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11778

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8554 (72.6%)
Target
6383 (54.2%)
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96 (0.8%)
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11778 (100.0%)

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Hasil Pencarian (11778)

Halaman 128 / 236
IQP-0528 DB14888
small molecule | CAS: 301297-45-0

IQP-0528 is under investigation in clinical trial NCT03082690 (ImQuest (IQP) DuoGel Phase 1 Pharmacokinetic Study).

Kategori:
Anti-HIV AgentsPyrimidines
Waktu Paruh-
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IR-901 DB17932
biotech | CAS: 146446-23-3

Deskripsi belum tersedia.

Waktu Paruh-
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Iratumumab DB05550
biotech | CAS: 640735-09-7

Immunoglobulin G1, anti-(human CD30 (antigen)) (human monoclonal MDX-060 heavy chain), disulfide with human monoclonal MDX-060 light chain, dimer. Molecular weight is approximately 170,000 daltons. In phase I/II clinical trials for treatment of CD30+ lymphoma…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Target Protein:
Tumor necrosis factor receptor superfamily member 8
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Irbesartan Approved DB01029
small molecule | CAS: 138402-11-6

Irbesartan is an angiotensin receptor blocker (ARB) indicated to treat hypertension or diabetic nephropathy.[L7456,L7459] It can also be used as part of a combination product with [hydrochlorothiazide] for patients not well controlled or not expected to be we…

Kategori:
Agents Acting on the Renin-Angiotensin SystemAgents causing hyperkalemiaAngiotensin 2 Receptor Blocker +24
Target Protein:
Type-1 angiotensin II receptorTranscription factor Jun
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensTotal plasma cleara…
Genetik -
Irinotecan Approved DB00762
small molecule | CAS: 97682-44-5

Irinotecan is a topoisomerase inhibitor used for chemotherapy. It is a water-soluble analogue of [camptothecin], which is extracted from the Chinese tree _Camptotheca acuminate_.[A263376] The bis-piperidine side chain in the structure of irinotecan bestows en…

Kategori:
AlkaloidsAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +29
Target Protein:
DNA topoisomerase I, mitochondrialDNA topoisomerase 1
Gen Terkait:
SLCO1B1 UGT1A1 UGT1A7 +2
Waktu ParuhAfter intravenous i…
Vol. DistribusiFollowing intraveno…
KlirensThe mean (± standar…
Genetik 5 Varian
Irofulven DB05786
small molecule | CAS: 158440-71-2

A novel anti-cancer compound synthesized by scientists at the University of California, San Diego more than a decade ago from toxins of the poisonous jack-o-lantern mushroom, has been granted “fast track” status by the U.S. Food and Drug Administration (FDA) …

Kategori:
Alkylating DrugsAntineoplastic AgentsAntineoplastic Agents, Alkylating +4
Target Protein:
Serine/threonine-protein kinase Chk2Far upstream element-binding protein 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iron Approved DB01592
small molecule | CAS: 7439-89-6

A metallic element found in certain minerals, in nearly all soils, and in mineral waters. It is an essential constituent of hemoglobin, cytochrome, and other components of respiratory enzyme systems. Its chief functions are in the transport of oxygen to tissu…

Kategori:
Alimentary Tract and MetabolismAntianemia DrugsAntianemic Preparations +14
Target Protein:
Hemoglobin subunit alphaTransferrin receptor protein 1Egl nine homolog 1 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 764-65-8

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicDicarboxylic AcidsOAT3/SLC22A8 Inhibitors
Target Protein:
Organic anion transporter 3
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Iron isomaltoside 1000 Approved DB12208
small molecule | CAS: 1370654-58-2

Iron isomaltoside 1000 is under investigation in Iron Deficiency Anaemia. Iron isomaltoside 1000 has been investigated for the treatment and basic science of Anemia, Gastric Cancer, Esophageal Cancer, Chronic Kidney Disease, and Anemia, Iron-Deficiency, among…

Kategori:
CarbohydratesHematinicsHematologic Agents +3
Waktu Paruh-
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Genetik -
small molecule | CAS: 53858-86-9

Deskripsi belum tersedia.

