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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Hasil Pencarian (16004)

Halaman 130 / 321
Droperidol Approved DB00450
small molecule | CAS: 548-73-2

A butyrophenone with general properties similar to those of haloperidol. It is used in conjunction with an opioid analgesic such as fentanyl to maintain the patient in a calm state of neuroleptanalgesia with indifference to surroundings but still able to coop…

Kategori:
Adjuvants, AnesthesiaAdrenergic alpha-1 Receptor AntagonistsAdrenergic alpha-Antagonists +27
Target Protein:
Alpha-1A adrenergic receptorD(2) dopamine receptor
Waktu ParuhBiphasic distributi…
Vol. Distribusi-
Klirens-
Genetik -
Dropropizine DB13785
small molecule | CAS: 17692-31-8

Deskripsi belum tersedia.

Kategori:
AlcoholsAntitussive AgentsCentral Nervous System Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drospirenone Approved DB01395
small molecule | CAS: 67392-87-4

Drospirenone is a synthetic progestin commonly found in the popular oral contraceptive, Yaz in combination with [Ethinyl estradiol].[L7973] Most recently, it was approved by both Health Canada and the FDA in combination with [Estetrol] as an oral contraceptiv…

Kategori:
Adrenal Cortex HormonesAgents causing hyperkalemiaAndrostanes +21
Target Protein:
Mineralocorticoid receptorAndrogen receptorProgesterone receptor +1
Waktu ParuhThe serum half-life…
Vol. DistribusiThe volume of distr…
KlirensDrospirenone is rap…
Genetik -
Drostanolone DB00858
small molecule | CAS: 58-19-5

Drostanolone (also known as dromostanolone) is a potent synthetic androgenic anabolic steroid similar to testosterone. Drostanolone is indicated in postmenopausal women with recurrent breast cancer, in a combined hormone therapy.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Target Protein:
Androgen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drostanolone propionate Approved DB14655
small molecule | CAS: 521-12-0

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drotaverine Approved DB06751
small molecule | CAS: 14009-24-6

Drotaverine is an antispasmodic drug that works by inhibiting phosphodiesterase-4 (PDE4).[A231619] It is a benzylisoquinoline derivative that is structurally related to [papaverine], although it displays more potent antispasmodic activities than papaverine. D…

Kategori:
Alimentary Tract and MetabolismAlkaloidsAnalgesics +15
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4AVoltage-dependent L-type calcium channel
Waktu ParuhFollowing oral admi…
Vol. DistribusiFollowing oral admi…
KlirensFollowing oral admi…
Genetik -
Drotebanol DB01547
small molecule | CAS: 3176-03-2

Deskripsi belum tersedia.

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drotrecogin alfa Approved DB00055
biotech | CAS: 98530-76-8

Drotrecogin alfa is activated human protein C that is synthesized by recombinant DNA technology. It is a glycoprotein of approximately 55 kilodalton molecular weight, consisting of a heavy chain and a light chain linked by a disulfide bond. Drotrecogin alfa w…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Infective AgentsAnticoagulants +14
Target Protein:
Coagulation factor VIIICoagulation factor VPlasminogen activator inhibitor 1 +7
Waktu Paruh5.5 hours (mammalia…
Vol. Distribusi-
Klirens* 40 L/hr [severe s…
Genetik -
Droxicam DB09215
small molecule | CAS: 90101-16-9

Droxicam is an oxicam non-steroidal anti-inflammatory drug and a prodrug of [DB00554]. It is used to reduce pain and inflammation in musculoskeletal disorders such as rheumatoid arthritis and osteoarthritis.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +13
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu ParuhData not available …
Vol. DistribusiData not available …
KlirensData not available …
Genetik -
Droxidopa Approved DB06262
small molecule | CAS: 23651-95-8

Droxidopa is a precursor of noradrenaline that is used in the treatment of Parkinsonism. It is approved for use in Japan and is currently in trials in the U.S. The racaemic form (dl-threo-3,4-dihydroxyphenylserine) has also been used, and has been investigate…

Kategori:
Adrenergic AgonistsAdrenergic alpha-1 Receptor AgonistsAdrenergic alpha-2 Receptor Agonists +23
Target Protein:
Alpha-1A adrenergic receptorAlpha-1B adrenergic receptorAlpha-1D adrenergic receptor +7
Waktu Paruh2-3 hours.
Vol. Distribusi-
Klirens-
Genetik -
Droxypropine DB13436
small molecule | CAS: 15599-26-5

