Hasil Filter

6694

Total database: 17430
Struktur (SMILES)
4518 (67.5%)
Target
3751 (56.0%)
Genomik
81 (1.2%)
Referensi
6694 (100.0%)

Tipe Molekul

Distribusi Wujud Zat

Status Regulasi

Hasil Pencarian (6694)

Halaman 126 / 134
Treamid DB16365
small molecule

Treamid, also known as bisamide derivative of dicarboxylic acid (BDDA), is a complexing agent that has been found to chelate metal ions, including calcium, copper, iron, magnesium, and zinc.[A225701] This drug has shown regenerative properties and restoration…

Kategori:
Acids, AcyclicDicarboxylic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trebananib DB12056
biotech | CAS: 894356-79-7

Trebananib is under investigation for the treatment of Ovarian Cancer, Peritoneal Cancer, and Fallopian Tube Cancer. Trebananib has been investigated for the treatment of Cancer, Oncology, Carcinoma, Metastases, and Colon Cancer, among others.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trelagliptin DB15323
small molecule | CAS: 865759-25-7

Trelagliptin is under investigation in clinical trial NCT03555591 (Specified Drug-Use Survey of Trelagliptin Tablets "Survey on Long-term Use in Patients With Type 2 Diabetes Mellitus").

Kategori:
PyrimidinesPyrimidinones
Target Protein:
Dipeptidyl peptidase 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tremelimumab Approved DB11771
biotech | CAS: 745013-59-6

Tremelimumab, formerly known as ticilimumab, is a fully human IgG2 monoclonal antibody directed against cytotoxic T-lymphocyte-associated antigen 4 (CTLA-4). CTLA-4 is a cell surface receptor expressed on activated T cells to act as a negative regulator for T…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +11
Target Protein:
Cytotoxic T-lymphocyte protein 4
Waktu ParuhThe geometric mean …
Vol. DistribusiThe geometric mean …
KlirensThe geometric mean …
Genetik -
biotech

Tremella fuciformis whole is a plant/plant extract used in some OTC (over-the-counter) products. It is not an approved drug.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Treprostinil Approved DB00374
small molecule | CAS: 81846-19-7

Treprostinil is a stable tricyclic analogue of prostacyclin[A248770] that promotes the vasodilation of pulmonary and systemic arterial vascular beds and the inhibition of platelet aggregation.[L41855,L41860,L41865] It reduces symptoms in patients with pulmona…

Kategori:
Antihypertensive AgentsAutacoidsBiological Factors +19
Target Protein:
Prostacyclin receptorProstaglandin E2 receptor EP2 subtypeProstaglandin D2 receptor +2
Waktu ParuhThe terminal elimin…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
small molecule | CAS: 1706528-83-7

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trestolone DB05830
small molecule | CAS: 3764-87-2

Trestolone (7?-methyl-19-nortestosterone) is a synthetic androgen developed by the Population Council as a potential candidate drug for use in hormonal male contraceptive methods. In males, regular administration of sufficient quantities of trestolone induces…

Kategori:
Adrenal Cortex HormonesContraceptive Agents, HormonalContraceptive Agents, Male +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 6157-87-5

Trestolone acetate is a synthetic and injected anabolic–androgenic steroid (AAS) and a derivative of nandrolone (19-nortestosterone) which was never marketed. It is an androgen ester – specifically, the C17 acetate ester of [DB05830].

Kategori:
EstranesEstrenesFused-Ring Compounds +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tretazicar DB04253
small molecule | CAS: 21919-05-1

Tretazicar is under investigation in clinical trial NCT00746590 (Study of Anti-tumour Effects and Safety of Prolarix™ in Hepatocellular Carcinoma).

