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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 127 / 282
Ferric maltol Approved DB15598
small molecule | CAS: 33725-54-1

Ferric maltol is an iron(III) atom complexed with 3 maltol molecules to increase the bioavailability compared to iron(II), without depositing it in the duodenum as insoluble ferric hydroxide and phosphate.[A189288] Ferric maltol has been described in literatu…

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansHematinics +8
Target Protein:
Integrin beta-3Natural resistance-associated macrophage protein 2
Waktu ParuhMaltol has a half l…
Vol. DistribusiData regarding the …
KlirensData regarding the …
Genetik -
Ferric oxide DB11576
small molecule | CAS: 1309-37-1

Iron(III) oxide or ferric oxide is the inorganic compound with the formula Fe2O3. It is one of the three main oxides of iron, the other two being iron(II) oxide (FeO) the rarer form, and iron(II,III) oxide (Fe3O4) which naturally as magnetite.

Kategori:
Contrast MediaIron CompoundsMagnetic Resonance Imaging Contrast Media +1
Waktu Paruh-
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Genetik -
small molecule | CAS: 20344-49-4

An antiferromagnetic material; constitutes the core of natural ferritin.

Kategori:
Iron CompoundsOrganometallic CompoundsPhosphate Binder +1
Waktu Paruh-
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Genetik -
Ferric pyrophosphate citrate Approved DB13995
small molecule | CAS: 1802359-96-1

Ferric pyrophosphate citrate is a soluble iron replacement product. Free iron presents several side effects as it can catalyze free radical formation and lipid peroxidation as well as the presence of interactions of iron in plasma. The ferric ion is strongly …

Kategori:
EnzymesEnzymes and CoenzymesHydrolases +3
Target Protein:
Ferritin light chainFerritin heavy chainHemoglobin subunit alpha +1
Waktu ParuhThe half-life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe mean clearance …
Genetik -
small molecule | CAS: 52031-09-1

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Preparations +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric subsulfate Approved DB13885
small molecule | CAS: 1310-45-8

Ferric subsulfate is a stypic or hemostatic agent that causes agglutination of surface proteins resulting in local hemostasis. It has the chemical formula Fe4(OH)2(SO4)5. It is used after superficial skin biopsies.

Kategori:
AnionsCoagulantsElectrolytes +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric sulfate Approved DB11171
small molecule | CAS: 10028-22-5

Ferric sulfate has the molecular formula of Fe2SO4, and it is a dark brown or yellow chemical agent with acidic properties. It is produced by the reaction of sulfuric acid and an oxidizing agent. It is used in different fields such as dermatology, dentistry a…

Kategori:
HematinicsIron Compounds
Waktu ParuhPharmacokinetic stu…
Vol. DistribusiPharmacokinetic stu…
KlirensPharmacokinetic stu…
Genetik -
biotech

Ferrimannitol-ovalbumin (FMOA) is an adduct between ovalbumin and the complex Fe(III)-mannitol.

Waktu Paruh-
Vol. Distribusi-
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Ferroheme DB18267
small molecule | CAS: 14875-96-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsCytochrome P-450 CYP3A InhibitorsCytochrome P-450 CYP3A4 Inhibitors +7
Target Protein:
Heme oxygenase 1Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2 +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferroheme C DB03317
small molecule | CAS: 26598-29-8

Deskripsi belum tersedia.

Kategori:
Biological FactorsHeterocyclic Compounds, Fused-RingMetalloporphyrins +2
Target Protein:
Nitrite reductaseHigh-molecular-weight cytochrome cCytochrome c'' +20
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous ascorbate Approved DB14490
small molecule | CAS: 24808-52-4

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicAntianemic PreparationsAntioxidants +15
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 75802-64-1

The use of ferrous acetate over ferrous sulfate is currently undergoing an investigation by a clinical trial [L5464]. It is also used for dying of fabric or leather and as a wood preservative.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Bivalent, Oral Preparations +1
Waktu Paruh-
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Ferrous bisglycinate Approved DB11210
small molecule | CAS: 20150-34-9

Ferrous bisglycinate is a chelate that is used as a source of dietary iron. Forming a ring structure when reacting with glycine, ferrous bisglycinate acts as both a chelate and a nutritionally functional [A27250]. It is found in foods for food enrichment or i…

Kategori:
Amino AcidsAmino Acids, Peptides, and ProteinsIron Compounds
Waktu Paruh-
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Genetik -
Ferrous cation DB14510
small molecule | CAS: 15438-31-0

Deskripsi belum tersedia.

