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2279

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Halaman 13 / 46
Danburstotug DB19064
biotech | CAS: 2307144-65-4

Danburstotug is under investigation in clinical trial NCT04809012 (Study of STI-3031 in Patients With Selected Relapsed or Refractory Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dapagliflozin Approved DB06292
small molecule | CAS: 461432-26-8

Dapagliflozin is a sodium-glucose cotransporter 2 (SGLT2) inhibitor, and it was the first SLGT2 inhibitor to be approved. indicated for managing diabetes mellitus type 2.[A261596] When combined with diet and exercise in adults, dapagliflozin helps to improve …

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesBlood Glucose Lowering Agents +19
Target Protein:
Sodium/glucose cotransporter 2
Waktu ParuhThe mean plasma ter…
Vol. DistribusiThe volume of distr…
KlirensOral plasma clearan…
Genetik -
Dapiclermin DB17979
biotech | CAS: 444069-80-1

Dapiclermin is a recombinant ciliary neurotrophic factor.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dapiglutide DB19182
biotech | CAS: 2296814-85-0

Dapiglutide is under investigation in clinical trial NCT05788601 (Dapiglutide for the Treatment of Obesity).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 1416147-64-2

Dapirolizumab pegol is under investigation in clinical trial NCT02804763 (A Phase 2 Efficacy and Safety Study of Dapirolizumab Pegol (DZP) in Systemic Lupus Erythematosus).

Kategori:
AlcoholsAmino Acids, Peptides, and ProteinsAntibodies, Monoclonal +14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Darbepoetin alfa Approved DB00012
biotech | CAS: 209810-58-2

Human erythropoietin with 2 aa substitutions to enhance glycosylation (5 N-linked chains), 165 residues (MW=37 kD). Produced in Chinese hamster ovary (CHO) cells by recombinant DNA technology.

Kategori:
Amino Acids, Peptides, and ProteinsAntianemic PreparationsBlood and Blood Forming Organs +10
Target Protein:
Erythropoietin receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Darunavir Approved DB01264
small molecule | CAS: 206361-99-1

Darunavir is a protease inhibitor used with other HIV protease inhibitor drugs as well as [ritonavir] for the effective management of HIV-1 infection.[L9227] As a second-generation protease inhibitor, darunavir is designed to combat resistance to standard HIV…

Kategori:
AmidesAnti-HIV AgentsAnti-Infective Agents +33
Target Protein:
Pol polyproteinGag-Pol polyprotein
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensDarunavir has a low…
Genetik -
Darvadstrocel Approved DB16581
biotech

Darvadstrocel is a suspension of expanded human allogeneic adipose-derived mesenchymal stem cells extracted from the subdermal adipose tissue of healthy donors via liposuction.[A244524] Darvadstrocel was first approved by the European Commission on March 23, …

Kategori:
Antineoplastic and Immunomodulating AgentsImmunomodulatory AgentsImmunosuppressive Agents +1
Waktu ParuhPharmacokinetic inf…
Vol. DistribusiIn preclinical tria…
KlirensPharmacokinetic inf…
Genetik -
Dasiglucagon Approved DB15226
biotech | CAS: 1544300-84-6

Dasiglucagon is a glucagon analog that acts to increase blood sugar levels.[L39190] It consists of 29 amino acids similar to endogenous glucagon; however, it contains seven substituted amino acids for improved physical and chemical stability in its drug formu…

Kategori:
Amino Acids, Peptides, and ProteinsAntihypertensive AgentsAntihypoglycemic Agent +10
Target Protein:
Glucagon receptor
Waktu ParuhThe half-life was a…
Vol. DistribusiThe mean apparent v…
Klirens-
Genetik -
Davunetide DB12613
small molecule | CAS: 211439-12-2

Davunetide has been used in trials studying the treatment of Progressive Nonfluent Aphasia, Progressive Supranuclear Palsy, Predicted Tauopathies, Including, Corticobasal Degeneration Syndrome, and Frontotemporal Dementia With Parkinsonism Linked to Chromosom…

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DaxibotulinumtoxinA Approved DB17929
biotech | CAS: 93384-43-1