Kategori:
Antineoplastic AgentsAzirinesProdrugs +1
Target Protein:
Ribosyldihydronicotinamide dehydrogenase [quinone]Oxygen-insensitive NAD(P)H nitroreductase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tretinoin Approved DB00755
small molecule | CAS: 302-79-4

Tretinoin, also known as all-trans-retinoic acid (ATRA), is a naturally occurring derivative of [vitamin A] (retinol).[A257474] It is an oxidation product in the physiological pathway of vitamin A metabolism.[A257689] In human circulation, tretinoin is normal…

Kategori:
Agents that produce hypertensionAlkenesAnti-Acne Preparations +37
Target Protein:
Retinoic acid receptor alphaRetinoic acid receptor betaRetinoic acid receptor gamma +13
Waktu ParuhThe terminal elimin…
Vol. DistribusiTretinoin is rapidl…
KlirensNo information is a…
Genetik -
Triamcinolone Approved DB00620
small molecule | CAS: 124-94-7

Triamcinolone is a corticosteroid used to treat various inflammatory conditions in the body from allergic rhinitis to acute exacerbations of multiple sclerosis.[L8255] Triamcinolone can be used as a one time adjunct treatment of osteoarthritic knee pain,[L826…

Kategori:
Adrenal Cortex HormonesAdrenalsAgents Causing Muscle Toxicity +44
Target Protein:
Glucocorticoid receptor
Waktu ParuhThe half life of tr…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of tr…
Genetik -
Triamterene Approved DB00384
small molecule | CAS: 396-01-0

Triamterene (2,4,7-triamino-6-phenylpteridine) is a potassium-sparing diuretic that is used in the management of hypertension. It works by promoting the excretion of sodium ions and water while decreasing the potassium excretion in the distal part of the neph…

Kategori:
Agents causing hyperkalemiaCardiovascular AgentsCytochrome P-450 CYP1A2 Substrates +15
Target Protein:
Amiloride-sensitive sodium channel subunit gammaAmiloride-sensitive sodium channel subunit alphaAmiloride-sensitive sodium channel subunit beta +1
Waktu ParuhThe half-life of th…
Vol. DistribusiIn a pharmacolineti…
KlirensThe total plasma cl…
Genetik -
Triazavirin DB15622
small molecule | CAS: 123606-06-4

Triazavirin is a guanine nucleotide analog antiviral originally developed in Russia that has shown efficacy against influenza A and B, including the H5N1 strain.[A191709,A191625,A191916] It appears that Triazavirin has shown promise in reducing influenza dise…

Kategori:
Antiviral AgentsExperimental Unapproved Treatments for COVID-19Guanine Nucleotides
Waktu ParuhIn rabbits, intraga…
Vol. DistribusiIn rabbits, intraga…
KlirensIn rabbits, intraga…
Genetik -
Tributyrin DB12709
small molecule | CAS: 60-01-5

Tributyrin has been used in trials studying the treatment of Prostate Cancer and Unspecified Adult Solid Tumor, Protocol Specific.

Kategori:
GlyceridesLipids
Target Protein:
Caspase-3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Tricaprylin DB12176
small molecule | CAS: 538-23-8

Tricaprilin has been used in trials studying the supportive care and treatment of Alzheimer's Disease.

Kategori:
Acids, AcyclicAlzheimer Disease, drug therapyCompounds used in a research, industrial, or household setting +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 99-14-9

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Aconitate hydratase, mitochondrial
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichloroacetate Approved DB11152
small molecule | CAS: 76-03-9

Trichloroacetate, or trichloroacetic acid, is a strong acid prepared by the reaction of chlorine with acetic acid in the presence of a suitable catalyst. In clinical chemistry and biochemistry, it is used as a precipitant of macromolecules including proteins,…

Kategori:
AcetatesAcids, AcyclicCaustics +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichloroethylene Approved DB13323
small molecule | CAS: 79-01-6

Trichloroethylene is a halocarbon commonly used as an industrial solvent, not to be confused with the similar 1,1,1-trichloroethane, also known as chlorothene. It has been sold under a variety of trade names including Trimar and Trilene and used as a volatile…

Kategori:
Agents that produce hypertensionAnestheticsAnesthetics, General +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trichothecium roseum Approved DB10696
biotech

Trichothecium roseum is a fungus which can provoke allergic reactions. Trichothecium roseum extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseIncreased IgG Production +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triciribine DB12405
small molecule | CAS: 35943-35-2

Triciribine has been used in trials studying the treatment of Leukemia, Ovarian Cancer, HER2/Neu Negative, Breast Adenocarcinoma, and Stage IV Breast Cancer, among others.