Waktu Paruh-
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Ferrous cysteine glycinate Approved DB11197
small molecule

Deskripsi belum tersedia.

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Ferrous fumarate Approved DB14491
small molecule | CAS: 141-01-5

Used in treatment of iron deficiency anemia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansDiet, Food, and Nutrition +9
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous gluconate Approved DB14488
small molecule | CAS: 299-29-6

Deskripsi belum tersedia.

Kategori:
Anemia, Iron-DeficiencyAntianemia DrugsAntianemic Preparations +8
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous glycine sulfate Approved DB14501
small molecule | CAS: 14729-84-1

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Bivalent, Oral Preparations +1
Target Protein:
Transferrin receptor protein 1Egl nine homolog 1Histone deacetylase 8 +10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferrous sulfate anhydrous Approved DB13257
small molecule | CAS: 7720-78-7

Iron deficiency anemia is a large public health concern worldwide, especially in young children, infants, and women of childbearing age.[A190804] This type of anemia occurs when iron intake, iron stores, and iron loss do not adequately support the formation o…

Kategori:
Anemia, Iron-DeficiencyDelayed-Action PreparationsHematinics +6
Target Protein:
Hemoglobin subunit alphaTransferrin receptor
Waktu ParuhThe half-life of or…
Vol. DistribusiAbout 60% of iron i…
Klirens-
Genetik -
small molecule | CAS: 2944-65-2

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Bivalent, Oral Preparations +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferulic acid DB07767
small molecule | CAS: 1135-24-6

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAnalgesicsAnalgesics, Non-Narcotic +17
Target Protein:
Carbonic anhydrase 12Carbonic anhydrase 2Carbonic anhydrase 14 +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule

Deskripsi belum tersedia.

Target Protein:
Catechol O-methyltransferase domain-containing protein 1
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Ferumoxytol Approved DB06215
small molecule | CAS: 722492-56-0

Ferumoxytol is an intravenously administered iron preparation indicated in the EU and the US for the treatment of iron deficiency anemia in adult patients with chronic kidney disease (CKD) [A32478]. It is comprised of superparamagnetic iron oxide nanoparti…

Kategori:
Compounds used in a research, industrial, or household settingFerric CompoundsFerrous Compounds +11
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiThe population mean…
KlirensSince there is no r…
Genetik -
Fesoterodine Approved DB06702
small molecule | CAS: 286930-02-7

Fesoterodine is an antimuscarinic prodrug for the treatment of overactive bladder syndrome.

Kategori:
Agents producing tachycardiaAnticholinergic AgentsBenzene Derivatives +14
Target Protein:
Muscarinic acetylcholine receptor M3Muscarinic acetylcholine receptor M4Muscarinic acetylcholine receptor M1 +2
Waktu Paruh7-8 hours for the a…
Vol. DistribusiIV, 5-HMT: 169 L
Klirens5-HMT, healthy subj…
Genetik -
FET F-18 DB15405
small molecule | CAS: 178433-03-9

FET F-18 is under investigation in clinical trial NCT01756352 (FET-PET for Evaluation of Response of Recurrent GBM to Avastin).

Kategori:
Diagnostic RadiopharmaceuticalsTumour Detection
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fevipiprant DB12011
small molecule | CAS: 872365-14-5

Fevipiprant has been used in trials studying the treatment of Asthma, Atopic Dermatitis, and Allergic Rhinitis.

Kategori:
Heterocyclic Compounds, Fused-RingIndoles
Target Protein:
Prostaglandin D2 receptor 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fexaramine DB02545
small molecule | CAS: 574013-66-4

Deskripsi belum tersedia.

