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14063

Total database: 17430
Struktur (SMILES)
10481 (74.5%)
Target
8038 (57.2%)
Genomik
107 (0.8%)
Referensi
14063 (100.0%)

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Hasil Pencarian (14063)

Halaman 126 / 282
fb-PMT DB17394
small molecule

Deskripsi belum tersedia.

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FCX-013 DB18218
biotech

FCX-013 consists of human dermal fibroblasts genetically modified with a lentiviral vector expressing metalloproteinase-1 (MMP-1).

Waktu Paruh-
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FDL169 DB16878
small molecule | CAS: 1628416-28-3

Deskripsi belum tersedia.

Waktu Paruh-
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Febantel DB11409
small molecule | CAS: 58306-30-2

Deskripsi belum tersedia.

Kategori:
AmidinesAnthelminticsAnti-Infective Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febarbamate DB13303
small molecule | CAS: 13246-02-1

Deskripsi belum tersedia.

Kategori:
Carbamic Acid EstersCentral Nervous System DepressantsMuscle Relaxants +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Febuxostat Approved DB04854
small molecule | CAS: 144060-53-7

Febuxostat is a non-purine xanthine oxidase (XO) inhibitor.[A39743] In early 2008, febuxostat was granted marketing authorization by the European Commission for the treatment of chronic hyperuricemia and gout.[A230548] In the following year, the FDA for appro…

Kategori:
Antigout PreparationsAntirheumatic AgentsBCRP/ABCG2 Inhibitors +15
Target Protein:
Xanthine dehydrogenase/oxidase
Waktu ParuhThe apparent mean t…
Vol. DistribusiThe apparent steady…
KlirensFollowing oral admi…
Genetik -
Fecal microbiota Approved DB17743
biotech

Fecal microbiota, given either as a rectal transplant or in an oral formulation of live spores, is an FDA-approved option to prevent the recurrence of _Clostridioides difficile_ infection (CDI) in patients given an antibacterial treatment for recurrent CDI.[A…

Kategori:
Miscellaneous Therapeutic Agents
Waktu ParuhNot available.
Vol. DistribusiNot available.
KlirensNot available.
Genetik -
Fedratinib Approved DB12500
small molecule | CAS: 936091-26-8

Fedratinib, also known as SAR302503 and TG101348, is a tyrosine kinase inhibitor used to treat intermediate-2 and high risk primary and secondary myelofibrosis.[A183176,L8090] It is an anilinopyrimidine derivative.[A183188] Fedratinib was granted FDA appro…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +25
Target Protein:
Tyrosine-protein kinase JAK2Receptor-type tyrosine-protein kinase FLT3Tyrosine-protein kinase JAK1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe apparent volume…
KlirensThe clearance of fe…
Genetik -
Fedrilate DB13825
small molecule | CAS: 23271-74-1

Deskripsi belum tersedia.

Kategori:
Cough and Cold Preparations
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Feladilimab DB16415
biotech

Feladilimab is under investigation in clinical trial NCT04128696 (Study of GSK3359609 and Pembrolizumab in Programmed Death Receptor 1-ligand 1 Positive Recurrent or Metastatic Head and Neck Squamous Cell Carcinoma).

Waktu Paruh-
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Felbamate Approved DB00949
small molecule | CAS: 25451-15-4

Felbamate is an anticonvulsant drug used in the treatment of epilepsy. In particular, in the adult patient population, it can be employed to treat partial seizures (with and without generalization). Alternatively, it is used to treat partial and generalized s…

Kategori:
Acids, AcyclicAlcoholsAnti-epileptic Agent +28
Target Protein:
Glutamate receptor ionotropic, NMDA 2BGlutamate receptor ionotropic, NMDA 2A
Waktu Paruh20-23 hours
Vol. Distribusi* 756±82 mL/kg
Klirens* 26 +/- 3 mL/hr/kg…
Genetik -
Felbinac DB07477
small molecule | CAS: 5728-52-9

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +12
Target Protein:
Prostaglandin G/H synthase 1Prostaglandin G/H synthase 2Procathepsin L
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felcisetrag DB12725
small molecule | CAS: 916075-84-8

Felcisetrag (TD-8954) has been used in trials studying the treatment of Enteral Feeding Intolerance and Gastrointestinal Motility Disorder.

