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12560

Total database: 17430
Struktur (SMILES)
9109 (72.5%)
Target
6912 (55.0%)
Genomik
109 (0.9%)
Referensi
12560 (100.0%)

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Hasil Pencarian (12560)

Halaman 129 / 252
Icapamespib DB18106
small molecule | CAS: 1000999-96-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icaridin DB14074
small molecule | CAS: 119515-38-7

Icaridin, also known as Picaridin or hydroxy-ethyl isobutyl piperidine carboxylate, is a cyclic amine and a member of the piperidine chemical family. Piperidines are structural components of [piperine], which is a plant extract from the genus _Piper _, or pep…

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingInsect Repellents +4
Target Protein:
Odorant binding protein
Waktu ParuhThe first eliminati…
Vol. DistribusiIn a rat study, der…
KlirensThere is no availab…
Genetik -
Icariin DB12052
small molecule | CAS: 489-32-7

Icariin has been investigated for the basic science of the Pharmacokinetic Profile of Icariin in Humans.

Kategori:
BenzopyransChromonesDrugs, Chinese Herbal +3
Target Protein:
cGMP-specific 3',5'-cyclic phosphodiesterase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icaritin DB12672
small molecule | CAS: 118525-40-9

Icaritin has been used in trials studying the treatment of Solid Tumors, Metastatic Breast Cancer, and Hepatocellular Carcinoma (HCC).

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icatibant Approved DB06196
biotech | CAS: 130308-48-4

Icatibant is a synthetic decapeptide with 5 nonproteinogenic amino acid antagonist targeting the B<sub>2</sub> receptors with a similar affinity to bradykinin. It is resistant to bradykinin-cleaving enzyme degradation and has a potency of 2-3 times higher tha…

Kategori:
Agents causing angioedemaAmino Acids, Peptides, and ProteinsAnalgesics +21
Target Protein:
B2 bradykinin receptorAminopeptidase N
Waktu ParuhFollowing subcutane…
Vol. DistribusiFollowing subcutane…
KlirensFollowing subcutane…
Genetik -
Icerguastat DB16932
small molecule | CAS: 951441-04-6

Deskripsi belum tersedia.

Kategori:
AmidinesGuanidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ICG-001 DB18024
small molecule | CAS: 780757-88-2

Deskripsi belum tersedia.

Kategori:
Pyrimidines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ichorcumab DB18930
biotech | CAS: 2589583-20-8

Ichorcumab is under investigation in clinical trial NCT03251482 (A Study to Evaluate the Safety and Efficacy of Intravenous JNJ-64179375 Versus Oral Apixaban in Participants Undergoing Elective Total Knee Replacement Surgery).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iclaprim DB06358
small molecule | CAS: 192314-93-5

Deskripsi belum tersedia.

Kategori:
Antibacterials for Systemic UseAntiinfectives for Systemic UseEnzyme Inhibitors +3
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iclepertin DB19058
small molecule | CAS: 1421936-85-7

Iclepertin is under investigation in clinical trial NCT05211947 (A Study to Test Long-term Safety of Iclepertin in People With Schizophrenia Who Took Part in a Previous CONNEX Study).

Target Protein:
Sodium- and chloride-dependent glycine transporter 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
iCo-007 DB05268
small molecule

iCo-007 (formerly known as ISIS 13650) is a second generation antisense compound being developed by iCo for the treatment of various eye diseases caused by the formation of new blood vessels (angiogenesis) such as age-related macular degeneration (AMD) and di…

Target Protein:
RAF proto-oncogene serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icodextrin Approved DB00702
small molecule | CAS: 337376-15-5

Icodextrin is an iso-osmotic peritoneal dialysis solution containing glucose polymers. It is used primarily for ambulatory peritoneal dialysis (CAPD) of diabetic patients and automated peritoneal dialysis (APD) for patients with end-stage renal disease. It is…

Kategori:
BiopolymersCarbohydratesCompounds used in a research, industrial, or household setting +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Icosabutate DB12990
small molecule | CAS: 1253909-57-7

Icosabutate is under investigation in clinical trial NCT02373176 ([14C] Icosabutate -A Phase I Absorption, Metabolism and Excretion Study).

