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13591

Total database: 17430
Struktur (SMILES)
10177 (74.9%)
Target
7625 (56.1%)
Genomik
104 (0.8%)
Referensi
13591 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

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Hasil Pencarian (13591)

Halaman 127 / 272
FP-1096 DB05310
small molecule

FP1096 reduced the painful symptoms of endometriosis in trial subjects with very minimal side effect.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR-234938 DB03220
small molecule | CAS: 256461-79-7

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR230513 DB03572
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR236913 DB02830
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FR239087 DB03370
small molecule

Deskripsi belum tersedia.

Target Protein:
Adenosine deaminase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fradafiban DB06472
small molecule | CAS: 148396-36-5

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesPlatelet Glycoprotein GPIIb-IIIa Complex, antagonists & inhibitors
Target Protein:
Integrin alpha-IIbIntegrin beta-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fraxinus americana pollen Approved DB10348
biotech

Fraxinus americana pollen is the pollen of the Fraxinus americana plant. Fraxinus americana pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fraxinus latifolia pollen Approved DB10723
biotech

Fraxinus latifolia pollen is the pollen of the Fraxinus latifolia plant. Fraxinus latifolia pollen is mainly used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fremanezumab Approved DB14041
biotech | CAS: 1655501-53-3

Fremanezumab is a humanized monoclonal antibody targeted against human calcitonin gene-related peptide (CGRP) for the prevention of migraine headaches.[L11749] It was developed by Teva Pharmaceuticals USA and approved by the FDA in September 2018.[L11779] Alo…

Kategori:
Amino Acids, Peptides, and ProteinsAnalgesicsAntibodies +12
Target Protein:
Calcitonin gene-related peptide 1Calcitonin gene-related peptide 2
Waktu ParuhThe mean half-life …
Vol. DistribusiFremanezumab has an…
KlirensThe apparent cleara…
Genetik -
Freneslerbart DB19080
biotech | CAS: 2453195-94-1

Freneslerbart is under investigation in clinical trial NCT04981717 (A Study to Examine the Efficacy and Safety of Anti-fel D 1 Antibodies Injections in Cat-allergic Adolescent and Adult Patients With Allergic Rhinitis Who Live With a Cat).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Freselestat DB03925
small molecule | CAS: 208848-19-5

Deskripsi belum tersedia.

Kategori:
Leukocyte Elastase, antagonists & inhibitorsOxazolesPyrimidines
Target Protein:
Chymotrypsin-like elastase family member 1Neutrophil elastase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fresolimumab DB12396
biotech | CAS: 948564-73-6

Fresolimumab has been used in trials studying the treatment of Primary Brain Tumors, Metastatic Breast Cancer, Diffuse Systemic Sclerosis, Pleural Malignant Mesothelioma, and Primary Focal Segmental Glomerulosclerosis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frexalimab DB18926
biotech | CAS: 2515463-86-0

Frexalimab is under investigation in clinical trial NCT06141486 (Efficacy and Safety Study of Frexalimab (SAR441344) in Adults With Nonrelapsing Secondary Progressive Multiple Sclerosis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Friulimicin B DB06087
small molecule | CAS: 239802-15-4

Friulimicin B is a naturally occurring antibiotic produced by a micro-organism, *Actinoplanes friuliensis*. It shows strong cidal activity against a number of Gram-positive pathogens which commonly cause serious infections in hospital patients and which are b…

Kategori:
Amino Acids, Peptides, and Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Froniglutide DB16178
biotech | CAS: 1417579-81-7

Glymera is under investigation in clinical trial NCT01658501 (Phase 2b Multicenter, Randomized, Double-blind, Placebo- and Active-controlled, Parallel-group Study to Assess the PD Response and Safety of Three Dose Levels of (PB1023) Injection Following 20 Wee…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frovocimab DB15089
biotech | CAS: 1643672-70-1

Frovocimab is under investigation in clinical trial NCT01671085 (A Study of LY3015014 in Healthy Participants With High Cholesterol).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fructose Approved DB04173
small molecule

Deskripsi belum tersedia.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDiet, Food, and Nutrition +12
Target Protein:
Maltoporin
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 643-13-0

Deskripsi belum tersedia.

Kategori:
CarbohydratesHexosephosphatesSugar Phosphates
Target Protein:
Fructose-1,6-bisphosphatase 1Fructose-1,6-bisphosphatase isozyme 26-phosphofructo-2-kinase/fructose-2,6-bisphosphatase 1 +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Frunexian DB18771
small molecule | CAS: 1803270-60-1

Deskripsi belum tersedia.