Kategori:
Antidepressive AgentsCentral Nervous System DepressantsHeterocyclic Compounds, Fused-Ring +4
Target Protein:
5-hydroxytryptamine receptor 4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felodipine Approved DB01023
small molecule | CAS: 72509-76-3

Felodipine is a long-acting 1,4-dihydropyridine calcium channel blocker (CCB)b. It acts primarily on vascular smooth muscle cells by stabilizing voltage-gated L-type calcium channels in their inactive conformation. By inhibiting the influx of calcium in smoot…

Kategori:
ACE Inhibitors and Calcium Channel BlockersAgents causing hyperkalemiaAntiarrhythmic agents +31
Target Protein:
Voltage-dependent L-type calcium channel subunit alpha-1CVoltage-dependent calcium channel subunit alpha-2/delta-1Voltage-dependent L-type calcium channel subunit beta-2 +10
Waktu Paruh17.5-31.5 hours in …
Vol. Distribusi* 10 L/kg
Klirens* 0.8 L/min [Young …
Genetik -
Felypressin DB00093
biotech | CAS: 56-59-7

A synthetic nonapeptide comprising cysteinyl, phenylalanyl, phenylalanyl, glutaminyl, asparaginyl, cysteinyl, prolyl, lysyl, and glycinamide residues in sequence, with a disulfide bridge joining the two cysteine residues. Its antidiuretic effects are less tha…

Kategori:
Amino Acids, Peptides, and ProteinsCardiovascular AgentsHormones +12
Target Protein:
Vasopressin V1a receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Felzartamab DB16375
biotech | CAS: 2197112-39-1

Felzartamab is under investigation in clinical trial NCT04145440 (Trial to Assess Safety and Efficacy of MOR202 in Anti-pla2r + Membranous Nephropathy (Amn)).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +8
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Fenamole DB12506
small molecule | CAS: 5467-78-7

Fenamole has been investigated for the supportive care of Side Effects and Dental Plaque.

Waktu Paruh-
Vol. Distribusi-
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Fenbendazole DB11410
small molecule | CAS: 43210-67-9

Fenbendazole is a benzimidazole that presents a wide spectrum anthelmintic effect. It is used against a number of gastrointestinal parasites including giardia, roundworms, hookworms, whipworms, the Taenia genus of tapeworms, pinworms, aelurostrongylus, parago…

Kategori:
Acids, AcyclicAnthelminticsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fencamfamin DB01463
small molecule | CAS: 1209-98-9

Fencamfamin (Glucoenergan, Reactivan) is a stimulant which was developed in the 1960s as an appetite suppressant, but was later withdrawn for this application due to problems with dependence and abuse. It is around half the potency of [dexamphetamine], and is…

Kategori:
Bridged-Ring CompoundsCentral Nervous System AgentsCentral Nervous System Depressants +7
Target Protein:
Sodium-dependent dopamine transporterD(2) dopamine receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fendiline DB08980
small molecule | CAS: 13042-18-7

Fendiline is a coronary vasodilator which inhibits calcium function in muscle cells in excitation-contraction coupling. It has been proposed as an antiarrhythmic and antianginal agent. Fendiline is non-selective.

Kategori:
Agents causing hyperkalemiaAminesAntiarrhythmic agents +15
Target Protein:
5-hydroxytryptamine receptor 2B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenethylline DB01482
small molecule | CAS: 3736-08-1

Deskripsi belum tersedia.

Kategori:
AlkaloidsAminesCentral Nervous System Agents +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
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Fenfluramine Approved DB00574
small molecule | CAS: 458-24-2

Dravet syndrome is a pediatric encephalopathy that typically manifests within the first year of life following exposure to elevated temperatures. It is characterized by recurrent pharmacoresistant seizures, which increase in frequency and severity with diseas…

Kategori:
Alimentary Tract and MetabolismAminesAnticonvulsants +27
Target Protein:
Sodium-dependent serotonin transporter5-hydroxytryptamine receptor 1D5-hydroxytryptamine receptor 2C +4
Waktu ParuhFenfluramine has an…
Vol. DistribusiFenfluramine has an…
KlirensFenfluramine has a …
Genetik -
Fenobam DB12931
small molecule | CAS: 57653-26-6

Fenobam is under investigation in clinical trial NCT00637221 (Open Label Study Investigating Safety and Efficacy of Fenobam anhydrous 50 mg - 150 mg on Prepulse Inhibition Tests and Continuous Performance Tasks, Adults With Fragile X Syndrome).

