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16004

Total database: 17430
Struktur (SMILES)
12010 (75.0%)
Target
9041 (56.5%)
Genomik
112 (0.7%)
Referensi
16004 (100.0%)

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Distribusi Wujud Zat

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Hasil Pencarian (16004)

Halaman 128 / 321
Dixanthogen DB13712
small molecule | CAS: 502-55-6

Deskripsi belum tersedia.

Kategori:
AnionsAntiparasitic Products, Insecticides and RepellentsEctoparasiticides, Incl. Scabicides +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dixyrazine DB13784
small molecule | CAS: 2470-73-7

Deskripsi belum tersedia.

Kategori:
AnalgesicsAnalgesics, Non-NarcoticAntiemetics +16
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha tocopheryl acetate Approved DB14477
small molecule | CAS: 52225-20-4

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-alpha-Tocopherol Approved DB14476
small molecule | CAS: 10191-41-0

Deskripsi belum tersedia.

Kategori:
Vitamin EVitaminsVitamins (Fat Soluble)
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 18656-38-7

A synthetic phospholipid used in liposomes and lipid bilayers for the study of biological membranes. It is used in commercial drug preparations to solubilize drugs for injection [A32711]

Kategori:
Compounds used in a research, industrial, or household settingGlycerophosphatesGlycerophospholipids +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61361-72-6

DL-dimyristoylphosphatidylglycerol is a phospholipid used in commercially available pharmaceutical preparations to solubilize drugs for injection.

Kategori:
GlycerophosphatesGlycerophospholipidsLipids +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DL-Methylephedrine Approved DB11278
small molecule | CAS: 1201-56-5

Methylephedrine is a sympathomimetic amine that appears in various over-the-counter cough and cold medications throughout the world [L2838], [L2839], [L2840]. The abuse of methylephedrine-containing medications has been reported in Japan. Methylephedrine is n…

Kategori:
Adrenergic AgonistsAdrenergic alpha-2 Receptor AgonistsAdrenergic alpha-Agonists +10
Target Protein:
Beta-1 adrenergic receptorAlpha-2A adrenergic receptorAlpha adrenergic receptor +1
Waktu Paruh3-6 hours (Ephedrin…
Vol. DistribusiEphedrine: 2.5-3.0 …
Klirens-
Genetik -
DM-1157 DB18600
small molecule | CAS: 1239953-66-2

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DMP-777 DB18488
small molecule | CAS: 157341-41-8

DMP-777 is a selective inhibitor of polymorphonuclear leukocyte (PMN) elastase.

Kategori:
AzetinesEnzyme InhibitorsPancreatic Elastase, antagonists & inhibitors
Target Protein:
Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNB-001 DB05757
small molecule

DNB-001 is a first-in-class oral therapy with dual mechanism of action, which is initially being developed for the treatment of glaucoma. In preclinical animal models, DNB-001 has demonstrated potent IOP- lowering effects as well as neuroprotective effects on…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DNL343 DB18678
small molecule | CAS: 2278265-85-1

DNL343 is under investigation in clinical trial NCT05842941 (HEALEY ALS Platform Trial - Regimen G DNL343).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dobesilic acid DB13529
small molecule | CAS: 88-46-0

Deskripsi belum tersedia.

Kategori:
Antivaricose TherapyArylsulfonatesArylsulfonic Acids +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dobutamine Approved DB00841
small molecule | CAS: 34368-04-2

A beta-1 agonist catecholamine that has cardiac stimulant action without evoking vasoconstriction or tachycardia. It is proposed as a cardiotonic after myocardial infarction or open heart surgery.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic alpha-1 Receptor Agonists +28
Target Protein:
Alpha-1 adrenergic receptorsBeta-1 adrenergic receptorBeta-2 adrenergic receptor +1
Waktu Paruh2 minutes
Vol. Distribusi-
Klirens-
Genetik -
Docaravimab DB17802
biotech | CAS: 2247196-23-0

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docarpamine DB18046
small molecule | CAS: 74639-40-0

Deskripsi belum tersedia.