Kategori:
AmidesAminesPyridines
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fruquintinib Approved DB11679
small molecule | CAS: 1194506-26-7

Fruquintinib is a novel small-molecule anti-VEGFR that targets VEGFR-1,-2, and -3 to inhibit angiogenesis. Tumor angiogenesis is one of the most critical biological processes for increasing oxygen and nutrient supply to cancer cells, and the VEGF/VEGFR pathwa…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsCytochrome P-450 CYP2C19 Substrates +10
Target Protein:
Vascular endothelial growth factor receptor 1Vascular endothelial growth factor receptor 2Vascular endothelial growth factor receptor 3
Waktu ParuhThe fruquintinib's …
Vol. DistribusiThe mean (SD) appar…
KlirensThe apparent cleara…
Genetik -
FT-1101 DB17553
small molecule | CAS: 1776060-36-6

FT-1101 is a novel Bromodomain and Extra-Terminal motif (BET) inhibitor.[A257301] FT-1101 is under investigation in clinical trial NCT02543879 (Study of a Novel BET Inhibitor FT-1101 in Patients With Relapsed or Refractory Hematologic Malignancies).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FT516 DB15732
biotech

FT516 is an investigational and engineered off-the-shelf natural killer (NK) cell therapy originating from induced pluripotent stem cells (iPSC). This compound expresses a high-affinity 158V, CD16 (hnCD16) Fc receptor that has an enhanced binding ability to t…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucitol DB03815
small molecule | CAS: 13074-06-1

Deskripsi belum tersedia.

Kategori:
AlcoholsCarbohydrates
Target Protein:
L-fucose isomerase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucose DB15236
small molecule | CAS: 2438-80-4

Fucose is under investigation in clinical trial NCT03354533 (Study of ORL-1F (L-fucose) in Patients With Leukocyte Adhesion Deficiency Type II).

Kategori:
CarbohydratesDeoxy Sugars
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fucoxanthin DB15462
small molecule | CAS: 3351-86-8

Fucoxanthin is under investigation in clinical trial NCT03613740 (Effect of Fucoxanthin on the Components of the Metabolic Syndrome, Insulin Sensitivity and Insulin Secretion). Fucoxanthin isis a marine carotenoid mainly found in brown algae, giving them a br…

Kategori:
AlkenesBiological FactorsCarotenoids +7
Target Protein:
NF-kappa-B inhibitor alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulacimstat DB15085
small molecule | CAS: 1488354-15-9

Fulacimstat is under investigation in clinical trial NCT02452515 (A Single-blind Pilot Study to Investigate Safety and Tolerability of the Chymase Inhibitor BAY1142524 in Clinically Stable Patients With Left-ventricular Dysfunction).

Kategori:
Enzyme Inhibitors
Target Protein:
Chymase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fulvestrant Approved DB00947
small molecule | CAS: 129453-61-8

Fulvestrant is a drug treatment of hormone receptor (HR)-positive metastatic breast cancer in post-menopausal women with disease progression following anti-estrogen therapy. It is an estrogen receptor antagonist with no agonist effects, which works both by do…

Kategori:
Anti-EstrogensAntineoplastic AgentsAntineoplastic Agents, Hormonal +20
Target Protein:
Estrogen receptor
Waktu Paruh40 days
Vol. Distribusi* 3 to 5 L/kg
Klirens-
Genetik -
Fumagillin DB02640
small molecule | CAS: 23110-15-8

Deskripsi belum tersedia.

Kategori:
Angiogenesis InhibitorsAngiogenesis Modulating AgentsAnti-Infective Agents +10
Target Protein:
Methionine aminopeptidase 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Funapide DB11769
small molecule | CAS: 1259933-16-8

Funapide has been used in trials studying the treatment of Pharmacokinetics, Postherpetic Neuralgia, and Osteoarthritis of the Knee.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Sodium channel protein type 9 subunit alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaltadone DB16567
small molecule | CAS: 139-91-3

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryFurans +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprevir DB12785
small molecule | CAS: 1435923-88-8

Furaprevir is under investigation in clinical trial NCT01523990 (A Study to Evaluate the Safety, Tolerability, and PK in Healthy Volunteers and HCV Genotype 1 Infected Patients).

Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furaprofen DB06499
small molecule | CAS: 67700-30-5

Deskripsi belum tersedia.

Kategori:
Heterocyclic Compounds, Fused-Ring
Target Protein:
Genome polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazabol DB01514
small molecule | CAS: 1239-29-8

Deskripsi belum tersedia.