Target Protein:
Metabotropic glutamate receptor 5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenofibrate Approved DB01039
small molecule | CAS: 49562-28-9

Fenofibrate is a fibric acid derivative like [clofibrate] and [gemfibrozil].[A185954] Fenofibrate is used to treat primary hypercholesterolemia, mixed dyslipidemia, severe hypertriglyceridemia.[L8588,L8591] Fenofibrate was granted FDA approval on 31 Decemb…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityBenzene Derivatives +39
Target Protein:
Peroxisome proliferator-activated receptor alphaNuclear receptor subfamily 1 group I member 2Matrix metalloproteinase-25
Waktu ParuhFenofibric acid, th…
Vol. DistribusiThe volume of distr…
KlirensThe oral clearance …
Genetik -
Fenofibric acid Approved DB13873
small molecule | CAS: 42017-89-0

Fenofibric acid is a lipid-lowering agent that is used in severe hypertriglyceridemia, primary hyperlipidemia, and mixed dyslipidemia. It works to decrease elevated low-density lipoprotein cholesterol, total cholesterol, triglycerides, apolipoprotein B, while…

Kategori:
Acids, AcyclicAgents Causing Muscle ToxicityAnticholesteremic Agents +17
Target Protein:
Peroxisome proliferator-activated receptor alphaFatty acid-binding protein, liverMatrix metalloproteinase-25 +3
Waktu ParuhFollowing once dail…
Vol. DistribusiThe volume of distr…
KlirensIn five elderly vol…
Genetik -
Fenoldopam Approved DB00800
small molecule | CAS: 67227-56-9

A dopamine D1 receptor agonist that is used as an antihypertensive agent. It lowers blood pressure through arteriolar vasodilation.

Kategori:
Adrenergic and Dopaminergic AgentsAntihypertensive AgentsAntihypertensive Agents Indicated for Hypertension +12
Target Protein:
D(1B) dopamine receptorD(1A) dopamine receptorAlpha-1B adrenergic receptor +5
Waktu ParuhThe elimination hal…
Vol. Distribusi-
Klirens-
Genetik -
Fenoprofen Approved DB00573
small molecule | CAS: 29679-58-1

An anti-inflammatory analgesic and antipyretic highly bound to plasma proteins. It is pharmacologically similar to aspirin, but causes less gastrointestinal bleeding.

Kategori:
Acids, CarbocyclicAgents causing hyperkalemiaAgents that produce hypertension +18
Target Protein:
Prostaglandin G/H synthase 2Prostaglandin G/H synthase 1Peroxisome proliferator-activated receptor alpha +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Fenoterol Approved DB01288
small molecule | CAS: 13392-18-2

Fenoterol is an adrenergic beta-2 agonist that is used as a bronchodilator and tocolytic.

Kategori:
Adrenergic AgentsAdrenergic AgonistsAdrenergic beta-2 Receptor Agonists +28
Target Protein:
Beta-2 adrenergic receptorBeta-1 adrenergic receptorBeta-3 adrenergic receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenoverine DB13042
small molecule | CAS: 37561-27-6

Fenoverine has been used in trials studying the treatment of Irritable Bowel Syndrome.

Kategori:
Alimentary Tract and MetabolismAutonomic AgentsDrugs for Functional Gastrointestinal Disorders +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 66441-23-4

Fenoxaprop-ethyl (organic nitrate combined with L-arginine), is an oral proprietary nitrate therapeutic shown to induce coronary vasodilation while overcoming the significant problem of drug tolerance. Fenoxaprop-ethyl has been investigated to treat chronic a…

Kategori:
Acids, AcyclicAgrochemicalsCompounds used in a research, industrial, or household setting +6
Target Protein:
Nitric oxide synthase 3Nitric oxide synthase, inducible
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenozolone DB13341
small molecule | CAS: 15302-16-6

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAgents that produce hypertensionAutonomic Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpiprane DB13439
small molecule | CAS: 3540-95-2

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismBenzene DerivativesDrugs for Functional Gastrointestinal Disorders
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpiverinium DB13759
small molecule | CAS: 258329-46-3

Deskripsi belum tersedia.

Kategori:
Agents producing tachycardiaAlimentary Tract and MetabolismAnticholinergic Agents +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenpropidin Approved DB12728
small molecule | CAS: 67306-00-7

Fenpropidin has been investigated for the treatment of Hernia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingFungicides, Industrial +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenproporex DB01550
small molecule | CAS: 16397-28-7

Fenproporex is an orally active stimulant drug, which was developed in the 1960s. It is used as an appetite suppressant and a treatment for obesity. It is listed as an illicit substance in many countries due to addiction issues and listed as a prohibited subs…

Kategori:
AminesDrugs that are Mainly Renally ExcretedEthylamines +2
Waktu Paruh-
Vol. Distribusi-
KlirensThe amphetamine met…
Genetik -
Fenpyroximate DB16164
small molecule | CAS: 134098-61-6

Fenpyroximate is under investigation in clinical trial NCT02533336 (The Effectiveness of Non-pyrethroid Insecticide-treated Durable Wall Liners as a Method for Malaria Control in Endemic Rural Tanzania).

Kategori:
Acids, CarbocyclicBenzene DerivativesElectron Transport Complex I, antagonists & inhibitors
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenquizone DB13708
small molecule | CAS: 20287-37-0

Deskripsi belum tersedia.

