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6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
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6694 (100.0%)

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Halaman 127 / 134
Trypan blue free acid Approved DB09158
small molecule | CAS: 2538-83-2

Trypan blue is a diazo dye used in ophthalmic cataract surgery to stain the anterior capsule in the presence of a mature cataract. This is done to aid in visualization before creating the continuous curvilinear capsulorhexis.

Kategori:
ArylsulfonatesArylsulfonic AcidsAzo Compounds +12
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
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Trypsin Approved DB11237
small molecule | CAS: 9002-07-7

Trypsin is a serine protease that plays an essential role in protein hydrolysis and absorption in mammals. When converted from its zymogen trypsinogen, trypsin is available as an active peptide hydrolase (EC 3.4.21.4) form to cleave peptide chains, mainly at …

Kategori:
Blood and Blood Forming OrgansDermatologicalsEndopeptidases +8
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Tryptophan Approved DB00150
small molecule | CAS: 73-22-3

An essential amino acid that is necessary for normal growth in infants and for nitrogen balance in adults. It is a precursor of indole alkaloids in plants. It is a precursor of serotonin (hence its use as an antidepressant and sleep aid). It can be a precurso…

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +14
Target Protein:
Indoleamine 2,3-dioxygenase 1Tryptophan--tRNA ligase, cytoplasmicTryptophan--tRNA ligase +1
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TSHA-101 DB18280
biotech

Deskripsi belum tersedia.

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TSHA-102 DB18599
biotech

TSHA-102 is a recombinant serotype 9 adeno-associated virus encoding a codon-optimized human MECP2 gene.

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TSHA-105 DB18328
biotech

TSHA-105 is an adeno-associated virus serotype 9 (AAV9) vector with an engineered transgene encoding the human SLC13A5 protein.

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TST10088 DB05151
small molecule

TST10088 is a recombinant variant of a plant toxin belonging to the family of class II ribosome inactivating proteins. These molecules efficiently kill cells by activating preprogrammed death pathways known as apoptosis. TST10088 has been designed and enginee…

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TT-232 DB12088
small molecule | CAS: 147159-51-1

Tln 232 is under investigation in clinical trial NCT00422786 (Phase II Study of CAP-232 in Patients With Refractory Metastatic Renal Cell Carcinoma).

Kategori:
Amino Acids, Peptides, and ProteinsHormonesHormones, Hormone Substitutes, and Hormone Antagonists +8
Target Protein:
Pyruvate kinase PKM
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TTP889 DB05131
small molecule

TTP889, an orally bioavailable selective inhibitor of the intrinsic coagulation pathway, is being developed as an anticoagulant for the treatment of thromboembolic disorders. TTP889 is the only known selective small molecule inhibitor of Factor IX, a key enzy…

Target Protein:
Coagulation factor IX
Waktu Paruh20 hours
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Tubercidin DB03172
small molecule | CAS: 69-33-0

An antibiotic purine ribonucleoside that readily substitutes for adenosine in the biological system, but its incorporation into DNA and RNA has an inhibitory effect on the metabolism of these nucleic acids.

Kategori:
Antibiotics, AntineoplasticAntimetabolitesAntineoplastic Agents +8
Target Protein:
Purine nucleoside phosphorylase DeoD-type
Waktu Paruh-
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biotech | CAS: 92129-86-7

Tuberculin Purified Protein Derivative (PPD) is a sterile aqueous solution of a purified protein fraction for intradermal administration as an aid in the diagnosis of tuberculosis. The diagnostic test is commonly referred to as the Mantoux test which serves t…

Kategori:
Amino Acids, Peptides, and ProteinsAntigensAntigens, Bacterial +12
Target Protein:
Toll-like receptor 2
Waktu Paruh-
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Tucatinib Approved DB11652
small molecule | CAS: 937263-43-9

Tucatinib is a kinase inhibitor drug used with [trastuzumab] and [capecitabine] in the treatment of unresectable or metastatic HER-2 positive breast cancer. It was developed by Seattle Genetics and approved by the FDA on April 17, 2020.[L12951] Tucatinib is a…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +18
Target Protein:
Receptor tyrosine-protein kinase erbB-2Receptor tyrosine-protein kinase erbB-3
Waktu ParuhA pharmacokinetic s…
Vol. DistribusiThe volume of distr…
KlirensThe apparent cleara…
Genetik -
Tucidinostat DB06334
small molecule | CAS: 1616493-44-7