Kategori:
AminesBenzene DerivativesBiogenic Amines +8
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docetaxel Approved DB01248
small molecule | CAS: 114977-28-5

Docetaxel is a clinically well established anti-mitotic chemotherapy medication used for the treatment of different types of cancer, including breast, ovarian, and non-small cell lung cancer. Docetaxel is a complex diterpenoid molecule and a semisynthetic ana…

Kategori:
Agents Causing Muscle ToxicityAntimitotic AgentsAntineoplastic Agents +32
Target Protein:
Tubulin beta-1 chainApoptosis regulator Bcl-2Nuclear receptor subfamily 1 group I member 2
Gen Terkait:
ABCC2
Waktu ParuhWith plasma samplin…
Vol. DistribusiDocetaxel has a ste…
KlirensAfter the administr…
Genetik 1 Varian
small molecule | CAS: 177021-00-0

Deskripsi belum tersedia.

Kategori:
AnticoagulantsCarbohydratesExperimental Unapproved Treatments for COVID-19 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doconexent Approved DB03756
small molecule | CAS: 6217-54-5

A mixture of fish oil and primrose oil, doconexent is used as a high-docosahexaenoic acid (DHA) supplement. DHA is a 22 carbon chain with 6 cis double bonds with anti-inflammatory effects. It can be biosythesized from alpha-linolenic acid or commercially manu…

Kategori:
Cytochrome P-450 CYP2C9 InhibitorsCytochrome P-450 CYP2C9 Inhibitors (strength unknown)Cytochrome P-450 CYP2C9 Substrates +11
Target Protein:
Peroxisome proliferator-activated receptor alphaProstaglandin G/H synthase 1Prostaglandin G/H synthase 2 +6
Waktu ParuhApproximately 20 ho…
Vol. DistribusiDHA is the most abu…
Klirens-
Genetik -
Docosanol Approved DB00632
small molecule | CAS: 661-19-8

Docosanol is a drug used for topical treatment for recurrent herpes simplex labialis episodes (episodes of cold sores or fever blisters). A saturated 22-carbon aliphatic alcohol, docosanol exhibits antiviral activity against many lipid enveloped viruses inclu…

Kategori:
AlcoholsAnti-Infective AgentsAntiviral Agents +2
Target Protein:
Envelope glycoprotein GP350Envelope glycoprotein GP340
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Docusate Approved DB11089
small molecule | CAS: 10041-19-7

Docusate, or dioctyl sulfosuccinate, is a stool softener indicated for the treatment of constipation[A32201]. Docusate acts by increasing the amount of water the stool absorbs in the gut, making the stool softer and easier to pass [L1801]. Docusate can be ora…

Kategori:
Alimentary Tract and MetabolismDrugs for ConstipationEnemas +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1442645-21-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dodecyl sulfate DB03967
small molecule | CAS: 151-41-7

Deskripsi belum tersedia.

Kategori:
AlcoholsAlkanesulfonatesAlkanesulfonic Acids +8
Target Protein:
Lysozyme CLipid A palmitoyltransferase PagP
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Retinoic acid receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dodecyl-Coa DB03264
small molecule

Deskripsi belum tersedia.

Target Protein:
3-oxoacyl-[acyl-carrier-protein] synthase 3Fatty acid metabolism regulator protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 1643-20-5

Deskripsi belum tersedia.

Kategori:
AminesCompounds used in a research, industrial, or household settingDetergents +3
Target Protein:
Dihydroorotate dehydrogenase (quinone), mitochondrialReaction center protein L chainReaction center protein M chain +47
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10182-91-9

Deskripsi belum tersedia.

Kategori:
AminesAmmonium CompoundsCompounds used in a research, industrial, or household setting +5
Target Protein:
Tyrosine-protein phosphatase non-receptor type 11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dofequidar DB14067
small molecule | CAS: 129716-58-1

Dofequidar is an antineoplastic agent.