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icosapent Approved DB00159
small molecule | CAS: 10417-94-4

Important polyunsaturated fatty acid found in fish oils. It serves as the precursor for the prostaglandin-3 and thromboxane-3 families. A diet rich in eicosapentaenoic acid lowers serum lipid concentration, reduces incidence of cardiovascular disorders, preve…

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnti-Inflammatory Agents +17
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor gamma +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Icosapent ethyl Approved DB08887
small molecule | CAS: 86227-47-6

Icosapent ethyl or ethyl eicosapentaenoic acid is a synthetic derivative of the omega-3 fatty acid eicosapentaenoic acid (EPA). It is used as an adjunct therapy for severe hypertriglyceridemia (TG levels > 500 mg/dL) and to reduce the risk of cardiovascular e…

Kategori:
Antiplatelet agentsDietary FatsDietary Fats, Unsaturated +12
Waktu ParuhThe half life of EP…
Vol. DistribusiSteady state volume…
KlirensTotal plasma cleara…
Genetik -
ICX-RHY DB05716
biotech

ICX-RHY is an investigational therapy comprised of cultured allogeneic fibroblasts. The drug was under investigation in clinical trials in the UK for the treatment of skin erosions in recessive dystrophic epidermolysis bulllosa.

Waktu Paruh-
Vol. Distribusi-
Klirens-
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Idalopirdine DB11957
small molecule | CAS: 467459-31-0

Idalopirdine has been used in trials studying the treatment of Cognition, Schizophrenia, and Alzheimer's Disease.

Kategori:
AminesAntidepressive AgentsBenzene Derivatives +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idanpramine DB13276
small molecule | CAS: 25466-44-8

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idarubicin Approved DB01177
small molecule | CAS: 58957-92-9

An orally administered anthracycline antineoplastic. The compound has shown activity against breast cancer, lymphomas and leukemias, together with the potential for reduced cardiac toxicity.

Kategori:
Anthracycline Topoisomerase InhibitorAnthracyclinesAnthracyclines and Related Substances +19
Target Protein:
DNA topoisomerase 2-betaDNADNA topoisomerase 2-alpha
Waktu Paruh22 hours
Vol. Distribusi-
Klirens-
Genetik -
Idarucizumab Approved DB09264
biotech | CAS: 1362509-93-0

Idarucizumab is a humanized monoclonal antibody fragment (Fab) derived from an immunoglobulin G1 isotype molecule that binds to and inactivates the oral anticoagulant dabigatran, thereby reversing its anticoagulant effect. As a direct acting oral anticoagulan…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +10
Waktu Paruhinitial half-life: …
Vol. Distribusi8.9 L
Klirens47.0 mL/min
Genetik -
Idasanutlin DB12325
small molecule | CAS: 1229705-06-9

Idasanutlin has been used in trials studying the treatment of Neoplasms, Non-Hodgkin's Lymphoma, Leukemia, Myeloid, Acute, Recurrent Plasma Cell Myeloma, and Neoplasms, Leukemia, Acute Myeloid Leukemia.

Kategori:
Acids, CarbocyclicAminobenzoatesBenzene Derivatives +2
Target Protein:
E3 ubiquitin-protein ligase Mdm2Receptor tyrosine-protein kinase erbB-4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idazoxan DB12551
small molecule | CAS: 79944-58-4

Idazoxan has been used in trials studying the basic science of Molecular Imaging, Alzheimer Disease, and Major Depressive Disorder.