Target Protein:
Bile acid receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fexinidazole Approved DB12265
small molecule | CAS: 59729-37-2

Human African trypanosomiasis (HAT, also colloquially referred to as sleeping sickness), caused by _T. brucei gambiense_ and _T. brucei rhodesiense_, remains a moderate risk (>1/10,000 inhabitants per year in endemic areas) despite focussed control efforts. T…

Kategori:
Agents Against Leishmaniasis and TrypanosomiasisAntiparasitic Products, Insecticides and RepellentsAntiprotozoals +43
Waktu ParuhFexinidazole, M1, a…
Vol. DistribusiFexinidazole has an…
KlirensFexinidazole has a …
Genetik -
Fexofenadine Approved DB00950
small molecule | CAS: 83799-24-0

Fexofenadine is an over-the-counter second-generation antihistamine used in the treatment of various allergic symptoms.[L4269] It is selective for the H<sub>1</sub> receptor, carries little-to-no activity at off-targets, and does not cross the blood-brain bar…

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseBenzene Derivatives +12
Target Protein:
Histamine H1 receptor
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Fezakinumab DB12344
biotech | CAS: 1007106-86-6

Fezakinumab has been used in trials studying the treatment of Atopic Dermatitis and Rheumatoid Arthritis.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fezolinetant Approved DB15669
small molecule | CAS: 1629229-37-3

Vasomotor symptoms (VMS), more colloquially known as hot flashes or night sweats, are some of the most common symptoms in menopause. With a median duration of 7.4 years, vasomotor symptoms are also the most common reasons why women seek treatments for menopau…

Kategori:
Cytochrome P-450 CYP1A2 SubstratesCytochrome P-450 CYP2C19 SubstratesCytochrome P-450 CYP2C9 Substrates +6
Target Protein:
Neuromedin-K receptor
Waktu ParuhThe effective half-…
Vol. DistribusiThe mean apparent v…
KlirensThe apparent cleara…
Genetik -
FF-10101-01 DB16050
small molecule | CAS: 1472797-69-5

FF-10101-01 is under investigation in clinical trial NCT03194685 (Study of FF-10101-01 in Patients With Relapsed or Refractory Acute Myeloid Leukemia).

Kategori:
Enzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
Receptor-type tyrosine-protein kinase FLT3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FF-10501-01 DB17554
small molecule

FF-10501-01 is a novel, selective inosine monophosphate dehydrogenase (IMPDH) inhibitor with anticancer activity.[A257306] FF-10501-01 is under investigation in clinical trial NCT03486353 (A Study of FF-10501-01 in Combination With Azacitidine in Patients Wit…

Waktu Paruh-
Vol. Distribusi-
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Genetik -
FG-2216 DB08687
small molecule | CAS: 223387-75-5

A orally active prolyl-hydroxylase inhibitor which can stabilize hypoxia-inducible transcription factor independent of oxygen availability. [A14422]

Target Protein:
Egl nine homolog 1Hypoxia-inducible factor 1-alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
FG-9041 DB03759
small molecule | CAS: 2379-57-9

Deskripsi belum tersedia.

Kategori:
Excitatory Amino Acid AgentsExcitatory Amino Acid AntagonistsHeterocyclic Compounds, Fused-Ring +1
Target Protein:
Glutamate receptor 1Glutamate receptor ionotropic, kainate 1Glutamate receptor ionotropic, NMDA 2B +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fiacitabine DB12901
small molecule | CAS: 69123-90-6

Fiacitabine has been used in trials studying the treatment of HIV Infections and Cytomegalovirus Infections.

Kategori:
Anti-Infective AgentsAntineoplastic AgentsAntiviral Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fialuridine DB15427
small molecule | CAS: 69123-98-4

Fialuridine is under investigation in clinical trial NCT01337466 (Biodistribution and Dosimetry Evaluation of [124I]FIAU).

Kategori:
Anti-Infective AgentsAntiviral AgentsArabinonucleosides +7
Target Protein:
DNA polymerase catalytic subunit
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fianlimab DB18858
biotech | CAS: 2126132-98-5

Fianlimab is under investigation in clinical trial NCT06190951 (A Trial to Learn if Fianlimab and Cemiplimab Are Safe and Work Better Than Anti-pd1 Alone in Adult Participants With Resectable Stage 3 or 4 Melanoma).