Kategori:
Antineoplastic AgentsHeterocyclic Compounds, Fused-RingP-glycoprotein inhibitors
Target Protein:
ATP-binding cassette sub-family B member 5ATP-dependent translocase ABCB1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dofetilide Approved DB00204
small molecule | CAS: 115256-11-6

Dofetilide is a class III antiarrhythmic agent that is approved by the Food and Drug Administration (FDA) for the maintenance of sinus rhythm in individuals prone to the formation of atrial fibrillation and flutter, and for the chemical cardioversion to sinus…

Kategori:
AmidesAminesAntiarrhythmic agents +17
Target Protein:
Voltage-gated inwardly rectifying potassium channel KCNH2Potassium channel subfamily K member 2ATP-sensitive inward rectifier potassium channel 12
Waktu Paruh10 hours
Vol. Distribusi* 3 L/kg
Klirens-
Genetik -
Dolasetron Approved DB00757
small molecule | CAS: 115956-12-2

Dolasetron is an antinauseant and antiemetic agent indicated for the prevention of nausea and vomiting associated with moderately-emetogenic cancer chemotherapy and for the prevention of postoperative nausea and vomiting. Dolasetron is a highly specific and s…

Kategori:
Alimentary Tract and MetabolismAntidepressive AgentsAntiemetic Serotonin 5-HT3 Receptor Antagonists +21
Target Protein:
5-hydroxytryptamine receptor 3A
Waktu Paruh8.1 hours
Vol. Distribusi* 5.8 L/kg [adults]
Klirens* Apparent cl=9.4 m…
Genetik -
Dolastatin 10 DB12730
small molecule | CAS: 110417-88-4

Dolastatin 10 has been used in trials studying the treatment of Sarcoma, Leukemia, Lymphoma, Liver Cancer, and Kidney Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAntimitotic AgentsAntineoplastic Agents +4
Target Protein:
Tubulin beta-2A chain
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolcanatide DB13112
biotech | CAS: 1092457-65-2

Dolcanatide has been investigated in Exposure.

Kategori:
Amino Acids, Peptides, and ProteinsEnzyme ActivatorsGastrointestinal Agents +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Dolichovespula maculata venom protein is an extract of Dolichovespula maculata venom. Dolichovespula maculata venom protein is used in allergenic testing.

Kategori:
Allergenic ExtractsBee and Wasp VenomCell-mediated Immunity +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dolutegravir Approved DB08930
small molecule | CAS: 1051375-16-6

Dolutegravir is an HIV-1 integrase inhibitor that blocks the strand transfer step of the integration of the viral genome into the host cell (INSTI).[A7514] The effect of this drug has no homology in human host cells, which gives it excellent tolerability and …

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAnti-Retroviral Agents +20
Target Protein:
Gag-Pol polyproteinIntegrase
Gen Terkait:
UGT1A1 UGT1A1 UGT1A1
Waktu ParuhThe half-life of do…
Vol. DistribusiThe administration …
KlirensThe apparent cleara…
Genetik 3 Varian
Domagrozumab DB15083
biotech | CAS: 1629605-31-7

Domagrozumab is under investigation in clinical trial NCT01616277 (A Phase 1 Study To Evaluate The Safety And Tolerability Of PF-06252616 In Healthy Subjects).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domatinostat DB17521
small molecule | CAS: 910462-43-0

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesBenzene Derivatives +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domiodol DB13768
small molecule | CAS: 61869-07-6

Deskripsi belum tersedia.

Kategori:
Cough and Cold PreparationsDioxolesExpectorants
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domiphen Approved DB11594
small molecule | CAS: 13900-14-6

Domiphen bromide is a quaternary ammonium compound that is predominantly employed as a topically administered antiseptic agent.

Kategori:
Alimentary Tract and MetabolismAminesAmmonium Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2382896-04-8

Domofenogene zalfaparvovec, formerly known as BMN-307, is an investigational AAV5-phenylalanine hydroxylase (PAH) gene therapy developed by BioMarin Pharmaceutical.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domoic Acid DB02852
small molecule | CAS: 14277-97-5

Deskripsi belum tersedia.

Kategori:
Central Nervous System DepressantsNeuromuscular AgentsNeurotoxins +2
Target Protein:
Glutamate receptor ionotropic, kainate 1Glutamate receptor ionotropic, kainate 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Domperidone Approved DB01184
small molecule | CAS: 57808-66-9

A specific blocker of dopamine receptors. It speeds gastrointestinal peristalsis, causes prolactin release, and is used as antiemetic and tool in the study of dopaminergic mechanisms.