Kategori:
Adrenergic AgentsAdrenergic alpha-2 Receptor AntagonistsAdrenergic alpha-Antagonists +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDD-1 DB05439
biotech

Lipids promote the fusion of liposomes to cells. Eladem (IDD-1) is a therapeutic vaccine consisting of dendritophages that are loaded in vitro with tumor antigens and then reinjected into the subject. As with other monoclonal antibodies, this process stimulat…

Waktu Paruh-
Vol. Distribusi-
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IDD-3 DB05427
biotech

IDD-3 is a therapeutic specific immunostimulant developed by IDM Pharma in partnership with sanofi-aventis. It consists of mature dendritic cells loaded with lysates from melanoma tumor cell lines. It includes Dendritophages that are dendritic cells, a type o…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDD552 DB02834
small molecule

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesHydrocarbons, FluorinatedHydrocarbons, Halogenated +1
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDD594 DB08084
small molecule

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAldehyde Reductase, antagonists & inhibitorsAmides +4
Target Protein:
Aldo-keto reductase family 1 member B1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idebenone Approved DB09081
small molecule | CAS: 58186-27-9

Idebenone is a synthetic analogue of ubiquinone (also known as Coenzyme Q10), a vital cell antioxidant and essential component of the Electron Transport Chain (ETC). It has been proposed that by interacting with the ETC, idebenone increases ATP production req…

Kategori:
AntioxidantsBenzoquinonesBiological Factors +9
Waktu Paruh-
Vol. DistribusiExperimental data h…
Klirens-
Genetik -
Idecabtagene vicleucel Approved DB16665
biotech

Multiple myeloma is a cancer where plasma cells rapidly divide out of control.[A232563] These cancerous cells generally express the B-cell maturation antigen, while it is rarely expressed on non-cancerous cells.[A232563] Multiple myeloma is typically treated …

Kategori:
Amino Acids, Peptides, and ProteinsAntineoplastic AgentsAntineoplastic Agents, Immunological +11
Target Protein:
Tumor necrosis factor receptor superfamily member 17
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idelalisib Approved DB09054
small molecule | CAS: 870281-82-6

Idelalisib is a phosphoinositide 3-kinase inhibitor indicated in the treatment of chronic lymphocytic leukemia (CLL), relapsed follicular B-cell non-Hodgkin lymphoma (FL), and relapsed small lymphocytic lymphoma (SLL). For the treatment of relapsed CLL, it is…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +47
Target Protein:
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
Waktu ParuhThe terminal elimin…
Vol. Distribusi23 L
Klirens14.9 L/hr
Genetik -
IDM-1 DB05292
small molecule

IDM-1 is IDM’s most advanced antibody-based Cell drug for the treatment of cancer. It is comprised of MAK(Monocytes-derived Activated Killer) cells associated with MDX-210, a bispecific anti-HER-2/neu antibody developed by Medarex Inc.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDM-2 DB05293
small molecule

IDM-2 is composed of Monocyte-derived Activated Killer (MAK) cells. IDM produces MAK cells from the patient's own white blood cells by activating these cells ex vivo to allow them to recognize and destroy tumor cells.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDM-4 DB05438
biotech

IDM-4 is an immuno-designed molecule that completed phase I/II of investigation for the treatment of Leukemia. It is a monoclonal antibody-specific antigen that can selectively target cancer-affected cells by coupling with tumor cell-killing MAK cells, which …

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDN-7314 DB18073
small molecule | CAS: 254750-11-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idoxuridine Approved DB00249
small molecule | CAS: 54-42-2

An analog of deoxyuridine that inhibits viral DNA synthesis. The drug is used as an antiviral agent.

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +15
Target Protein:
DNAThymidine kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idraparinux DB06406
small molecule | CAS: 162610-17-5

Idraparinux, a synthetic pentasaccharide is an antithrombin-dependent inhibitor of activated factor X. It was developed for the treatment and prevention of thromboembolic events. However, clinical trials have revealed that idraparinux had lead to bleeding. As…

Kategori:
AnticoagulantsAntithrombinsCarbohydrates +6
Target Protein:
Coagulation factor X
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idrevloride DB18042
small molecule | CAS: 1416973-63-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idronoxil DB04915
small molecule | CAS: 81267-65-4

Idronoxil is a substance that is being studied in the treatment of cancer. It belongs to the family of drugs called signal transduction inhibitors.