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAmidesAmines +7
Target Protein:
Histone deacetylase 1
Waktu Paruh-
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Tulathromycin A DB11474
small molecule | CAS: 217500-96-4

Tulathromycin is a macrolide antibiotic used to treat bovine respiratory disease in cattle and swine respiratory disease in pigs. It is marketed by Pfizer Inc. under the tradename Draxxin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsCarbohydrates +4
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Tuna Approved DB10574
biotech

Tuna allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
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Tunicamycin DB13172
small molecule | CAS: 11089-65-9

Tunicamycin is a mixture of homologous nucleoside antibiotics that inhibits the UDP-HexNAc: polyprenol-P HexNAc-1-P family of enzymes. One member of this family is the enzyme GlcNAc phosphotransferase (GPT), which catalyzes the transfer of N-acetylglucosamine…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsNucleic Acids, Nucleotides, and Nucleosides +3
Waktu Paruh-
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Tuparstobart DB19118
biotech | CAS: 2649466-03-3

Tuparstobart is under investigation in clinical trial NCT05287113 (Study of Retinfanlimab in Combination With INCAGN02385 and INCAGN02390 as First-line Treatment in Participants With Pd-l1-positive (CPS ? 1) Recurrent/metastatic Squamous Cell Carcinoma of the…

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Turoctocog alfa Approved DB09109
biotech | CAS: 1192451-26-5

Turoctocog alfa is a recombinant factor VIII (rFVIII) with a truncated B-domain made from the sequence coding for 10 amino acids from the N-terminus and 11 amino acids from the C-terminus of the naturally occurring B-domain. Turoctocog alfa is produced in Chi…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin
Waktu ParuhIn pre-clinical stu…
Vol. DistribusiIn pre-clinical stu…
KlirensIn pre-clinical stu…
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Turoctocog alfa pegol Approved DB14738
biotech | CAS: 1309086-46-1

Turoctocog alfa pegol is a pegylated version of [turoctocog alfa]. Novo Nordisk's brand name Esperoct (turoctocog alfa pegol, N8-GP) was approved by the US FDA on February 19, 2019. Fundamentally, the N8-GP moiety is identical to [turoctocog alfa], a recom…

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsBlood Coagulation Factors +5
Target Protein:
Coagulation factor IXCoagulation factor XProthrombin +1
Waktu ParuhThe mean plasma hal…
Vol. DistribusiThe mean volume of …
KlirensThe mean clearance …
Genetik -
biotech | CAS: 2254086-60-5

Tusamitamab ravtansine is an antibody-drug conjugate that targets carcinoembryonic antigen-related cell adhesion molecule-5 (CEACAM5).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsGlobulins +4
Waktu Paruh-
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Ty800 DB04989
biotech

Ty800 is a vaccine designed to offer rapid, oral, single-dose protection against <i>Salmonella typhi</i>, the cause of typhoid fever. The Ty800 vaccine was developed using genetic techniques to delete specific genes known to be essential to the virulence of <…

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Tylosin DB11475
small molecule | CAS: 1401-69-0

Tylosin is a bacteriostatic macrolide antibiotic and feed additive used in veterinary medicine. It has a broad spectrum of activity against Gram-positive organisms and a limited range of Gram-negative organisms. Tylosin is produced as a fermentation product o…

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsLactones +1
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Typhoid vaccine Approved DB14022
biotech

Deskripsi belum tersedia.

Kategori:
Bacterial VaccinesBiological ProductsComplex Mixtures +3
Waktu Paruh-
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Typhoid Vaccine Live Approved DB11050
biotech

Salmonella typhi Ty21a live antigen is a live attenuated vaccine for oral administration only. It contains the attenuated strain *Salmonella typhi* Ty21a. The vaccine prevents the development of typhoid fever, an acute, febrile enteric disease caused by *Salm…

Kategori:
Actively Acquired ImmunityInactivated Salmonella Typhi VaccineLive Attenuated Salmonella Typhi Vaccine +2
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biotech

Typhoid Vi polysaccharide vaccine is a vaccine that is administered intramuscularly. It is an active immunization for the prevention of typhoid fever caused by S typhi and is approved for use in persons two years of age or older. The vaccine contains the puri…

Kategori:
Actively Acquired ImmunityAntiinfectives for Systemic UseBacterial Vaccines +3
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Tyramine DB08841
small molecule | CAS: 51-67-2

