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15718

Total database: 17430
Struktur (SMILES)
10762 (68.5%)
Target
7957 (50.6%)
Genomik
112 (0.7%)
Referensi
15718 (100.0%)

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Hasil Pencarian (15718)

Halaman 126 / 315
Encaleret DB18096
small molecule | CAS: 787583-71-5

Deskripsi belum tersedia.

Kategori:
Acids, CarbocyclicAlcoholsAmines +3
Target Protein:
Extracellular calcium-sensing receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encenicline DB11726
small molecule | CAS: 550999-75-2

Encenicline has been investigated for the treatment of Cognition, Schizophrenia, Alzheimer's Disease, Cardiac Repolarization, and Central Nervous System Diseases.

Kategori:
Nicotinic AgonistsSulfur Compounds
Target Protein:
Neuronal acetylcholine receptor subunit alpha-7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enclomiphene DB06735
small molecule | CAS: 15690-57-0

Deskripsi belum tersedia.

Kategori:
Benzene DerivativesBenzylidene CompoundsClomiphene +11
Target Protein:
Estrogen receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Encorafenib Approved DB11718
small molecule | CAS: 1269440-17-6

Encorafenib, also known as _BRAFTOVI_, is a kinase inhibitor. Encorafenib inhibits BRAF gene, which encodes for B-raf protein, which is a proto-oncogene involved in various genetic mutations.[L12216] This protein plays a role in regulating the MAP kinase/E…

Kategori:
AmidesAntineoplastic AgentsAntineoplastic and Immunomodulating Agents +47
Target Protein:
Serine/threonine-protein kinase B-rafG1/S-specific cyclin-D1RAF proto-oncogene serine/threonine-protein kinase +7
Waktu ParuhThe mean (CV%) term…
Vol. DistribusiThe blood-to-plasma…
KlirensThe apparent cleara…
Genetik -
Endostar DB11727
biotech

Endostar is under investigation for the treatment of Nasopharyngeal Carcinoma. Endostar has been investigated for the treatment of Non-small Cell Lung Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endostatin DB06423
biotech | CAS: 187888-07-9

Deskripsi belum tersedia.

Kategori:
Amino Acids, Peptides, and ProteinsAngiogenesis InhibitorsAngiogenesis Modulating Agents +15
Target Protein:
72 kDa type IV collagenaseMatrix metalloproteinase-9Collagenase 3 +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endothelin-1 DB12652
biotech | CAS: 117399-94-7

Endothelin 1 is under investigation in clinical trial NCT00745693 (The Effects of Diesel Exhaust Inhalation on Vascular Function - the Role of Endothelin).

Kategori:
Amino Acids, Peptides, and ProteinsBiological FactorsEndothelin-1, antagonists & inhibitors +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Endralazine DB13435
small molecule | CAS: 39715-02-1

Deskripsi belum tersedia.

Kategori:
Antihypertensive AgentsArteriolar Smooth Muscle, Agents Acting OnCardiovascular Agents +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eneboparatide DB18207
biotech | CAS: 1349298-00-5

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enecadin DB13032
small molecule | CAS: 259525-01-4

Enecadin has been investigated for the treatment of Stroke.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enflurane Approved DB00228
small molecule | CAS: 13838-16-9

Enflurane is a halogenated inhalational anesthetic initially approved by the FDA in 1972. Since this date, it has been withdrawn from the US market.[L13646,L13649] Unlike its other inhalational anesthetic counterparts including [isoflurane] and [halothane], e…

Kategori:
Agents that reduce seizure thresholdAnestheticsAnesthetics, General +8
Target Protein:
GABA(A) ReceptorVoltage-dependent calcium channelGlycine receptor subunit alpha-1 +4
Waktu Paruh-
Vol. DistribusiEnflurane distribut…
Klirens-
Genetik -
Enfortumab vedotin Approved DB13007
biotech | CAS: 1346452-25-2

Enfortumab vedotin is an antibody-drug conjugate used in the treatment of patients with advanced, treatment-resistant urothelial cancers.[L10836] It is comprised of a fully human monoclonal antibody targeted against Nectin-4 and a microtubule-disrupting chemo…

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +19
Target Protein:
Nectin-4
Waktu ParuhThe elimination hal…
Vol. DistribusiThe estimated stead…
KlirensThe mean clearance …
Genetik -
Enfuvirtide Approved DB00109
biotech | CAS: 159519-65-0