Kategori:
Nucleic Acids, Nucleotides, and NucleosidesNucleosides
Target Protein:
Gag-Pol polyprotein
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 61966-08-3

Deskripsi belum tersedia.

Kategori:
NaphthalenesNucleic Acids, Nucleotides, and NucleosidesNucleotides
Target Protein:
RAC-gamma serine/threonine-protein kinase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triclabendazole Approved DB12245
small molecule | CAS: 68786-66-3

Triclabendazole, manufactured by Novartis pharmaceuticals, is an antihelminthic drug that was approved by the FDA in February 2019 for the treatment of fascioliasis in humans.[FDA label, L5452] Fascioliasis is a parasitic infection often caused by the helmi…

Kategori:
AnthelminticsAnti-Infective AgentsAntihelminthic +34
Target Protein:
CruzipainExcretory Secretory (ES) proteins
Waktu ParuhThe plasma eliminat…
Vol. DistribusiThe apparent volume…
Klirens-
Genetik -
small molecule | CAS: 2433-96-7

Deskripsi belum tersedia.

Kategori:
Fatty AcidsLipids
Target Protein:
Lipase 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 77-93-0

Deskripsi belum tersedia.

Kategori:
Acids, AcyclicTricarboxylic Acids
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 78-40-0

Deskripsi belum tersedia.

Kategori:
Organophosphorus Compounds
Target Protein:
Parathion hydrolaseCellular tumor antigen p53Parathion hydrolase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triethylenetetramine Approved DB06824
small molecule | CAS: 112-24-3

Triethylenetatramine (TETA), also known as trientine, is a potent and selective copper (II)-selective chelator. It is a structural analog of linear polyamine compounds, [spermidine] and [spermine]. TETA was first developed in Germany in 1861 and its chelating…

Kategori:
Alimentary Tract and MetabolismAminesChelating Agents +11
Target Protein:
Carbonic anhydrase 14
Waktu ParuhThe mean terminal h…
Vol. DistribusiTETA is widely dist…
KlirensIn healthy adult vo…
Genetik -
Trifluridine Approved DB00432
small molecule | CAS: 70-00-8

Trifluridine is a fluorinated pyrimidine nucleoside that is structurally related to [idoxuridine] [A35271]. It is an active antiviral agent in ophthalmic solutions used mainly in the treatment of primary keratoconjunctivitis and recurrent epithelial keratitis…

Kategori:
Anti-Infective AgentsAntimetabolitesAntineoplastic Agents +20
Target Protein:
Thymidylate synthaseDNAThymidylate synthase
Waktu ParuhAfter administratio…
Vol. DistribusiFollowing a single …
KlirensFollowing a single …
Genetik -
Triflusal Approved DB08814
small molecule | CAS: 322-79-2

Triflusal is a 2-acetoxy-4-trifluoromethylbenzoic acid and it is an aspirin chemically-related molecule but not a derivative. The benefits of this agent are the lack of action over the arachidonic acid pathway, the driven production of nitric oxide and the in…

Kategori:
Acids, CarbocyclicAnticoagulantsAntiplatelet agents +8
Target Protein:
Prostaglandin G/H synthase 1Nuclear factor NF-kappa-B p105 subunitNitric oxide synthase, inducible +1
Waktu ParuhIn the healthy huma…
Vol. DistribusiThe reported volume…
KlirensRenal clearance is …
Genetik -
Triheptanoin Approved DB11677
small molecule | CAS: 620-67-7

Triheptanoin is a source of heptanoate fatty acids, which can be metabolized without the enzymes of long chain fatty acid oxidation.[L14612] In clinical trials, patients with long chain fatty acid oxidation disorders (lc-FAODs) treated with triheptanoin are l…

Kategori:
Alimentary Tract and MetabolismCaloric AgentsGlycerides +5
Waktu ParuhDue to multiple pea…
Vol. Distribusi-
KlirensA single dose of 0.…
Genetik -
Trilaciclib Approved DB15442
small molecule | CAS: 1374743-00-6

Trilaciclib, or G1T28, is a CDK4 and CDK6 inhibitor, indicated to reduce the incidence of chemotherapy induced myelosuppression in patients before topotecan-containing or platinum and etoposide-containing chemotherapy for extensive stage small cell lung cance…