Kategori:
HematinicsHematologic AgentsIron Compounds +1
Waktu Paruh-
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Iron protein succinylate Approved DB11209
small molecule | CAS: 250705-13-6

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAmino Acids, Peptides, and ProteinsAntianemic Preparations +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iron sucrose Approved DB09146
small molecule | CAS: 8047-67-4

Iron sucrose (sucroferric oxyhydroxide or iron saccharate) is used as a source of iron in patients with iron deficiency anemia with chronic kidney disease (CKD), including those who are undergoing dialysis (hemodialysis or peritoneal) and those who do not req…

Kategori:
Acids, AcyclicCarbohydratesDisaccharides +12
Waktu Paruh6 hours.
Vol. DistribusiVd is 7.3 L
KlirensTotal body clearanc…
Genetik -
Irosustat DB02292
small molecule | CAS: 288628-05-7

Irosustat has been investigated for the treatment of Metastatic Breast Cancer and Locally Advanced Breast Cancer.

Kategori:
AcidsAcids, NoncarboxylicSteryl-Sulfatase, antagonists & inhibitors +2
Target Protein:
Steryl-sulfataseCarbonic anhydrase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iroxanadine DB05444
small molecule | CAS: 276690-58-5

BRX-235 (iroxanadine) is a a novel small molecule synthesized by Biorex, Hungary that acts as a cardioprotective agent. It induces phosphorylation of p38 SAPK, which plays an important role in EC homeostasis. endothelial cell (EC). EC function plays a central…

Target Protein:
Heat shock 70 kDa protein 1AHeat shock 70 kDa protein 1B
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Irpagratinib DB18732
small molecule | CAS: 2230974-62-4

Irpagratinib (ABSK011) is a highly selective inhibitor of fibroblast growth factor receptor (FGFR) 4.

Waktu Paruh-
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Irsenontrine DB19044
small molecule | CAS: 1429509-82-9

Irsenontrine is under investigation in clinical trial NCT03467152 (Study to Evaluate the Efficacy, Safety and Tolerability of E2027 (Hereinafter Referred to as Irsenontrine) in Participants With Dementia With Lewy Bodies).

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Irsogladine DB13056
small molecule | CAS: 57381-26-7

Irsogladine is under investigation in clinical trial NCT02581696 (The Drug-drug Interaction and Safety of Lafutidine and Irsogladine Maleate in Healthy Adult Volunteers).

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAnticarcinogenic Agents +6
Waktu Paruh-
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Iruplinalkib DB17494
small molecule | CAS: 1854943-32-0

Deskripsi belum tersedia.

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IRX-2 DB05643
biotech | CAS: 951209-71-5

IRX-2 contains a human leukocyte-derived cytokine mixture. It is being investigated to promote or enhance an anti-cancer immune response.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsIntercellular Signaling Peptides and Proteins +2
Waktu Paruh-
Vol. Distribusi-
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IRX-5183 DB05653
small molecule | CAS: 367273-07-2

Deskripsi belum tersedia.

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
Retinoic acid receptor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ISA101b DB18694
biotech

ISA101b (peltopepimut-S) is a therapeutic vaccine against the HPV-specific E6/E7 oncoproteins.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
biotech | CAS: 2378601-29-5

Isaralgagene civaparvovec, formerly known as ST-920, is liver-tropic rAAV 2/6 vector carrying the cDNA for human alpha-galactosidase A (?-Gal A) enzyme. It is developed by Sangamo Therapeutics and investigated in Fabry Disease.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
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Isatoribine DB04860
small molecule | CAS: 122970-40-5

Isatoribine is a selective agonist of TLR7.