Enfuvirtide is a 36 amino acid biomimetic peptide that is structurally similar to the HIV proteins that are responsible for the fusion of the virus to cell membranes and subsequent intracellular uptake. The first agent in the novel class of antiretroviral dru…

Kategori:
Amino Acids, Peptides, and ProteinsAnti-HIV AgentsAnti-Infective Agents +31
Target Protein:
Envelope glycoprotein
Waktu Paruh3.8 +/- 0.6 hrs
Vol. Distribusi* 5.5 ± 1.1 L
Klirens* 24.8 +/- 4.1 mL/h…
Genetik -
biotech | CAS: 2567881-77-8

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Engensis DB17931
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
English sole Approved DB10904
biotech

English sole allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
English walnut Approved DB10577
biotech

English walnut allergenic extract is used in allergenic testing.

Kategori:
Cell-mediated ImmunityIncreased Histamine ReleaseNon-Standardized Food Allergenic Extract
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Englitazone DB14035
small molecule | CAS: 109229-58-5

Englitazone is a hypoglycemic agent.

Kategori:
Blood Glucose Lowering AgentsHeterocyclic Compounds, Fused-RingPyrans +2
Target Protein:
Peroxisome proliferator-activated receptor gamma
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
biotech | CAS: 2417199-08-5

Englumafusp alfa is under investigation in clinical trial NCT04077723 (A Study to Evaluate the Safety, Pharmacokinetics and Preliminary Anti-tumor Activity of Englumafusp Alfa in Combination With Obinutuzumab and in Combination With Glofitamab Following a Pre…

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibarcimab DB16730
biotech | CAS: 2305638-98-4

Enibarcimab is under investigation in clinical trial NCT03989531 (Adrecizumab in Cardiogenic Shock).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +6
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enibomal DB13229
small molecule | CAS: 125-55-3

Deskripsi belum tersedia.

Kategori:
AnestheticsAnesthetics, GeneralNervous System +2
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Eniluracil DB03516
small molecule | CAS: 59989-18-3

Eniluracil, which was previously under development by GlaxoSmithKline (GSK), is being developed by Adherex to enhance the therapeutic value and effectiveness of 5-fluorouracil (5-FU), one of the world’s most widely-used oncology agents. 5-FU is widely used i…

Kategori:
Enzyme InhibitorsPyrimidinesPyrimidinones
Target Protein:
Dihydropyrimidine dehydrogenase [NADP(+)]Aldehyde oxidaseXanthine dehydrogenase/oxidase
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enisoprost DB19319
small molecule | CAS: 81026-63-3

Deskripsi belum tersedia.

Kategori:
Anti-Ulcer AgentsAutacoidsBiological Factors +11
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enitociclib DB17297
small molecule | CAS: 1610408-97-3

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-1198 DB05959
small molecule | CAS: 864668-87-1

Deskripsi belum tersedia.

Kategori:
EstranesFused-Ring CompoundsSteroids
Target Protein:
Hypoxia-inducible factor 1-alphaTumor necrosis factor receptor superfamily member 11ASignal transducer and activator of transcription 3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
ENMD-981693 DB16891
small molecule | CAS: 934353-76-1

Deskripsi belum tersedia.

Kategori:
Protein Kinase Inhibitors
Target Protein:
Aurora kinase A
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enmetazobactam Approved DB18716
small molecule | CAS: 1001404-83-6

Enmetazobactam is a penicillanic acid sulfone extended-spectrum beta (?)-lactamase (ESBL) inhibitor.[A263266] Because ESBL enzymes can hydrolyze important antibiotics such as penicillins, broad-spectrum cephalosporins and monobactams, ESBL-producing bacteria …

Kategori:
Anti-Bacterial AgentsAnti-Infective AgentsAza Compounds +7
Target Protein:
Extended-spectrum beta-lactamase PER-1Beta-lactamase
Waktu ParuhThe mean (SD) half-…
Vol. DistribusiMean (SD) steady st…
KlirensThe mean (SD) clear…
Genetik -
Enoblituzumab DB15017
biotech | CAS: 1353485-38-7

Enoblituzumab is under investigation in clinical trial NCT02982941 (Enoblituzumab (MGA271) in Children With B7-H3-expressing Solid Tumors).

Kategori:
Amino Acids, Peptides, and ProteinsAntibodies, MonoclonalAntibodies, Monoclonal, Humanized +4
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enobosarm DB12078
small molecule | CAS: 841205-47-8

Enobosarm has been used in trials studying the treatment of Stress Urinary Incontinence and Triple Negative Breast Cancer.