Kategori:
BCRP/ABCG2 SubstratesCyclin-dependent Kinase 4 InhibitorsCyclin-dependent Kinase 6 Inhibitors +16
Target Protein:
Cyclin-dependent kinase 4Cyclin-dependent kinase 6Cyclin-dependent kinase 9 +3
Waktu ParuhThe mean terminal h…
Vol. DistribusiThe volume of distr…
KlirensThe clearance of tr…
Genetik -
Trimesic acid DB08632
small molecule | CAS: 554-95-0

Deskripsi belum tersedia.

Kategori:
Acids, Acyclic
Target Protein:
Hemoglobin subunit alphaHemoglobin subunit beta
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetazidine Approved DB09069
small molecule | CAS: 5011-34-7

Trimetazidine is a piperazine derivative indicated for the symptomatic treatment of stable angina pectoris in patients inadequately controlled or intolerant to first line therapies.[L33015] Trimetazidine has been studied as a treatment for angina pectoris sin…

Kategori:
Cardiac TherapyCardiovascular AgentsPiperazines +1
Target Protein:
3-ketoacyl-CoA thiolase, mitochondrial
Waktu ParuhIn young, healthy s…
Vol. DistribusiThe volume of distr…
KlirensTrimetazidine clear…
Genetik -
Trimethadione Approved DB00347
small molecule | CAS: 127-48-0

An anticonvulsant effective in absence seizures, but generally reserved for refractory cases because of its toxicity. (From AMA Drug Evaluations Annual, 1994, p378)

Kategori:
Agents causing hyperkalemiaAnti-epileptic AgentAntiarrhythmic agents +18
Target Protein:
Voltage-dependent T-type calcium channel subunit alpha-1G
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimethoprim Approved DB00440
small molecule | CAS: 738-70-5

Trimethoprim is an antifolate antibacterial agent that inhibits bacterial dihydrofolate reductase (DHFR), a critical enzyme that catalyzes the formation of tetrahydrofolic acid (THF) - in doing so, it prevents the synthesis of bacterial DNA and ultimately con…

Kategori:
Agents causing hyperkalemiaAgents Causing Muscle ToxicityAnti-Infective Agents +32
Target Protein:
Dihydrofolate reductaseDihydrofolate reductase
Waktu ParuhTrimethoprim half-l…
Vol. DistribusiTrimethoprim is ext…
KlirensFollowing oral admi…
Genetik -
Trimethyllysine DB03977
small molecule | CAS: 19253-88-4

Deskripsi belum tersedia.

Kategori:
Amino AcidsAmino Acids, BasicAmino Acids, Diamino +3
Target Protein:
Calmodulin-2Calmodulin-1Calmodulin-3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trimetrexate Approved DB01157
small molecule | CAS: 52128-35-5

A nonclassical folic acid inhibitor through its inhibition of the enzyme dihydrofolate reductase. It is being tested for efficacy as an antineoplastic agent and as an antiparasitic agent against pneumocystis pneumonia in AIDS patients. Myelosuppression is its…

Kategori:
Acids, AcyclicAcids, AldehydicAnti-Infective Agents +18
Target Protein:
Peptide deformylase, mitochondrialDihydrofolate reductase
Waktu Paruh11 to 20 hours
Vol. Distribusi* 20 ± 8 L/m2 * 36…
Klirens* 38 +/- 15 mL/min/…
Genetik -
Trioxsalen Approved DB04571
small molecule | CAS: 3902-71-4

Trioxsalen (trimethylpsoralen, trioxysalen or trisoralen) is a furanocoumarin and a psoralen derivative obtained from several plants, mainly Psoralea corylifolia. Like other psoralens it causes photosensitization of the skin. It is administered either topical…

Kategori:
AntipsoriaticsAntipsoriatics for Systemic UseAntipsoriatics for Topical Use +11
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 10380-08-2

Used as water softener, peptizing agent, emulsifier & dispersing agent; ingredient of cleansers; meat preservative.