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Drozitumab DB19106
biotech | CAS: 912628-39-8

Drozitumab is a human monoclonal antibody directed against tumor necrosis factor receptor superfamily member 10B (TNFRSF10B), a member of tumor necrosis factor related apoptosis-inducing ligand (TRAIL). It was developed by Genentech as a drug for the treatmen…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DS-1211 DB17837
small molecule | CAS: 19764-30-8

DS-1211 is a potent and selective novel small molecule tissue-nonspecific alkaline phosphatase (TNAP) inhibitor.[A259786]

Target Protein:
Alkaline phosphatase, tissue-nonspecific isozyme
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DS-2325a DB18134
biotech

DS-2325a is an inhibitor of kallikrein 5 under development for the treatment of Netherton Syndrome.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DSM-265 DB12397
small molecule | CAS: 1282041-94-4

DSM265 has been used in trials studying the prevention and treatment of Malaria.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DSP-5336 DB18514
small molecule | CAS: 2412555-70-3

DSP-5336 is a menin inhibitor.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DSP107 DB17501
biotech

DSP107 is a bi-functional, trimeric, fusion protein composed of sequences from the extracellular domain of SIRP? and 4-1BBL.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DT-DEC01 DB19433
biotech

DT-DEC01 is a novel Dystrophin Expressing Chimeric (DEC) cell therapy being investigated by Dystrogen Therapeutics Corporation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DT2216 DB18020
small molecule | CAS: 2365172-42-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DTP-348 DB12741
small molecule | CAS: 1383370-92-0

Dtp348 has been used in trials studying the treatment of Solid Tumors and Head and Neck Neoplasms.

Target Protein:
Carbonic anhydrase 9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DTS-201 DB06071
small molecule

DTS-201 is a prodrug of doxorubicin, a widely used anti-cancer drug that Diatos intends to develop for the treatment of various solid tumors. It is activated in the tumor environment. DTS-201 may be suitable for the treatment of many types of solid tumors, i…

Kategori:
AnthracyclinesCarbohydratesGlycosides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DTX-101 DB17699
biotech

DTX-101 is an investigational gene therapy consisting of an adeno-associated virus serotype Rh10 vector encoding the human Factor Ix gene. It was previously investigated for the treatment of hemophilia B; however, the clinical development of DTX-101 was disco…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DTx-1252 DB18086
small molecule

DTx-1252 is a siRNA therapeutic under investigation for the treatment of Charcot-Marie-Tooth Disease type 1A (CMTD1A).[L48096]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DU125530 DB16040
small molecule | CAS: 161611-99-0

DU125530 is under investigation in clinical trial NCT01119430 (Fluoxetine Versus Fluoxetine Plus DU125530 in Major Depressive Disorder).

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsSerotonin 5-HT1 Receptor Antagonists +4
Target Protein:
5-hydroxytryptamine receptor 1A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dubermatinib DB15187
small molecule | CAS: 1341200-45-0

Dubermatinib is under investigation in clinical trial NCT03572634 (Phase 1/2 Study of TP-0903 (an Inhibitor of AXL Kinase) in Patients With Previously Treated CLL).

Kategori:
AmidesBenzene DerivativesSulfonamides +2
Target Protein:
Tyrosine-protein kinase receptor UFO
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dulaglutide Approved DB09045
biotech | CAS: 923950-08-7

Dulaglutide, marketed by Eli Lilly as Trulicity, is a once-weekly subcutaneous glucagon-like peptide-1 (GLP-1) receptor agonist designed using recombinant DNA technology; it has been approved as an adjunct therapy to diet and exercise in the management of 2 …

Kategori:
Alimentary Tract and MetabolismAmino Acids, Peptides, and ProteinsBlood Glucose Lowering Agents +21
Target Protein:
Glucagon-like peptide 1 receptor
Waktu ParuhIn a pharmacokineti…
Vol. DistribusiThe apparent volume…
KlirensThe apparent popula…
Genetik -
Dulanermin DB12349
biotech | CAS: 867153-61-5

Dulanermin has been used in trials studying the treatment of Colorectal Cancer, Non-Hodgkin's Lymphoma, and Metastatic Colorectal Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Duligotuzumab DB12142
biotech | CAS: 1314238-96-4

Duligotuzumab has been used in trials studying the treatment of Neoplasms, Colorectal Cancer, Head and Neck Cancer, and Epithelial Tumors, Malignant.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Duloxetine Approved DB00476
small molecule | CAS: 116539-59-4

