under the EUA granted in February 2021, etesevimab is used in combinatio…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Target Protein:
Spike glycoprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Etevritamab DB17211
biotech | CAS: 2329692-74-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethacizine DB13645
small molecule | CAS: 33414-33-4

Deskripsi belum tersedia.

Kategori:
Antiarrhythmic agentsAntiarrhythmics, Class IAntiarrhythmics, Class Ic +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethacridine DB13190
small molecule | CAS: 442-16-0

Deskripsi belum tersedia.

Kategori:
Acridine DerivativesAcridinesAminoacridines +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethadione DB13799
small molecule | CAS: 520-77-4

Deskripsi belum tersedia.

Kategori:
AnticonvulsantsCentral Nervous System DepressantsNervous System +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethambutol Approved DB00330
small molecule | CAS: 74-55-5

Ethambutol is a bacteriostatic agent indicated alongside medications such as [isoniazid], [rifampin], and [pyrazinamide] in the treatment of pulmonary tuberculosis.[L31743] Ethambutol was first described in the literature in 1961.[A229048] It was developed ou…

Kategori:
AminesAnti-Bacterial AgentsAnti-Infective Agents +23
Target Protein:
Probable arabinosyltransferase CProbable arabinosyltransferase BProbable arabinosyltransferase A
Waktu ParuhEthambutol has a ha…
Vol. DistribusiPatients coinfected…
KlirensPatients coinfected…
Genetik -
small molecule | CAS: 594-45-6

Deskripsi belum tersedia.

Kategori:
AlkanesAlkanesulfonic AcidsHydrocarbons, Acyclic +3
Target Protein:
Platelet basic proteinPhosphonoacetaldehyde hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethanol Approved DB00898
small molecule | CAS: 64-17-5

A clear, colorless liquid rapidly absorbed from the gastrointestinal tract and distributed throughout the body. It has bactericidal activity and is used often as a topical disinfectant. It is widely used as a solvent and preservative in pharmaceutical prepara…

Kategori:
Agents Causing Muscle ToxicityAlcoholsAnti-Infective Agents +34
Target Protein:
Gamma-aminobutyric acid receptor subunit alpha-1Glutamate receptor ionotropic, NMDA 3AGlycine receptor subunit alpha-1 +51
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethanolamine DB03994
small molecule | CAS: 141-43-5

A viscous, hygroscopic amino alcohol with an ammoniacal odor. It is widely distributed in biological tissue and is a component of lecithin. It is used as a surfactant, fluorimetric reagent, and to remove CO2 and H2S from natural gas and other gases.

Kategori:
AlcoholsAminesAmino Alcohols +4
Target Protein:
Surface protein AAnnexin A3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethanolamine oleate Approved DB06689
small molecule | CAS: 2272-11-9

Ethanolamine oleate is a mild sclerosing agent. It is composed of ethanolamine, a basic substance, which when combined with oleic acid forms a clear, straw to pale yellow colored, deliquescent oleate.

Kategori:
Antivaricose TherapyCardiovascular AgentsCompounds used in a research, industrial, or household setting +10
Target Protein:
Calcium ionsCoagulation factor XII
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ethaselen DB15051
small molecule | CAS: 217798-39-5

Ethaselen is under investigation in clinical trial NCT02166242 (Ethaselen for the Treatment of Thioredoxin Reductase High Expression Advanced Non-small Cell Lung Cancers).

Kategori:
Selenium Compounds
Waktu Paruh-
Vol. Distribusi-
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Ethchlorvynol Approved DB00189
small molecule | CAS: 113-18-8

Ethchlorvynol is a sedative and hypnotic drug. It has been used to treat insomnia, but has been largely superseded and is only offered where an intolerance or allergy to other drugs exists.

Kategori:
AlcoholsCentral Nervous System AgentsCentral Nervous System Depressants +4
Target Protein:
Gamma-aminobutyric acid receptor subunit beta-2Gamma-aminobutyric acid receptor subunit alpha-1GABA(A) Receptor
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Ethenzamide DB13544
small molecule | CAS: 938-73-8

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAmides +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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