Kategori:
AcidsAcids, NoncarboxylicAnions +5
Target Protein:
Poly(A) polymerase alpha
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Triprolidine Approved DB00427
small molecule | CAS: 486-12-4

First generation histamine H1 antagonist used in allergic rhinitis; asthma; and urticaria. It is a component of cough and cold medicines. It may cause drowsiness.

Kategori:
Anti-Allergic AgentsAntihistamines for Systemic UseCentral Nervous System Depressants +7
Target Protein:
Histamine H1 receptor
Waktu Paruh4 to 6 hours.
Vol. Distribusi-
Klirens-
Genetik -
TRK-001 DB18577
biotech

TRK-001 is an autologous regulatory T-cell therapy. It is being investigated for the prevention of graft rejection following solid organ transplantation.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troclosene DB15960
small molecule | CAS: 2782-57-2

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntiviral Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trofinetide Approved DB06045
small molecule | CAS: 853400-76-7

Trofinetide is a novel synthetic analog of [glypromate], also known as glycine–proline–glutamate (GPE), a naturally occurring protein in the brain and the N-terminal tripeptide of insulin-like growth factor 1 (IGF-1).[A258438] Trofinetide was approved by the …

Kategori:
Amino AcidsAmino Acids, AcidicAmino Acids, Dicarboxylic +11
Waktu ParuhThe effective elimi…
Vol. DistribusiFollowing oral admi…
KlirensNo information is a…
Genetik -
Troglitazone Approved DB00197
small molecule | CAS: 97322-87-7

Troglitazone was withdrawn in 2000 due to risk of hepatotoxicity. It was superseded by [pioglitazone] and [rosiglitazone].

Kategori:
Alimentary Tract and MetabolismBenzopyransBlood Glucose Lowering Agents +38
Target Protein:
Peroxisome proliferator-activated receptor gammaEstrogen-related receptor gammaSteroid hormone receptor ERR1 +6
Waktu Paruh16-34 hours
Vol. Distribusi-
Klirens-
Genetik -
Trolamine salicylate Approved DB11079
small molecule | CAS: 2174-16-5

Trolamine salicylate is an organic compound or a salt formed between triethanolamine and salicylic acid. Triethanolamine neutralizes the acidity of the salicylic acid. It is a topical analgesic used for temporary relief of minor pain associated with arthritis…

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAnti-Inflammatory Agents +11
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2
Waktu Paruh-
Vol. DistribusiTopical administrat…
Klirens-
Genetik -
Troleandomycin Approved DB13179
small molecule | CAS: 2751-09-9

A macrolide antibiotic that is similar to erythromycin.

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAntibacterials for Systemic Use +18
Target Protein:
50S ribosomal protein L3250S ribosomal protein L4Nuclear receptor subfamily 1 group I member 2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Trovafloxacin Approved DB00685
small molecule | CAS: 147059-72-1

Trovafloxacin is a broad spectrum antibiotic that has been commonly marketed under the brand name Trovan by Pfizer. It exerts its antibacterial activity by inhibiting the uncoiling of supercoiled DNA in various bacteria by blocking the activity of DNA gyrase …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +16
Target Protein:
DNA gyrase subunit ADNA gyrase subunit BDNA gyrase subunit A +2
Waktu ParuhFollowing oral admi…
Vol. Distribusi-
Klirens-
Genetik -
Troxacitabine DB04961
small molecule | CAS: 145918-75-8

Troxacitabine is a nucleoside analog with antineoplastic activity. There has been growing interest in its development for the treatment of patients with refractory lymphoproliferative conditions.

Kategori:
Anti-HIV AgentsAnti-Infective AgentsAntineoplastic Agents +3
Target Protein:
DNA
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Troxerutin DB13124
small molecule | CAS: 7085-55-4

Troxerutin has been used in trials studying the treatment of Chronic Venous Insufficiency.

Kategori:
AnticoagulantsBenzopyransCapillary Stabilizing Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
TRX-E-002-1 DB17264
small molecule | CAS: 1803036-93-2

Deskripsi belum tersedia.

Kategori:
BenzopyransChromonesHeterocyclic Compounds, Fused-Ring +1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Menampilkan 6251–6300 dari 6694
Sebelumnya Halaman 126 / 134 Berikutnya