Tyramine (4-hydroxyphenethylamine; para-tyramine, mydrial or uteramin) is a naturally occurring monoamine compound and trace amine derived from the amino acid tyrosine. Tyramine acts by inducing the release of catecholamine. An important characteristic of thi…

Kategori:
Adrenergic AgentsAgents producing tachycardiaAgents that produce hypertension +9
Target Protein:
Trace amine-associated receptor 1
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Tyropanoic acid Approved DB09340
small molecule | CAS: 27293-82-9

Tyropanoic acid is a radiocontrast agent used in cholecystography, the X-ray diagnosis of gallstones under the trade names include Bilopaque, Lumopaque, Tyropaque, and Bilopac. The molecule contains three heavy iodine atoms which obstruct X-rays in the same w…

Kategori:
Benzene DerivativesCompounds used in a research, industrial, or household settingContrast Media +6
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Tyroserleutide DB17300
small molecule | CAS: 138168-48-6

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsPeptides
Waktu Paruh-
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Tyrosinase DB16626
biotech | CAS: 9002-10-2

Tyrosinase is a multi-copper-containing multifunctional metalloenzyme with 4 possible oxidation states.[A231829, A231834, A231839] It is responsible for producing melanin pigment across the phylogenetic spectrum.[A231829, A231834, A231839] Within mammals, …

Kategori:
Catechol OxidaseEnzymesEnzymes and Coenzymes +6
Waktu Paruh-
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Tyrosine Approved DB00135
small molecule | CAS: 60-18-4

Tyrosine is a non-essential amino acid. In animals it is synthesized from [phenylalanine]. It is also the precursor of [epinephrine], thyroid hormones, and melanin.

Kategori:
Amino AcidsAmino Acids, AromaticAmino Acids, Cyclic +4
Target Protein:
Tyrosine 3-monooxygenaseTyrosine--tRNA ligase, mitochondrialTyrosine--tRNA ligase, cytoplasmic +1
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Tyrothricin Approved DB13503
small molecule | CAS: 1404-88-2

Tyrothricin is an antibiotic peptide complex produced and extracted from the aerobic Gram-positive bacillus Brevibacillus parabrevis [L4019, L4021, A32851] which was previously categorized as Bacillus brevis and Bacillus aneurinolyticus [A36353]. This complex…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +9
Target Protein:
Phospholipid membraneAcetylcholinesteraseBeta-galactosidase
Waktu Paruh-
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Tyrphostin B48 DB16774
small molecule | CAS: 133550-35-3

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
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TZP-102 DB16129
small molecule | CAS: 1008993-65-4

TZP-102 is under investigation in clinical trial NCT01452815 (Affects of Once-daily Oral Administration of TZP-102 on the Treatment of Symptoms Associated With Diabetic Gastroparesis).

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UB-612 DB16444
biotech

The UB-612 COVID-19 vaccine was developed by United Biomedical Inc Asia in Taipei as the first COVID-19 “multi-tope” protein-peptide vaccine made up of eight rationally designed components[L30653]. The vaccine incorporates a strong S1-RBD component linked to …

Kategori:
Biological ProductsComplex MixturesVaccines +1
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Ubamatamab DB18875
biotech | CAS: 2305629-50-7

Ubamatamab is under investigation in clinical trial NCT03564340 (Study of REGN4018 Administered Alone or in Combination With Cemiplimab in Adult Patients With Recurrent Ovarian Cancer or Other Recurrent Mucin-16 Expressing (MUC16+) Cancers).

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Ublituximab Approved DB11850
biotech | CAS: 1174014-05-1

CD20, an antigen expressed by various B and T cells, is an attractive therapeutic target in various cancers and autoimmune conditions.[A244195, A244200, A244205] Monoclonal antibodies for B cell depletion rely on their binding affinity and ability to clear bo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
B-lymphocyte antigen CD20
Waktu ParuhThe estimated mean …
Vol. DistribusiThe estimated centr…
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Ubrogepant Approved DB15328
small molecule | CAS: 1374248-77-7

Ubrogepant is indicated for the acute treatment of migraine headaches with or without aura in adults.[L10926] It was approved by the FDA on December 23, 2019, and is the first oral calcitonin gene-related peptide (CGRP) receptor antagonist approved for the ac…

Kategori:
AnalgesicsAntimigraine PreparationsBCRP/ABCG2 Substrates +23
Target Protein:
Calcitonin gene-related peptide type 1 receptor
Waktu ParuhUbrogepant has an e…
Vol. DistribusiThe apparent centra…
KlirensThe apparent oral c…
Genetik -
UC-781 DB05871
small molecule | CAS: 178870-32-1

UC-781 is a thiocarboxanilide non-nucleoside reverse transcriptase inhibitor (NNRTI). It is a topical microbicide targeted against the AIDS virus.