Kategori:
Heterocyclic Compounds, Fused-RingNucleic Acids, Nucleotides, and NucleosidesNucleosides +3
Target Protein:
Toll-like receptor 7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isatuximab Approved DB14811
biotech | CAS: 1461640-62-9

Isatuximab (formerly SAR650984) is a humanized, IgG1-derived monoclonal antibody (mAb) produced from a Chinese hamster ovary (CHO) cell line.[L12099,A191799] Structurally, isatuximab is comprised of two identical immunoglobulin kappa light chains and two iden…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +16
Target Protein:
ADP-ribosyl cyclase/cyclic ADP-ribose hydrolase 1
Waktu Paruh-
Vol. DistribusiThe predicted volum…
KlirensTotal clearance dec…
Genetik -
Isavuconazole Approved DB11633
small molecule | CAS: 241479-67-4

Isavuconazole is an triazole antifungal with broad spectrum of activity and good safety profile [A32026]. It is approved by the FDA and EMA for the treatment of invasive aspergillosis and mucormycosis. It works by inhibiting fungal cell membrane synthesis. In…

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiinfectives for Systemic Use +38
Target Protein:
Lanosterol 14-alpha demethylaseVoltage-gated inwardly rectifying potassium channel KCNH2Voltage-dependent L-type calcium channel subunit alpha-1C +7
Waktu ParuhBased on a populati…
Vol. DistribusiThe mean steady sta…
KlirensThe clearance (CL) …
Genetik -
Isavuconazonium Approved DB06636
small molecule | CAS: 742049-41-8

Isavuconazonium is a second-generation triazole antifungal approved on March 6, 2015 by the FDA and July 2015 by the EMA for the treatment of adults with invasive aspergillosis and invasive mucormycosis, marketed by Astellas under the brand Cresemba.[A38834] …

Kategori:
Anti-Infective AgentsAntifungal AgentsAzole Antifungals +31
Target Protein:
Lanosterol 14-alpha demethylase
Waktu ParuhBased on a populati…
Vol. DistribusiIsavuconazole is ex…
KlirensIn healthy subjects…
Genetik -
ISB 1342 DB17251
biotech

ISB 1342 is a bispecific antibody simultaneously targeting CD38 and CD3.

Waktu Paruh-
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Genetik -
ISB 1442 DB18475
biotech

ISB 1442 is a bispecific, biparatopic antibody targeting CD38 and CD47

Waktu Paruh-
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Genetik -
ISB 2001 DB18570
biotech

ISB 2001 is a T cell-engaging antibody that targets BCMA, CD38, and CD3.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iscotrizinol DB15468
small molecule | CAS: 154702-15-5

Deskripsi belum tersedia.

Kategori:
Sunscreen Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Iseganan DB16010
biotech | CAS: 257277-05-7

Iseganan is under investigation in clinical trial NCT00022373 (Iseganan Hydrochloride in Preventing Oral Mucositis in Patients Who Are Undergoing Radiation Therapy for Head and Neck Cancer).

Kategori:
Amino Acids, Peptides, and ProteinsAntimicrobial PeptidesMembrane Proteins +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Isepamicin DB13540
small molecule | CAS: 58152-03-7

Deskripsi belum tersedia.

Kategori:
Agents that produce neuromuscular block (indirect)Aminoglycoside AntibacterialsAnti-Bacterial Agents +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ISIS 104838 DB16201
biotech | CAS: 250755-32-9

ISIS 104838 is under investigation in clinical trial NCT00048321 (ISIS 104838, an Inhibitor of Tumor Necrosis Factor, for Active Rheumatoid Arthritis).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
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ISIS 113715 DB05506
small molecule

ISIS 113715 is our second-generation antisense inhibitor of protein tyrosine phosphatase 1b, or PTP?1b, for the treatment of type 2 diabetes. In early trials, ISIS 113715 induced statistically significant improvements in multiple measures of glucose control a…

Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ISIS 2503 DB16181
biotech | CAS: 149957-14-2

ISIS 2503 is under investigation in clinical trial NCT00004193 (ISIS 2503 in Treating Patients With Metastatic And/or Locally Recurrent Colorectal Cancer).