DaxibotulinumtoxinA is an acetylcholine release inhibitor and neuromuscular blocking agent. It is a botulinum toxin without accessory proteins purified from the bacterium _Clostridium botulinum_ type A,[L47840] the gram-positive anaerobic bacterium primarily …

Kategori:
Acetylcholine Release InhibitorsBotulinum ToxinsBotulinum Toxins, Type A +6
Target Protein:
Synaptosomal-associated protein 25
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dazodalibep DB19025
biotech | CAS: 2245953-10-8

Dazodalibep is under investigation in clinical trial NCT06104124 (A Study to Evaluate the Efficacy and Safety of Dazodalibep in Participants With Sjögren's Syndrome (SS) With Moderate-to-severe Systemic Disease Activity).

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Dazukibart DB18429
biotech | CAS: 2639474-65-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DCLL-9718S DB17392
biotech

DCLL9718S is an antibody-drug conjugate targeting C-type lectin-like molecule-1 (CLL-1). DCLL9718S is under investigation in clinical trial NCT03298516 (A Study of DCLL9718S in Participants With Relapsed or Refractory Acute Myeloid Leukemia (AML) or DCLL9718S…

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DCN-tCRK DB18262
biotech

DCN-tCRK is a recombinant, multi-functional fusion protein consisting of human decorin fused to the C-terminal vascular homing peptide tCRK.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Debrisoquine Approved DB04840
small molecule | CAS: 1131-64-2

An adrenergic neuron-blocking drug similar in effects to guanethidine. It is also noteworthy in being a substrate for a polymorphic cytochrome P-450 enzyme. Persons with certain isoforms of this enzyme are unable to properly metabolize this and many other cli…

Kategori:
Adrenergic AgentsAntiadrenergic Agents, Peripherally ActingAntihypertensive Agents +12
Target Protein:
Sodium-dependent noradrenaline transporter
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deflazacort Approved DB11921
small molecule | CAS: 14484-47-0

Deflazacort, also known as Emflaza, is a corticosteroid prodrug used as an agent to manage Duchenne Muscular Dystrophy (DMD). It is marketed by Marathon Pharmaceuticals and was approved in February 2017 by the FDA.[L6694,FDA label] Duchenne Muscular Dystro…

Kategori:
Adrenal Cortex HormonesAnti-Inflammatory AgentsCorticosteroid Hormone Receptor Agonists +18
Target Protein:
Glucocorticoid receptor
Waktu ParuhThe half-life of de…
Vol. DistribusiOne study determine…
Klirens114 ±27 L/h, accord…
Genetik -
small molecule | CAS: 490-83-5

Dehydroascorbic acid is made from the oxidation of ascorbic acid. This reaction is reversible, but dehydroascorbic acid can instead undergo irreversible hydrolysis to 2,3-diketogulonic acid. Dehydroascorbic acid as well as ascorbic acid are both termed Vitami…

Kategori:
Acids, AcyclicCarbohydratesDiet, Food, and Nutrition +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Delamanid Approved DB11637
small molecule | CAS: 681492-22-8

Delamanid is an anti-tuberculosis agent derived from the nitro-dihydro-imidazooxazole class of compounds that inhibits mycolic acid synthesis of bacterial cell wall [A31965]. It is used in the treatment of multidrug-resistant and extensively drug-resistant tu…

Kategori:
Antiinfectives for Systemic UseAntimycobacterialsCytochrome P-450 CYP3A Substrates +7
Waktu ParuhThe half life range…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
biotech | CAS: 2061938-98-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

The recombinant chimeric DC vaccine is a subunit-based vaccine candidate investigated for safety and effectiveness against SARS-CoV-2-induced pneumonia. With a better safety profile than inactivated and live-attenuated virus and virus-vector vaccines, the rec…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denecimig DB18426
biotech | CAS: 2488745-86-2

Delpacibart is a humanized, bispecific, bivalent monoclonal antibody against coagulation factor 9.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denenicokin DB12908
biotech | CAS: 716840-32-3