Duloxetine is a dual serotonin and norepinephrine reuptake inhibitor.[label] It was originally discovered in 1993 and developed by Eli Lilly and Company as LY248686.[A178741] Duloxetine first received approval from the FDA in August, 2004 as Cymbalta for the …

Kategori:
Agents producing tachycardiaAnalgesicsAntidepressive Agents +39
Target Protein:
Sodium-dependent serotonin transporterSodium-dependent noradrenaline transporterSodium-dependent dopamine transporter
Waktu ParuhMean of 12 h with a…
Vol. DistribusiApparent Vd of 1620…
KlirensThere is a large de…
Genetik -
Dupilumab Approved DB12159
biotech | CAS: 1190264-60-8

Dupilumab is a fully human monoclonal antibody of the immunoglobulin G4 subclass that binds to the interleukin-4 (IL-4) receptor, inhibiting the receptor signaling pathways.[A180478] As an interleukin-4 receptor alpha antagonist, dupilumab inhibits the signal…

Kategori:
Agents for Dermatitis, Excluding CorticosteroidsAmino Acids, Peptides, and ProteinsAnti-Asthmatic Agents +13
Target Protein:
Interleukin-4 receptor subunit alphaInterleukin-13Interleukin-4
Waktu ParuhThere is limited hu…
Vol. DistribusiThe estimated volum…
KlirensThere is limited da…
Genetik -
Durlobactam Approved DB16704
small molecule | CAS: 1467829-71-5

Durlobactam is a diazabicyclooctane non-beta-lactam, beta-lactamase inhibitor. It is typically given in combination with [sulbactam] to protect it from degradation by certain serine-beta-lactamases.[L47336] The combination product of durlobactam and sulbactam…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +3
Target Protein:
Beta-lactamase CTX-M
Waktu ParuhThe elimination hal…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of du…
Genetik -
Duroquinone DB01927
small molecule | CAS: 527-17-3

Deskripsi belum tersedia.

Kategori:
Quinones
Target Protein:
NAD(P)H dehydrogenase [quinone] 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Durvalumab Approved DB11714
biotech | CAS: 1428935-60-7

Durvalumab is a human immunoglobulin G1 kappa (IgG1?) monoclonal antibody and a novel immune-checkpoint inhibitor for cancer treatment.[A192789] Produced by recombinant DNA technology in Chinese Hamster Ovary (CHO) cell suspension culture,[L12621] durvalumab …

Kategori:
Amino Acids, Peptides, and ProteinsAntibiotics, AntineoplasticAntibodies +20
Target Protein:
Programmed cell death 1 ligand 1Programmed cell death protein 1
Waktu ParuhBased on baseline c…
Vol. DistribusiIn patients receivi…
KlirensClearance of durval…
Genetik -
Dusigitumab DB12363
biotech | CAS: 1204390-13-5

Dusigitumab has been used in trials studying the treatment of Cancer, Advanced Solid Malignancies, Unresectable or Metastatic Hepatocellular Carcinoma (HCC), and Hormone-sensitive, HER-2 Negative Metastatic Breast Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dusquetide DB11879
small molecule | CAS: 931395-42-5

Dusquetide has been used in trials studying the treatment of Oral Mucositis.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dutasteride Approved DB01126
small molecule | CAS: 164656-23-9

Dutasteride is an oral synthetic 4-azasteroid commonly marketed under the trade name Avodart. It is a novel dual 5?-reductase inhibitor that works by blocking both isoforms of 5?-reductase enzymes in a potent, selective, and irreversible manner.[A1909] Type I…

Kategori:
5-alpha Reductase InhibitorsAdrenergic alpha-AntagonistsAdrenergic Antagonists +14
Target Protein:
3-oxo-5-alpha-steroid 4-dehydrogenase 1Polyprenal reductase3-oxo-5-alpha-steroid 4-dehydrogenase 2
Waktu ParuhThe terminal elimin…
Vol. DistribusiDutasteride display…
KlirensIn a study of healt…
Genetik -
Dutogliptin DB11723
small molecule | CAS: 852329-66-9

Dutogliptin has been investigated for the treatment of Diabetes Mellitus, Type II.