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ISIS 325568 DB06099
small molecule

ISIS 325568 is a generation 2.2 antisense drug that targets the glucagon receptor (GCGR). It was under investigation in clinical trial NCT00519727 (Safety Study of ISIS 325568 in Healthy Volunteers) for lowering blood glucose and helping control type 2 diabet…

Target Protein:
Glucagon receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ISIS-333611 DB17978
biotech | CAS: 937407-37-9

Deskripsi belum tersedia.

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Genetik -
ISO-1 F-18 DB14900
small molecule | CAS: 945992-47-2

ISO-1 F-18 is under investigation in clinical trial NCT00968656 (Assessment of Cellular Proliferation in Tumors by Positron Emission Tomography (PET) Using [18F]ISO-1).

Target Protein:
Sigma intracellular receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoaminile Approved DB08944
small molecule | CAS: 77-51-0

Isoaminile, an antitussive drug with a structure similar to methadone, is also an anticholinergic with both antimuscarinic and antinicotinic properties.

Kategori:
Antitussive AgentsCentral Nervous System AgentsCough and Cold Preparations +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isobromindione DB13545
small molecule | CAS: 1470-35-5

Deskripsi belum tersedia.

Kategori:
Antigout PreparationsMusculo-Skeletal SystemPreparations Increasing Uric Acid Excretion
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isobutyramide DB17705
small molecule | CAS: 563-83-7

Deskripsi belum tersedia.

Kategori:
Antineoplastic Agents
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isobutyric acid DB02531
small molecule | CAS: 79-31-2

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicButyratesFatty Acids +2
Target Protein:
Free fatty acid receptor 22-hydroxy-6-oxo-7-methylocta-2,4-dienoate hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isocaproic acid DB03993
small molecule | CAS: 646-07-1

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicFatty AcidsFatty Acids, Volatile +1
Target Protein:
Branched-chain-amino-acid aminotransferase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isocarboxazid Approved DB01247
small molecule | CAS: 59-63-2

Isocarboxazid has the formula 1-benzyl-2-(5-methyl-3-isoxazolylcarbonyl)hydrazine-isocarboxazid. It is a monoamine oxidase inhibitor.[A31930] It is used in the treatment of major depression, dysthymic disorder, atypical disorder, panic disorder and the phobic…

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAntidepressive Agents +17
Target Protein:
Amine oxidase [flavin-containing] AAmine oxidase [flavin-containing] B
Waktu ParuhThe pharmacokinetic…
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 22642-82-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicCyclohexanecarboxylic AcidsCyclohexanes +3
Target Protein:
Phenazine biosynthesis protein PhzD
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isocitric Acid DB01727
small molecule | CAS: 320-77-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicCitratesTricarboxylic Acids
Target Protein:
Isocitrate dehydrogenase [NADP]Isocitrate dehydrogenase [NADP]Aconitate hydratase, mitochondrial +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoconazole Approved DB08943
small molecule | CAS: 27523-40-6

Isoconazole is an azole antifungal drug that has similar effectiveness to clotrimazole in the treatment of foot and vaginal infections.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +9
Target Protein:
Steroid 17-alpha-hydroxylase/17,20 lyase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isocyanomethane DB04337
small molecule | CAS: 593-75-9

Deskripsi belum tersedia.

Target Protein:
Myoglobin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoetharine Approved DB00221
small molecule | CAS: 79490-84-9

Isoetharine is a relatively selective beta-2 adrenergic agonist. It is a catechol-like agent. Isoetharine is a fast-acting bronchodilator used for emphysema, bronchitis and asthma.[A330]

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +16
Target Protein:
Beta-1 adrenergic receptorBeta-2 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Isoeugenol Approved DB14188
small molecule | CAS: 97-54-1

Isoeugenol is a commonly used fragrance added to many commercially available products, and occurs naturally in the essential oils of plants such as ylang-ylang. It is also a significant dermatologic sensitizer and allergen, and as a result has been restricted…

Kategori:
Acids, CarbocyclicAlkenesAllyl Compounds +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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