Kategori:
AmidesAnti-Infective AgentsAnti-Retroviral Agents +2
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
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UCART22 DB17466
biotech

UCART22 are allogeneic CD22-specific universal CAR-expressing T lymphocytes.

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UCB7362 DB17096
small molecule

UCB7362 is an orally active plasmepsin X (PMX) inhibitor currently investigated for the treatment of malaria.[A254222] Plasmepsins are aspartyl proteases produced by the malaria parasite _Plasmodium falciparum_, and PMX is considered to be essential for paras…

Target Protein:
Plasmepsin XPlasmepsin X
Waktu Paruh-
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Udifitimod DB19053
small molecule | CAS: 1883345-06-9

Udifitimod is under investigation in clinical trial NCT05014438 (A Study of BMS-986166 or Branebrutinib for the Treatment of Participants With Atopic Dermatitis).

Kategori:
Naphthalenes
Waktu Paruh-
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Udonitrectag DB18013
small molecule | CAS: 1458063-04-1

Deskripsi belum tersedia.

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small molecule | CAS: 2616-64-0

A nucleoside diphosphate sugar which serves as a source of glucuronic acid for polysaccharide biosynthesis. It may also be epimerized to UDP iduronic acid, which donates iduronic acid to polysaccharides. In animals, UDP glucuronic acid is used for formation o…

Kategori:
CarbohydratesGlycosidesNucleic Acids, Nucleotides, and Nucleosides +8
Target Protein:
UDP-glucose 4-epimeraseGalactosylgalactosylxylosylprotein 3-beta-glucuronosyltransferase 3UDP-glucose 6-dehydrogenase
Waktu Paruh-
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small molecule | CAS: 3616-06-6

The decarboxylation product of UDPglucuronic acid, which is used for formation of the xylosides of seryl hydroxyl groups in mucoprotein synthesis. Also forms plant xylans.

Target Protein:
UDP-glucose 6-dehydrogenase
Waktu Paruh-
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UK-396,082 DB12099
small molecule | CAS: 400044-47-5

UK-396,082 has been used in trials studying the basic science of Safety, Phase 1, Toleration, Multiple Dose, and Pharmacokinetic.

Kategori:
Amino Acids, Peptides, and Proteins
Target Protein:
Carboxypeptidase B2
Waktu Paruh-
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Ularitide DB05034
small molecule | CAS: 118812-69-4

Ularitide is a synthetic form of urodilatin, a naturally occurring human natriuretic peptide that is involved in regulating blood pressure and the excretion of water and sodium from the kidneys. Urodilatin is produced in the kidney and excreted into the urine…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Asthmatic AgentsAutonomic Agents +10
Target Protein:
Atrial natriuretic peptide receptor 1
Waktu Paruh-
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Ulenistamab DB18291
biotech | CAS: 2415259-90-2

Deskripsi belum tersedia.

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Ulipristal Approved DB08867
small molecule | CAS: 159811-51-5

Ulipristal is a selective progesterone receptor modulator used for the purposes of emergency contraception (Ella) and for the treatment of uterine fibroids (Fibristal). It is a derivative of 19-norprogesterone and has both antagonistic and partial agonist ac…

Kategori:
Adrenal Cortex HormonesContraceptive Agents, FemaleContraceptive Agents, Hormonal +16
Target Protein:
Progesterone receptorGlucocorticoid receptorAndrogen receptor
Waktu ParuhMean elimination ha…
Vol. Distribusi-
KlirensMean oral clearance…
Genetik -
Ulodesine DB12353
small molecule | CAS: 548486-59-5

Ulodesine has been used in trials studying the treatment of Gout, Arthritis, Hyperuricemia, and Joint Disease.

Kategori:
CarbohydratesIminesImino Sugars +3
Target Protein:
Purine nucleoside phosphorylase
Waktu Paruh-
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Genetik -
biotech

The use of umbilical cord blood (UCB) for therapies is advantageous because of its ease of access, non-invasive collection procedures, and more plasticity for multi-differentiation. UCB contains a large source of hematopoietic stem cells (HSCs) that are capab…

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Menampilkan 6301–6350 dari 6694
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