Denenicokin is under investigation in clinical trial NCT01152788 (Phase II Study of Interleukin-21 (rIL-21) vs Dacarbazine (DTIC) in Patients With Metastatic or Recurrent Melanoma).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Denileukin diftitox Approved DB00004
biotech | CAS: 173146-27-5

Denileukin diftitox is an IL2-receptor-directed cytotoxin, is a recombinant DNA-derived fusion protein composed of the amino acid sequences for diphtheria toxin fragments A and B (Met<sub>1</sub>-Thr<sub>387</sub>)-His and the sequence for human interleukin-2…

Kategori:
ADP Ribose TransferasesAmino Acids, Peptides, and ProteinsAntineoplastic Agents +15
Target Protein:
Interleukin-2 receptor subunit alphaInterleukin-2 receptor subunit beta
Waktu ParuhThe arithmetic mean…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Denosumab Approved DB06643
biotech | CAS: 615258-40-7

Denosumab is a novel, fully human IgG2 monoclonal antibody specific to receptor activator of nuclear factor kappa-B ligand (RANKL), suppresses bone resorption via inhibiting RANK-mediated activation of osteoclasts. It is the first and currently the only RANKL…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
Tumor necrosis factor ligand superfamily member 11
Waktu ParuhAfter C<sub>max</su…
Vol. DistribusiThe central volume …
KlirensNo information is a…
Genetik -
biotech

Dental pulp is a soft, connective tissue present in the dental crown of both third molar and first premolar teeth. Dental pulp stem cells (DPSCs) exhibit fibro-blast like plasticity and adherent properties. They are harvested through surgical extraction of wi…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deoxyribonuclease I (DNase I) is a human enzyme responsible for the digestion of extracellular DNA7[A227723]. It is normally found in saliva, urine, pancreatic secretions, and blood[A227723]. Because of the hypothesis that increased concentrations of high-mol…

Kategori:
Deoxyribonuclease I, antagonists & inhibitorsDeoxyribonucleasesEndodeoxyribonucleases +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Depelestat DB17873
biotech | CAS: 506433-25-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsLeukocyte Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Depemokimab DB18846
biotech | CAS: 2243274-14-6

Depemokimab is under investigation in clinical trial NCT05274750 (Efficacy and Safety of Depemokimab (GSK3511294) in Participants With Chronic Rhinosinusitis With Nasal Polyps).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desirudin Approved DB11095
biotech | CAS: 120993-53-5

Desirudin is a direct inhibitor of human thrombin. It has a protein structure that is similar to that of hirudin, the naturally occurring anticoagulant present in the peripharyngeal glands in the medicinal leech, Hirudo medicinalis. Hirudin is a single polype…

Kategori:
Amino Acids, Peptides, and ProteinsAnticoagulantsAntithrombin Proteins +12
Waktu Paruh~2 hours.
Vol. Distribusi0.25 L/kg.
Klirens1.5 to 2.7 mL/min/k…
Genetik -
small molecule | CAS: 13147-09-6

Desmethylprodine, a derivative of meperidine, is an opioid analgesic with the potency of morphine. It has been listed as a Schedule I controlled drug in the United States, and thus is not used clinically. It is known to be a designer drug, synthesized in 1977…

Kategori:
Isonipecotic AcidsPiperidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Desoxyribonuclease Approved DB09551
biotech | CAS: 9003-98-9

Desoxyribonuclease is a crystalline enzyme that aids in the digestion of the thymus nucleic acid. The mechanism of action of the enzyme involves the splitting of thymus nucleic acid into fragments approaching the size of tetranucleotides without the release o…

Kategori:
Blood and Blood Forming OrgansDeoxyribonucleasesEnzymes +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Deutetrabenazine Approved DB12161
small molecule | CAS: 1392826-25-3

Deutetrabenazine is a novel, highly selective vesicular monoamine transporter 2 (VMAT2) inhibitor indicated for the management of chorea associated with Huntington’s disease. It is a hexahydro-dimethoxybenzoquinolizine derivative and a deuterated [DB04844] [A…