Kategori:
AndrostanesFused-Ring CompoundsSteroids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazidin DB13475
small molecule | CAS: 1672-88-4

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAnti-Infective Agents, UrinaryAntibacterials for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furazolidone DB00614
small molecule | CAS: 67-45-8

A nitrofuran derivative with antiprotozoal and antibacterial activity. Furazolidone binds bacterial DNA which leads to the gradual inhibition of monoamine oxidase. (From Martindale, The Extra Pharmacopoeia, 30th ed, p514)

Kategori:
Agents that produce hypertensionAgents that reduce seizure thresholdAnti-Infective Agents +20
Target Protein:
DNA
Waktu Paruh10 minutes
Vol. Distribusi-
Klirens-
Genetik -
Furethidine DB01464
small molecule | CAS: 2385-81-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furosemide Approved DB00695
small molecule | CAS: 54-31-9

Furosemide is a potent loop diuretic that acts on the kidneys to ultimately increase water loss from the body. It is an anthranilic acid derivative.[L7958] Furosemide is used for edema secondary to various clinical conditions, such as congestive heart failure…

Kategori:
Acids, CarbocyclicAmidesAmines +30
Target Protein:
Solute carrier family 12 member 1Carbonic anhydrase 2G-protein coupled receptor 35
Waktu ParuhThe half-life from …
Vol. DistribusiThe volume of distr…
KlirensFollowing intraveno…
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fursultiamine Approved DB08966
small molecule | CAS: 804-30-8

Compound used for therapy of thiamine deficiency. It has also been suggested for several non-deficiency disorders but has not yet proven useful. Fursultiamine is a vitamin B1 derivative.

Kategori:
MicronutrientsPyrimidinesSulfur Compounds +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Furvina DB16547
small molecule | CAS: 189935-72-6

Furvina (G1) is an antimicrobial agent active against Gram-positive and Gram-negative bacteria, yeasts, and filamentous fungi. Furvina is marketed in Cuba as Dermofural®, an ointment containing G1 as the only active principle ingredient. It is used to treat d…

Kategori:
AlkenesAnti-Infective AgentsHydrocarbons, Acyclic
Target Protein:
30S ribosomal protein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusafungine Approved DB08965
small molecule | CAS: 1393-87-9

Fusafungine is an antibiotic from Fusarium lateririum, and is used for the treatment of respiratory infections.

Kategori:
Amino Acids, Peptides, and ProteinsAnti-Bacterial AgentsAnti-Infective Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusarium graminearum Approved DB13907
biotech

Fusarium graminearum allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech

Fusarium oxysporum vasinfectum is a fungus which can provoke allergic reactions. Fusarium oxysporum vasinfectum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusicoccin DB01780
small molecule | CAS: 20108-30-9

Deskripsi belum tersedia.

Kategori:
CarbohydratesMycotoxins
Target Protein:
14-3-3 protein epsilon
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fusidic acid Approved DB02703
small molecule | CAS: 6990-06-3

An antibiotic isolated from the fermentation broth of Fusidium coccineum. (From Merck Index, 11th ed) It acts by inhibiting translocation during protein synthesis. It is often used topically in creams and eyedrops but is available in systemic formulations inc…

Kategori:
Agents Causing Muscle ToxicityAnti-Bacterial AgentsAnti-Infective Agents +35
Target Protein:
Elongation factor GChloramphenicol acetyltransferaseChloramphenicol acetyltransferase 3
Waktu ParuhApproximately 5 to …
Vol. Distribusi-
Klirens-
Genetik -
Futibatinib Approved DB15149
small molecule | CAS: 1448169-71-8

Futibatinib is an inhibitor of Fibroblast Growth Factor receptor (FGFR), which comprises a group of receptor tyrosine kinases that play a key role in cell proliferation, differentiation, migration, and survival. FGFR was investigated in oncology as a therapeu…

Kategori:
Antineoplastic AgentsAntineoplastic and Immunomodulating AgentsBCRP/ABCG2 Substrates +10
Target Protein:
Fibroblast growth factor receptor 1Fibroblast growth factor receptor 2Fibroblast growth factor receptor 3 +1
Waktu ParuhThe mean (CV%) elim…
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
Futuximab DB15262
biotech | CAS: 1310460-85-5

Futuximab is under investigation in clinical trial NCT01955473 (Japanese Phase 1 Trial of Sym004 in Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fx-1006A DB05352
small molecule

Fx-1006A is a small molecule compound with the potential to treat genetic disorders, such as familial amyloid cardiomyopathy (FAC) and familial amyloid polyneuropathy (FAP).

Kategori:
Heterocyclic Compounds, Fused-Ring
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G305 DB17292
biotech

G305 is a [recombinant NY-ESO-1 protein] plus glucopyranosyl lipid A (GLA) in a stable emulsion (SE). G305 is an active component of CMB305 along with [LV305].[L47346]

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
G4460 DB06359
biotech

Deskripsi belum tersedia.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleotidesOligonucleotides +1
Target Protein:
Transcriptional activator Myb
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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