Kategori:
AmidesAminesAniline Compounds
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enokizumab DB05555
biotech | CAS: 909875-08-7

A humanized immunoglobulin G1k anti-interleukin-9 mAb.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesAntibodies, Monoclonal +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enoxacin Approved DB00467
small molecule | CAS: 74011-58-8

A broad-spectrum 6-fluoronaphthyridinone antibacterial agent (fluoroquinolones) structurally related to nalidixic acid.

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +14
Target Protein:
DNA topoisomerase 2-betaDNA gyrase subunit ADNA topoisomerase 4 subunit A +1
Waktu ParuhPlasma half-life is…
Vol. Distribusi-
Klirens-
Genetik -
Enoxaparin Approved DB01225
small molecule | CAS: 9005-49-6

Enoxaparin is a common low-molecular-weight heparin (LMWH) used in the prevention and management of various thromboembolic disorders. Initially approved by the FDA in 1993, it is administered by a subcutaneous or intravenous injection and marketed by several …

Kategori:
Agents causing hyperkalemiaAnticoagulantsBlood and Blood Forming Organs +7
Target Protein:
Antithrombin-IIICoagulation factor XProthrombin
Waktu ParuhThe half-life of en…
Vol. DistribusiThe volume of distr…
KlirensThe mean clearance …
Genetik -
Enoximone Approved DB04880
small molecule | CAS: 77671-31-9

Enoximone is a selective phosphodiesterase inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. It is used in patients with congestive heart failure. Trials were halted in the U.S., but the …

Kategori:
Cardiac Stimulants Excl. Cardiac GlycosidesCardiac TherapyCardiotonic Agents +10
Target Protein:
cGMP-inhibited 3',5'-cyclic phosphodiesterase 3A
Waktu Paruh4-10 hours
Vol. Distribusi-
Klirens-
Genetik -
Enoxolone DB13089
small molecule | CAS: 471-53-4

Enoxolone (glycyrrhetic acid) has been investigated for the basic science of Apparent Mineralocorticoid Excess (AME).

Kategori:
Anti-Inflammatory AgentsCicatrizantsDermatologicals +4
Target Protein:
Tyrosine-protein phosphatase non-receptor type 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enpatoran DB16501
small molecule | CAS: 2101938-42-3

Enpatoran (M5049) was under investigation in clinical trials for various conditions. It was investigated for systemic lupus erythematosus and cutaneous lupus erythematosus in completed trials (NCT04647708 and NCT05162586) and in a recruiting trial (NCT0554032…

Kategori:
Experimental Unapproved Treatments for COVID-19
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enprofylline Approved DB00824
small molecule | CAS: 41078-02-8

Enprofylline is a derivative of theophylline which shares bronchodilator properties. Enprofylline is used in asthma, chronic obstructive pulmonary disease, and in the management of cerebrovascular insufficiency, sickle cell disease, and diabetic neuropathy. L…

Kategori:
Adenosine A2 Receptor AntagonistsAlkaloidsAnti-Asthmatic Agents +11
Target Protein:
3',5'-cyclic-AMP phosphodiesterase 4B5'-nucleotidaseAdenosine receptor A2b +4
Waktu Paruh1.9 hours
Vol. Distribusi-
Klirens-
Genetik -
Enprostil DB13824
small molecule | CAS: 73121-56-9

Deskripsi belum tersedia.

Kategori:
Alimentary Tract and MetabolismAnti-Ulcer AgentsAutacoids +12
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enrasentan DB06460
small molecule | CAS: 167256-08-8

Deskripsi belum tersedia.

Kategori:
Endothelin Receptor AntagonistsIndenes
Target Protein:
Endothelin-1 receptorEndothelin receptor type B
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Enrofloxacin DB11404
small molecule | CAS: 93106-60-6

Enrofloxacin is an antibiotic agent from the fluoroquinolone family produced by the Bayer Corporation. Enrofloxacin is approved by the FDA for its veterinary use. Due to the identification of fluoroquinolone-resistant strains of _Campylobacter_, in September …

Kategori:
4-QuinolonesAnti-Bacterial AgentsAnti-Infective Agents +7
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensartinib DB14860
small molecule | CAS: 1370651-20-9

Ensartinib is under investigation in clinical trial NCT03420508 (Treating Patients With Melanoma and ALK Alterations With Ensartinib).