Kategori:
AcidsAcids, NoncarboxylicAgents causing angioedema +3
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh10-13 hours
Vol. Distribusi-
Klirens-
Genetik -
Duvakitug DB19444
biotech | CAS: 2750005-84-4

Duvakitug is under investigation in clinical trial NCT05668013 (A Study to Evaluate the Long-term Effect of TEV-48574 in Moderate to Severe Ulcerative Colitis or Crohn's Disease).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Duvelisib Approved DB11952
small molecule | CAS: 1201438-56-3

Duvelisib, also known as IPI-145 and INK-1197, is a small-molecule inhibitor of phosphoinositide-3 kinases that was designed initially to prove that simultaneous inhibition of the isoforms delta and gamma can produce a broad adaptative and innate immune cell …

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe reported half-l…
Vol. DistribusiThe volume of distr…
KlirensDuvelisib clearance…
Genetik -
Duvoglustat DB03206
small molecule | CAS: 19130-96-2

An alpha-glucosidase inhibitor with antiviral action. Derivatives of deoxynojirimycin may have anti-HIV activity.

Kategori:
AlkaloidsAmino SugarsAnti-Infective Agents +7
Target Protein:
Maltase-glucoamylaseLysosomal alpha-glucosidaseNeutral alpha-glucosidase AB +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Duvortuxizumab DB15211
biotech | CAS: 1831098-91-9

Duvortuxizumab is under investigation in clinical trial NCT02743546 (Study of the Safety, Pharmacokinetics, Pharmacodynamics, and Efficacy of Duvortuxizumab (JNJ-64052781) Plus Ibrutinib in Lymphoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dyclonine Approved DB00645
small molecule | CAS: 586-60-7

Dyclonine is an oral anaesthetic found in Sucrets, an over the counter throat lozenge. It may also be found in some Cepacol sore throat spray products.

Kategori:
AnestheticsAnesthetics, LocalCentral Nervous System Agents +6
Target Protein:
Sodium channel protein type 10 subunit alphaSodium channel protein type 5 subunit alpha
Waktu ParuhApproximately 30 to…
Vol. Distribusi-
Klirens-
Genetik -
Dydrogesterone Approved DB00378
small molecule | CAS: 152-62-5

A synthetic progestational hormone with no androgenic or estrogenic properties. Unlike many other progestational compounds, dydrogesterone produces no increase in temperature and does not inhibit ovulation.

Kategori:
Adrenal Cortex HormonesCytochrome P-450 CYP3A SubstratesCytochrome P-450 CYP3A4 Substrates +12
Target Protein:
Progesterone receptor
Waktu ParuhDydrogesterone: 5-7…
Vol. Distribusi-
Klirens-
Genetik -
DYN-101 DB17921
biotech

DYN-101 is an antisense product candidate designed to reduce the expression of dynamin 2 protein.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dynasore DB15964
small molecule | CAS: 304448-55-3

Deskripsi belum tersedia.

Kategori:
Dynamins, antagonists & inhibitorsHydrazines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DYNE-251 DB18130
biotech

DYNE-251 is a phosphorodiamidate morpholino oligomer (PMO) conjugated to a fragment antibody (Fab) that binds to the transferrin receptor 1 (TfR1). It is being investigated for the treatment of Duchenne muscular dystrophy (DMD) in patients who are amenable to…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dynorphin DB16146
small molecule | CAS: 80448-90-4

Dynorphin is under investigation in clinical trial NCT00000244 (Effects of Dynorphin 1-13 on Heroin Addiction - 1).

Kategori:
Amino Acids, Peptides, and ProteinsNerve Tissue ProteinsNeuropeptides +4
Target Protein:
Kappa-type opioid receptorMu-type opioid receptorDelta-type opioid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dyphylline Approved DB00651
small molecule | CAS: 479-18-5

Dyphylline is a theophylline derivative with broncho- and vasodilator properties. It is typically used in the management of asthma, cardiac dyspnea, and bronchitis.

Kategori:
Anti-Asthmatic AgentsAutonomic AgentsBronchodilator Agents +13
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidase3',5'-cyclic-AMP phosphodiesterase 4A +4
Waktu Paruh2 hours (range 1.8 …
Vol. Distribusi-
Klirens-
Genetik -
E-2012 DB05171
small molecule | CAS: 870843-42-8

E-2012 is a gamma secretase modulator that is being evaluated as a potential new treatment for Alzheimer's disease.

Kategori:
Amyloid Precursor Protein SecretasesEnzyme InhibitorsGamma Secretase Inhibitors and Modulators
Target Protein:
Gamma-secretase subunit APH-1BNicastrinPresenilin-1 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
E-52862 DB16881
small molecule | CAS: 878141-96-9

Deskripsi belum tersedia.

Kategori:
OxazinesReceptors, sigma, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6451–6500 dari 16004
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