Kategori:
DiureticsHeterocyclic Compounds, Fused-RingLow-Ceiling Diuretics, Excl. Thiazides +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fentanyl Approved DB00813
small molecule | CAS: 437-38-7

Fentanyl, a potent opioid agonist, was developed in the 1950s to fill a need for strong and rapid analgesia.[A179542] Because of these characteristics, fentanyl is commonly used to treat chronic cancer pain or in anesthesia.[Label,L6598,L6601,L6604,L6607,L922…

Kategori:
AdjuvantsAdjuvants, AnesthesiaAgents that produce hypertension +32
Target Protein:
Mu-type opioid receptorDelta-type opioid receptorKappa-type opioid receptor +1
Waktu ParuhThe half life of fe…
Vol. DistribusiThe intravenous vol…
KlirensTotal plasma cleara…
Genetik -
Fenthion DB11412
small molecule | CAS: 55-38-9

Fenthion is an _organothiophosphate_ drug used as an insecticide, avicide, and acaricide. Its mode of action is explained by cholinesterase enzyme inhibition, which is similar to other organophosphates. Fenthion is listed as a restricted use compound by the U…

Kategori:
AgrochemicalsCholinergic AgentsCholinesterase Inhibitors +13
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fentiazac DB13217
small molecule | CAS: 18046-21-4

Deskripsi belum tersedia.

Kategori:
Acetic Acid Derivatives and Related SubstancesAcids, AcyclicAgents causing hyperkalemia +19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenticonazole DB13434
small molecule | CAS: 72479-26-6

Deskripsi belum tersedia.

Kategori:
Anti-Infective AgentsAntifungal AgentsAntifungals for Dermatological Use +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fenvalerate DB18391
small molecule | CAS: 51630-58-1

Deskripsi belum tersedia.

Kategori:
AgrochemicalsCompounds used in a research, industrial, or household settingCyclopentane Monoterpenes +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fepixnebart DB19079
biotech | CAS: 1799706-87-8

Fepixnebart is under investigation in clinical trial NCT04456686 (Chronic Pain Master Protocol (CPMP): A Study of LY3016859 in Participants With Osteoarthritis).

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Fepradinol DB15902
small molecule | CAS: 36981-91-6

Deskripsi belum tersedia.

Kategori:
AlcoholsAminesAmino Alcohols +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Feprazone DB13364
small molecule | CAS: 30748-29-9

Deskripsi belum tersedia.

Kategori:
Agents causing hyperkalemiaAgents that produce hypertensionAnalgesics +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
small molecule | CAS: 54063-42-2

Deskripsi belum tersedia.

Kategori:
Diagnostic RadiopharmaceuticalsVarious Diagnostic Radiopharmaceuticals
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ferric carboxymaltose Approved DB08917
small molecule | CAS: 9007-72-1

Ferric carboxymaltose is an iron replacement product and, chemically, an iron-carbohydrate complex. It was FDA approved on July 25, 2013.

Kategori:
CarbohydratesCompounds used in a research, industrial, or household settingDisaccharides +5
Waktu ParuhThe terminal half-l…
Vol. DistribusiThe estimated volum…
Klirens-
Genetik -
Ferric cation Approved DB13949
small molecule | CAS: 20074-52-6

Iron is a transition metal with a symbol Fe and atomic number 26. By mass, it is the most common element on Earth. Iron is an essential element involved in various metabolic processes, including oxygen transport, deoxyribonucleic acid (DNA) synthesis, and ene…

Kategori:
Iron CompoundsParenteral Iron ReplacementPhosphate Binder +2
Target Protein:
Transferrin receptor protein 1Iron(3+)-hydroxamate-binding protein FhuD
Waktu ParuhThe pharmacokinetic…
Vol. DistribusiLess than 65% of ir…
KlirensThe rate of iron lo…
Genetik -
Ferric derisomaltose Approved DB15617
small molecule | CAS: 1345510-43-1

Iron deficiency is an extremely common condition and is the most frequent cause of anemia worldwide. Iron deficiency results when iron intake, iron stores, and loss of iron from the body do not adequately support production of erythrocytes, also known as red …

Kategori:
Anemia, Iron-DeficiencyAntianemia DrugsAntianemic Preparations +6
Target Protein:
Hemoglobin subunit alphaTransferrin receptor
Waktu ParuhThe plasma-half liv…
Vol. DistribusiFerric derisomaltos…
KlirensIntravenous iron is…
Genetik -
small molecule | CAS: 1309-33-7

Deskripsi belum tersedia.

Kategori:
Antianemic PreparationsBlood and Blood Forming OrgansIron Compounds +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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