Kategori:
Alimentary Tract and MetabolismAntiemeticsAutonomic Agents +25
Target Protein:
D(3) dopamine receptorD(2) dopamine receptor
Waktu Paruh7 hours
Vol. Distribusi-
Klirens-
Genetik -
Domvanalimab DB18848
biotech | CAS: 2368219-35-4

Domvanalimab is under investigation in clinical trial NCT05502237 (Zimberelimab and Domvanalimab in Combination With Chemotherapy Versus Pembrolizumab With Chemotherapy in Patients With Untreated Metastatic Non-small Cell Lung Cancer).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Donanemab Approved DB16647
biotech | CAS: 1931944-80-7

Donanemab is a humanized immunoglobulin gamma 1 (IgG1) monoclonal antibody directed against insoluble N-truncated pyroglutamate amyloid beta (A?), [L50978] which is found in the brain amyloid plaques that contribute to the pathophysiology of Alzheimer's Disea…

Kategori:
Alzheimer Disease, drug therapyAmino Acids, Peptides, and ProteinsAmyloid Beta-directed Antibodies +11
Target Protein:
Beta amyloid plaque
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe central volume …
KlirensThe clearance is ab…
Genetik -
Donepezil Approved DB00843
small molecule | CAS: 120014-06-4

In 2016, the global burden of dementia was estimated to be 43.8 million, demonstrating a significant increase from a global prevalence of 20.2 million in 1990.[A182411] Donepezil, also known as Aricept, is a piperidine derivative acetylcholinesterase inhibito…

Kategori:
Anti-Dementia DrugsBCRP/ABCG2 SubstratesBradycardia-Causing Agents +20
Target Protein:
Acetylcholinesterase5-hydroxytryptamine receptor 2ACholinesterase +5
Gen Terkait:
CYP2D6
Waktu ParuhThe average elimina…
Vol. DistribusiThe volume of distr…
KlirensAccording to the FD…
Genetik 1 Varian
Donidalorsen DB18751
biotech | CAS: 2304692-48-4

Donidalorsen is under investigation in clinical trial NCT05392114 to assess the long-term safety and efficacy of donidalorsen in the prophylactic treatment of hereditary angioedema (HAE)

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesPolynucleotides
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
DONU DB12968
small molecule | CAS: 58484-17-6

Donu has been used in trials studying the treatment of Psychosis.

Kategori:
AmidesNitroso Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dopamine Approved DB00988
small molecule | CAS: 51-61-6

One of the catecholamine neurotransmitters in the brain. It is derived from tyrosine and is the precursor to norepinephrine and epinephrine. Dopamine is a major transmitter in the extrapyramidal system of the brain, and important in regulating movement. A fa…

Kategori:
Adrenergic and Dopaminergic AgentsAgents producing tachycardiaAgents that produce hypertension +26
Target Protein:
D(2) dopamine receptorD(1A) dopamine receptorD(1B) dopamine receptor +13
Waktu Paruh2 minutes
Vol. Distribusi-
Klirens-
Genetik -
Dopastatin DB16144
small molecule | CAS: 868562-36-1

Dopastatin is under investigation in clinical trial NCT04335357 (TBR-760 in Adult Patients With Non-functioning Pituitary Adenomas).

Kategori:
AminesAmino Acids, Peptides, and ProteinsBenzene Derivatives +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Dopexamine Approved DB12313
small molecule | CAS: 86197-47-9

Dopexamine has been used in trials studying the diagnostic and treatment of Free Flap, Oral Cancer, Hypotension, Septic Shock, and Head and Neck Cancer.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic and Dopaminergic Agents +18
Target Protein:
D(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Doramapimod DB03044
small molecule | CAS: 285983-48-4

Doramapimod is a P38 MAP kinase inhibitor.

Kategori:
AmidesBenzene DerivativesProtein Kinase Inhibitors
Target Protein:
Tyrosine-protein kinase HCKMitogen-activated protein kinase 14
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6351–6400 dari 16004
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