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2D6 SubstratesCytochrome P-450 CYP3A Substrates +11
Target Protein:
Synaptic vesicular amine transporter
Waktu ParuhThe half-life of to…
Vol. DistribusiThe median volume o…
KlirensIn patients with Hu…
Genetik -
Dexelvucitabine DB12470
small molecule | CAS: 134379-77-4

Dexelvucitabine has been used in trials studying the treatment of HIV Infections and Human Immunodeficiency Virus.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +13
Target Protein:
Reverse transcriptase/RNaseH
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dexfenfluramine Approved DB01191
small molecule | CAS: 3239-44-9

Dexfenfluramine, also marketed under the name Redux, is a serotoninergic anorectic drug. For a fairly limited time during the middle of the nineties, the US FDA had approved it for use in managing weight loss. However, following multiple concerns about the ca…

Kategori:
Alimentary Tract and MetabolismAminesAntidepressive Agents +17
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 2C
Waktu Paruh17-20 hours
Vol. Distribusi-
Klirens-
Genetik -
Dexlansoprazole Approved DB05351
small molecule | CAS: 138530-94-6

Dexlansoprazole is a new-generation proton pump inhibitor (PPI) used for the management of symptoms associated with gastroesophageal reflux disease (GERD) and erosive esophagitis. Dexlansoprazole is the R-enantiomer of [DB00448], which is composed of a racemi…

Kategori:
2-PyridinylmethylsulfinylbenzimidazolesAcid ReducersAlimentary Tract and Metabolism +20
Target Protein:
Potassium-transporting ATPase alpha chain 1Potassium-transporting ATPase subunit betaN(G),N(G)-dimethylarginine dimethylaminohydrolase 1
Waktu ParuhDexlansoprazole is …
Vol. DistribusiThe apparent volume…
KlirensApparent clearance …
Genetik -
Dexpanthenol Approved DB09357
small molecule | CAS: 81-13-0

Dexpanthenol is an alcohol derivative of pantothenic acid, a component of the B complex vitamins and an essential component of a normally functioning epithelium. Dexpanthenol is enzymatically cleaved to form pantothenic acid, which is an essential component o…

Kategori:
AlanineAlimentary Tract and MetabolismAmino Acids +13
Waktu ParuhHalf life have not …
Vol. DistribusiDexpanthenol is rea…
Klirens-
Genetik -
Dextran Approved DB09255
small molecule | CAS: 9004-54-0

Dextran is a polysaccharide that differs from others in that its glucose units are joined together 1:6 glucoside links. The main chain of glucose has short branches at frequent intervals which are probably joined by 1:3 and 1:4 glucoside links. The chains can…

Kategori:
AnticoagulantsBiopolymersBlood and Blood Forming Organs +16
Waktu ParuhThe elimination hal…
Vol. DistribusiThe reported volume…
Klirens-
Genetik -
Dextropropoxyphene Approved DB00647
small molecule | CAS: 469-62-5

Dextropropoxyphene is an opioid analgesic manufactured by Eli Lilly and Company. It is used in the symptomatic treatment of mild pain. It displays antitussive and local anaesthetic actions. Due to the risk of cardiac arrhythmias and overdose, possibly leading…

Kategori:
Acids, AcyclicAgents that reduce seizure thresholdAnalgesics +22
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +2
Waktu Paruh6-12 hours
Vol. Distribusi* 16 L/kg
Klirens* 2.6 L/min
Genetik -
Dextrose, unspecified form Approved DB09341
small molecule

Glucose is a simple sugar (monosaccharide) generated during phosynthesis involving water, carbon and sunlight in plants. It is produced in humans via hepatic gluconeogenesis and breakdown of polymeric glucose forms (glycogenolysis). It circulates in human cir…

Kategori:
Caloric AgentsCardiac FunctionCompounds used in a research, industrial, or household setting +4
Waktu ParuhThe approximate hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean metabolic …
Genetik -
Dezamizumab DB15153
biotech | CAS: 1662664-56-3

Dezamizumab is under investigation in clinical trial NCT03417830 (Biodistribution of 89Zirconium-labelled GSK2398852 Using PET Imaging).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dezocine Approved DB01209
small molecule | CAS: 53648-55-8

Dezocine is a partial opiate drug and is used for pain management. Dezocine is a very effective alternative to fentanyl when administered during outpatient laparoscopy, although is associated with an increased incidence of postoperative nausea.