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Fibrinogen human Approved DB09222
biotech | CAS: 9001-32-5

Fibrinogen concentrate (human) is a hematological agent. It works by replacing a specific protein in the blood, fibrinogen (factor I), that helps with blood clotting. It is a soluble plasma glycoprotein with a molecular weight of about 340 kDa and is a physi…

Kategori:
Acute-Phase ProteinsAmino Acids, Peptides, and ProteinsBiological Factors +8
Waktu Paruh-
Vol. Distribusi-
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Fibrinolysin DB05254
biotech | CAS: 9004-09-5

Fibrinolysin consists of two polypeptide chains, one light and one heavy, linked by a disulfide bond. The light chain has a molecular weight of approximately 27,000 Da and contains the active center of Fibrinolysin; the heavy chain has a molecular weight of a…

Kategori:
AnticoagulantsBlood and Blood Forming OrgansCardiovascular Agents +11
Target Protein:
Plasminogen activator inhibitor 1Urokinase-type plasminogen activator
Waktu ParuhAlmost completely i…
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 106096-92-8

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsFibroblast Growth Factor 1 +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fibronectin DB15150
biotech

Fibronectin is under investigation in clinical trial NCT01812239 (Vaginal Progesterone in Twins With Short Cervix).

Kategori:
Amino Acids, Peptides, and ProteinsBlood ProteinsCarbohydrates +9
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ficonalkib DB18774
small molecule | CAS: 2233574-95-1

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Fidanacogene elaparvovec Approved DB16783
biotech | CAS: 1954659-47-2

Fidanacogene elaparvovec is a liver-specific adeno-associated virus (AAV) vector containing a codon-optimized human coagulation FIX gene that was investigated as a potential treatment for hemophilia B.[L46691] Hemophilia B is a rare X-linked genetic disorder …

Kategori:
Adeno-associated Viral Vector TherapiesHepatotoxic Agents
Target Protein:
Coagulation factor IX (F9)
Waktu Paruh-
Vol. DistribusiIn a monkey biodist…
KlirensClearance of vector…
Genetik -
Fidarestat DB02021
small molecule | CAS: 136087-85-9

Deskripsi belum tersedia.

Kategori:
Aldehyde Reductase, antagonists & inhibitorsImidazoles
Target Protein:
Aldo-keto reductase family 1 member B1Aldo-keto reductase family 1 member B10
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fidaxomicin Approved DB08874
small molecule | CAS: 873857-62-6

Fidaxomicin is a novel macrolide antibiotic used in the treatment of diarrhea caused by _Clostridioides_ (formerly _Clostridium_) _difficile_ in adult and pediatric patients over the age of 6 months.[L11575] Fidaxomicin is a naturally-occurring 18-member macr…

Kategori:
Alimentary Tract and MetabolismAnti-Bacterial AgentsAnti-Infective Agents +13
Target Protein:
RNA polymerase sigma factor SigA
Waktu ParuhFollowing oral admi…
Vol. DistribusiFidaxomicin is main…
KlirensThere is limited in…
Genetik -
Fidrisertib DB18064
small molecule | CAS: 2141955-96-4

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
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Genetik -
Figopitant DB12122
small molecule | CAS: 502422-74-4

Figopitant is under investigation in clinical trial NCT02209714 (Safety, Tolerability and Pharmacodynamics After Oral Administration of BIIF 1149 BS in Healthy Male Volunteers).

Kategori:
AcetamidesAmidesBenzene Derivatives
Target Protein:
Substance-P receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Filaminast DB02660
small molecule | CAS: 141184-34-1

Filaminast is a phosphodiesterase 4 inhibitor (PDE4 inhibitor). As such, has potential in the treatment of asthma and chronic obstructive pulmonary disease (COPD).

Kategori:
AminesHydroxylamines
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B
Waktu Paruh-
Vol. Distribusi-
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Genetik -
Filgotinib Approved DB14845
small molecule | CAS: 1206161-97-8

Rheumatoid arthritis (RA) is a chronic, autoimmune, systemic, and inflammatory disease that causes synovial joint symptoms and can limit range of motion in severe cases.[A221451,A221456] The disease is associated with extra-articular manifestations, progressi…

Kategori:
Antineoplastic and Immunomodulating AgentsArthritis, Rheumatoid, drug therapyImmunosuppressive Agents +5
Target Protein:
Tyrosine-protein kinase JAK1
Waktu ParuhThe half-life of fi…
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6301–6350 dari 14063
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