Kategori:
Antineoplastic AgentsEnzyme InhibitorsProtein Kinase Inhibitors
Target Protein:
ALK tyrosine kinase receptor
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensifentrine Approved DB16157
small molecule | CAS: 1884461-72-6

Ensifentrine is a first-in-class, selective dual inhibitor of the phosphodiesterase 3 (PDE3) and phosphodiesterase 4 (PDE4) enzymes.[L50903] On June 26, 2024, the FDA announced the approval of an inhaled product of ensifentrine for the treatment of chronic o…

Kategori:
BCRP/ABCG2 SubstratesCytochrome P-450 CYP2C9 SubstratesCytochrome P-450 CYP2D6 Substrates +6
Target Protein:
Phosphodiesterase 3Phosphodiesterase 4
Waktu ParuhFollowing twice-dai…
Vol. DistribusiApparent central an…
Klirens-
Genetik -
Ensitrelvir DB18834
small molecule | CAS: 2647530-73-0

Ensitrelvir is under investigation in clinical trial NCT05605093 (Strategies and Treatments for Respiratory Infections & Viral Emergencies (STRIVE): Shionogi Protease Inhibitor (Ensitrelvir)).

Kategori:
Antiinfectives for Systemic UseAntiviral AgentsAntivirals for Systemic Use +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensituximab DB12342
biotech | CAS: 1092658-06-4

Ensituximab has been used in trials studying the treatment of Pancreatic Cancer, Adult, Metastatic Colorectal Cancer, and Metastatic Pancreatic Cancer.

Kategori:
Amino Acids, Peptides, and ProteinsAntibodiesBlood Proteins +5
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensovibep DB19078
biotech | CAS: 2451126-06-8

Ensovibep is under investigation in clinical trial NCT04501978 (ACTIV-3: Therapeutics for Inpatients With COVID-19).

Kategori:
Amino Acids, Peptides, and ProteinsProteinsRecombinant Proteins
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Ensulizole Approved DB11115
small molecule | CAS: 27503-81-7

Ensulizole, also known as 2-phenylbenzimidazole-5-sulfonic acid, is a water-soluble sunscreen agent that absorbs strongly at UV-B wavelengths. It is commonly found in cosmetic products and sunscreen formulas in combination with other UV filter compounds due t…

Kategori:
AcidsAcids, NoncarboxylicHeterocyclic Compounds, Fused-Ring +3
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entacapone Approved DB00494
small molecule | CAS: 130929-57-6

Entacapone is a selective, reversible catechol-O-methyl transferase (COMT) inhibitor for the treatment of Parkinson's disease. It is a member of the class of nitrocatechols. When administered concomittantly with levodopa and a decarboxylase inhibitor (e.g., c…

Kategori:
Anti-Dyskinesia AgentsAnti-Parkinson DrugsBenzene Derivatives +11
Target Protein:
Catechol O-methyltransferase
Waktu Paruh0.4-0.7 hour
Vol. Distribusi* 20 L
Klirens* 850 mL/min
Genetik -
biotech | CAS: 2247971-01-1

Deskripsi belum tersedia.

Kategori:
Adeno-associated Viral Vector Therapies
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entecavir Approved DB00442
small molecule | CAS: 142217-69-4

Entecavir is an oral antiviral drug used in the treatment of hepatitis B infection. It is marketed under the trade name Baraclude (BMS). Entecavir is a guanine analogue that inhibits all three steps in the viral replication process, and the manufacturer cl…

Kategori:
Anti-Infective AgentsAntiinfectives for Systemic UseAntiviral Agents +12
Target Protein:
DNA
Waktu ParuhAfter reaching peak…
Vol. Distribusi-
Klirens* renal cl=383.2 +/…
Genetik -
biotech

Deskripsi belum tersedia.

Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
Entinostat DB11841
small molecule | CAS: 209783-80-2

Entinostat is under investigation for the treatment and other of Volunteers, Breast Cancer, Human Volunteers, and Normal Volunteers. Entinostat has been investigated for the treatment of Non-Small Lung Cancer, Epigenetic Therapy.

Kategori:
Acids, CarbocyclicAmidesAntineoplastic Agents +8
Target Protein:
Histone deacetylaseHistone deacetylase 1
Waktu Paruh-
Vol. Distribusi-
Klirens-
Genetik -
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