Kategori:
AnalgesicsCentral Nervous System AgentsCentral Nervous System Depressants +8
Target Protein:
Mu-type opioid receptorKappa-type opioid receptor
Waktu ParuhElimination half-li…
Vol. Distribusi-
Klirens-
Genetik -
DF-1001 DB18231
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Transferon is comprised of several peptides mixed from human dialyzable leucocyte extracts and acts as an immunomodulator. It is thought to have widespread effects on the immune system, and effective in treating infections and immunological issues.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsCytokines +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Diamorphine Approved DB01452
small molecule | CAS: 561-27-3

Diamorphine (heroin) is a narcotic analgesic that may be habit-forming. It is a controlled substance (opium derivative) listed in the U.S. Code of Federal Regulations, Title 21 Parts 329.1, 1308.11 (1987). Sale is forbidden in the United States by Federal sta…

Kategori:
AlkaloidsAnalgesicsCentral Nervous System Agents +16
Target Protein:
Mu-type opioid receptorKappa-type opioid receptorDelta-type opioid receptor +1
Waktu ParuhIn humans, administ…
Vol. DistribusiData regarding the …
KlirensSome studies have d…
Genetik -
Diazepam Approved DB00829
small molecule | CAS: 439-14-5

A benzodiazepine with anticonvulsant, anxiolytic, sedative, muscle relaxant, and amnesic properties and a long duration of action. Its actions are mediated by enhancement of gamma-aminobutyric acid activity. It is used in the treatment of severe anxiety disor…

Kategori:
Adjuvants, AnesthesiaAnestheticsAnesthetics, General +40
Target Protein:
Translocator proteinGABA(A) ReceptorGABA(A) Receptor Benzodiazepine Binding Site
Waktu ParuhDiazepam has a biph…
Vol. DistribusiIn young healthy ma…
KlirensThe clearance of di…
Genetik -
Dibotermin alfa Approved DB11639
biotech | CAS: 246539-15-1

Dibotermin alfa is a recombinant human bone morphogenetic protein-2 (rhBMP-2) derived from a recombinant Chinese Hamster Ovary (CHO) cell line [FDA Label]. It is implanted in patients undergoing bone surgeries or those with fractures. BMPs are subfamily of th…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBone Morphogenetic Proteins +7
Target Protein:
Bone morphogenetic protein receptor type-2Bone morphogenetic protein receptor type-1A
Waktu ParuhWhen injected intra…
Vol. Distribusi-
KlirensAt the site of impl…
Genetik -
Dichlorvos DB11397
small molecule | CAS: 62-73-7

Dichlorvos or 2,2-dichlorovinyl dimethyl phosphate is a drug of the _organophosphate_ class, frequently used as an insecticide for the control of indoor pests and for the protection of stored products from insect infestations. The compound has been available…

Kategori:
AgrochemicalsAnthelminticsAnti-Infective Agents +13
Target Protein:
SerotransferrinCholinesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 302776-68-7

Diethylamino hydroxybenzoyl hexyl benzoate is a UV filter with high absorption in the UV-A range. Minimizing the overexposure of human skin to ultraviolet radiation that may lead to acute and chronic photodamage, diethylamino hydroxybenzoyl hexyl benzoate is …

Kategori:
AminesAniline CompoundsBenzene Derivatives +3
Waktu ParuhNo pharmacokinetic …
Vol. DistribusiNo pharmacokinetic …
KlirensNo pharmacokinetic …
Genetik -
Diethyltoluamide Approved DB11282
small molecule | CAS: 134-62-3

Diethyltoluamide (DEET) is the common active ingredient in many insect repellent products. It is widely used to repel biting pests such as mosquitoes and ticks. Every year, DEET formulations are used to protect populations from mosquito-borne illnesses like W…

Kategori:
Acids, CarbocyclicAgrochemicalsAmides +11
Waktu ParuhThe elimination hal…
Vol. DistribusiAfter dermal applic…
KlirensReadily accessible …
Genetik -
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