Kategori:
BenzopyransChromonesFlavonoids +2
Target Protein:
E3 ubiquitin-protein ligase XIAPSphingosine kinase 1Ecto-NOX disulfide-thiol exchanger 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 56472-29-8

Deskripsi belum tersedia.

Kategori:
Fatty AcidsFatty Acids, MonounsaturatedFatty Acids, Unsaturated +1
Target Protein:
Phosphatidylcholine:ceramide cholinephosphotransferase 1Phosphatidylcholine:ceramide cholinephosphotransferase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IDRX-42 DB18087
small molecule | CAS: 2590556-80-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Idursulfase Approved DB01271
biotech | CAS: 50936-59-9

Idursulfase is a purified form of human iduronate-2-sulfatase, a lysosomal enzyme. Idursulfase is produced by recombinant DNA technology in a human cell line. Idursulfase is an enzyme that hydrolyzes the 2-sulfate esters of terminal iduronate sulfate residues…

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes +4
Target Protein:
Dermatan sulfateHeparan sulfatePerilipin-3
Waktu Paruh44 &plusmn; 19 minu…
Vol. Distribusi-
Klirens* 3 mL/min/kg [Pati…
Genetik -
biotech | CAS: 1271734-34-9

Idursulfase beta is under investigation in clinical trial NCT01645189 (Safety and Efficacy of Hunterase).

Kategori:
Alimentary Tract and MetabolismEnzymesEnzymes and Coenzymes
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ieramilimab DB16419
biotech | CAS: 2137049-37-5

Ieramilimab is under investigation in clinical trial NCT02460224 (Safety and Efficacy of LAG525 Single Agent and in Combination With PDR001 in Patients With Advanced Malignancies.).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifebemtinib DB17570
small molecule | CAS: 1227948-82-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifenprodil DB08954
small molecule | CAS: 23210-56-2

N-methyl-D-aspartate (NMDA) receptors (NMDARs) are members of the ionotropic glutamate receptor family, with key roles in brain development and neurological function.[A220118, A220128] NMDARs are heterotetramers that typically involve a dimer of dimers of bot…

Kategori:
Adrenergic AgentsAdrenergic alpha-AntagonistsAdrenergic Antagonists +12
Target Protein:
Glutamate receptor ionotropic, NMDA 2BChymotrypsin-like elastase family member 1Glutamate receptor ionotropic, NMDA 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iferanserin DB11686
small molecule | CAS: 58754-46-4

Iferanserin has been investigated for the treatment of Hemorrhoids.

Kategori:
Acids, CarbocyclicAntidepressive AgentsCentral Nervous System Depressants +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2407582-19-6

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ifidancitinib DB16191
small molecule | CAS: 1236667-40-5

Ifidancitinib is under investigation in clinical trial NCT03585296 (A Study of ATI-502 Topical Solution for the Treatment of Atopic Dermatitis).

Kategori:
Adrenal Cortex HormonesFused-Ring CompoundsNorpregnanes +4
Target Protein:
Tyrosine-protein kinase JAK3Tyrosine-protein kinase JAK1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2484870-92-8

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IFx-Hu2.0 DB18396
biotech

IFx-Hu2.0 is an investigational cancer vaccine. It is composed of plasmid DNA encoding the streptococcal membrane protein, Emm55, contained within a cationic polymer.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
IGN101 DB06500
biotech

IGN101 is an antibody-based cancer vaccine directed against epithelial cancers. It consists of 500 ug 17-1A antibody adsorbed on aluminum hydroxide.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
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